HDAC6

>Q9UBN7
MTSTGQDSTT TRQRRSRQNP QSPPQDSSVT SKRNIKKGAV PRSIPNLAEV KKKGKMKKLG
QAMEEDLIVG LQGMDLNLEA EALAGTGLVL DEQLNEFHCL WDDSFPEGPE RLHAIKEQLI
QEGLLDRCVS FQARFAEKEE LMLVHSLEYI DLMETTQYMN EGELRVLADT YDSVYLHPNS
YSCACLASGS VLRLVDAVLG AEIRNGMAII RPPGHHAQHS LMDGYCMFNH VAVAARYAQQ
KHRIRRVLIV DWDVHHGQGT QFTFDQDPSV LYFSIHRYEQ GRFWPHLKAS NWSTTGFGQG
QGYTINVPWN QVGMRDADYI AAFLHVLLPV ALEFQPQLVL VAAGFDALQG DPKGEMAATP
AGFAQLTHLL MGLAGGKLIL SLEGGYNLRA LAEGVSASLH TLLGDPCPML ESPGAPCRSA
QASVSCALEA LEPFWEVLVR STETVERDNM EEDNVEESEE EGPWEPPVLP ILTWPVLQSR
TGLVYDQNMM NHCNLWDSHH PEVPQRILRI MCRLEELGLA GRCLTLTPRP ATEAELLTCH
SAEYVGHLRA TEKMKTRELH RESSNFDSIY ICPSTFACAQ LATGAACRLV EAVLSGEVLN
GAAVVRPPGH HAEQDAACGF CFFNSVAVAA RHAQTISGHA LRILIVDWDV HHGNGTQHMF
EDDPSVLYVS LHRYDHGTFF PMGDEGASSQ IGRAAGTGFT VNVAWNGPRM GDADYLAAWH
RLVLPIAYEF NPELVLVSAG FDAARGDPLG GCQVSPEGYA HLTHLLMGLA SGRIILILEG
GYNLTSISES MAACTRSLLG DPPPLLTLPR PPLSGALASI TETIQVHRRY WRSLRVMKVE
DREGPSSSKL VTKKAPQPAK PRLAERMTTR EKKVLEAGMG KVTSASFGEE STPGQTNSET
AVVALTQDQP SEAATGGATL AQTISEAAIG GAMLGQTTSE EAVGGATPDQ TTSEETVGGA
ILDQTTSEDA VGGATLGQTT SEEAVGGATL AQTTSEAAME GATLDQTTSE EAPGGTELIQ
TPLASSTDHQ TPPTSPVQGT TPQISPSTLI GSLRTLELGS ESQGASESQA PGEENLLGEA
AGGQDMADSM LMQGSRGLTD QAIFYAVTPL PWCPHLVAVC PIPAAGLDVT QPCGDCGTIQ
ENWVCLSCYQ VYCGRYINGH MLQHHGNSGH PLVLSYIDLS AWCYYCQAYV HHQALLDVKN
IAHQNKFGED MPHPH

The same domains may appear in multiple rows, following InterPro convention.

Start	End	Type	Name	InterPro	Source
79	463	Homologous_superfamily	Histone deacetylase domain superfamily	IPR037138	G3DSA:3.40.800.20
86	417	Homologous_superfamily	Ureohydrolase domain superfamily	IPR023696	SSF52768
106	401	Domain	Histone deacetylase domain	IPR023801	PF00850
475	851	Homologous_superfamily	Histone deacetylase domain superfamily	IPR037138	G3DSA:3.40.800.20
478	834	Homologous_superfamily	Ureohydrolase domain superfamily	IPR023696	SSF52768
479	912	Family	Histone deacetylase class II, eukaryotic-type	IPR017320	PTHR45364
500	797	Domain	Histone deacetylase domain	IPR023801	PF00850
607	630	Family	Histone deacetylase family	IPR000286	PR01270
642	657	Family	Histone deacetylase family	IPR000286	PR01270
732	742	Family	Histone deacetylase family	IPR000286	PR01270
1107	1213	Homologous_superfamily	Zinc finger, RING/FYVE/PHD-type	IPR013083	G3DSA:3.30.40.10
1111	1209	Domain	Zinc finger, UBP-type	IPR001607	PS50271
1132	1181	Domain	Zinc finger, UBP-type	IPR001607	SM00290
1133	1193	Domain	Zinc finger, UBP-type	IPR001607	PF02148

GO term	Name	Ontology	Evidence	Reference
GO:0006325	chromatin organization	Biological Process	IEA	GO_REF:0000043
GO:0006950	response to stress	Biological Process	IEA	GO_REF:0000117
GO:0016236	macroautophagy	Biological Process	IEA	GO_REF:0000117
GO:0032886	regulation of microtubule-based process	Biological Process	IEA	GO_REF:0000117
GO:0051129	negative regulation of cellular component organization	Biological Process	IEA	GO_REF:0000117
GO:0051130	positive regulation of cellular component organization	Biological Process	IEA	GO_REF:0000117
GO:0051646	mitochondrion localization	Biological Process	IEA	GO_REF:0000117
GO:0065008	regulation of biological quality	Biological Process	IEA	GO_REF:0000117
GO:0098732	macromolecule deacylation	Biological Process	IEA	GO_REF:0000117
GO:0106047	polyamine deacetylation	Biological Process	IDA	PMID:28516954
GO:0106048	spermidine deacetylation	Biological Process	IDA	PMID:28516954
GO:0033148	positive regulation of intracellular estrogen receptor signaling pathway	Biological Process	IMP	PMID:18316616
GO:0000209	protein polyubiquitination	Biological Process	IEA	GO_REF:0000107
GO:0006511	ubiquitin-dependent protein catabolic process	Biological Process	IEA	GO_REF:0000107
GO:0007015	actin filament organization	Biological Process	IEA	GO_REF:0000107
GO:0007026	negative regulation of microtubule depolymerization	Biological Process	IEA	GO_REF:0000107
GO:0032984	protein-containing complex disassembly	Biological Process	IEA	GO_REF:0000107
GO:0035973	aggrephagy	Biological Process	IDA	PMID:17580304
GO:0043131	erythrocyte enucleation	Biological Process	IEA	GO_REF:0000107
GO:0043162	ubiquitin-dependent protein catabolic process via the multivesicular body sorting pathway	Biological Process	IEA	GO_REF:0000107
GO:0045598	regulation of fat cell differentiation	Biological Process	IEA	GO_REF:0000107
GO:0048668	collateral sprouting	Biological Process	IEA	GO_REF:0000107
GO:0060997	dendritic spine morphogenesis	Biological Process	IEA	GO_REF:0000107
GO:0070201	regulation of establishment of protein localization	Biological Process	IEA	GO_REF:0000107
GO:0070842	aggresome assembly	Biological Process	IEA	GO_REF:0000107
GO:0071211	protein targeting to vacuole involved in autophagy	Biological Process	IDA	PMID:37802024
GO:0071218	cellular response to misfolded protein	Biological Process	IEA	GO_REF:0000107
GO:0140694	membraneless organelle assembly	Biological Process	IDA	PMID:29343546
GO:0001975	response to amphetamine	Biological Process	IEA	GO_REF:0000107
GO:0006476	protein deacetylation	Biological Process	IDA	PMID:28516954
GO:0006515	protein quality control for misfolded or incompletely synthesized proteins	Biological Process	IMP	PMID:14675537
GO:0006886	intracellular protein transport	Biological Process	IMP	PMID:16192271
GO:0006914	autophagy	Biological Process	IEA	GO_REF:0000043
GO:0007173	epidermal growth factor receptor signaling pathway	Biological Process	IMP	PMID:18356165
GO:0010506	regulation of autophagy	Biological Process	TAS	PMID:25548531
GO:0010634	positive regulation of epithelial cell migration	Biological Process	IMP	PMID:12024216
GO:0010727	negative regulation of hydrogen peroxide metabolic process	Biological Process	IMP	PMID:18606987
GO:0010821	regulation of mitochondrion organization	Biological Process	IEA	GO_REF:0000107
GO:0010977	negative regulation of neuron projection development	Biological Process	IEA	GO_REF:0000107
GO:0016241	regulation of macroautophagy	Biological Process	IMP	PMID:16192271
GO:0019896	axonal transport of mitochondrion	Biological Process	IEA	GO_REF:0000107
GO:0030182	neuron differentiation	Biological Process	IEA	GO_REF:0000107
GO:0031333	negative regulation of protein-containing complex assembly	Biological Process	IMP	PMID:23962722
GO:0031647	regulation of protein stability	Biological Process	IMP	PMID:23580651
GO:0031648	protein destabilization	Biological Process	IEA	GO_REF:0000107
GO:0032418	lysosome localization	Biological Process	IMP	PMID:16192271
GO:0032461	positive regulation of protein oligomerization	Biological Process	IEA	GO_REF:0000107
GO:0034605	cellular response to heat	Biological Process	TAS	Reactome:R-HSA-3371511
GO:0035902	response to immobilization stress	Biological Process	IEA	GO_REF:0000107
GO:0035967	cellular response to topologically incorrect protein	Biological Process	IMP	PMID:16192271
GO:0043242	negative regulation of protein-containing complex disassembly	Biological Process	IMP	PMID:15916966
GO:0045814	negative regulation of gene expression, epigenetic	Biological Process	IMP	PMID:24413532
GO:0045861	negative regulation of proteolysis	Biological Process	IMP	PMID:18356165
GO:0045892	negative regulation of DNA-templated transcription	Biological Process	ISS	PMID:11861901
GO:0048843	negative regulation of axon extension involved in axon guidance	Biological Process	IEA	GO_REF:0000107
GO:0050775	positive regulation of dendrite morphogenesis	Biological Process	IEA	GO_REF:0000107
GO:0051412	response to corticosterone	Biological Process	IEA	GO_REF:0000107
GO:0051788	response to misfolded protein	Biological Process	IMP	PMID:14675537
GO:0051968	positive regulation of synaptic transmission, glutamatergic	Biological Process	IEA	GO_REF:0000107
GO:0060271	cilium assembly	Biological Process	TAS	Reactome:R-HSA-5617833
GO:0060632	regulation of microtubule-based movement	Biological Process	IC	PMID:19228685
GO:0060765	regulation of androgen receptor signaling pathway	Biological Process	TAS	PMID:18852123
GO:0061523	cilium disassembly	Biological Process	IMP	PMID:17604723
GO:0061734	type 2 mitophagy	Biological Process	IGI	PMID:20457763
GO:0070301	cellular response to hydrogen peroxide	Biological Process	IMP	PMID:18606987
GO:0070507	regulation of microtubule cytoskeleton organization	Biological Process	IEA	GO_REF:0000107
GO:0070845	polyubiquitinated misfolded protein transport	Biological Process	IMP	PMID:14675537
GO:0071374	cellular response to parathyroid hormone stimulus	Biological Process	IEA	GO_REF:0000107
GO:0071548	response to dexamethasone	Biological Process	IEA	GO_REF:0000107
GO:0090042	tubulin deacetylation	Biological Process	ISS	GO_REF:0000024
GO:1900409	positive regulation of cellular response to oxidative stress	Biological Process	IEA	GO_REF:0000107
GO:1903146	regulation of autophagy of mitochondrion	Biological Process	TAS	PMID:25548531
GO:1904056	positive regulation of cholangiocyte proliferation	Biological Process	IEA	GO_REF:0000107
GO:1905091	positive regulation of type 2 mitophagy	Biological Process	IEA	GO_REF:0000107
GO:1905336	negative regulation of aggrephagy	Biological Process	IDA	PMID:31857589
GO:0005634	nucleus	Cellular Component	IEA	GO_REF:0000120
GO:0005654	nucleoplasm	Cellular Component	IDA	GO_REF:0000052
GO:0005737	cytoplasm	Cellular Component	IEA	GO_REF:0000043
GO:0005813	centrosome	Cellular Component	IEA	GO_REF:0000044
GO:0005829	cytosol	Cellular Component	IDA	GO_REF:0000052
GO:0005856	cytoskeleton	Cellular Component	IEA	GO_REF:0000043
GO:0015630	microtubule cytoskeleton	Cellular Component	IEA	GO_REF:0000117
GO:0030424	axon	Cellular Component	IEA	GO_REF:0000044
GO:0030425	dendrite	Cellular Component	IEA	GO_REF:0000044
GO:0042995	cell projection	Cellular Component	IEA	GO_REF:0000043
GO:0043204	perikaryon	Cellular Component	IEA	GO_REF:0000044
GO:0120025	plasma membrane bounded cell projection	Cellular Component	IEA	GO_REF:0000117
GO:0000118	histone deacetylase complex	Cellular Component	IEA	GO_REF:0000117
GO:0005771	multivesicular body	Cellular Component	TAS	PMID:25548531
GO:0005874	microtubule	Cellular Component	IDA	PMID:12620231
GO:0005901	caveola	Cellular Component	IDA	PMID:18356165
GO:0005929	cilium	Cellular Component	IEA	GO_REF:0000044
GO:0016234	inclusion body	Cellular Component	IDA	PMID:16192271
GO:0016235	aggresome	Cellular Component	IDA	PMID:14675537
GO:0031252	cell leading edge	Cellular Component	IDA	PMID:12024216
GO:0036064	ciliary basal body	Cellular Component	IDA	PMID:17604723
GO:0043005	neuron projection	Cellular Component	IEA	GO_REF:0000107
GO:0043025	neuronal cell body	Cellular Component	IEA	GO_REF:0000107
GO:0048471	perinuclear region of cytoplasm	Cellular Component	IDA	PMID:12024216
GO:1904115	axon cytoplasm	Cellular Component	IEA	GO_REF:0000108
GO:0005875	microtubule associated complex	Cellular Component	IDA	PMID:19228685
GO:0032991	protein-containing complex	Cellular Component	IEA	GO_REF:0000107
GO:0003779	actin binding	Molecular Function	IEA	GO_REF:0000043
GO:0004407	histone deacetylase activity	Molecular Function	IEA	GO_REF:0000117
GO:0008270	zinc ion binding	Molecular Function	IEA	GO_REF:0000120
GO:0016740	transferase activity	Molecular Function	IEA	GO_REF:0000043
GO:0016787	hydrolase activity	Molecular Function	IEA	GO_REF:0000043
GO:0046872	metal ion binding	Molecular Function	IEA	GO_REF:0000043
GO:0047611	acetylspermidine deacetylase activity	Molecular Function	IDA	PMID:28516954
GO:0000978	RNA polymerase II cis-regulatory region sequence-specific DNA binding	Molecular Function	IDA	PMID:24413532
GO:0001222	transcription corepressor binding	Molecular Function	IPI	PMID:12535528
GO:0005515	protein binding	Molecular Function	IPI	PMID:16919237
GO:0008013	beta-catenin binding	Molecular Function	IPI	PMID:18356165
GO:0008017	microtubule binding	Molecular Function	ISS	GO_REF:0000024
GO:0019213	deacetylase activity	Molecular Function	IBA	GO_REF:0000033
GO:0019899	enzyme binding	Molecular Function	ISS	PMID:11861901
GO:0031593	polyubiquitin modification-dependent protein binding	Molecular Function	IDA	PMID:14675537
GO:0031625	ubiquitin protein ligase binding	Molecular Function	IPI	PMID:21753002
GO:0033558	protein lysine deacetylase activity	Molecular Function	IEA	GO_REF:0000120
GO:0036479	peroxidase inhibitor activity	Molecular Function	IMP	PMID:18606987
GO:0042030	ATPase inhibitor activity	Molecular Function	IMP	PMID:15916966
GO:0042826	histone deacetylase binding	Molecular Function	IPI	PMID:12620231
GO:0042903	tubulin deacetylase activity	Molecular Function	ISS	GO_REF:0000024
GO:0043014	alpha-tubulin binding	Molecular Function	IDA	PMID:19228685
GO:0043130	ubiquitin binding	Molecular Function	IEA	GO_REF:0000107
GO:0048156	tau protein binding	Molecular Function	IEA	GO_REF:0000107
GO:0048487	beta-tubulin binding	Molecular Function	IEA	GO_REF:0000107
GO:0051787	misfolded protein binding	Molecular Function	EXP	PMID:17785525
GO:0051879	Hsp90 protein binding	Molecular Function	IDA	PMID:15916966
GO:0070840	dynein complex binding	Molecular Function	IDA	PMID:14675537
GO:0141221	histone deacetylase activity, hydrolytic mechanism	Molecular Function	IEA	GO_REF:0000003

Substrate	Name	Known ESI (UbiBrowser)	Known ESI (UbiNet)	PPI (IntAct direct) PSI-MI score ≥ 0.5	PPI (IntAct indirect) PSI-MI scores ≥ 0.5 for both PPIs	PubMed Ref.	IntAct Ref.	Substrate Specificity

Type	ChEMBL Compound ID	Source	pChEMBL	PDB Compound ID	PDB Codes	SMILES
E3 Binder	CHEMBL5285777	ChEMBL	6.96	—	—	O=C(CCCO/N=C1C(=C2/C(=O)N(Cc3cn(CCOCCNc4cccc5c4C(=O)C(N4CCC(=O)NC4=O)C5=O)nn3)c3ccccc32)/Nc2ccccc2/1)NO
E3 Binder	CHEMBL3940017	ChEMBL	7.0	—	—	C#CCCCn1c(Sc2cccc(OCC(=O)NO)c2)nc2c(N)ncnc21
E3 Binder	CHEMBL5177240	ChEMBL	7.22	—	—	C#CCN(C)CCCOc1cc(NC(=O)CCCCCCC(=O)NO)c(Cl)cc1Cl
E3 Binder	CHEMBL5170598	ChEMBL	8.0	—	—	C#CCN(C)CCCOc1cc(NC(=O)CCCCCCC(=O)NO)ccc1Cl
E3 Binder	CHEMBL5187984	ChEMBL	7.1	—	—	C#CCN(C)CCCOc1cc(NC(=O)CCCCCCCC(=O)NO)ccc1Cl
E3 Binder	CHEMBL5200566	ChEMBL	6.8	—	—	C#CCN(C)CCCOc1cc(NC(=O)CCCCCCCCC(=O)NO)ccc1Cl
E3 Binder	CHEMBL5191350	ChEMBL	7.0	—	—	C#CCN(C)CCCOc1cc(NCc2ccc(/C=C/C(=O)NO)cc2)ccc1Cl
E3 Binder	CHEMBL5178014	ChEMBL	8.0	—	—	C#CCN(C)CCCOc1cc(NCc2ccc(C(=O)NO)cc2)ccc1Cl
E3 Binder	CHEMBL5182215	ChEMBL	8.22	—	—	C#CCN(C)CCCOc1ccc(NC(=O)CCCCCCC(=O)NO)cc1Cl
E3 Binder	CHEMBL5193384	ChEMBL	7.05	—	—	C#CCN(C)CCCOc1cccc(NC(=O)CCCCCCC(=O)NO)c1Cl
E3 Binder	CHEMBL5171489	ChEMBL	7.7	—	—	C#CCN(C)Cc1cccc(NC(=O)CCCCCCC(=O)NO)c1
E3 Binder	CHEMBL4785871	ChEMBL	7.08	—	—	C#CCn1c(=O)c(OCc2ccc(C(=O)NO)cc2)c(-c2ccccc2)c2ccccc21
E3 Binder	CHEMBL598798	ChEMBL	8.47	—	—	C#Cc1cc(Nc2ncnc3cc(OC)c(OCCCCCCC(=O)NO)cc23)ccc1F
E3 Binder	CHEMBL3704923	ChEMBL	7.47	—	—	C#Cc1ccc(CNC(=O)O[C@H]2C[C@@H](C)C=C3C=C[C@H](C)[C@H](CC[C@@H]4C[C@@H](O[Si](C)(C)C(C)(C)C)CC(=O)O4)[C@H]32)cc1
E3 Binder	CHEMBL3704922	ChEMBL	6.89	—	—	C#Cc1ccc(NC(=O)O[C@H]2C[C@@H](C)C=C3C=C[C@H](C)[C@H](CC[C@@H]4C[C@@H](O[Si](C)(C)C(C)(C)C)CC(=O)O4)[C@H]32)cc1
E3 Binder	CHEMBL2047028	ChEMBL	6.25	—	—	C#Cc1cccc(NC(=O)c2cc(NC(=O)CCCCCC(=O)NO)ccc2OC)c1
E3 Binder	CHEMBL4060174	ChEMBL	7.67	—	—	C#Cc1cccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c1
E3 Binder	CHEMBL3217996	ChEMBL	6.7	—	—	C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)cc4)ccc23)c1
E3 Binder	CHEMBL3217995	ChEMBL	6.29	—	—	C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)nc4)ccc23)c1
E3 Binder	CHEMBL3217994	ChEMBL	6.42	—	—	C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)s4)ccc23)c1
E3 Binder	CHEMBL3939206	ChEMBL	7.0	—	—	C#Cc1cccc(Nc2ncnc3cc(OC)c(NC(=O)CCCC(=O)NO)cc23)c1
E3 Binder	CHEMBL3898372	ChEMBL	7.0	—	—	C#Cc1cccc(Nc2ncnc3cc(OC)c(NC(=O)CCCCC(=O)NO)cc23)c1
E3 Binder	CHEMBL3941197	ChEMBL	7.0	—	—	C#Cc1cccc(Nc2ncnc3cc(OC)c(OCCCC(=O)NO)cc23)c1
E3 Binder	CHEMBL599398	ChEMBL	7.0	—	—	C#Cc1cccc(Nc2ncnc3cc(OC)c(OCCCCC(=O)NO)cc23)c1
E3 Binder	CHEMBL598164	ChEMBL	7.88	—	—	C#Cc1cccc(Nc2ncnc3cc(OC)c(OCCCCCC(=O)NO)cc23)c1
E3 Binder	CHEMBL598797	ChEMBL	8.36	—	—	C#Cc1cccc(Nc2ncnc3cc(OC)c(OCCCCCCC(=O)NO)cc23)c1
E3 Binder	CHEMBL598611	ChEMBL	7.47	—	—	C#Cc1cccc(Nc2ncnc3cc(OCCCCCCC(=O)NO)c(OC)cc23)c1
E3 Binder	CHEMBL3979482	ChEMBL	6.0	—	—	C#Cc1cccc(Nc2ncnc3ccc(OCCCC(=O)NO)cc23)c1
E3 Binder	CHEMBL3218000	ChEMBL	6.7	—	—	C#Cc1cccc(Nc2ncnc3ccc(OCc4ccc(C(=O)Nc5ccccc5N)cc4)cc23)c1
E3 Binder	CHEMBL3218002	ChEMBL	8.19	—	—	C#Cc1cccc(Nc2ncnc3ccc(S(=O)(=O)n4ccc(/C=C/C(=O)NO)c4)cc23)c1
E3 Binder	CHEMBL5181479	ChEMBL	6.8	—	—	C#Cc1nc(/C=C/C(=O)NO)cs1
E3 Binder	CHEMBL5170140	ChEMBL	6.8	—	—	C#Cc1nc(/C=C/C=C/C(=O)NO)cs1
E3 Binder	CHEMBL5186798	ChEMBL	8.0	—	—	C#Cc1nc(/C=C/CCCCCC(=O)NO)cs1
E3 Binder	CHEMBL5181798	ChEMBL	7.6	—	—	C#Cc1nc(/C=C\CCCCCC(=O)NO)cs1
E3 Binder	CHEMBL5209294	ChEMBL	9.0	—	—	C#Cc1nc(C(=O)NCCCCCCC(=O)NO)cs1
E3 Binder	CHEMBL5267651	ChEMBL	7.55	—	—	C/C(=C\c1ccc(C(=O)NO)cc1)CNc1cnc2c(Br)cccc2c1
E3 Binder	CHEMBL3763386	ChEMBL	7.01	—	—	C/C(=N\N(C)C(=O)c1ccc(N(C)C)cc1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3764728	ChEMBL	7.25	—	—	C/C(=N\NC(=O)c1ccc(N(C)C)cc1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4785327	ChEMBL	7.46	—	—	C/C(=N\NC(=S)NCCCCCC(=O)NO)c1ccc(Br)cc1
E3 Binder	CHEMBL4749226	ChEMBL	7.2	—	—	C/C(=N\NC(=S)NCCCCCC(=O)NO)c1ccc(F)cc1
E3 Binder	CHEMBL4791832	ChEMBL	7.42	—	—	C/C(=N\NC(=S)NCCCCCC(=O)NO)c1cccc(Br)c1
E3 Binder	CHEMBL4877805	ChEMBL	7.97	—	—	C/C(=N\O)c1ccc2c(c1)N(Cc1ccc(C(=O)NO)cc1)c1ccccc1S2
E3 Binder	CHEMBL4846564	ChEMBL	7.81	—	—	C/C(=N\O)c1ccc2c(c1)N(Cc1ccc(C(=O)NO)cc1)c1ccccc1[S+]2[O-]
E3 Binder	CHEMBL3287266	ChEMBL	6.42	—	—	C/C=C/c1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO
E3 Binder	CHEMBL3925574	ChEMBL	6.33	—	—	C/C=C/c1sc(-c2nccs2)nc1C(=O)NCCCNC(=O)CS
E3 Binder	CHEMBL146250	ChEMBL	6.83	—	—	C/C=C1\NC(=O)[C@@H](CS)NC(=O)[C@@H](C(C)C)NC(=O)C[C@@H](/C=C/CCS)OC(=O)[C@H](C(C)C)NC1=O
E3 Binder	CHEMBL4061025	ChEMBL	6.1	—	—	C/C=C1\NC(=O)[C@H](CS)NC(=O)[C@@H](C(C)C)NC(=O)C[C@@H](/C=C/CS)OC(=O)[C@H](C(C)C)NC1=O
E3 Binder	CHEMBL3310505	ChEMBL	9.0	—	—	C/C=C1\NC(=O)[C@H]2CSSCC/C=C/[C@@H](CC(=O)N[C@H](C(C)C)C(=O)N2)OC(=O)[C@H](C(C)C)NC1=O
E3 Binder	CHEMBL343448	ChEMBL	8.44	—	—	C/C=C1\NC(=O)[C@H]2CSSCC/C=C/[C@H](CC(=O)N[C@H](C(C)C)C(=O)N2)OC(=O)[C@H](C(C)C)NC1=O
E3 Binder	CHEMBL3622729	ChEMBL	6.48	—	—	C/C=C1\NC(=O)c2csc(n2)CNC(=O)C[C@@H](/C=C/CCS)OC(=O)[C@H](C(C)C)NC1=O
E3 Binder	CHEMBL5076242	ChEMBL	7.16	—	—	C/C=C1\NC(=O)c2csc(n2)CNC(=O)C[C@@H](/C=C/CCSSCCCCCCC)OC(=O)[C@H](CCCCNC(=O)CCCCC[N+]2=C(/C=C/C=C/C=C3/N(CC)c4ccc5c(S(=O)(=O)O)cc(S(=O)(=O)O)cc5c4C3(C)C)C(C)(C)c3c2ccc2c(S(=O)(=O)[O-])cc(S(=O)(=O)O)cc32)NC1=O
E3 Binder	CHEMBL3622727	ChEMBL	6.34	—	—	C/C=C1\NC(=O)c2csc(n2)[C@@H](C(C)C)NC(=O)C[C@@H](/C=C/CCS)OC(=O)[C@H](C(C)C)NC1=O
E3 Binder	CHEMBL1796688	ChEMBL	8.48	—	—	C=C(C)[C@H]1NC(=O)[C@H]2CSSCC/C=C/[C@H](CC(=O)N[C@H](C)C(=O)N2)OC(=O)C[C@@H]1O
E3 Binder	CHEMBL1808167	ChEMBL	7.05	—	—	C=CCC(/C=C/c1ccccc1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL2046608	ChEMBL	6.41	—	—	C=CCCC(=O)Nc1ccc(C(=O)N2CCc3nc(C(=O)NO)sc3C2)cc1
E3 Binder	CHEMBL3681868	ChEMBL	6.51	—	—	C=CCCCNc1cc(/C=C/C(=O)NO)ccc1SCCN(CC)CC
E3 Binder	CHEMBL4247128	ChEMBL	9.6	—	—	C=CCCn1cc(-c2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc3[nH]ccc23)cn1
E3 Binder	CHEMBL2018442	ChEMBL	9.01	—	—	C=CCN1CCc2c(c3ccccc3n2Cc2ccc(C(=O)NO)cc2)C1
E3 Binder	CHEMBL3681864	ChEMBL	6.46	—	—	C=CCNc1cc(/C=C/C(=O)NO)ccc1SCCN(CC)CC
E3 Binder	CHEMBL5289013	ChEMBL	7.59	—	—	C=CN1C(=O)CN(Cc2ccc(C(=O)NO)cc2)C(=O)C1Cc1ccccc1
E3 Binder	CHEMBL3287267	ChEMBL	6.75	—	—	C=Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO
E3 Binder	CHEMBL3959685	ChEMBL	6.16	—	—	C=Cc1sc(-c2nccs2)nc1C(=O)NCCCNC(=O)CS
E3 Binder	CHEMBL26159	ChEMBL	8.74	—	—	CC(/C=C/C(=O)NO)=C\C(C)C(=O)c1ccc(N(C)C)cc1
E3 Binder	CHEMBL99	ChEMBL	9.89	TSN	—	CC(/C=C/C(=O)NO)=C\[C@@H](C)C(=O)c1ccc(N(C)C)cc1
E3 Binder	CHEMBL1164992	ChEMBL	6.24	—	—	CC(/C=C/C(=O)NO)=C\[C@@H](C)[C@H]1CC[C@H]2/C(=C/C=C3\C[C@@H](O)C[C@@H](O)C3)CCC[C@]12C
E3 Binder	CHEMBL164868	ChEMBL	7.66	E1Z	—	CC(/C=C/C(=O)NO)=C\[C@H](C)C(=O)c1ccc(N(C)C)cc1
E3 Binder	CHEMBL81522	ChEMBL	6.52	—	—	CC(/C=C/C(=O)NO)=C\c1ccc(Cl)cc1
E3 Binder	CHEMBL82989	ChEMBL	6.1	—	—	CC(/C=C/C(=O)NO)=C\c1ccc(N(C)C)cc1
E3 Binder	CHEMBL316183	ChEMBL	7.31	—	—	CC(/C=C/C(=O)NO)=C\c1ccc(NS(=O)(=O)c2ccc(Cl)cc2)cc1
E3 Binder	CHEMBL4744603	ChEMBL	6.32	—	—	CC(/C=C/C(=O)NO)=C\c1ccc(NS(=O)(=O)c2ccc(N(CCCl)CCCl)cc2)cc1
E3 Binder	CHEMBL314643	ChEMBL	6.76	—	—	CC(/C=C/C(=O)NO)=C\c1ccc(NS(=O)(=O)c2ccccc2)cc1
E3 Binder	CHEMBL490018	ChEMBL	8.46	—	—	CC(/C=C/c1ccccc1)=C\C(=O)NCCCCCC(=O)NO
E3 Binder	CHEMBL595908	ChEMBL	8.77	—	—	CC(/C=C/c1ccccc1)N1CCN(c2ncc(C(=O)NO)cn2)CC1
E3 Binder	CHEMBL1807693	ChEMBL	7.21	—	—	CC(/C=C/c1ccccc1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL217651	ChEMBL	7.89	—	—	CC(=O)CCCCC[C@H](NC(=O)C1CCCCN1C)C(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL468513	ChEMBL	8.0	—	—	CC(=O)CCCCC[C@H](NC(=O)C1CCN(C)CC1)c1ncc(-c2ccc3ccccc3c2)[nH]1
E3 Binder	CHEMBL272401	ChEMBL	7.89	—	—	CC(=O)CCCCC[C@H](NC1CCCCN1C)C(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL4565296	ChEMBL	7.15	—	—	CC(=O)N(Cc1ccc(C(C)(C)C)cc1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4639051	ChEMBL	6.93	—	—	CC(=O)N(Cc1cccc(C(F)(F)F)c1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3693751	ChEMBL	7.6	—	—	CC(=O)N(c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1)c1c(C)cccc1C
E3 Binder	CHEMBL3693742	ChEMBL	7.66	—	—	CC(=O)N(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1c(C)cccc1C
E3 Binder	CHEMBL3693750	ChEMBL	7.43	—	—	CC(=O)N(c1ccccc1)c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693730	ChEMBL	8.52	—	—	CC(=O)N(c1ccccc1)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3759970	ChEMBL	6.31	—	—	CC(=O)N1CC2(CC(=O)c3cc(/C=C/C(=O)NO)ccc3O2)C1
E3 Binder	CHEMBL3916917	ChEMBL	8.23	—	—	CC(=O)N1CCC(Nc2ncc(C(=O)NO)cn2)(C(C)C)CC1
E3 Binder	CHEMBL3929319	ChEMBL	8.8	—	—	CC(=O)N1CCC(Nc2ncc(C(=O)NO)cn2)(c2ccccc2)CC1
E3 Binder	CHEMBL3759596	ChEMBL	6.02	—	—	CC(=O)N1CCC2(CC(=O)c3cc(/C=C/C(=O)NO)ccc3O2)C1
E3 Binder	CHEMBL1938431	ChEMBL	6.19	—	—	CC(=O)N1CCC2(CC1)CC(=O)c1cc(/C=C/C(=O)NO)ccc1O2
E3 Binder	CHEMBL4295221	ChEMBL	7.2	—	—	CC(=O)N1CCC2(CC1)CN(Cc1ccc(C(=O)NO)cc1)c1ccccc12
E3 Binder	CHEMBL3758807	ChEMBL	6.68	—	—	CC(=O)N1CCCC2(CC(=O)c3cc(/C=C/C(=O)NO)ccc3O2)C1
E3 Binder	CHEMBL3759508	ChEMBL	6.49	—	—	CC(=O)N1CCCC2(CC1)CC(=O)c1cc(/C=C/C(=O)NO)ccc1O2
E3 Binder	CHEMBL4562244	ChEMBL	7.1	—	—	CC(=O)N1CCc2c(c3ccccc3n2Cc2ccc(C(=O)NO)cc2)C1
E3 Binder	CHEMBL3220922	ChEMBL	6.63	—	—	CC(=O)N1c2ccc(-c3ccc(NC(=O)CCCCCCC(=O)NO)cc3)cc2[C@H](NC(=O)OC(C)C)C[C@@H]1C
E3 Binder	CHEMBL3220925	ChEMBL	6.01	—	—	CC(=O)N1c2ccc(NC(=O)CCCCCCC(=O)NO)cc2[C@H](Nc2ccccc2)C[C@@H]1C
E3 Binder	CHEMBL569174	ChEMBL	7.77	—	—	CC(=O)NCCCCC[C@@H]1NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2cccc3ccccc23)NC(=O)[C@H](CCCCCC(=O)O)NC1=O
E3 Binder	CHEMBL3936740	ChEMBL	7.33	—	—	CC(=O)NCCCc1nc2ccccc2n1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5271183	ChEMBL	6.51	—	—	CC(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H]1CC[S+](C)Cc2cccc(c2)C[S+](C)CC[C@@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CC(C)C)C(=O)NCCCCCC(=O)NO)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(=N)N)NC1=O
E3 Binder	CHEMBL468842	ChEMBL	8.17	—	—	CC(=O)Nc1ccc(-c2cc(C(=O)NCCCCCCC(=O)NO)no2)cc1
E3 Binder	CHEMBL5274303	ChEMBL	7.7	—	—	CC(=O)Nc1ccc(-c2ccnc(NCc3ccc(OCCCCCC(=O)NO)cc3)n2)cc1
E3 Binder	CHEMBL4282471	ChEMBL	6.93	—	—	CC(=O)Nc1ccc(-c2ccnc(Nc3ccc(NC(=O)CCCCC(=O)NO)cc3)n2)cc1.O=C(O)C(F)(F)F
E3 Binder	CHEMBL4290831	ChEMBL	10.0	—	—	CC(=O)Nc1ccc(-c2ccnc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)n2)cc1.Cl
E3 Binder	CHEMBL4290748	ChEMBL	8.89	—	—	CC(=O)Nc1ccc(-c2ccnc(Nc3ccc(OCCCCCC(=O)NO)cc3)n2)cc1.Cl
E3 Binder	CHEMBL4283921	ChEMBL	8.52	—	—	CC(=O)Nc1ccc(-c2ccnc(Nc3ccc(OCCCCCCC(=O)NO)cc3)n2)cc1.Cl
E3 Binder	CHEMBL4291781	ChEMBL	7.85	—	—	CC(=O)Nc1ccc(-c2ccnc(Nc3ccc(OCCCCCCCC(=O)NO)cc3)n2)cc1.Cl
E3 Binder	CHEMBL4284388	ChEMBL	8.34	—	—	CC(=O)Nc1ccc(-c2ccnc(Nc3cccc(NC(=O)CCCCC(=O)NO)c3)n2)cc1.O=C(O)C(F)(F)F
E3 Binder	CHEMBL4282456	ChEMBL	9.09	—	—	CC(=O)Nc1ccc(-c2ccnc(Nc3cccc(NC(=O)CCCCCCC(=O)NO)c3)n2)cc1.Cl
E3 Binder	CHEMBL4280540	ChEMBL	8.62	—	—	CC(=O)Nc1ccc(-c2ccnc(Nc3cccc(OCCCCCC(=O)NO)c3)n2)cc1
E3 Binder	CHEMBL4294153	ChEMBL	8.74	—	—	CC(=O)Nc1ccc(-c2ccnc(Nc3cccc(OCCCCCCC(=O)NO)c3)n2)cc1
E3 Binder	CHEMBL4278591	ChEMBL	8.17	—	—	CC(=O)Nc1ccc(-c2ccnc(Nc3cccc(OCCCCCCCC(=O)NO)c3)n2)cc1.Cl
E3 Binder	CHEMBL4280050	ChEMBL	8.46	—	—	CC(=O)Nc1ccc(-c2nc(Nc3ccc(OCCCCCC(=O)NO)cc3)ncc2C)cc1
E3 Binder	CHEMBL4295224	ChEMBL	8.21	—	—	CC(=O)Nc1ccc(-c2nc(Nc3cccc(OCCCCCCC(=O)NO)c3)ncc2C)cc1
E3 Binder	CHEMBL4290689	ChEMBL	8.01	—	—	CC(=O)Nc1ccc(-c2nc(Nc3cccc(OCCCCCCCC(=O)NO)c3)ncc2C)cc1
E3 Binder	CHEMBL4448978	ChEMBL	6.79	—	—	CC(=O)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4862508	ChEMBL	7.24	—	—	CC(=O)Nc1ccc(C(=O)NO)cc1F
E3 Binder	CHEMBL235842	ChEMBL	6.69	20Y	—	CC(=O)Nc1ccc(C(=O)Nc2cc(-c3cccs3)ccc2N)cc1
E3 Binder	CHEMBL250397	ChEMBL	6.09	—	—	CC(=O)Nc1ccc(CN2CCC=C(CCC(=O)NO)C2=O)cc1
E3 Binder	CHEMBL1401	ChEMBL	6.0	NTI	—	CC(=O)Oc1ccccc1C(=O)Nc1ncc([N+](=O)[O-])s1
E3 Binder	CHEMBL272613	ChEMBL	7.09	—	—	CC(=O)SCC(=O)CCCCCCC(=O)Nc1ccccc1
E3 Binder	CHEMBL454749	ChEMBL	7.0	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(C)cc2)cc1
E3 Binder	CHEMBL480560	ChEMBL	6.38	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(Cl)c(Cl)c2)cc1
E3 Binder	CHEMBL480562	ChEMBL	6.55	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(Cl)cc2)cc1
E3 Binder	CHEMBL521243	ChEMBL	6.02	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1
E3 Binder	CHEMBL480589	ChEMBL	6.7	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OC(F)(F)F)cc2)cc1
E3 Binder	CHEMBL527425	ChEMBL	6.96	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OC3CCCN(C)C3)cc2)nc1
E3 Binder	CHEMBL488585	ChEMBL	7.36	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OC3CCN(C)CC3)cc2)nc1
E3 Binder	CHEMBL487966	ChEMBL	7.54	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OCCCCN(C)C)cc2)nc1
E3 Binder	CHEMBL488583	ChEMBL	7.6	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OCCCN(C)C)cc2)nc1
E3 Binder	CHEMBL488167	ChEMBL	7.21	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OCCCN3CCCC3)cc2)nc1
E3 Binder	CHEMBL519901	ChEMBL	7.28	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OCCCN3CCCCC3)cc2)nc1
E3 Binder	CHEMBL487354	ChEMBL	7.17	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OCCCN3CCOCC3)cc2)nc1
E3 Binder	CHEMBL487180	ChEMBL	6.96	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OCCCO)cc2)nc1
E3 Binder	CHEMBL528766	ChEMBL	6.66	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OCCCc3ccccn3)cc2)nc1
E3 Binder	CHEMBL487181	ChEMBL	7.03	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OCCN(C)C)cc2)nc1
E3 Binder	CHEMBL488169	ChEMBL	6.72	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OCCc3ccccn3)cc2)nc1
E3 Binder	CHEMBL519262	ChEMBL	6.66	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(OCc3ccccn3)cc2)nc1
E3 Binder	CHEMBL514325	ChEMBL	7.23	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3[nH]ccc3c2)cc1
E3 Binder	CHEMBL474428	ChEMBL	6.8	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)CCN3)cc1
E3 Binder	CHEMBL475624	ChEMBL	7.09	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)CCO3)cc1
E3 Binder	CHEMBL473821	ChEMBL	7.02	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)CCO3)nc1
E3 Binder	CHEMBL487965	ChEMBL	7.42	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)COOC3)nc1
E3 Binder	CHEMBL473616	ChEMBL	7.04	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)N(C(C)=O)CC3)cc1
E3 Binder	CHEMBL473615	ChEMBL	7.33	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)NCC3)cc1
E3 Binder	CHEMBL514179	ChEMBL	7.0	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)OCCN3C)cc1
E3 Binder	CHEMBL515103	ChEMBL	6.82	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)OCCN3C)nc1
E3 Binder	CHEMBL515291	ChEMBL	7.58	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)OCCO3)cc1
E3 Binder	CHEMBL475468	ChEMBL	7.06	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)OCO3)cc1
E3 Binder	CHEMBL474987	ChEMBL	6.44	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)OCO3)nc1
E3 Binder	CHEMBL455757	ChEMBL	7.42	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)ncn3C)cc1
E3 Binder	CHEMBL473820	ChEMBL	6.62	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3c(c2)ncn3C)nc1
E3 Binder	CHEMBL475788	ChEMBL	7.36	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3cc[nH]c3c2)cc1
E3 Binder	CHEMBL474427	ChEMBL	7.54	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3ccccc3c2)cc1
E3 Binder	CHEMBL475631	ChEMBL	7.38	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccc3ccccc3c2)nc1
E3 Binder	CHEMBL482346	ChEMBL	6.82	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2cccc(Cl)c2)cc1
E3 Binder	CHEMBL480561	ChEMBL	6.34	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2cccc(F)c2)cc1
E3 Binder	CHEMBL480588	ChEMBL	6.1	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2cccc(OC(F)(F)F)c2)cc1
E3 Binder	CHEMBL520079	ChEMBL	6.48	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccccc2)cc1
E3 Binder	CHEMBL475469	ChEMBL	6.82	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccccc2)nc1
E3 Binder	CHEMBL482345	ChEMBL	6.07	—	—	CC(=O)SCC(=O)c1ccc(NS(=O)(=O)c2ccccc2Cl)cc1
E3 Binder	CHEMBL482165	ChEMBL	6.0	—	—	CC(=O)SCC(=O)c1ccc(S(=O)(=O)Nc2ccc(OC(F)(F)F)cc2)cc1
E3 Binder	CHEMBL235300	ChEMBL	6.62	—	—	CC(=O)SCC/C=C/[C@@H]1CC(=O)N[C@H](C)C(=O)N[C@H](C)C(=O)N[C@H](C(C)C)C(=O)NCC(=O)O1
E3 Binder	CHEMBL4551751	ChEMBL	7.47	—	—	CC(=O)SCCCCCC(NC(=O)OCc1ccccc1)C(=O)Nc1cccc2cccnc12
E3 Binder	CHEMBL3356948	ChEMBL	7.51	—	—	CC(=O)SCCCCC[C@H](NC(=O)[C@@H]1CC(=O)N1)C(=O)Nc1ccccc1
E3 Binder	CHEMBL3356940	ChEMBL	7.0	—	—	CC(=O)SCCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)Nc1ccccc1
E3 Binder	CHEMBL3353926	ChEMBL	8.3	—	—	CC(=O)SCCCCC[C@H](NC(=O)[C@H]1CCC(=O)N1)C(=O)Nc1ccccc1
E3 Binder	CHEMBL570589	ChEMBL	7.54	—	—	CC(=O)c1ccc(-c2ccc(C(=O)C(F)(F)F)s2)cc1
E3 Binder	CHEMBL15870	ChEMBL	6.29	—	—	CC(C(=O)O)c1ccc(N2Cc3ccccc3C2=O)cc1
E3 Binder	CHEMBL190727	ChEMBL	7.01	—	—	CC(C)(C(=O)Nc1ccc(C(=O)NO)cc1)c1ccccc1
E3 Binder	CHEMBL1808163	ChEMBL	7.75	—	—	CC(C)(C)C(/C=C/c1ccccc1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL4290685	ChEMBL	7.22	—	—	CC(C)(C)C(=O)N1CCC2(CC1)CN(Cc1ccc(C(=O)NO)cc1)c1ccccc12
E3 Binder	CHEMBL2431913	ChEMBL	6.31	—	—	CC(C)(C)C(=O)N1CCCc2cc(C(=O)NO)ccc2C1
E3 Binder	CHEMBL2431902	ChEMBL	7.28	—	—	CC(C)(C)C(=O)N1CCc2cc(C(=O)NO)ccc2C1
E3 Binder	CHEMBL2431917	ChEMBL	7.46	—	—	CC(C)(C)C(=O)N1CCc2cc(C(=O)NO)sc2C1
E3 Binder	CHEMBL2431909	ChEMBL	6.92	—	—	CC(C)(C)C(=O)N1CCc2ccc(C(=O)NO)cc2CC1
E3 Binder	CHEMBL2431920	ChEMBL	7.33	—	—	CC(C)(C)C(=O)N1CCc2sc(C(=O)NO)cc2C1
E3 Binder	CHEMBL2431907	ChEMBL	7.05	—	—	CC(C)(C)C(=O)N1Cc2ccc(C(=O)NO)cc2C1
E3 Binder	CHEMBL2431863	ChEMBL	7.1	—	—	CC(C)(C)C(=O)NCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5204510	ChEMBL	7.57	—	—	CC(C)(C)NC(=O)CN(Cc1ccc(C(=O)NO)cc1F)C(=O)c1ccccc1C(F)(F)F
E3 Binder	CHEMBL5197066	ChEMBL	7.68	—	—	CC(C)(C)NC(=O)CN(Cc1ccc(C(=O)NO)cc1F)C(=O)c1ccccc1Cl
E3 Binder	CHEMBL5189667	ChEMBL	7.58	—	—	CC(C)(C)NC(=O)CN(Cc1ccc(C(=O)NO)cc1F)C(=O)c1ccccc1F
E3 Binder	CHEMBL4227494	ChEMBL	6.78	—	—	CC(C)(C)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)/C=C/c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4559559	ChEMBL	7.55	—	—	CC(C)(C)OC(=O)N(Cc1ccc(C(C)(C)C)cc1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4291778	ChEMBL	7.38	—	—	CC(C)(C)OC(=O)N1CCC2(CC1)CN(Cc1ccc(C(=O)NO)cc1)c1ccccc12
E3 Binder	CHEMBL4294088	ChEMBL	6.14	—	—	CC(C)(C)OC(=O)N1CCC2(CC1)CN(Cc1ccc(C(=O)NO)s1)c1ccccc12
E3 Binder	CHEMBL5267454	ChEMBL	6.82	—	—	CC(C)(C)OC(=O)N1CCC2(CC1)c1ccccc1N(Cc1ccc(C(=O)NO)cc1)C2c1cccnc1
E3 Binder	CHEMBL2018303	ChEMBL	8.65	—	—	CC(C)(C)OC(=O)N1CCc2c(c3ccccc3n2Cc2ccc(C(=O)NO)cc2)C1
E3 Binder	CHEMBL3233683	ChEMBL	7.01	—	—	CC(C)(C)OC(=O)NCC(=O)N[C@H](COc1ccc(/C=C/C(=O)NO)cc1)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL3354907	ChEMBL	6.05	—	—	CC(C)(C)OC(=O)NCC(=O)N[C@H](COc1cccc(/C=C/C(=O)NO)c1)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL480729	ChEMBL	7.4	—	—	CC(C)(C)OC(=O)NCCCC[C@@H]1C(=O)Nc2ccccc2N1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4534503	ChEMBL	7.1	—	—	CC(C)(C)OC(=O)NCc1cn(Cc2ccc(C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL3968356	ChEMBL	6.25	—	—	CC(C)(C)OC(=O)NCc1nc(-c2nc(C(=O)NCCCCCC(=O)NO)cs2)cs1
E3 Binder	CHEMBL1289931	ChEMBL	7.58	—	—	CC(C)(C)OC(=O)N[C@@H](CCCCCC(=O)NO)C(=O)NC1CCCC1
E3 Binder	CHEMBL1289498	ChEMBL	6.62	—	—	CC(C)(C)OC(=O)N[C@@H](CCCCCO)C(=O)NC1CCCC1
E3 Binder	CHEMBL213934	ChEMBL	7.54	—	—	CC(C)(C)OC(=O)N[C@@H](CCCCCS)C(=O)NC1CCCC1
E3 Binder	CHEMBL209551	ChEMBL	7.44	—	—	CC(C)(C)OC(=O)N[C@@H](CCCCCS)C(=O)NC1CCCCC1
E3 Binder	CHEMBL379049	ChEMBL	7.64	—	—	CC(C)(C)OC(=O)N[C@@H](CCCCCS)C(=O)NC1CCCCCC1
E3 Binder	CHEMBL3233685	ChEMBL	7.01	—	—	CC(C)(C)OC(=O)N[C@H](CO)C(=O)N[C@H](COc1ccc(/C=C/C(=O)NO)cc1)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL3233681	ChEMBL	6.28	—	—	CC(C)(C)OC(=O)N[C@H](COc1ccc(/C=C/C(=O)NO)cc1)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL3354906	ChEMBL	6.04	—	—	CC(C)(C)OC(=O)N[C@H](COc1cccc(/C=C/C(=O)NO)c1)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL467792	ChEMBL	7.5	—	—	CC(C)(C)OC(=O)Nc1ccc(-c2cc(C(=O)NCCCCC(=O)NO)no2)cc1
E3 Binder	CHEMBL511749	ChEMBL	9.49	—	—	CC(C)(C)OC(=O)Nc1ccc(-c2cc(C(=O)NCCCCCCC(=O)NO)no2)cc1
E3 Binder	CHEMBL4554511	ChEMBL	8.22	—	—	CC(C)(C)OC(=O)Nc1ccc(-c2cc(C(=O)NCCc3cc(C(=O)NO)no3)no2)cc1
E3 Binder	CHEMBL4126811	ChEMBL	9.48	—	—	CC(C)(C)OC(=O)Nc1ccc(-c2cc(C(=O)NCc3ccc(C(=O)NO)cc3)no2)cc1
E3 Binder	CHEMBL5093602	ChEMBL	7.17	—	—	CC(C)(C)OC(=O)Nc1ccc(-c2ncc(C(=O)NCCCCCCC(=O)NO)s2)cc1
E3 Binder	CHEMBL469275	ChEMBL	8.4	—	—	CC(C)(C)OC(=O)Nc1cccc(-c2cc(C(=O)NCCCCC(=O)NO)no2)c1
E3 Binder	CHEMBL5173000	ChEMBL	8.11	—	—	CC(C)(C)OC(=O)Nc1cccc(-c2cc(C(=O)NCCc3cc(C(=O)NO)no3)no2)c1
E3 Binder	CHEMBL4542499	ChEMBL	8.0	—	—	CC(C)(C)OC(=O)Nc1cccc(C(=O)/C=C/c2ccc(/C=C/C(=O)NO)cc2)c1
E3 Binder	CHEMBL521431	ChEMBL	7.3	—	—	CC(C)(C)Oc1ccc(C[C@@H]2C(=O)Nc3ccccc3N2Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL244811	ChEMBL	6.9	—	—	CC(C)(C)SC(=S)SCC(=O)c1ccc(Cl)c(Cl)c1
E3 Binder	CHEMBL1093335	ChEMBL	6.96	—	—	CC(C)(C)c1[nH]c2ccccc2c1[C@@H]1CCCN(Cc2ccc(/C=C/C(=O)NO)cc2F)C1
E3 Binder	CHEMBL1093033	ChEMBL	6.93	—	—	CC(C)(C)c1[nH]c2ccccc2c1[C@H]1CCCN(Cc2ccc(/C=C/C(=O)NO)cc2F)C1
E3 Binder	CHEMBL4645307	ChEMBL	6.03	—	—	CC(C)(C)c1cc(C(=O)NOCCCCCC(=O)NO)cc(C(C)(C)C)c1
E3 Binder	CHEMBL4637127	ChEMBL	6.72	—	—	CC(C)(C)c1cc(C(=O)Nc2ccc(C(=O)NO)cc2)cc(C(C)(C)C)c1
E3 Binder	CHEMBL4646090	ChEMBL	6.12	—	—	CC(C)(C)c1cc(CN(C(=O)c2cccc(C(F)(F)F)c2)c2ccc(C(=O)NO)cc2)cc(C(C)(C)C)c1
E3 Binder	CHEMBL474991	ChEMBL	6.28	—	—	CC(C)(C)c1ccc(-c2nc3c(N4CCN(Cc5ccc6nccnc6c5)CC4)cccc3[nH]2)cc1
E3 Binder	CHEMBL4303368	ChEMBL	6.53	—	—	CC(C)(C)c1ccc(-c2nc3ccccc3[nH]2)cc1
E3 Binder	CHEMBL4755326	ChEMBL	7.68	—	—	CC(C)(C)c1ccc(C(=O)N(Cc2ccc(C(=O)NO)cc2)C2CC2)cc1
E3 Binder	CHEMBL4799423	ChEMBL	7.49	—	—	CC(C)(C)c1ccc(C(=O)NCc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4452620	ChEMBL	7.62	—	—	CC(C)(C)c1ccc(C(=O)Nc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4755724	ChEMBL	7.89	—	—	CC(C)(C)c1ccc(CC(=O)Nc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4855750	ChEMBL	6.94	—	—	CC(C)(C)c1ccc(CC2(c3ccccc3)NC(=O)N(Cc3ccc(C(=O)NO)cc3)C2=O)cc1
E3 Binder	CHEMBL3427663	ChEMBL	6.42	—	—	CC(C)(C)c1ccc(CCCn2cccc(/C=C/C(=O)NO)c2=O)cc1
E3 Binder	CHEMBL3427652	ChEMBL	6.96	—	—	CC(C)(C)c1ccc(CCn2cccc(/C=C/C(=O)NO)c2=O)cc1
E3 Binder	CHEMBL4520400	ChEMBL	6.72	—	—	CC(C)(C)c1ccc(CN(C(=O)CN(Cc2c(F)c(F)c(F)c(F)c2F)S(=O)(=O)c2ccc(F)cc2)c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4437895	ChEMBL	7.56	—	—	CC(C)(C)c1ccc(CN(C(=O)CN(Cc2c(F)c(F)c(F)c(F)c2F)S(C)(=O)=O)c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4534860	ChEMBL	6.44	—	—	CC(C)(C)c1ccc(CN(C(=O)CN(Cc2ccccc2C(F)(F)F)S(=O)(=O)c2ccc(F)c(F)c2)c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4546897	ChEMBL	6.64	—	—	CC(C)(C)c1ccc(CN(C(=O)CN(Cc2ccccc2C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4580317	ChEMBL	6.54	—	—	CC(C)(C)c1ccc(CN(C(=O)CN(Cc2ccccc2C(F)(F)F)S(=O)(=O)c2ccc(F)cc2F)c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4560533	ChEMBL	7.28	—	—	CC(C)(C)c1ccc(CN(C(=O)CNS(=O)(=O)c2ccc(F)cc2)c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL5085755	ChEMBL	7.38	—	—	CC(C)(C)c1ccc(CN(Cc2ccc(C(=O)NO)cc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL4868120	ChEMBL	6.86	—	—	CC(C)(C)c1ccc(CN2C(=O)N(Cc3ccc(C(=O)NO)cc3)C(=O)C2Cc2ccccc2)cc1
E3 Binder	CHEMBL4853389	ChEMBL	7.39	—	—	CC(C)(C)c1ccc(CN2CC(=O)N(Cc3ccc(C(=O)NO)cc3)C2=O)cc1
E3 Binder	CHEMBL247218	ChEMBL	6.0	—	—	CC(C)(C)c1ccc(CN2Cc3ccc(/C=C/C(=O)NO)cc3C2=O)cc1
E3 Binder	CHEMBL4472310	ChEMBL	6.96	—	—	CC(C)(C)c1ccc(CNc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL5269353	ChEMBL	6.73	—	—	CC(C)(C)c1ccc(COc2cccc3ccc(C(=O)NCCCCCC(=O)NO)nc23)cc1
E3 Binder	CHEMBL3427642	ChEMBL	7.05	—	—	CC(C)(C)c1ccc(Cn2cccc(/C=C/C(=O)NO)c2=O)cc1
E3 Binder	CHEMBL4742241	ChEMBL	7.98	—	—	CC(C)(C)c1ccc(NC(=O)c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4760053	ChEMBL	7.76	—	—	CC(C)(C)c1ccc(NS(=O)(=O)c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4758855	ChEMBL	7.38	—	—	CC(C)(C)c1ccc(S(=O)(=O)NCc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4798826	ChEMBL	8.7	—	—	CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4638377	ChEMBL	7.18	—	—	CC(C)(C)c1cccc(C(=O)Nc2ccc(C(=O)NO)cc2)c1
E3 Binder	CHEMBL4639383	ChEMBL	6.38	—	—	CC(C)(C)c1cccc(NC(=O)c2ccc(C(=O)NO)cc2)c1
E3 Binder	CHEMBL4082059	ChEMBL	7.25	—	—	CC(C)(C)c1cccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c1
E3 Binder	CHEMBL3899708	ChEMBL	6.0	—	—	CC(C)(C)c1cnc(CSc2cnc(NC(=O)C3CCN(CCCCC(=O)NO)CC3)s2)o1
E3 Binder	CHEMBL3931285	ChEMBL	6.0	—	—	CC(C)(C)c1cnc(CSc2cnc(NC(=O)C3CCN(CCCCCC(=O)NO)CC3)s2)o1
E3 Binder	CHEMBL3912995	ChEMBL	7.0	—	—	CC(C)(C)c1cnc(CSc2cnc(NC(=O)C3CCN(CCCCCCC(=O)NO)CC3)s2)o1
E3 Binder	CHEMBL3922737	ChEMBL	7.0	—	—	CC(C)(C)c1cnc(CSc2cnc(NC(=O)CCCC(=O)NO)s2)o1
E3 Binder	CHEMBL3957562	ChEMBL	7.0	—	—	CC(C)(C)c1cnc(CSc2cnc(NC(=O)CCCCC(=O)NO)s2)o1
E3 Binder	CHEMBL3913135	ChEMBL	7.0	—	—	CC(C)(C)c1cnc(CSc2cnc(NC(=O)CCCCCCC(=O)NO)s2)o1
E3 Binder	CHEMBL3944861	ChEMBL	7.0	—	—	CC(C)(C)c1cnc(CSc2cnc(NC(=O)Cc3ccc(OCCCC(=O)NO)cc3)s2)o1
E3 Binder	CHEMBL3982819	ChEMBL	7.0	—	—	CC(C)(C)c1cnc(CSc2cnc(NC(=O)Cc3ccc(OCCCCC(=O)NO)cc3)s2)o1
E3 Binder	CHEMBL475862	ChEMBL	6.08	—	—	CC(C)(C)c1csc(NC(=O)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc2ccccc2)n1
E3 Binder	CHEMBL4754795	ChEMBL	6.48	—	—	CC(C)(C)n1nnnc1CNCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4241370	ChEMBL	6.89	—	—	CC(C)(CCCCC(=O)NO)Nc1c(Nc2ccc(C(F)(F)F)cc2)c(=O)c1=O
E3 Binder	CHEMBL189137	ChEMBL	7.6	—	—	CC(C)(CCc1ccccc1)C(=O)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5091589	ChEMBL	6.76	—	—	CC(C)(F)CN1CCc2cc(O)ccc2C1c1ccc(OC2CN(CC(=O)NO)C2)cc1
E3 Binder	CHEMBL5078131	ChEMBL	7.18	—	—	CC(C)(F)CN1CCc2cc(O)ccc2C1c1ccc(OCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL5090940	ChEMBL	7.2	—	—	CC(C)(F)CN1CCc2cc(O)ccc2C1c1ccc(OCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL4539071	ChEMBL	6.83	—	—	CC(C)(NC(=O)c1nc(-c2nccs2)sc1C1CC1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4762877	ChEMBL	9.19	—	—	CC(C)(Nc1ncc(C(=O)NO)cc1F)c1ccccc1
E3 Binder	CHEMBL4777764	ChEMBL	9.22	—	—	CC(C)(Nc1ncc(C(=O)NO)cc1F)c1ccccn1
E3 Binder	CHEMBL3655969	ChEMBL	7.48	—	—	CC(C)(Nc1ncc(C(=O)NO)cn1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1
E3 Binder	CHEMBL3655951	ChEMBL	8.22	—	—	CC(C)(Nc1ncc(C(=O)NO)cn1)c1ccc(C(F)(F)F)cc1
E3 Binder	CHEMBL3655963	ChEMBL	7.89	—	—	CC(C)(Nc1ncc(C(=O)NO)cn1)c1ccc(C(F)(F)F)cc1F
E3 Binder	CHEMBL3655957	ChEMBL	8.7	—	—	CC(C)(Nc1ncc(C(=O)NO)cn1)c1ccc(Cl)c(Cl)c1
E3 Binder	CHEMBL3655960	ChEMBL	8.52	—	—	CC(C)(Nc1ncc(C(=O)NO)cn1)c1ccc(Cl)cc1F
E3 Binder	CHEMBL3655953	ChEMBL	8.4	—	—	CC(C)(Nc1ncc(C(=O)NO)cn1)c1ccc(F)c(F)c1
E3 Binder	CHEMBL3639548	ChEMBL	8.52	—	—	CC(C)(Nc1ncc(C(=O)NO)cn1)c1ccc(F)cc1
E3 Binder	CHEMBL3655947	ChEMBL	8.52	—	—	CC(C)(Nc1ncc(C(=O)NO)cn1)c1ccc(F)cc1F
E3 Binder	CHEMBL3655952	ChEMBL	8.52	—	—	CC(C)(Nc1ncc(C(=O)NO)cn1)c1cccc(F)c1
E3 Binder	CHEMBL3655933	ChEMBL	8.4	—	—	CC(C)(Nc1ncc(C(=O)NO)cn1)c1ccccc1
E3 Binder	CHEMBL3655948	ChEMBL	8.7	—	—	CC(C)(Nc1ncc(C(=O)NO)cn1)c1ccccc1F
E3 Binder	CHEMBL3287268	ChEMBL	6.78	—	—	CC(C)/C=C/c1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO
E3 Binder	CHEMBL3953198	ChEMBL	6.67	—	—	CC(C)/C=C/c1sc(-c2nccs2)nc1C(=O)NCCCNC(=O)CS
E3 Binder	CHEMBL3287264	ChEMBL	6.75	—	—	CC(C)=Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO
E3 Binder	CHEMBL3984885	ChEMBL	6.74	—	—	CC(C)=Cc1sc(-c2nccs2)nc1C(=O)NCCCNC(=O)CS
E3 Binder	CHEMBL1808162	ChEMBL	7.66	—	—	CC(C)C(/C=C/c1ccccc1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL3693752	ChEMBL	7.17	—	—	CC(C)C(=O)N(c1ccccc1)c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL191091	ChEMBL	7.52	—	—	CC(C)C(C(=O)Nc1ccc(C(=O)NO)cc1)c1ccccc1
E3 Binder	CHEMBL3953441	ChEMBL	6.91	—	—	CC(C)C(c1ccc(C(=O)NO)cc1)C(C)C
E3 Binder	CHEMBL2036475	ChEMBL	7.64	—	—	CC(C)C(c1nc2ccccc2o1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL2036476	ChEMBL	8.3	—	—	CC(C)C(c1nc2ccccc2s1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL3891741	ChEMBL	8.29	—	—	CC(C)C1(Nc2ncc(C(=O)NO)cn2)CCN(C(=O)OCc2ccccc2)CC1
E3 Binder	CHEMBL3287269	ChEMBL	6.73	—	—	CC(C)C1CC1c1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO
E3 Binder	CHEMBL1808164	ChEMBL	6.08	—	—	CC(C)CC(/C=C/c1ccccc1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL2036479	ChEMBL	7.72	—	—	CC(C)CC(c1nc2ccccc2o1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL4868785	ChEMBL	6.6	—	—	CC(C)CC1C(=O)N(Cc2ccc(C(=O)NO)cc2)C(=O)N1C
E3 Binder	CHEMBL4875843	ChEMBL	6.89	—	—	CC(C)CC1C(=O)N(Cc2ccc(C(=O)NO)cc2)C(=O)N1Cc1ccccc1
E3 Binder	CHEMBL4170617	ChEMBL	9.19	—	—	CC(C)CCN(CCCCCCC(=O)NO)c1ncc(C(=O)NCCCn2ccnc2)s1
E3 Binder	CHEMBL4282004	ChEMBL	7.62	—	—	CC(C)CCN1CC(=O)N2Cc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)CC2C1=O
E3 Binder	CHEMBL1822040	ChEMBL	6.37	—	—	CC(C)CCc1c(OCCCCC(=O)NO)ccc(CCC(=O)NO)c1O
E3 Binder	CHEMBL1822048	ChEMBL	6.15	—	—	CC(C)CCc1c(OCCCCC(=O)NO)ccc2c1OC(=O)CC2
E3 Binder	CHEMBL1822044	ChEMBL	6.28	—	—	CC(C)CCc1c(OCCCCC(=O)NO)ccc2ccc(=O)oc12
E3 Binder	CHEMBL1822041	ChEMBL	6.68	—	—	CC(C)CCc1c(OCCCCCC(=O)NO)ccc(CCC(=O)NO)c1O
E3 Binder	CHEMBL1822049	ChEMBL	6.37	—	—	CC(C)CCc1c(OCCCCCC(=O)NO)ccc2c1OC(=O)CC2
E3 Binder	CHEMBL1822045	ChEMBL	6.89	—	—	CC(C)CCc1c(OCCCCCC(=O)NO)ccc2ccc(=O)oc12
E3 Binder	CHEMBL1822042	ChEMBL	7.8	—	—	CC(C)CCc1c(OCCCCCCC(=O)NO)ccc(CCC(=O)NO)c1O
E3 Binder	CHEMBL1822050	ChEMBL	7.62	—	—	CC(C)CCc1c(OCCCCCCC(=O)NO)ccc2c1OC(=O)CC2
E3 Binder	CHEMBL1822046	ChEMBL	7.82	—	—	CC(C)CCc1c(OCCCCCCC(=O)NO)ccc2ccc(=O)oc12
E3 Binder	CHEMBL1822043	ChEMBL	7.85	—	—	CC(C)CCc1c(OCCCCCCCC(=O)NO)ccc(CCC(=O)NO)c1O
E3 Binder	CHEMBL1822051	ChEMBL	6.95	—	—	CC(C)CCc1c(OCCCCCCCC(=O)NO)ccc2c1OC(=O)CC2
E3 Binder	CHEMBL1822047	ChEMBL	7.41	—	—	CC(C)CCc1c(OCCCCCCCC(=O)NO)ccc2ccc(=O)oc12
E3 Binder	CHEMBL4518616	ChEMBL	7.08	—	—	CC(C)CCc1c(OCCCCOc2ccc(/C=C/C(=O)NO)cc2)ccc2c1OC(=O)CC2
E3 Binder	CHEMBL4451082	ChEMBL	7.92	—	—	CC(C)CCc1c(OCCCOc2cccc(/C=C/C(=O)NO)c2)ccc2c1OC(=O)CC2
E3 Binder	CHEMBL4468518	ChEMBL	7.25	—	—	CC(C)CCc1c(OCCOc2ccc(/C=C/C(=O)NO)cc2)ccc2c1OC(=O)CC2
E3 Binder	CHEMBL4456028	ChEMBL	8.2	—	—	CC(C)CCc1c(OCCOc2cccc(/C=C/C(=O)NO)c2)ccc2c1OC(=O)CC2
E3 Binder	CHEMBL3601774	ChEMBL	7.27	—	—	CC(C)CCn1ccc2ccc(NC(=O)CCCCCCC(=O)NO)cc2c1=O
E3 Binder	CHEMBL4174193	ChEMBL	7.92	—	—	CC(C)CN(Cc1ccc(C(=O)NO)cc1)C(=O)Nc1ccccc1
E3 Binder	CHEMBL5202595	ChEMBL	7.61	—	—	CC(C)CN(Cc1ccc(C(=O)NO)cc1)S(=O)(=O)c1cc(F)c(F)c(F)c1F
E3 Binder	CHEMBL4284297	ChEMBL	8.42	—	—	CC(C)CN1CC(=O)N2Cc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)CC2C1=O
E3 Binder	CHEMBL4518933	ChEMBL	6.82	—	—	CC(C)CNC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4225960	ChEMBL	6.51	—	—	CC(C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)/C=C/c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4113844	ChEMBL	7.92	—	—	CC(C)C[C@@H](C(=O)N1CCC(Nc2ncc(C(=O)NO)cn2)(c2ccccc2)CC1)c1ccccc1
E3 Binder	CHEMBL318616	ChEMBL	6.19	—	—	CC(C)C[C@@H]1CC(=O)N([C@@H](CC2CCCCC2)C(=O)NCCCCCC(=O)NO)C1=O
E3 Binder	CHEMBL98748	ChEMBL	7.0	—	—	CC(C)C[C@@H]1CC(=O)N([C@@H](Cc2ccccc2)C(=O)NCCCCCC(=O)NO)C1=O
E3 Binder	CHEMBL253309	ChEMBL	6.64	—	—	CC(C)C[C@@H]1NC(=O)C(C)(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
E3 Binder	CHEMBL3907413	ChEMBL	7.96	—	—	CC(C)C[C@H](C(=O)N1CCC(Nc2ncc(C(=O)NO)cn2)(c2ccccc2)CC1)c1ccccc1
E3 Binder	CHEMBL4576202	ChEMBL	6.89	—	—	CC(C)C[C@H](NC(=O)CNC(=O)c1cccc(/C=C/C(=O)NO)c1)B1O[C@@H]2[C@@H]3C[C@H](C[C@]2(C)O1)C3(C)C
E3 Binder	CHEMBL4459294	ChEMBL	6.5	A6I	—	CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)C(=O)NCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL317734	ChEMBL	7.18	—	—	CC(C)C[C@H]1C(=O)N([C@@H](Cc2ccccc2)C(=O)NCCCCCC(=O)NO)C(=O)C12CCCC2
E3 Binder	CHEMBL329977	ChEMBL	7.42	—	—	CC(C)C[C@H]1C(=O)N2C[C@@H]1CCCCCOc1ccc(cc1)C[C@H]2C(=O)NCCCCCC(=O)NO
E3 Binder	CHEMBL569446	ChEMBL	6.3	—	—	CC(C)C[C@H]1CC(=O)NC(C)(C)C(=O)N[C@@H](CCCCCC(=O)O)C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N1
E3 Binder	CHEMBL585939	ChEMBL	8.52	—	—	CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(=O)NO)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1
E3 Binder	CHEMBL570490	ChEMBL	6.49	—	—	CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(=O)O)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1
E3 Binder	CHEMBL570041	ChEMBL	6.69	—	—	CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(=O)O)C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N1
E3 Binder	CHEMBL570419	ChEMBL	6.27	—	—	CC(C)C[C@H]1CC(=O)N[C@@H](C)C(=O)N[C@@H](CCCCCC(=O)O)C(=O)N[C@@H](Cc2ccccc2)C(=O)N1
E3 Binder	CHEMBL566637	ChEMBL	7.16	—	—	CC(C)C[C@H]1CC(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](CCCCCC(=O)NO)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N1
E3 Binder	CHEMBL569211	ChEMBL	6.6	—	—	CC(C)C[C@H]1CC(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](CCCCCC(=O)O)C(=O)N[C@@H](Cc2cccc3ccccc23)C(=O)N1
E3 Binder	CHEMBL95881	ChEMBL	8.68	—	—	CC(C)C[C@H]1CN[C@H](C(=O)NCCCCCC(=O)NO)Cc2ccc(cc2)OCCCCC[C@H]1C(=O)OC(C)(C)C
E3 Binder	CHEMBL5270345	ChEMBL	8.22	—	—	CC(C)Cc1c(OCCOc2cccc(/C=C/C(=O)NO)c2)ccc2c1OC(=O)CC2
E3 Binder	CHEMBL3771366	ChEMBL	7.05	—	—	CC(C)Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)C(F)(F)F
E3 Binder	CHEMBL3287250	ChEMBL	6.91	—	—	CC(C)Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO
E3 Binder	CHEMBL3939120	ChEMBL	6.3	—	—	CC(C)Cc1sc(-c2nccs2)nc1C(=O)NCCCCCC(=O)NO
E3 Binder	CHEMBL3933626	ChEMBL	6.24	—	—	CC(C)Cc1sc(-c2nccs2)nc1C(=O)NCCCCCCCC(=O)NO
E3 Binder	CHEMBL3947538	ChEMBL	6.72	—	—	CC(C)Cc1sc(-c2nccs2)nc1C(=O)NCCCCCNC(=O)CS
E3 Binder	CHEMBL3971832	ChEMBL	6.06	—	—	CC(C)Cc1sc(-c2nccs2)nc1C(=O)NCCCCNC(=O)CS
E3 Binder	CHEMBL3968415	ChEMBL	7.06	—	—	CC(C)Cc1sc(-c2nccs2)nc1C(=O)NCCCNC(=O)CS
E3 Binder	CHEMBL4535745	ChEMBL	6.51	—	—	CC(C)Cc1sc(-c2nccs2)nc1C(=O)Nc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL3935445	ChEMBL	6.53	—	—	CC(C)Cc1sc(-c2nccs2)nc1C(=O)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3891163	ChEMBL	6.52	—	—	CC(C)Cc1sc(-c2nccs2)nc1C(=O)Nc1cccc(/C=C/C(=O)NO)c1
E3 Binder	CHEMBL142992	ChEMBL	7.64	—	—	CC(C)N(CCc1c[nH]c2ccccc12)Cc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL1096022	ChEMBL	7.0	—	—	CC(C)N(CCn1c(-c2cccc(/C=C/C(=O)NO)c2)nc2ccccc21)C(C)C
E3 Binder	CHEMBL4763401	ChEMBL	7.85	—	—	CC(C)N(Cc1ccc(C(=O)NO)cc1)C(=O)c1c(F)c(F)c(F)c(F)c1F
E3 Binder	CHEMBL3899275	ChEMBL	6.91	—	—	CC(C)N(Cc1ccc(C(=O)NO)cc1)C(C)C
E3 Binder	CHEMBL5173782	ChEMBL	7.79	—	—	CC(C)N(Cc1ccc(C(=O)NO)cc1)Cc1cc(F)c(F)c(F)c1F
E3 Binder	CHEMBL5179295	ChEMBL	8.4	—	—	CC(C)N(Cc1ccc(C(=O)NO)cc1)S(=O)(=O)c1c(F)c(F)c(F)c(F)c1F
E3 Binder	CHEMBL5177475	ChEMBL	8.39	O2L	—	CC(C)N(Cc1ccc(C(=O)NO)cc1)S(=O)(=O)c1cc(F)c(F)c(F)c1F
E3 Binder	CHEMBL5195141	ChEMBL	6.92	—	—	CC(C)N(Cc1ccc(C(=O)NO)cn1)S(=O)(=O)c1cc(F)c(F)c(F)c1F
E3 Binder	CHEMBL5184540	ChEMBL	6.84	—	—	CC(C)N(Cc1ccc(CC(=O)NO)cc1)S(=O)(=O)c1cc(F)c(F)c(F)c1F
E3 Binder	CHEMBL2413318	ChEMBL	6.75	—	—	CC(C)N(Cc1ccccc1)Cc1ccc(/C=C/C(=O)NO)o1
E3 Binder	CHEMBL3601341	ChEMBL	7.6	—	—	CC(C)N1CCN(c2nccc3ccc(NC(=O)CCCCCCC(=O)NO)cc23)CC1
E3 Binder	CHEMBL2018441	ChEMBL	8.05	—	—	CC(C)N1CCc2c(c3ccccc3n2Cc2ccc(C(=O)NO)cc2)C1
E3 Binder	CHEMBL2385381	ChEMBL	6.67	—	—	CC(C)Nc1nc2c(s1)Cc1cc(/C=C/C(=O)NO)ccc1-2
E3 Binder	CHEMBL515408	ChEMBL	6.17	—	—	CC(C)Nc1nc2cc(Cl)c(Cl)cc2n1[C@H]1O[C@@H](CO)[C@H](O)[C@@H]1O
E3 Binder	CHEMBL4166504	ChEMBL	7.28	—	—	CC(C)OC(=O)N(CCc1ccccc1)Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4755061	ChEMBL	8.27	—	—	CC(C)Oc1ccc(C(C)(C)O)cc1-c1cn(C)c(=O)c2[nH]c(C(=O)NCCCCCCC(=O)NO)cc12
E3 Binder	CHEMBL4753908	ChEMBL	7.28	—	—	CC(C)Oc1ccc(C(C)(C)O)cc1-c1cn(C)c(=O)c2[nH]c(C(=O)NCc3ccc(C(=O)NO)cc3)cc12
E3 Binder	CHEMBL165790	ChEMBL	6.04	—	—	CC(C)Oc1ccc2c(=O)c(-c3ccccc3)coc2c1
E3 Binder	CHEMBL4208584	ChEMBL	7.11	—	—	CC(C)Oc1cccc(-c2ccc3c(NC(=O)c4ccc(C(=O)NO)cc4)n[nH]c3c2)c1
E3 Binder	CHEMBL4849606	ChEMBL	8.17	—	—	CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(C(=O)NCCCCCCC(=O)NO)cc2)ncc1Cl
E3 Binder	CHEMBL4855319	ChEMBL	8.36	—	—	CC(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)ncc1Cl
E3 Binder	CHEMBL242684	ChEMBL	7.0	—	—	CC(C)SC(=S)SCC(=O)c1ccc(Cl)c(Cl)c1
E3 Binder	CHEMBL4649745	ChEMBL	6.38	—	—	CC(C)[C@@H](C#Cc1ccc(C(=O)NO)cc1)NC(=O)C1Cc2ccccc2O1
E3 Binder	CHEMBL4106624	ChEMBL	7.89	—	—	CC(C)[C@@H](C(=O)N1CCC(Nc2ncc(C(=O)NO)cn2)(c2ccccc2)CC1)c1ccccc1
E3 Binder	CHEMBL191483	ChEMBL	7.08	—	—	CC(C)[C@@H](C(=O)Nc1ccc(C(=O)NO)cc1)c1ccccc1
E3 Binder	CHEMBL2036482	ChEMBL	8.15	—	—	CC(C)[C@@H](c1nc2ccccc2o1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL4111331	ChEMBL	7.65	—	—	CC(C)[C@@H]1C(=O)N(c2ccccc2)C(=O)N1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3593409	ChEMBL	7.31	—	—	CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2cccc(n2)CNC(=O)C[C@@H](/C=C/CCS)OC1=O
E3 Binder	CHEMBL3593411	ChEMBL	7.45	—	—	CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2ccnc(c2)CNC(=O)C[C@@H](/C=C/CCS)OC1=O
E3 Binder	CHEMBL2436595	ChEMBL	7.01	—	—	CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2coc(n2)CNC(=O)C[C@@H](/C=C/CCS)OC1=O
E3 Binder	CHEMBL2436596	ChEMBL	7.3	—	—	CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2coc(n2)CNC(=O)C[C@@H](/C=C/CCSSCC/C=C/[C@@H]2CC(=O)NCc3nc(co3)C3=N[C@@](C)(CS3)C(=O)N[C@@H](C(C)C)C(=O)O2)OC1=O
E3 Binder	CHEMBL4099942	ChEMBL	6.22	—	—	CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(n2)CNC(=O)C[C@@H](/C=C/CCC(=O)NO)OC1=O
E3 Binder	CHEMBL3593407	ChEMBL	6.99	L6G	—	CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(n2)CNC(=O)C[C@@H](/C=C/CCS)NC1=O
E3 Binder	CHEMBL3593247	ChEMBL	7.55	—	—	CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(n2)CNC(=O)C[C@@H](/C=C/CCS)OC1=O
E3 Binder	CHEMBL3329621	ChEMBL	7.21	—	—	CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(n2)CNC(=O)C[C@@H](/C=C/CCSSCC/C=C/[C@@H]2CC(=O)NCc3nc(cs3)C3=N[C@@](C)(CS3)C(=O)N[C@@H](C(C)C)C(=O)O2)OC1=O
E3 Binder	CHEMBL3329622	ChEMBL	6.87	—	—	CC(C)[C@@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(n2)CNC(=O)C[C@@H](/C=C/CCSSC[C@H](NC(=O)OC(C)(C)C)C(=O)OC(C)(C)C)OC1=O
E3 Binder	CHEMBL3916246	ChEMBL	8.3	—	—	CC(C)[C@H](C(=O)N1CCC(Nc2ncc(C(=O)NO)cn2)(c2ccccc2)CC1)c1ccccc1
E3 Binder	CHEMBL191482	ChEMBL	8.18	QCP	—	CC(C)[C@H](C(=O)Nc1ccc(C(=O)NO)cc1)c1ccccc1
E3 Binder	CHEMBL573899	ChEMBL	6.24	—	—	CC(C)[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)CC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)CNC(=O)CCCc1cn(-c2ccc(-c3cn(CCCCCC(=O)NO)nn3)cc2)nn1)C(=O)NCC(=O)NCC(N)=O
E3 Binder	CHEMBL582926	ChEMBL	6.14	—	—	CC(C)[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)CC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)CNC(=O)CCCc1cn(-c2ccc(-c3cn(CCCCCCC(=O)NO)nn3)cc2)nn1)C(=O)NCC(=O)NCC(N)=O
E3 Binder	CHEMBL573900	ChEMBL	6.15	—	—	CC(C)[C@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)CC(=O)[C@H](CCCCN)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)CNC(=O)CCCc1cn(-c2ccc(-c3cn(CCCCCCCC(=O)NO)nn3)cc2)nn1)C(=O)NCC(=O)NCC(N)=O
E3 Binder	CHEMBL4538450	ChEMBL	7.85	—	—	CC(C)[C@H](NC(=O)c1nc(-c2nccs2)sc1C1CC1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL2036469	ChEMBL	7.51	—	—	CC(C)[C@H](c1nc2ccccc2o1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL235082	ChEMBL	8.14	—	—	CC(C)[C@H]1NC(=O)C[C@H]2/C=C/CCSSC[C@@H](NC1=O)C(=O)N[C@H](C(C)C)C(=O)NCC(=O)O2
E3 Binder	CHEMBL393361	ChEMBL	8.15	—	—	CC(C)[C@H]1NC(=O)[C@@H](C)NC(=O)[C@@H](C)NC(=O)C[C@@H](/C=C/CCS)OC(=O)CNC1=O
E3 Binder	CHEMBL255714	ChEMBL	7.35	—	—	CC(C)[C@H]1NC(=O)[C@@H](C)[C@@H](C/C=C\CCC(N)=O)NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@@H](C)NC1=O
E3 Binder	CHEMBL393360	ChEMBL	7.82	—	—	CC(C)[C@H]1NC(=O)[C@H]2CSSCC/C=C/[C@H](CC(=O)N[C@H](C)C(=O)N2)OC(=O)CNC1=O
E3 Binder	CHEMBL1796689	ChEMBL	7.46	—	—	CC(C)[C@H]1NC(=O)[C@]2(C)CSC(=N2)c2csc(n2)CNC(=O)C[C@@H](/C=C/CCS)OC1=O
E3 Binder	CHEMBL2347008	ChEMBL	7.08	—	—	CC(C)c1c(C(=O)Nc2ccccc2)c(-c2ccccc2)c(-c2ccc(F)cc2)n1CC[C@@H](O)C[C@@H](O)CC(=O)NO
E3 Binder	CHEMBL3235118	ChEMBL	7.92	—	—	CC(C)c1cc(-n2nnc(C(=O)NCCCCCCC(=O)NO)c2-c2ccc(CN3CCOCC3)cc2)c(O)cc1O
E3 Binder	CHEMBL5174143	ChEMBL	6.97	—	—	CC(C)c1cc(C(=O)N(C)Cc2ccc(C(=O)NO)cc2)c(O)cc1O
E3 Binder	CHEMBL4514330	ChEMBL	7.4	—	—	CC(C)c1cc(C(=O)N(C)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c(O)cc1O
E3 Binder	CHEMBL4448385	ChEMBL	6.5	—	—	CC(C)c1cc(C(=O)N(C)c2ccc(NC(=O)CCCCCCCC(=O)NO)cc2)c(O)cc1O
E3 Binder	CHEMBL4241177	ChEMBL	6.06	—	—	CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCC(=O)NO)ccc32)c(O)cc1O
E3 Binder	CHEMBL4237454	ChEMBL	7.06	—	—	CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCCC(=O)NO)ccc32)c(O)cc1O
E3 Binder	CHEMBL4241615	ChEMBL	7.21	—	—	CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCCCC(=O)NO)ccc32)c(O)cc1O
E3 Binder	CHEMBL4247905	ChEMBL	6.76	—	—	CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCCCCC(=O)NO)ccc32)c(O)cc1O
E3 Binder	CHEMBL4237899	ChEMBL	6.98	—	—	CC(C)c1cc(C(=O)N2CCc3cc(NC(=O)CCCCCCCCC(=O)NO)ccc32)c(O)cc1O
E3 Binder	CHEMBL3233755	ChEMBL	8.39	—	—	CC(C)c1cc(C(=O)N2CCc3onc(C(=O)NCCCCCCC(=O)NO)c3C2)c(O)cc1O
E3 Binder	CHEMBL4747757	ChEMBL	6.52	—	—	CC(C)c1cc(C(=O)N2Cc3ccc(/C=C/C(=O)NO)cc3C2)c(O)cc1O
E3 Binder	CHEMBL4740842	ChEMBL	7.16	—	—	CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCC(=O)NO)cc3C2)c(O)cc1O
E3 Binder	CHEMBL4741850	ChEMBL	6.48	—	—	CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCC(=O)NO)cc3C2)c(O)cc1O
E3 Binder	CHEMBL4798549	ChEMBL	8.03	—	—	CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCCC(=O)NO)cc3C2)c(O)cc1O
E3 Binder	CHEMBL4790559	ChEMBL	6.66	—	—	CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCCCC(=O)NO)cc3C2)c(O)cc1O
E3 Binder	CHEMBL4790152	ChEMBL	8.67	—	—	CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCCCCC(=O)NO)cc3C2)c(O)cc1O
E3 Binder	CHEMBL4789155	ChEMBL	6.41	—	—	CC(C)c1cc(C(=O)N2Cc3ccc(NC(=O)CCCCCCCCC(=O)NO)cc3C2)c(O)cc1O
E3 Binder	CHEMBL4782478	ChEMBL	7.48	—	—	CC(C)c1cc(C(=O)N2Cc3ccc(NCc4ccc(C(=O)NO)cc4)cc3C2)c(O)cc1O
E3 Binder	CHEMBL4862927	ChEMBL	6.6	—	—	CC(C)c1ccc(C(=O)N(CC(=O)NC23CC4CC(CC(C4)C2)C3)Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4858841	ChEMBL	6.57	—	—	CC(C)c1ccc(C(=O)N(Cc2ccc(C(=O)NO)cc2)C(C)(C)C(=O)NC2CCCCC2)cc1
E3 Binder	CHEMBL4878499	ChEMBL	7.22	—	—	CC(C)c1ccc(C(=O)N(Cc2ccc(C(=O)NO)cc2)C(C)(C)C(=O)NCc2ccccc2)cc1
E3 Binder	CHEMBL4761974	ChEMBL	6.5	—	—	CC(C)c1ccc(C(=O)N(Cc2ccc(C(=O)NO)cc2)Cc2nnnn2Cc2ccccc2)cc1
E3 Binder	CHEMBL2312163	ChEMBL	6.3	—	—	CC(C)c1ccc(C(=O)NOCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL5279301	ChEMBL	6.7	—	—	CC(C)c1ccc(C(C)c2nnc(NC(=O)CCC(=O)NO)s2)cc1
E3 Binder	CHEMBL4548143	ChEMBL	6.68	—	—	CC(C)c1ccc(C/C(=N\O)C(=O)NCCSSCCNC(=O)/C(Cc2ccc(C(C)C)cc2)=N/O)cc1
E3 Binder	CHEMBL4873978	ChEMBL	7.4	—	—	CC(C)c1ccc(CC(=O)N(CC(=O)NC2CCCCC2)Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4873872	ChEMBL	7.7	—	—	CC(C)c1ccc(CC(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4090841	ChEMBL	7.44	—	—	CC(C)c1ccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)cc1
E3 Binder	CHEMBL1909943	ChEMBL	6.27	—	—	CC(C)c1ccc(S(=O)(=O)N2CCC(CCCC(=O)NO)CC2)cc1
E3 Binder	CHEMBL3693707	ChEMBL	7.35	—	—	CC(C)c1cccc(C(C)C)c1N(C)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693761	ChEMBL	6.96	—	—	CC(C)c1cccc(C(C)C)c1Nc1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693709	ChEMBL	7.7	—	—	CC(C)c1cccc(C(C)C)c1Nc1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693771	ChEMBL	7.29	—	—	CC(C)c1cccc(C(C)C)c1Nc1ncc(C(=O)N(C)CCCCCCC(=O)NO)cn1
E3 Binder	CHEMBL4068828	ChEMBL	7.45	—	—	CC(C)c1cccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c1
E3 Binder	CHEMBL5170634	ChEMBL	7.38	—	—	CC(C)c1ccccc1C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(C(=O)NO)cc1F
E3 Binder	CHEMBL3693718	ChEMBL	7.3	—	—	CC(C)c1ccccc1N(C)c1ncc(C(=O)N(C)CCCCCCC(=O)NO)cn1
E3 Binder	CHEMBL3693710	ChEMBL	8.15	—	—	CC(C)c1ccccc1N(C)c1ncc(C(=O)NCCCCCCC(=O)NO)cn1
E3 Binder	CHEMBL2347009	ChEMBL	6.88	—	—	CC(C)c1nc(N(C)S(C)(=O)=O)nc(-c2ccc(F)cc2)c1/C=C/[C@@H](O)C[C@@H](O)CC(=O)NO
E3 Binder	CHEMBL2425964	ChEMBL	7.89	—	—	CC(C)c1nc2cc(/C=C/C(=O)NO)ccc2c(=O)n1CCc1ccccc1
E3 Binder	CHEMBL3926575	ChEMBL	7.33	—	—	CC(C)c1nc2ccccc2n1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL1097017	ChEMBL	7.0	—	—	CC(C)n1c(-c2cccc(/C=C/C(=O)NO)c2)nc2ccccc21
E3 Binder	CHEMBL5268599	ChEMBL	6.56	—	—	CC(C)n1cnc2c(-c3ccc(COCC(=O)NO)cc3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5291062	ChEMBL	6.56	—	—	CC(C)n1cnc2c(-c3ccc(COCCCCC(=O)NO)cc3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5290191	ChEMBL	6.56	—	—	CC(C)n1cnc2c(-c3ccc(COCCCCCC(=O)NO)cc3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5266821	ChEMBL	6.56	—	—	CC(C)n1cnc2c(-c3ccc(COCCCCCCC(=O)NO)cc3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5266294	ChEMBL	6.56	—	—	CC(C)n1cnc2c(-c3ccc(COCCCCCCCC(=O)NO)cc3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5265991	ChEMBL	6.56	—	—	CC(C)n1cnc2c(-c3ccc(OCC(=O)NO)cc3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5269926	ChEMBL	6.56	—	—	CC(C)n1cnc2c(-c3ccc(OCCCCC(=O)NO)cc3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5280085	ChEMBL	6.56	—	—	CC(C)n1cnc2c(-c3ccc(OCCCCCC(=O)NO)cc3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5278900	ChEMBL	6.56	—	—	CC(C)n1cnc2c(-c3ccc(OCCCCCCC(=O)NO)cc3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5285774	ChEMBL	6.56	—	—	CC(C)n1cnc2c(-c3ccc(OCCCCCCCC(=O)NO)cc3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5285531	ChEMBL	7.46	—	—	CC(C)n1cnc2c(-c3cccc(COCC(=O)NO)c3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5284588	ChEMBL	7.46	—	—	CC(C)n1cnc2c(-c3cccc(COCCCCC(=O)NO)c3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5287278	ChEMBL	7.46	—	—	CC(C)n1cnc2c(-c3cccc(COCCCCCC(=O)NO)c3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5278517	ChEMBL	7.46	—	—	CC(C)n1cnc2c(-c3cccc(COCCCCCCC(=O)NO)c3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5266822	ChEMBL	7.46	—	—	CC(C)n1cnc2c(-c3cccc(COCCCCCCCC(=O)NO)c3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5270770	ChEMBL	7.46	—	—	CC(C)n1cnc2c(-c3cccc(OCC(=O)NO)c3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5201623	ChEMBL	7.62	—	—	CC(C)n1cnc2c(-c3cccc(OCCCC(=O)NO)c3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5290567	ChEMBL	7.46	—	—	CC(C)n1cnc2c(-c3cccc(OCCCCC(=O)NO)c3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5277242	ChEMBL	7.46	—	—	CC(C)n1cnc2c(-c3cccc(OCCCCCC(=O)NO)c3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5287597	ChEMBL	7.46	—	—	CC(C)n1cnc2c(-c3cccc(OCCCCCCC(=O)NO)c3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL5281219	ChEMBL	7.46	—	—	CC(C)n1cnc2c(-c3cccc(OCCCCCCCC(=O)NO)c3)nc(N3CCOCC3)nc21
E3 Binder	CHEMBL2204667	ChEMBL	6.46	—	—	CC(CCCCC(=O)NO)CC(=O)Nc1ccccc1
E3 Binder	CHEMBL1835673	ChEMBL	6.46	—	—	CC(CCCCC(=O)Nc1ccccc1)CC(=O)NO
E3 Binder	CHEMBL4095596	ChEMBL	9.0	—	—	CC(CCCCCC(=O)NO)n1cc(-c2ncnc3[nH]ccc23)cn1
E3 Binder	CHEMBL4549965	ChEMBL	6.55	—	—	CC(CNC(=O)c1ccc(/C=C/C(=O)NO)cc1)Oc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
E3 Binder	CHEMBL140088	ChEMBL	7.62	—	—	CC(Cc1c[nH]c2ccccc12)NCc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL3354908	ChEMBL	6.07	—	—	CC(NC(=O)OC(C)(C)C)C(=O)N[C@H](COc1cccc(/C=C/C(=O)NO)c1)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL485967	ChEMBL	6.44	—	—	CC(NC(=O)c1ccc(C(=O)C(F)(F)F)s1)c1cccc2ccccc12
E3 Binder	CHEMBL485968	ChEMBL	6.58	—	—	CC(NC(=O)c1ccc(C(=O)C(F)(F)F)s1)c1ccncc1
E3 Binder	CHEMBL4527843	ChEMBL	7.38	—	—	CC(NC(=O)c1nc(-c2nccs2)sc1C1CC1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL140566	ChEMBL	7.64	—	—	CC(NCCc1c[nH]c2ccccc12)c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4244764	ChEMBL	6.89	—	—	CC(Nc1c(NCCCCCC(=O)NO)c(=O)c1=O)C12CC3CC(CC(C3)C1)C2
E3 Binder	CHEMBL3655973	ChEMBL	8.05	—	—	CC(Nc1ncc(C(=O)NO)cn1)(c1ccc(F)cc1)c1ccc(F)cc1
E3 Binder	CHEMBL3655956	ChEMBL	8.22	—	—	CC(Nc1ncc(C(=O)NO)cn1)(c1ccccc1)c1ccccc1
E3 Binder	CHEMBL3655915	ChEMBL	8.7	—	—	CC(Nc1ncc(C(=O)NO)cn1)c1ccccc1
E3 Binder	CHEMBL3655962	ChEMBL	8.4	—	—	CC(Nc1ncc(C(=O)NO)cn1)c1ccncc1
E3 Binder	CHEMBL3693808	ChEMBL	8.15	—	—	CC(O)(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1ccccn1
E3 Binder	CHEMBL3693798	ChEMBL	8.52	—	—	CC(O)(c1ccc(F)cc1)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3233686	ChEMBL	7.07	—	—	CC(O)[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](COc1ccc(/C=C/C(=O)NO)cc1)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL4281611	ChEMBL	6.06	—	—	CC(c1ccc(C(=O)NO)cc1)n1[se]c2ccccc2c1=O
E3 Binder	CHEMBL2036474	ChEMBL	7.07	—	—	CC(c1nc2ccccc2o1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL4248952	ChEMBL	6.29	—	—	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C)cc1)c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4240593	ChEMBL	6.32	—	—	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C)cc1)c1ccc(CCC(=O)NO)cc1
E3 Binder	CHEMBL4237922	ChEMBL	6.52	—	—	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C)cc1)c1ccc(CCCCC(=O)NO)cc1
E3 Binder	CHEMBL2401848	ChEMBL	6.25	—	—	CC/C(=C(\c1ccccc1)c1ccc(OCCN(C)Cc2ccc(-c3cn(CCCCCC(=O)NO)nn3)cc2)cc1)c1ccccc1
E3 Binder	CHEMBL2401849	ChEMBL	6.66	—	—	CC/C(=C(\c1ccccc1)c1ccc(OCCN(C)Cc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)cc1)c1ccccc1
E3 Binder	CHEMBL1830536	ChEMBL	8.4	—	—	CC/C=C\CCc1nc2cc(/C=C/C(=O)NO)ccc2n1CCNCC
E3 Binder	CHEMBL4749523	ChEMBL	6.43	—	—	CC1(C)C(=O)C(C#N)=C[C@]2(C)[C@H]3C(=O)C=C4[C@@H]5C[C@@](C)(C(=O)N6CCN(c7ccc(NC(=O)CCCCCCC(=O)NO)cc7)CC6)CC[C@]5(C)CC[C@@]4(C)[C@]3(C)CC[C@@H]12
E3 Binder	CHEMBL4448523	ChEMBL	6.16	—	—	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=O)N1Cc1ccc(-c2cn(CCCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL3983635	ChEMBL	7.44	—	—	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)NCCCCCC(=O)NO)c(F)c1
E3 Binder	CHEMBL3966165	ChEMBL	6.3	—	—	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)NCCOCCC(=O)NO)c(F)c1
E3 Binder	CHEMBL3894825	ChEMBL	8.7	—	—	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)OCCCCCC(=O)NO)c(F)c1
E3 Binder	CHEMBL5280445	ChEMBL	8.82	—	—	CC1(C)CC(=O)Nc2ccc(C(=O)NCC3CCC(/C=C/C(=O)NO)CC3)cc21
E3 Binder	CHEMBL3311473	ChEMBL	7.04	—	—	CC1(C)CC(=O)Nc2ccc(C(=O)NCCCCCCC(=O)NO)cc21
E3 Binder	CHEMBL3309299	ChEMBL	6.14	—	—	CC1(C)CC(=O)Nc2ccc(C(=O)NC[C@H]3CC[C@@H](/C=C/C(=O)NO)CC3)cc21
E3 Binder	CHEMBL3309300	ChEMBL	6.28	—	—	CC1(C)CC(=O)Nc2ccc(C(=O)NC[C@H]3CC[C@@H](CCC(=O)NO)CC3)cc21
E3 Binder	CHEMBL3309297	ChEMBL	7.24	—	—	CC1(C)CC(=O)Nc2ccc(C(=O)NC[C@H]3CC[C@H](/C=C/C(=O)NO)CC3)cc21
E3 Binder	CHEMBL3309298	ChEMBL	6.36	—	—	CC1(C)CC(=O)Nc2ccc(C(=O)NC[C@H]3CC[C@H](CCC(=O)NO)CC3)cc21
E3 Binder	CHEMBL3309291	ChEMBL	6.96	—	—	CC1(C)CC(=O)Nc2ccc(C(=O)NCc3ccc(/C=C/C(=O)NO)cc3)cc21
E3 Binder	CHEMBL3309290	ChEMBL	6.54	—	—	CC1(C)CC(=O)Nc2ccc(C(=O)NCc3cccc(/C=C/C(=O)NO)c3)cc21
E3 Binder	CHEMBL3311466	ChEMBL	6.26	—	—	CC1(C)CC(=O)Nc2ccc(NC(=O)CCCCCCC(=O)NO)cc21
E3 Binder	CHEMBL4579774	ChEMBL	7.55	—	—	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCCCCCC(=O)NO)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(Cl)cc2)C1
E3 Binder	CHEMBL4469267	ChEMBL	7.55	—	—	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCCCCCCC(=O)NO)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(Cl)cc2)C1
E3 Binder	CHEMBL4592343	ChEMBL	7.72	—	—	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCCCCCCCC(=O)NO)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(Cl)cc2)C1
E3 Binder	CHEMBL567457	ChEMBL	6.0	—	—	CC1(C)NC(=O)C[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2cccc3ccccc23)NC(=O)[C@H](CCCCCC(=O)O)NC1=O
E3 Binder	CHEMBL360194	ChEMBL	7.4	—	—	CC1(C)NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O
E3 Binder	CHEMBL238829	ChEMBL	6.39	—	—	CC1(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O
E3 Binder	CHEMBL4285950	ChEMBL	6.46	—	—	CC1(C)OB(c2ccc(CONC(=O)/C=C/c3cccc(S(=O)(=O)Nc4ccccc4)c3)cc2)OC1(C)C
E3 Binder	CHEMBL4571732	ChEMBL	6.83	P7J	—	CC1(C)[C@@H]2CC[C@@H](CNCc3ccc(C(=O)NO)cc3)[C@H]1C2
E3 Binder	CHEMBL5276718	ChEMBL	6.78	—	—	CC1(C)c2ccccc2N(Cc2ccc(C(=O)NO)cc2)C1c1ccccc1
E3 Binder	CHEMBL5283402	ChEMBL	7.38	—	—	CC1(C)c2ccccc2N(Cc2ccc(C(=O)NO)cc2)C1c1cccnc1
E3 Binder	CHEMBL5289038	ChEMBL	7.21	—	—	CC1(C)c2ccccc2N(Cc2ccc(C(=O)NO)cc2)C1c1ccncc1
E3 Binder	CHEMBL5276531	ChEMBL	7.15	—	—	CC1(C)c2ccccc2N(Cc2ccc(C(=O)NO)cc2)[C@@H]1c1cccnc1
E3 Binder	CHEMBL5281527	ChEMBL	7.04	—	—	CC1(C)c2ccccc2N(Cc2ccc(C(=O)NO)cc2)[C@H]1c1cccnc1
E3 Binder	CHEMBL5267435	ChEMBL	6.09	—	—	CC1(C)c2ccccc2N(Cc2ccc(C(=O)NO)s2)C1c1cccnc1
E3 Binder	CHEMBL5286210	ChEMBL	6.21	—	—	CC1(C)c2ccccc2N(Cc2ccc(OCCCC(=O)NO)cc2)C1c1cccnc1
E3 Binder	CHEMBL5178702	ChEMBL	7.03	—	—	CC1(NC(=O)CC(=O)NCc2ccc(/C=C/C(=O)NO)cc2)CCN(c2cnc(-c3cccc(Cl)c3Cl)c(N)n2)CC1
E3 Binder	CHEMBL5187828	ChEMBL	6.35	—	—	CC1(NC(=O)CC(=O)NCc2cccc(/C=C/C(=O)NO)c2)CCN(c2cnc(-c3cccc(Cl)c3Cl)c(N)n2)CC1
E3 Binder	CHEMBL5204351	ChEMBL	7.45	—	—	CC1(NC(=O)CCCC(=O)NO)CCN(c2cnc(-c3cccc(Cl)c3Cl)c(N)n2)CC1
E3 Binder	CHEMBL5199132	ChEMBL	6.35	—	—	CC1(NC(=O)CCCCCC(=O)NO)CCN(c2cnc(-c3cccc(Cl)c3Cl)c(N)n2)CC1
E3 Binder	CHEMBL5205784	ChEMBL	6.44	—	—	CC1(NC(=O)CCCCCCC(=O)NO)CCN(c2cnc(-c3cccc(Cl)c3Cl)c(N)n2)CC1
E3 Binder	CHEMBL5206963	ChEMBL	6.04	—	—	CC1(NC(=O)CNC(=O)c2ccc(C(=O)NO)cc2)CCN(c2cnc(-c3cccc(Cl)c3Cl)c(N)n2)CC1
E3 Binder	CHEMBL5190008	ChEMBL	6.49	—	—	CC1(NC(=O)c2ccc(C(=O)NO)cc2)CCN(c2cnc(-c3cccc(Cl)c3Cl)c(N)n2)CC1
E3 Binder	CHEMBL5198194	ChEMBL	7.31	—	—	CC1(NCC(=O)NCc2ccc(/C=C/C(=O)NO)cc2)CCN(c2cnc(-c3cccc(Cl)c3Cl)c(N)n2)CC1
E3 Binder	CHEMBL5175565	ChEMBL	7.07	—	—	CC1(NCC(=O)Nc2ccc(/C=C/C(=O)NO)cc2)CCN(c2cnc(-c3cccc(Cl)c3Cl)c(N)n2)CC1
E3 Binder	CHEMBL5174636	ChEMBL	6.55	—	—	CC1(NCc2ccc(/C=C/C(=O)NO)cc2)CCN(c2cnc(-c3cccc(Cl)c3Cl)c(N)n2)CC1
E3 Binder	CHEMBL5189911	ChEMBL	7.57	—	—	CC1(NCc2ccc(C(=O)NCc3ccc(/C=C/C(=O)NO)cc3)cc2)CCN(c2cnc(-c3cccc(Cl)c3Cl)c(N)n2)CC1
E3 Binder	CHEMBL5186922	ChEMBL	6.64	—	—	CC1(NCc2ccc(C(=O)Nc3ccc(/C=C/C(=O)NO)cc3)cc2)CCN(c2cnc(-c3cccc(Cl)c3Cl)c(N)n2)CC1
E3 Binder	CHEMBL3415627	ChEMBL	7.68	—	—	CC1(Nc2ccc(C(=O)NO)cc2)CCN(c2ccc(Cl)cc2)C1=O
E3 Binder	CHEMBL3415628	ChEMBL	7.75	—	—	CC1(Nc2ccc(C(=O)NO)cc2)CCN(c2ccc3ncccc3c2)C1=O
E3 Binder	CHEMBL3415626	ChEMBL	6.34	—	—	CC1(Nc2ccc(C(=O)NO)cc2)CCN(c2ccccc2)C1=O
E3 Binder	CHEMBL3655987	ChEMBL	7.39	—	—	CC1(Nc2ncc(C(=O)NO)cn2)CCCCC1
E3 Binder	CHEMBL4868079	ChEMBL	7.13	—	—	CC1(c2ccccc2)NC(=O)N(Cc2ccc(C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL5184678	ChEMBL	6.75	—	—	CC12CC3CC(C)(C1)CC(NC(=O)/C=C/c1ccc(C(=O)NO)cc1)(C3)C2
E3 Binder	CHEMBL4848719	ChEMBL	6.69	—	—	CC12CC3CC(C)(C1)CC(NC(=O)CCCCCC(=O)NO)(C3)C2
E3 Binder	CHEMBL4851084	ChEMBL	6.44	—	—	CC12CC3CC(C)(C1)CC(NC(=O)CCCCCCC(=O)NO)(C3)C2
E3 Binder	CHEMBL4871275	ChEMBL	6.64	—	—	CC12CC3CC(C)(C1)CC(NC(=O)CCCCCCCC(=O)NO)(C3)C2
E3 Binder	CHEMBL4872595	ChEMBL	6.57	—	—	CC12CC3CC(C)(C1)CC(NC(=O)CCCCCCCCC(=O)NO)(C3)C2
E3 Binder	CHEMBL4872337	ChEMBL	7.11	—	—	CC12CC3CC(C)(C1)CC(NCc1ccc(/C=C/C(=O)NO)cc1)(C3)C2
E3 Binder	CHEMBL4871938	ChEMBL	8.27	—	—	CC12CC3CC(C)(C1)CC(NCc1ccc(NC(=O)CCCCCCC(=O)NO)cc1)(C3)C2
E3 Binder	CHEMBL4860287	ChEMBL	7.12	—	—	CC12CC3CC(C)(C1)CC(NCc1ccc(NCc4ccc(C(=O)NO)cc4)cc1)(C3)C2
E3 Binder	CHEMBL4868381	ChEMBL	7.22	—	—	CC12CC3CC(C)(C1)CC(NCc1cccc(NC(=O)CCCCCCC(=O)NO)c1)(C3)C2
E3 Binder	CHEMBL4870114	ChEMBL	6.99	—	—	CC12CC3CC(C)(C1)CC(NS(=O)(=O)c1ccc(/C=C/C(=O)NO)cc1)(C3)C2
E3 Binder	CHEMBL4872845	ChEMBL	7.03	—	—	CC12CC3CC(C)(C1)CC(NS(=O)(=O)c1cccc(/C=C/C(=O)NO)c1)(C3)C2
E3 Binder	CHEMBL3577298	ChEMBL	7.64	—	—	CC1=C(C)C(=O)C(CONC(=O)CCCCCCC(=O)Nc2ccccc2)=C(C)C1=O
E3 Binder	CHEMBL56770	ChEMBL	6.13	—	—	CC1c2ccccc2CC1C(=O)NCCCCCCC(=O)NO
E3 Binder	CHEMBL1807694	ChEMBL	7.26	—	—	CCC(/C=C/c1ccccc1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL1793820	ChEMBL	7.75	—	—	CCC(=O)C(=O)CCCC[C@@H]1NC(=O)[C@H]2CCCCN2CC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC1=O
E3 Binder	CHEMBL2371002	ChEMBL	6.96	—	—	CCC(=O)C(F)CCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC1=O
E3 Binder	CHEMBL1793826	ChEMBL	6.96	—	—	CCC(=O)C(F)CCCC[C@@H]1NC(=O)[C@H]2CCCCN2CC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC1=O
E3 Binder	CHEMBL1793825	ChEMBL	7.41	—	—	CCC(=O)C(O)CCCC[C@@H]1NC(=O)[C@H]2CCCCN2CC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC1=O
E3 Binder	CHEMBL1793941	ChEMBL	8.3	—	—	CCC(=O)C1OC1CCC[C@@H]1NC(=O)[C@H]2CCCCN2CC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC1=O
E3 Binder	CHEMBL1793814	ChEMBL	7.07	—	—	CCC(=O)CCCCC[C@@H]1/N=C(\S)[C@H]2CCCCN2CC(=O)[C@H]([C@@H](C)CC)/N=C(\S)[C@H](Cc2cn(OC)c3ccccc23)NC1=O
E3 Binder	CHEMBL1164046	ChEMBL	7.72	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)CNC(=O)C[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cc3ccccc3[nH]2)NC1=O
E3 Binder	CHEMBL2170186	ChEMBL	6.0	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](C)N(C)C(=O)CCN(CC(C)C)C(=O)CN(CCc2c[nH]c3ccccc23)C1=O
E3 Binder	CHEMBL2012813	ChEMBL	7.4	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](C)N(C)C(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O
E3 Binder	CHEMBL583130	ChEMBL	7.72	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O
E3 Binder	CHEMBL1165336	ChEMBL	7.4	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cc3ccccc3[nH]2)NC1=O
E3 Binder	CHEMBL2170018	ChEMBL	6.68	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](CCCCNC(C)=O)NC(=O)CCN(CC(C)C)C(=O)CN(CCc2c[nH]c3ccccc23)C1=O
E3 Binder	CHEMBL2170019	ChEMBL	7.22	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](CCCNC(=N)N)NC(=O)CCN(CC(C)C)C(=O)CN(CCc2c[nH]c3ccccc23)C1=O
E3 Binder	CHEMBL2170017	ChEMBL	6.6	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H](CCCNC(=N)N)NC(=O)CCN(CC=C(C)C)C(=O)CN(CCc2c[nH]c3ccccc23)C1=O
E3 Binder	CHEMBL4878197	ChEMBL	6.66	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC23CCN(CCCCCCCCn2ccc4cc(c(OC)cc4c2=O)-c2cnc1[nH]2)CC3
E3 Binder	CHEMBL4863325	ChEMBL	6.07	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CC23CCN(CCCCCn2c(=O)ccc4cc(ccc42)-c2cnc1o2)CC3
E3 Binder	CHEMBL1793969	ChEMBL	6.59	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@@H](C(=O)Cc2ccccc2)NC1=O
E3 Binder	CHEMBL1793983	ChEMBL	7.17	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@@H](c2cnc3ccccc3c2Cl)NC1=O
E3 Binder	CHEMBL1793982	ChEMBL	7.89	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@@H](c2cnc3ccccc3c2N2CCCCC2)NC1=O
E3 Binder	CHEMBL1793981	ChEMBL	6.35	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CC(=O)C(C)(C)C)NC1=O
E3 Binder	CHEMBL1793978	ChEMBL	6.38	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CC(=O)Cc2ccccc2)NC1=O
E3 Binder	CHEMBL1793968	ChEMBL	7.04	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CC(=O)c2ccccc2[N+](=O)[O-])NC1=O
E3 Binder	CHEMBL1793974	ChEMBL	7.47	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CCOc2ccccc2)NC1=O
E3 Binder	CHEMBL1793985	ChEMBL	9.7	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2c(-c3cc(OC)cc(OC)c3)[nH]c3ccccc23)NC1=O
E3 Binder	CHEMBL1793984	ChEMBL	8.4	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2c(-c3ccccc3)[nH]c3ccccc23)NC1=O
E3 Binder	CHEMBL1793989	ChEMBL	8.7	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O
E3 Binder	CHEMBL4467135	ChEMBL	9.0	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cc3ccccc3n2OC)CC1=O
E3 Binder	CHEMBL1793992	ChEMBL	8.89	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(CCN)c3ccccc23)NC1=O
E3 Binder	CHEMBL1793991	ChEMBL	9.7	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(CN3CCCC3)c3ccccc23)NC1=O
E3 Binder	CHEMBL430060	ChEMBL	9.0	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC1=O
E3 Binder	CHEMBL1793972	ChEMBL	6.48	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](c2cn(CC)c3ccccc3c2=O)NC1=O
E3 Binder	CHEMBL1793973	ChEMBL	7.07	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](c2cn(OC)c3ccccc3c2=O)NC1=O
E3 Binder	CHEMBL1791401	ChEMBL	6.64	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@H](C)CC)NC(=O)[C@H](Cc2cn(CC(=O)NCCCCCCNC(=O)CCSSCCNC(=O)C(CCCCNC(=O)CCCCC3SCC4NC(=O)NC43)NC(=O)c3ccc(N=[N+]=[N-])cc3)c3ccccc23)NC1=O
E3 Binder	CHEMBL1791134	ChEMBL	6.67	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)[C@H]([C@H](C)CC)NC(=O)[C@H](c2cn(C)c3ccccc3c2=O)NC1=O
E3 Binder	CHEMBL1793815	ChEMBL	7.07	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2CC(=O)[C@H]([C@@H](C)CC)/N=C(\S)[C@H](Cc2cn(OC)c3ccccc23)N=C1S
E3 Binder	CHEMBL1793943	ChEMBL	7.07	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2CC(=O)[C@H]([C@@H](C)CC)/N=C(\S)[C@H](Cc2cn(OC)c3ccccc23)NC1=O
E3 Binder	CHEMBL1793810	ChEMBL	9.0	—	—	CCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2CC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC1=O
E3 Binder	CHEMBL5270878	ChEMBL	6.21	—	—	CCC(=O)CCCCC[C@H](NC(=O)C(=O)N1CCOCC1)c1ncc(-c2cc3ccccc3nc2OC)o1
E3 Binder	CHEMBL5269165	ChEMBL	7.82	—	—	CCC(=O)CCCCC[C@H](NC(=O)C(C)(C)N(C)C)c1ncc(-c2cc3ccccc3nc2OC)o1
E3 Binder	CHEMBL5268361	ChEMBL	6.37	—	—	CCC(=O)CCCCC[C@H](NC(=O)C1(F)CN(C)C1)c1ncc(-c2cc3ccccc3nc2OC)o1
E3 Binder	CHEMBL5282110	ChEMBL	7.37	—	—	CCC(=O)CCCCC[C@H](NC(=O)C12CCN(CC1)CC2)c1ncc(-c2cc3ccccc3nc2OC)o1
E3 Binder	CHEMBL467678	ChEMBL	6.1	—	—	CCC(=O)CCCCC[C@H](NC(=O)C1CCN(C)CC1)c1ncc(-c2ccc3ccccc3c2)[nH]1
E3 Binder	CHEMBL5279520	ChEMBL	7.03	—	—	CCC(=O)CCCCC[C@H](NC(=O)C1CN(C)C1)c1ncc(-c2cc3ccccc3[nH]c2=O)o1
E3 Binder	CHEMBL2448576	ChEMBL	6.17	—	—	CCC(=O)CCCCC[C@H](NC(=O)C1CN(C)C1)c1ncc(-c2cc3ccccc3nc2OC)[nH]1
E3 Binder	CHEMBL5271471	ChEMBL	7.3	—	—	CCC(=O)CCCCC[C@H](NC(=O)C1CN(C)C1)c1ncc(-c2cc3ccccc3nc2OC)o1
E3 Binder	CHEMBL5285293	ChEMBL	6.9	—	—	CCC(=O)CCCCC[C@H](NC(=O)C1CN(C)C1)c1ncc(-c2ccc3ccccc3c2)[nH]1
E3 Binder	CHEMBL5273223	ChEMBL	6.06	—	—	CCC(=O)CCCCC[C@H](NC(=O)C1CN(C)C1)c1ncc(-c2ccc3ccccc3c2)o1
E3 Binder	CHEMBL5285433	ChEMBL	6.68	—	—	CCC(=O)CCCCC[C@H](NC(=O)C1CNC(=O)C1)c1ncc(-c2cc3ccccc3nc2OC)o1
E3 Binder	CHEMBL501319	ChEMBL	7.36	—	—	CCC(=O)CCCCC[C@H](NC(=O)Cc1c(C)[nH]c2ccc(OC)cc12)c1ncc(-c2ccc3ccccc3c2)[nH]1
E3 Binder	CHEMBL5285266	ChEMBL	6.38	—	—	CCC(=O)CCCCC[C@H](NC(=O)Cc1c(C)[nH]c2ccc(OC)cc12)c1ncc(-c2ccc3ccccc3c2)o1
E3 Binder	CHEMBL5285418	ChEMBL	6.86	—	—	CCC(=O)CCCCC[C@H](NC(=O)Cn1ccnn1)c1ncc(-c2cc3ccccc3nc2OC)o1
E3 Binder	CHEMBL5218854	ChEMBL	6.34	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C(C)C)CC2)c1ncc(-c2cc3ccc(C)nc3cc2OC)[nH]1
E3 Binder	CHEMBL5219409	ChEMBL	6.5	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C)CC2)c1ncc(-c2cc3ccc(C)nc3cc2OC)[nH]1
E3 Binder	CHEMBL5220278	ChEMBL	6.34	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C)CC2)c1ncc(-c2cc3ccc(C)nc3cc2OC)o1
E3 Binder	CHEMBL4861271	ChEMBL	7.35	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C)CC2)c1ncc(-c2cc3ccc(N4CCCC4)nc3cc2OC)[nH]1
E3 Binder	CHEMBL5220844	ChEMBL	6.26	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C)CC2)c1ncc(-c2cc3ccccc3[nH]c2=O)[nH]1
E3 Binder	CHEMBL5219590	ChEMBL	6.18	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C)CC2)c1ncc(-c2cc3ccccc3n(C)c2=O)[nH]1
E3 Binder	CHEMBL5218586	ChEMBL	6.7	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C)CC2)c1ncc(-c2cc3cccnc3cc2OC)[nH]1
E3 Binder	CHEMBL4862556	ChEMBL	7.13	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C)CC2)c1ncc(-c2cc3cccnc3cc2OC)o1
E3 Binder	CHEMBL5219039	ChEMBL	6.12	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C)CC2)c1ncc(-c2cc3ccncc3nc2OC)[nH]1
E3 Binder	CHEMBL5218535	ChEMBL	6.16	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C)CC2)c1ncc(-c2ccc3ncccc3c2)[nH]1
E3 Binder	CHEMBL5219811	ChEMBL	7.08	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C)CC2)c1ncc(-c2ccc3nccnc3c2)[nH]1
E3 Binder	CHEMBL5218749	ChEMBL	6.35	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C)CC2)c1ncc(-c2cn(C)c3ccccc3c2=O)[nH]1
E3 Binder	CHEMBL5219825	ChEMBL	6.51	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(C1CCC1)CC2)c1ncc(-c2cc3ccc(C)nc3cc2OC)[nH]1
E3 Binder	CHEMBL5220454	ChEMBL	6.51	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2cc3ccc(=O)n(C)c3cc2OC)o1
E3 Binder	CHEMBL5220926	ChEMBL	6.46	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2cc3ccc(C)nc3cc2OC)[nH]1
E3 Binder	CHEMBL5218693	ChEMBL	6.66	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2cc3ccc(C)nc3cc2OC)o1
E3 Binder	CHEMBL4864510	ChEMBL	6.84	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2cc3cccnc3cc2OC)[nH]1
E3 Binder	CHEMBL4873493	ChEMBL	7.08	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2cc3cccnc3cc2OC)o1
E3 Binder	CHEMBL5220715	ChEMBL	7.08	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2cc3cccnc3nc2OC)o1
E3 Binder	CHEMBL5218767	ChEMBL	6.01	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2cc3ccn(CC)c(=O)c3cc2OC)o1
E3 Binder	CHEMBL5219490	ChEMBL	6.52	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2cc3ccncc3nc2OC)o1
E3 Binder	CHEMBL5221097	ChEMBL	6.25	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2cc3cn(C)nc3cc2OC)[nH]1
E3 Binder	CHEMBL5218487	ChEMBL	6.8	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2cc3cn(C)nc3cc2OC)o1
E3 Binder	CHEMBL5220576	ChEMBL	6.51	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2cc3nccnc3cc2OC)[nH]1
E3 Binder	CHEMBL5220120	ChEMBL	6.58	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2ccc3ccncc3c2)[nH]1
E3 Binder	CHEMBL5218553	ChEMBL	6.0	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC)CC2)c1ncc(-c2ccc3cnccc3c2)[nH]1
E3 Binder	CHEMBL5219294	ChEMBL	6.57	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC1CC1)CC2)c1ncc(-c2cc3ccc(C)nc3cc2OC)[nH]1
E3 Binder	CHEMBL4862152	ChEMBL	6.95	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC1CC1)CC2)c1ncc(-c2cc3ccc(C)nc3cc2OC)o1
E3 Binder	CHEMBL5220360	ChEMBL	6.21	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC1CC1)CC2)c1ncc(-c2cc3ccc(C4CC4)nc3cc2OC)[nH]1
E3 Binder	CHEMBL5219875	ChEMBL	6.52	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC1CC1)CC2)c1ncc(-c2cc3ccc(CC)nc3cc2OC)[nH]1
E3 Binder	CHEMBL4861467	ChEMBL	7.12	—	—	CCC(=O)CCCCC[C@H](NC(=O)[C@H]1CC12CCN(CC1CC1)CC2)c1ncc(-c2cc3cccnc3cc2OC)[nH]1
E3 Binder	CHEMBL5199116	ChEMBL	9.52	—	—	CCC(=O)CCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)C([C@@H](C)CC)NC(=O)C(Cc2c[nH]c3ccccc23)NC1=O
E3 Binder	CHEMBL569812	ChEMBL	7.27	—	—	CCC(=O)CCCSC[C@@H]1NC(=O)[C@H](C)NC(=O)C[C@H](CC(C)C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O
E3 Binder	CHEMBL189929	ChEMBL	7.27	—	—	CCC(C(=O)Nc1ccc(C(=O)NO)cc1)c1ccccc1
E3 Binder	CHEMBL2347007	ChEMBL	7.17	—	—	CCC(C)(C)C(=O)O[C@H]1C[C@@H](C)C=C2C=C[C@H](C)[C@H](CC[C@@H](O)C[C@@H](O)CC(=O)NO)[C@H]21
E3 Binder	CHEMBL3970138	ChEMBL	7.3	—	—	CCC(C)C(=O)OC1C[C@@H](C)C=C2C=C[C@H](C)[C@H](CC[C@@H](O)C[C@@H](O)CC(=O)NO)[C@H]21
E3 Binder	CHEMBL2036478	ChEMBL	8.4	—	—	CCC(C)C(c1nc2ccccc2o1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL2313364	ChEMBL	8.66	—	—	CCC(C)[C@H]1NC(=O)[C@H]2CSSCC/C=C/[C@H](CC(=O)N[C@H](C)C(=O)N2)OC(=O)C[C@@H]1O
E3 Binder	CHEMBL3909252	ChEMBL	6.25	—	—	CCC(CC)(c1ccc(C(=O)NCCCCCC(=O)NO)cc1)c1ccc(OCC(O)C(C)(C)C)c(C)c1
E3 Binder	CHEMBL3233691	ChEMBL	6.88	—	—	CCC(CC)C(=O)N[C@H](COc1ccc(/C=C/C(=O)NO)cc1)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL4288220	ChEMBL	6.8	—	—	CCC(CCCC(=O)Nc1ccccc1)CCC(=O)NO
E3 Binder	CHEMBL1793944	ChEMBL	7.14	—	—	CCC(CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2CC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC1=O)SC(C)=O
E3 Binder	CHEMBL1793808	ChEMBL	6.84	—	—	CCC(N)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2CC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC1=O
E3 Binder	CHEMBL429416	ChEMBL	7.02	—	—	CCC(c1ccc(/C=C/C(=O)NO)cc1)c1nc2ccccc2n1CC
E3 Binder	CHEMBL1808160	ChEMBL	6.88	—	—	CCCC(/C=C/c1ccccc1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL1793947	ChEMBL	9.0	—	—	CCCC(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2CC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC1=O
E3 Binder	CHEMBL482765	ChEMBL	7.64	—	—	CCCC(=S)SCC(=O)c1ccc(NC(C)=O)cc1
E3 Binder	CHEMBL445518	ChEMBL	6.96	—	—	CCCC(=S)SCC(=O)c1ccc(OC)cc1
E3 Binder	CHEMBL3233692	ChEMBL	6.01	—	—	CCCC(CCC)C(=O)N[C@H](COc1ccc(/C=C/C(=O)NO)cc1)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL2336043	ChEMBL	6.42	—	—	CCCC(CCC)C(=O)N[C@H](COc1ccc(/C=C/C(=O)NO)cc1OC)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL4859396	ChEMBL	7.29	—	—	CCCC1(c2ccccc2)NC(=O)N(Cc2ccc(C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL5206179	ChEMBL	7.24	—	—	CCCC1=C(Nc2ccc(C(=O)NO)cc2)C2N=CC=CC2=N1
E3 Binder	CHEMBL1808161	ChEMBL	6.86	—	—	CCCCC(/C=C/c1ccccc1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL2204665	ChEMBL	6.34	—	—	CCCCC(CC)CC(CCCCC(=O)NO)CC(=O)Nc1ccccc1
E3 Binder	CHEMBL4086409	ChEMBL	6.5	—	—	CCCCC(CCCC(=O)NO)CCC(=O)Nc1ccccc1
E3 Binder	CHEMBL4285869	ChEMBL	7.06	—	—	CCCCC(CCCC(=O)Nc1ccccc1)CCC(=O)NO
E3 Binder	CHEMBL4756672	ChEMBL	6.92	—	—	CCCCC(NCc1ccc(C(=O)NO)cc1)c1nnnn1Cc1ccccc1
E3 Binder	CHEMBL3953547	ChEMBL	6.07	—	—	CCCCCC(CCCCCC(=O)Nc1ccccc1)C(=O)NO
E3 Binder	CHEMBL4064944	ChEMBL	6.39	—	—	CCCCCCC(CCCC(=O)NO)CCC(=O)Nc1ccccc1
E3 Binder	CHEMBL4277951	ChEMBL	6.85	—	—	CCCCCCC(CCCC(=O)Nc1ccccc1)CCC(=O)NO
E3 Binder	CHEMBL3982264	ChEMBL	6.22	—	—	CCCCCCC(CCCCCC(=O)Nc1ccccc1)C(=O)NO
E3 Binder	CHEMBL1173445	ChEMBL	6.78	—	—	CCCCCCCC(=O)SCC/C=C/[C@@H]1CC(=O)NCc2nc(cs2)C2=N[C@@](C)(CS2)C(=O)N[C@@H](C(C)C)C(=O)O1
E3 Binder	CHEMBL1793807	ChEMBL	7.21	—	—	CCCCCCCC[C@@H]1NC(=O)[C@H]2CCCCN2CC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC1=O
E3 Binder	CHEMBL2440719	ChEMBL	6.39	—	—	CCCCCCCNC(=O)Nc1cc(/C=C/C(=O)NO)ccc1OCCN(CC)CC
E3 Binder	CHEMBL2440718	ChEMBL	6.52	—	—	CCCCCCNC(=O)Nc1cc(/C=C/C(=O)NO)ccc1OCCN(CC)CC
E3 Binder	CHEMBL2440723	ChEMBL	6.73	—	—	CCCCCCNC(=S)Nc1cc(/C=C/C(=O)NO)ccc1OCCN(CC)CC
E3 Binder	CHEMBL1830424	ChEMBL	6.52	—	—	CCCCCCc1nc2cc(/C=C/C(=O)NO)ccc2n1CCN(C)C
E3 Binder	CHEMBL1830422	ChEMBL	6.46	—	—	CCCCCCc1nc2cc(/C=C/C(=O)NO)ccc2n1CCNC(C)C
E3 Binder	CHEMBL1830420	ChEMBL	6.55	—	—	CCCCCCc1nc2cc(/C=C/C(=O)NO)ccc2n1CCNCC
E3 Binder	CHEMBL2440717	ChEMBL	6.73	—	—	CCCCCNC(=O)Nc1cc(/C=C/C(=O)NO)ccc1OCCN(CC)CC
E3 Binder	CHEMBL2440712	ChEMBL	6.7	—	—	CCCCCNC(=O)Nc1cc(/C=C/C(=O)NO)ccc1SCCN(CC)CC
E3 Binder	CHEMBL2440722	ChEMBL	6.67	—	—	CCCCCNC(=S)Nc1cc(/C=C/C(=O)NO)ccc1OCCN(CC)CC
E3 Binder	CHEMBL3681859	ChEMBL	6.24	—	—	CCCCCNc1cc(/C=C/C(=O)NO)ccc1SCCN(CC)CC
E3 Binder	CHEMBL589906	ChEMBL	6.47	—	—	CCCCC[C@@H]1NC(=O)[C@@H](CCCCC)NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCCN2C1=O
E3 Binder	CHEMBL1830537	ChEMBL	6.64	—	—	CCCCCc1nc2cc(/C=C/C(=O)NO)ccc2n1CCNC(C)C
E3 Binder	CHEMBL2179244	ChEMBL	7.6	—	—	CCCCN(C(=O)NCc1ccc(C(=O)NO)cc1)c1ccccc1
E3 Binder	CHEMBL5192895	ChEMBL	6.88	—	—	CCCCN(Cc1ccc(C(=O)NNCC)cc1)C(=O)Nc1ccccc1
E3 Binder	CHEMBL5181667	ChEMBL	6.72	—	—	CCCCN(Cc1ccc(C(=O)NNCC)cc1)C(=O)c1ccccc1
E3 Binder	CHEMBL4159465	ChEMBL	7.13	—	—	CCCCN(Cc1ccc(C(=O)NO)cc1)C(=O)NCCN1CCCC1
E3 Binder	CHEMBL4167374	ChEMBL	7.37	—	—	CCCCN(Cc1ccc(C(=O)NO)cc1)C(=O)Nc1cc(C)ccn1
E3 Binder	CHEMBL4759584	ChEMBL	9.05	—	—	CCCCN(Cc1ccc(C(=O)NO)cc1)C(=O)Nc1ccc(CN)cc1
E3 Binder	CHEMBL4170768	ChEMBL	8.8	—	—	CCCCN(Cc1ccc(C(=O)NO)cc1)C(=O)Nc1ccc2cn[nH]c2c1
E3 Binder	CHEMBL4166281	ChEMBL	8.77	—	—	CCCCN(Cc1ccc(C(=O)NO)cc1)C(=O)Nc1cccc(N(C)C)c1
E3 Binder	CHEMBL2179618	ChEMBL	8.8	N4R	—	CCCCN(Cc1ccc(C(=O)NO)cc1)C(=O)Nc1ccccc1
E3 Binder	CHEMBL4162826	ChEMBL	8.22	—	—	CCCCN(Cc1ccc(C(=O)NO)cc1)C(=O)Nc1ncccn1
E3 Binder	CHEMBL4278868	ChEMBL	6.43	—	—	CCCCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2c([nH]c3ccccc32)c(-c2cccc(OC)c2)n1
E3 Binder	CHEMBL4287197	ChEMBL	6.47	—	—	CCCCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2c([nH]c3ccccc32)c(-c2ccccc2OC)n1
E3 Binder	CHEMBL4280382	ChEMBL	6.03	—	—	CCCCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2c([nH]c3ccccc32)c(C)n1
E3 Binder	CHEMBL2413319	ChEMBL	6.64	—	—	CCCCN(Cc1ccccc1)Cc1ccc(/C=C/C(=O)NO)o1
E3 Binder	CHEMBL4281183	ChEMBL	8.03	—	—	CCCCN1C(=O)C2Cc3c(n(Cc4ccc(C(=O)NO)cc4)c4ccccc34)CN2C1=O
E3 Binder	CHEMBL4292205	ChEMBL	8.49	—	—	CCCCN1CC(=O)N2Cc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)CC2C1=O
E3 Binder	CHEMBL4553537	ChEMBL	7.1	—	—	CCCCNC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4059953	ChEMBL	6.1	—	—	CCCCNC(=O)CN(CCCCCC(=O)NO)C(=O)c1ccc(N(C)C)cc1
E3 Binder	CHEMBL2440711	ChEMBL	6.76	—	—	CCCCNC(=O)Nc1cc(/C=C/C(=O)NO)ccc1SCCN(CC)CC
E3 Binder	CHEMBL4225111	ChEMBL	7.07	—	—	CCCCNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)/C=C/c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL2440721	ChEMBL	6.89	—	—	CCCCNC(=S)Nc1cc(/C=C/C(=O)NO)ccc1OCCN(CC)CC
E3 Binder	CHEMBL5169697	ChEMBL	6.02	—	—	CCCCNc1nc(Cl)nc2c1ncn2CCCC(=O)NCc1ccc(C(=O)Nc2ccccc2N)cc1
E3 Binder	CHEMBL5193978	ChEMBL	6.0	—	—	CCCCNc1nc(Cl)nc2c1ncn2Cc1ccc(C(=O)Nc2ccc(C)cc2N)cc1
E3 Binder	CHEMBL5196817	ChEMBL	7.56	—	—	CCCCNc1nc(Cl)nc2c1ncn2Cc1ccc(C(=O)Nc2ccccc2N)cc1
E3 Binder	CHEMBL401837	ChEMBL	6.55	—	—	CCCC[C@@H]1NC(=O)C(C)(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
E3 Binder	CHEMBL5203249	ChEMBL	7.77	—	—	CCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](CCCCCS)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](C)NC(=O)[C@H](CCCCN)NC1=O
E3 Binder	CHEMBL1836042	ChEMBL	6.21	—	—	CCCC[C@H]1NC(=O)C[C@@H](/C=C/CCS)OC(=O)C[C@H](O)[C@@H]([C@@H](C)CC)NC(=O)[C@@H](CS)NC1=O
E3 Binder	CHEMBL3218562	ChEMBL	6.03	—	—	CCCC[C@H]1NC(=O)C[C@H]2/C=C/CCSSC[C@@H](NC1=O)C(=O)N[C@H](C(C)C)[C@@H](O)CC(=O)O2
E3 Binder	CHEMBL1801245	ChEMBL	7.66	—	—	CCCCc1ccc(CN[C@H]2[C@@H]3CN(c4ncc(C(=O)NO)cn4)C[C@@H]32)cc1
E3 Binder	CHEMBL1851943	ChEMBL	7.03	—	—	CCCCc1nc2cc(/C=C/C(=O)NO)ccc2n1CCN(CC)CC
E3 Binder	CHEMBL3215861	ChEMBL	6.61	—	—	CCCCc1nc2cc(/C=C/C(=O)NO)ccc2n1CCN(CC)CC.Cl.Cl
E3 Binder	CHEMBL1830396	ChEMBL	6.65	—	—	CCCCc1nc2cc(/C=C/C(=O)NO)ccc2n1CCNC(C)C
E3 Binder	CHEMBL3287254	ChEMBL	6.21	—	—	CCCCc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO
E3 Binder	CHEMBL3601343	ChEMBL	7.49	—	—	CCCCn1ccc2ccc(NC(=O)CCCCCCC(=O)NO)cc2c1=O
E3 Binder	CHEMBL4536420	ChEMBL	6.58	—	—	CCCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2c([nH]c3ccccc32)c(-c2ccc(OC)cc2)n1
E3 Binder	CHEMBL4289542	ChEMBL	6.64	—	—	CCCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2c([nH]c3ccccc32)c(-c2cccc(OC)c2)n1
E3 Binder	CHEMBL4279273	ChEMBL	6.58	—	—	CCCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2c([nH]c3ccccc32)c(-c2ccccc2OC)n1
E3 Binder	CHEMBL4291022	ChEMBL	6.07	—	—	CCCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2c([nH]c3ccccc32)c(C)n1
E3 Binder	CHEMBL4849709	ChEMBL	6.99	—	—	CCCN(Cc1ccc(C(=O)NO)cn1)C12CC3C[C@@](C)(C1)C[C@](C)(C3)C2
E3 Binder	CHEMBL2413317	ChEMBL	6.77	—	—	CCCN(Cc1ccccc1)Cc1ccc(/C=C/C(=O)NO)o1
E3 Binder	CHEMBL4287618	ChEMBL	8.0	—	—	CCCN1C(=O)C2Cc3c(n(Cc4ccc(C(=O)NO)cc4)c4ccccc34)CN2C1=O
E3 Binder	CHEMBL4856388	ChEMBL	6.76	—	—	CCCN1C(=O)N(Cc2ccc(C(=O)NO)cc2)C(=O)C1CC(C)C
E3 Binder	CHEMBL4851633	ChEMBL	7.25	—	—	CCCN1C(=O)N(Cc2ccc(C(=O)NO)cc2)C(=O)C1Cc1ccccc1
E3 Binder	CHEMBL4458308	ChEMBL	7.9	—	—	CCCN1C(=O)N(c2ccc(Cl)cc2)C(=O)C1CCC(=O)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4854023	ChEMBL	7.27	—	—	CCCN1CC(=O)N(Cc2ccc(C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL4277484	ChEMBL	9.05	—	—	CCCN1CC(=O)N2Cc3c(c4cc(O)ccc4n3Cc3ccc(C(=O)NO)cc3)CC2C1=O
E3 Binder	CHEMBL4285431	ChEMBL	8.78	—	—	CCCN1CC(=O)N2Cc3c(c4cc(OC)ccc4n3Cc3ccc(C(=O)NO)cc3)CC2C1=O
E3 Binder	CHEMBL4292609	ChEMBL	8.9	—	—	CCCN1CC(=O)N2Cc3c(c4cc(OCc5ccccc5)ccc4n3Cc3ccc(C(=O)NO)cc3)CC2C1=O
E3 Binder	CHEMBL4280893	ChEMBL	8.43	—	—	CCCN1CC(=O)N2Cc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)CC2C1=O
E3 Binder	CHEMBL4283931	ChEMBL	7.08	—	—	CCCN1CC(=O)N2[C@@H](Cc3c(n(Cc4ccc(C(=O)NO)cc4)c4ccccc34)[C@@H]2C)C1=O
E3 Binder	CHEMBL4281792	ChEMBL	7.22	—	—	CCCN1CC(=O)N2[C@H](C)c3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)C[C@H]2C1=O
E3 Binder	CHEMBL4294514	ChEMBL	8.74	—	—	CCCN1CC(=O)N2[C@H](Cc3c(n(Cc4ccc(C(=O)NO)cc4)c4ccccc34)[C@@H]2C)C1=O
E3 Binder	CHEMBL4277718	ChEMBL	7.73	—	—	CCCN1CC(=O)N2[C@H](Cc3c(n(Cc4ccc(C(=O)NO)cc4)c4ccccc34)[C@H]2C)C1=O
E3 Binder	CHEMBL2440715	ChEMBL	6.63	—	—	CCCNC(=O)Nc1cc(/C=C/C(=O)NO)ccc1OCCN(CC)CC
E3 Binder	CHEMBL2440710	ChEMBL	6.7	—	—	CCCNC(=O)Nc1cc(/C=C/C(=O)NO)ccc1SCCN(CC)CC
E3 Binder	CHEMBL2440720	ChEMBL	6.68	—	—	CCCNC(=S)Nc1cc(/C=C/C(=O)NO)ccc1OCCN(CC)CC
E3 Binder	CHEMBL3681860	ChEMBL	6.18	—	—	CCCNc1cc(/C=C/C(=O)NO)ccc1SCCN(CC)CC
E3 Binder	CHEMBL4475116	ChEMBL	8.32	—	—	CCCNc1ccc2c3c(cccc13)C(=O)N(CCCCCC(=O)NO)C2=O
E3 Binder	CHEMBL5179973	ChEMBL	6.24	—	—	CCCNc1nc(Cl)nc2c1ncn2Cc1ccc(C(=O)Nc2ccccc2N)cc1
E3 Binder	CHEMBL4469297	ChEMBL	7.58	—	—	CCCNc1nc(Nc2cnn(CCCCCCC(=O)NO)c2)ncc1Cl
E3 Binder	CHEMBL4202659	ChEMBL	6.46	—	—	CCCOc1cccc(-c2ccc3c(NC(=O)c4ccc(C(=O)NO)cc4)n[nH]c3c2)c1
E3 Binder	CHEMBL471173	ChEMBL	6.62	—	—	CCCS(=O)(=O)Cc1noc(-c2ccc(C(=O)C(F)(F)F)s2)n1
E3 Binder	CHEMBL510856	ChEMBL	7.36	—	—	CCCSC(=S)SCC(=O)c1ccc(C(=O)N[C@H](C)c2ccccc2)s1
E3 Binder	CHEMBL317614	ChEMBL	7.42	—	—	CCC[C@H]1C(=O)N([C@@H](Cc2ccc(OC)cc2)C(=O)NCCCCCC(=O)NO)C(=O)[C@@H]1CC(C)C
E3 Binder	CHEMBL328819	ChEMBL	7.29	—	—	CCC[C@H]1C(=O)N([C@@H](Cc2ccccc2)C(=O)NCCCCCC(=O)NO)C(=O)[C@@H]1CC(C)C
E3 Binder	CHEMBL4225760	ChEMBL	6.78	—	—	CCCc1cc(-c2ccc(F)cc2)n(Cc2ccc(C(=O)NO)cc2)n1
E3 Binder	CHEMBL4228210	ChEMBL	6.97	—	—	CCCc1cc(-c2ccc(F)cc2)nn1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4873778	ChEMBL	7.92	—	—	CCCc1ccc2c(c1)CCC(=O)N2Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4209220	ChEMBL	6.49	—	—	CCCc1nc(C)c2c(=O)[nH]c(-c3cc(-c4ccc(C(=O)NO)cc4)ccc3OCC)nn12
E3 Binder	CHEMBL4208487	ChEMBL	6.96	—	—	CCCc1nc(C)c2c(=O)[nH]c(-c3cc(CC4CC(C(=O)NO)C4)ccc3OCC)nn12
E3 Binder	CHEMBL4213615	ChEMBL	6.59	—	—	CCCc1nc(C)c2c(=O)[nH]c(-c3cc(Cc4ccc(C(=O)NO)cc4)ccc3OCC)nn12
E3 Binder	CHEMBL4214135	ChEMBL	7.01	—	—	CCCc1nc(C)c2c(=O)[nH]c(-c3cc(Cc4ccc(C(=O)NO)s4)ccc3OCC)nn12
E3 Binder	CHEMBL4216635	ChEMBL	7.38	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(-c4ccc(C(=O)NO)cc4)ccc3OCC)nc12
E3 Binder	CHEMBL4202521	ChEMBL	7.43	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(-c4ccc(C(=O)NO)s4)ccc3OCC)nc12
E3 Binder	CHEMBL4204952	ChEMBL	6.09	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(-c4ccc(CC(=O)NO)cc4)ccc3OCC)nc12
E3 Binder	CHEMBL4217166	ChEMBL	6.72	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(C(=O)c4ccc(C(=O)NO)s4)ccc3OCC)nc12
E3 Binder	CHEMBL4212445	ChEMBL	7.05	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(C(O)c4ccc(C(=O)NO)cc4)ccc3OCC)nc12
E3 Binder	CHEMBL4207538	ChEMBL	7.11	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(C(OC)c4ccc(C(=O)NO)cc4)ccc3OCC)nc12
E3 Binder	CHEMBL4207409	ChEMBL	6.47	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(C4=CCC(C(=O)NO)CC4)ccc3OCC)nc12
E3 Binder	CHEMBL4210653	ChEMBL	6.66	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(C4=CCC(CC(=O)NO)CC4)ccc3OCC)nc12
E3 Binder	CHEMBL4217364	ChEMBL	7.09	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(CC4CC(C(=O)NO)C4)ccc3OCC)nc12
E3 Binder	CHEMBL4209025	ChEMBL	6.85	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(Cc4ccc(C(=O)NO)c(F)c4)ccc3OCC)nc12
E3 Binder	CHEMBL4217821	ChEMBL	7.21	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(Cc4ccc(C(=O)NO)cc4)ccc3OCC)nc12
E3 Binder	CHEMBL4204146	ChEMBL	7.06	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(Cc4ccc(C(=O)NO)cc4F)ccc3OCC)nc12
E3 Binder	CHEMBL4214699	ChEMBL	6.78	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(Cc4ccc(C(=O)NO)o4)ccc3OCC)nc12
E3 Binder	CHEMBL4212186	ChEMBL	7.82	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(Cc4ccc(C(=O)NO)s4)ccc3OCC)nc12
E3 Binder	CHEMBL4212866	ChEMBL	6.79	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(Cc4ccc(CC(=O)NO)cc4)ccc3OCC)nc12
E3 Binder	CHEMBL3979179	ChEMBL	6.23	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(N(C)C4CCN(c5ncc(C(=O)NO)cn5)CC4)ccc3OCC)nc12
E3 Binder	CHEMBL3907730	ChEMBL	6.36	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(NC4CCN(c5ncc(C(=O)NO)cn5)CC4)ccc3OCC)nc12
E3 Binder	CHEMBL3978271	ChEMBL	6.15	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(NCC4CCN(c5ncc(C(=O)NO)cn5)CC4)ccc3OCC)nc12
E3 Binder	CHEMBL4203481	ChEMBL	7.18	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(Nc4ccc(C(=O)NO)cc4)ccc3OCC)nc12
E3 Binder	CHEMBL4207836	ChEMBL	7.48	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(OCc4ccc(C(=O)NO)cc4)ccc3OCC)nc12
E3 Binder	CHEMBL3954968	ChEMBL	7.06	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)N4CCC(CCC(=O)NO)CC4)ccc3OCC)nc12
E3 Binder	CHEMBL3926754	ChEMBL	6.44	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)N4CCN(CCCC(=O)NO)CC4)ccc3OCC)nc12
E3 Binder	CHEMBL3899814	ChEMBL	7.05	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)N4CCN(Cc5ccc(/C=C/C(=O)NO)cc5)CC4)ccc3OCC)nc12
E3 Binder	CHEMBL3970984	ChEMBL	6.57	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)N4CCN(c5ncc(C(=O)NO)cn5)CC4)ccc3OCC)nc12
E3 Binder	CHEMBL3986487	ChEMBL	7.23	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)NC4CCN(c5ncc(C(=O)NO)cn5)CC4)ccc3OCC)nc12
E3 Binder	CHEMBL3925737	ChEMBL	7.08	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc(S(=O)(=O)Nc4ccc(/C=C/C(=O)NO)cc4)ccc3OCC)nc12
E3 Binder	CHEMBL4206296	ChEMBL	7.32	—	—	CCCc1nn(C)c2c(=O)[nH]c(-c3cc([C@H]4CC[C@@H](C(=O)NO)CC4)ccc3OCC)nc12
E3 Binder	CHEMBL4243458	ChEMBL	8.8	—	—	CCCn1cc(-c2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc3[nH]ccc23)cn1
E3 Binder	CHEMBL1793990	ChEMBL	7.82	—	—	CCCn1cc(C(=O)[C@H]2NC(=O)[C@H](CCCCCC(=O)CC)NC(=O)[C@H]3CCCCN3C(=O)[C@H]([C@@H](C)CC)NC2=O)c2ccccc21
E3 Binder	CHEMBL1791140	ChEMBL	6.64	—	—	CCCn1cc([C@@H]2NC(=O)[C@H](CCCCCC(=O)CC)NC(=O)[C@H]3CCCCN3C(=O)[C@H]([C@H](C)CC)NC2=O)c(=O)c2ccccc21
E3 Binder	CHEMBL2179246	ChEMBL	7.39	—	—	CCN(C(=O)NCc1ccc(C(=O)NO)cc1)c1ccccc1
E3 Binder	CHEMBL4633453	ChEMBL	6.09	—	—	CCN(C(=O)c1ccccc1C(F)(F)F)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5090521	ChEMBL	6.8	—	—	CCN(CC)CCCNC(=O)c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL4542853	ChEMBL	6.92	—	—	CCN(CC)CCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2c([nH]c3ccccc32)c(-c2ccc(OC)cc2)n1
E3 Binder	CHEMBL4084499	ChEMBL	6.77	—	—	CCN(CC)CCNC(=O)c1ccc(-c2cn(CCCCCC(=O)NO)nn2)cn1
E3 Binder	CHEMBL4096623	ChEMBL	7.8	—	—	CCN(CC)CCNC(=O)c1ccc(-c2cn(CCCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL4092997	ChEMBL	7.47	—	—	CCN(CC)CCNC(=O)c1ccc(-c2cn(CCCCCCC(=O)NO)nn2)cn1
E3 Binder	CHEMBL4102456	ChEMBL	7.57	—	—	CCN(CC)CCNC(=O)c1ccc(-c2cn(CCCCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL5093179	ChEMBL	7.85	—	—	CCN(CC)CCNC(=O)c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3681866	ChEMBL	6.53	—	—	CCN(CC)CCSc1ccc(/C=C/C(=O)NO)cc1N
E3 Binder	CHEMBL3681865	ChEMBL	6.1	—	—	CCN(CC)CCSc1ccc(/C=C/C(=O)NO)cc1NC
E3 Binder	CHEMBL3681869	ChEMBL	6.5	—	—	CCN(CC)CCSc1ccc(/C=C/C(=O)NO)cc1NC(=O)C(Cl)Cl
E3 Binder	CHEMBL3681861	ChEMBL	6.45	—	—	CCN(CC)CCSc1ccc(/C=C/C(=O)NO)cc1NC(C)=O
E3 Binder	CHEMBL3681858	ChEMBL	6.2	—	—	CCN(CC)CCSc1ccc(/C=C/C(=O)NO)cc1NCCCc1ccccc1
E3 Binder	CHEMBL3681863	ChEMBL	6.56	—	—	CCN(CC)CCSc1ccc(/C=C/C(=O)NO)cc1NCc1ccccc1
E3 Binder	CHEMBL3681867	ChEMBL	6.61	—	—	CCN(CC)CCSc1ccc(/C=C/C(=O)NO)cc1NS(=O)(=O)c1ccc(C)cc1
E3 Binder	CHEMBL3681862	ChEMBL	6.5	—	—	CCN(CC)CCSc1ccc(/C=C/C(=O)NO)cc1[N+](=O)[O-]
E3 Binder	CHEMBL1095711	ChEMBL	7.1	—	—	CCN(CC)CCn1c(-c2cccc(/C=C/C(=O)NO)c2)nc2ccccc21
E3 Binder	CHEMBL3329994	ChEMBL	8.14	—	—	CCN(CC)CCn1c(C)c(CCNS(=O)(=O)c2ccc(/C=C/C(=O)NO)cc2)c2ccccc21
E3 Binder	CHEMBL3601344	ChEMBL	7.41	—	—	CCN(CC)CCn1ccc2ccc(NC(=O)CCCCCCC(=O)NO)cc2c1=O
E3 Binder	CHEMBL4757504	ChEMBL	8.16	—	—	CCN(CC)Cc1ccc(Cn2c(=O)c(OCc3ccc(C(=O)NO)cc3)c(-c3ccccc3)c3ccccc32)cc1
E3 Binder	CHEMBL4744710	ChEMBL	7.94	—	—	CCN(CC)Cc1ccc(Cn2c(=O)c(OCc3ccc(C(=O)NO)cc3)c(-c3cccnc3)c3ccccc32)cc1
E3 Binder	CHEMBL4870227	ChEMBL	8.0	—	—	CCN(CC)Cc1ccc2cc(COC(=O)Nc3c(F)cc(C(=O)NO)cc3F)ccc2c1
E3 Binder	CHEMBL1213492	ChEMBL	8.38	QCM	—	CCN(CC)Cc1ccc2cc(COC(=O)Nc3ccc(C(=O)NO)cc3)ccc2c1
E3 Binder	CHEMBL4454663	ChEMBL	8.05	—	—	CCN(CC)S(=O)(=O)c1cccc(-c2nnc(Sc3ccc(C(=O)NO)cc3)n2N)c1
E3 Binder	CHEMBL1773685	ChEMBL	6.28	—	—	CCN(CC)c1ccc(-n2nc3cc(C)c(N)cc3n2)cc1
E3 Binder	CHEMBL5078298	ChEMBL	6.68	—	—	CCN(CC)c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3339027	ChEMBL	7.37	—	—	CCN(CC)c1ccc(Nc2ncnc3sc(NC(=O)CCCCCCC(=O)NO)cc23)cc1
E3 Binder	CHEMBL3339028	ChEMBL	8.46	—	—	CCN(CC)c1ccc(Nc2ncnc3sc(NC(=O)CCCCCCC(=O)NO)cc23)cc1F
E3 Binder	CHEMBL3931061	ChEMBL	6.0	—	—	CCN(CCNC(=O)c1ccc(N)cc1)C(=O)CCCCC(=O)NO
E3 Binder	CHEMBL3329996	ChEMBL	7.53	—	—	CCN(CCc1c(C)[nH]c2ccccc12)S(=O)(=O)c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL5087228	ChEMBL	7.66	—	—	CCN(CCc1ccc(C(=O)NO)cc1)c1nc(N)n2nc(-c3ccco3)nc2n1
E3 Binder	CHEMBL2413311	ChEMBL	6.32	—	—	CCN(CCc1ccc2c(c1)OCO2)Cc1ccc(/C=C/C(=O)NO)o1
E3 Binder	CHEMBL2413299	ChEMBL	6.08	—	—	CCN(Cc1ccc(-c2ccccc2)cc1)Cc1ccc(/C=C/C(=O)NO)o1
E3 Binder	CHEMBL4286217	ChEMBL	6.08	—	—	CCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cc2c([nH]c3ccccc32)c(-c2ccccc2OC)n1
E3 Binder	CHEMBL2413316	ChEMBL	6.89	—	—	CCN(Cc1ccccc1)Cc1ccc(/C=C/C(=O)NO)o1
E3 Binder	CHEMBL3693721	ChEMBL	8.22	—	—	CCN(c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1)c1ccccc1C(F)(F)F
E3 Binder	CHEMBL3693715	ChEMBL	8.1	—	—	CCN(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1c(Cl)cccc1Cl
E3 Binder	CHEMBL3693712	ChEMBL	8.3	—	—	CCN(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1ccccc1C(F)(F)F
E3 Binder	CHEMBL3693727	ChEMBL	7.96	—	—	CCN(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1cnccn1
E3 Binder	CHEMBL4640819	ChEMBL	6.06	—	—	CCN(c1ccc(C(=O)NO)cc1)S(=O)(=O)c1cccc(C(C)(C)C)c1
E3 Binder	CHEMBL4643791	ChEMBL	6.15	—	—	CCN(c1ccc(C(=O)NO)cc1)S(=O)(=O)c1cccc(C(F)(F)F)c1
E3 Binder	CHEMBL4279707	ChEMBL	8.34	—	—	CCN1C(=O)C2Cc3c(n(Cc4ccc(C(=O)NO)cc4)c4ccccc34)CN2C1=O
E3 Binder	CHEMBL4288791	ChEMBL	8.1	—	—	CCN1CC(=O)N2Cc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)CC2C1=O
E3 Binder	CHEMBL1095764	ChEMBL	7.1	—	—	CCN1CCCC(n2c(-c3cccc(/C=C/C(=O)NO)c3)nc3ccccc32)C1
E3 Binder	CHEMBL1095136	ChEMBL	7.0	—	—	CCN1CCC[C@@H](n2c(-c3cccc(/C=C/C(=O)NO)c3)nc(-c3ccccc3)c2C)C1
E3 Binder	CHEMBL1095119	ChEMBL	7.1	—	—	CCN1CCC[C@@H](n2c(-c3cccc(/C=C/C(=O)NO)c3)nc(C)c2-c2ccccc2)C1
E3 Binder	CHEMBL1096033	ChEMBL	6.92	—	—	CCN1CCC[C@@H](n2c(-c3cccc(/C=C/C(=O)NO)c3)nc(C)c2C)C1
E3 Binder	CHEMBL1094077	ChEMBL	7.0	—	—	CCN1CCC[C@@H](n2c(-c3cccc(/C=C/C(=O)NO)c3)nc(Cc3ccccc3)c2C)C1
E3 Binder	CHEMBL1095765	ChEMBL	7.1	—	—	CCN1CCC[C@@H](n2c(-c3cccc(/C=C/C(=O)NO)c3)nc3ccccc32)C1
E3 Binder	CHEMBL1099065	ChEMBL	6.2	—	—	CCN1CCC[C@@H](n2c(-c3ccccc3)nc(C)c2-c2cccc(/C=C/C(=O)NO)c2)C1
E3 Binder	CHEMBL1095085	ChEMBL	6.4	—	—	CCN1CCC[C@@H](n2c(C)nc(C)c2-c2cccc(/C=C/C(=O)NO)c2)C1
E3 Binder	CHEMBL1098067	ChEMBL	6.3	—	—	CCN1CCC[C@@H](n2c(Cc3ccccc3)nc(C)c2-c2cccc(/C=C/C(=O)NO)c2)C1
E3 Binder	CHEMBL1095135	ChEMBL	7.1	—	—	CCN1CCC[C@H](n2c(-c3cccc(/C=C/C(=O)NO)c3)nc3ccccc32)C1
E3 Binder	CHEMBL2018305	ChEMBL	8.52	—	—	CCN1CCc2c(c3ccccc3n2Cc2ccc(C(=O)NO)cc2)C1
E3 Binder	CHEMBL471044	ChEMBL	6.94	—	—	CCNC(=O)SCC(=O)c1ccc(OC)cc1
E3 Binder	CHEMBL4228723	ChEMBL	6.95	—	—	CCNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)/C=C/c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4228653	ChEMBL	8.1	—	—	CCNC(=O)c1cc2c(-c3cccc(OCCCCCCOc4ccc(Nc5nc(-c6cnn(CCCCCCC(=O)NO)c6)c6cc[nH]c6n5)cc4)c3)nc(N)nc2s1
E3 Binder	CHEMBL462146	ChEMBL	6.51	—	—	CCNC(=O)c1ccc(C(=O)C(F)(F)F)s1
E3 Binder	CHEMBL3921290	ChEMBL	6.0	—	—	CCNC(=O)c1noc(-c2cc(Cl)c(O)cc2O)c1-c1ccc(OCCCC(=O)NO)cc1
E3 Binder	CHEMBL3942950	ChEMBL	7.0	—	—	CCNC(=O)c1noc(-c2cc(Cl)c(O)cc2O)c1-c1ccc(OCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3920405	ChEMBL	7.0	—	—	CCNC(=O)c1noc(-c2cc(Cl)c(O)cc2O)c1-c1ccc(OCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3956162	ChEMBL	7.0	—	—	CCNC(=O)c1noc(-c2cc(Cl)c(O)cc2O)c1-c1ccc(OCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL481297	ChEMBL	7.75	—	—	CCNC(=S)SCC(=O)c1ccc(NC(C)=O)cc1
E3 Binder	CHEMBL487615	ChEMBL	7.03	—	—	CCNC(=S)SCC(=O)c1ccc(OC)cc1
E3 Binder	CHEMBL5189799	ChEMBL	6.76	—	—	CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3ccc(C(F)(F)F)cc32)cc1
E3 Binder	CHEMBL5169915	ChEMBL	7.12	—	—	CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3ccc(C)cc32)cc1
E3 Binder	CHEMBL5200063	ChEMBL	7.43	—	—	CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3ccc(F)cc32)cc1
E3 Binder	CHEMBL5201672	ChEMBL	7.38	—	—	CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3ccccc32)cc1
E3 Binder	CHEMBL5173493	ChEMBL	8.52	—	—	CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3ccncc32)cc1
E3 Binder	CHEMBL5203278	ChEMBL	7.33	—	—	CCNNC(=O)c1ccc(CN2c3ccccc3C=Cc3nc(C)nc(C)c32)cc1
E3 Binder	CHEMBL5198893	ChEMBL	6.98	—	—	CCNNC(=O)c1ccc(CN2c3ccccc3CC(=O)c3ccccc32)cc1
E3 Binder	CHEMBL5205184	ChEMBL	6.6	—	—	CCNNC(=O)c1ccc(CN2c3ccccc3CCc3ccccc32)cc1
E3 Binder	CHEMBL5208188	ChEMBL	6.63	—	—	CCNNC(=O)c1ccc(CN2c3ccccc3Cc3ccccc32)cc1
E3 Binder	CHEMBL5172937	ChEMBL	6.07	—	—	CCNNC(=O)c1ccc(CN2c3ccccc3Oc3ccccc32)cc1
E3 Binder	CHEMBL5174152	ChEMBL	6.76	—	—	CCNNC(=O)c1ccc(CN2c3ccccc3Sc3ccccc32)cc1
E3 Binder	CHEMBL5191436	ChEMBL	7.21	—	—	CCNNC(=O)c1ccc(CN2c3ccccc3Sc3cccnc32)cc1
E3 Binder	CHEMBL5189990	ChEMBL	7.47	—	—	CCNNC(=O)c1ccc(CNC(=O)Nc2cccc3cccnc23)cc1
E3 Binder	CHEMBL4104334	ChEMBL	6.41	—	—	CCNNC(=O)c1ccc(CNC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(OC)cc2)cc1
E3 Binder	CHEMBL4752015	ChEMBL	7.11	—	—	CCNNC(=O)c1ccc(CNC(=O)c2ccccc2)cc1
E3 Binder	CHEMBL5177971	ChEMBL	7.39	—	—	CCNNC(=O)c1ccc(CNc2cccc3cccnc23)cc1
E3 Binder	CHEMBL5188941	ChEMBL	6.84	—	—	CCNNC(=O)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3ccccc32)cc1
E3 Binder	CHEMBL5184034	ChEMBL	6.34	—	—	CCNNC(=O)c1ccc(Cn2c3c(c4ccccc42)CCCC3)cc1
E3 Binder	CHEMBL5197272	ChEMBL	6.44	—	—	CCNNC(=O)c1ccc(Cn2c3ccccc3c3ccccc32)cc1
E3 Binder	CHEMBL5206738	ChEMBL	7.43	—	—	CCNNC(=O)c1ccc(Cn2c3ccccc3c3cccnc32)cc1
E3 Binder	CHEMBL5180229	ChEMBL	7.14	—	—	CCNNC(=O)c1ccc(Cn2c3ccccc3c3ccncc32)cc1
E3 Binder	CHEMBL5200361	ChEMBL	6.96	—	—	CCNNC(=O)c1ccc(Cn2c3ccccc3c3cnccc32)cc1
E3 Binder	CHEMBL5195924	ChEMBL	6.35	—	—	CCNNC(=O)c1ccc(Cn2ccc3cc(C(=O)c4ccc(OC)cc4)ccc32)cc1
E3 Binder	CHEMBL5197503	ChEMBL	7.8	—	—	CCNNC(=O)c1ccc(Cn2nnnc2-c2cccs2)cc1
E3 Binder	CHEMBL3759250	ChEMBL	6.54	—	—	CCOC(=O)N1CC2(CC(=O)c3cc(/C=C/C(=O)NO)ccc3O2)C1
E3 Binder	CHEMBL3758904	ChEMBL	6.82	—	—	CCOC(=O)N1CCC2(CC(=O)c3cc(/C=C/C(=O)NO)ccc3O2)C1
E3 Binder	CHEMBL1938432	ChEMBL	6.85	—	—	CCOC(=O)N1CCC2(CC1)CC(=O)c1cc(/C=C/C(=O)NO)ccc1O2
E3 Binder	CHEMBL1938438	ChEMBL	6.39	—	—	CCOC(=O)N1CCC2(CC1)CC(=O)c1ccc(/C=C/C(=O)NO)cc1O2
E3 Binder	CHEMBL3759450	ChEMBL	6.63	—	—	CCOC(=O)N1CCCC2(CC(=O)c3cc(/C=C/C(=O)NO)ccc3O2)C1
E3 Binder	CHEMBL3760116	ChEMBL	6.52	—	—	CCOC(=O)N1CCCC2(CC1)CC(=O)c1cc(/C=C/C(=O)NO)ccc1O2
E3 Binder	CHEMBL3086767	ChEMBL	6.36	—	—	CCOC(=O)NCCCC(=O)NCCc1ccccc1
E3 Binder	CHEMBL147134	ChEMBL	7.1	—	—	CCOC(=O)NCCSSCCNC(=O)/C(Cc1ccc(O)c(Br)c1)=N/O
E3 Binder	CHEMBL515411	ChEMBL	6.7	—	—	CCOC(=O)N[C@@H](CCCCNS(N)(=O)=O)C(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL4464421	ChEMBL	9.1	—	—	CCOC(=O)Nc1cccc(-c2csc(NC(=O)CCCCCC(=O)NO)n2)c1
E3 Binder	CHEMBL3943242	ChEMBL	8.3	—	—	CCOC(=O)Nc1cccc(-c2csc(NC(=O)CCCCCCC(=O)NO)n2)c1
E3 Binder	CHEMBL244831	ChEMBL	6.7	—	—	CCOC(=O)Nc1cccc(C(=O)CSC(=S)SCC)c1
E3 Binder	CHEMBL496703	ChEMBL	6.26	—	—	CCOC(=O)c1ccc(C(=O)C(F)(F)F)o1
E3 Binder	CHEMBL447397	ChEMBL	6.26	—	—	CCOC(=O)c1ccc(C(=O)C(F)(F)F)s1
E3 Binder	CHEMBL475042	ChEMBL	6.24	—	—	CCOC(=O)c1csc(NC(=O)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc2ccccc2)n1
E3 Binder	CHEMBL481136	ChEMBL	7.05	—	—	CCOC(=S)SCC(=O)c1ccc(NC(C)=O)cc1
E3 Binder	CHEMBL493249	ChEMBL	6.35	—	—	CCOC(=S)SCC(=O)c1ccc(OC)cc1
E3 Binder	CHEMBL3693801	ChEMBL	7.35	—	—	CCOC(c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1)(c1ccccn1)c1ccccn1
E3 Binder	CHEMBL3693800	ChEMBL	8.22	—	—	CCOC(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)(c1ccccn1)c1ccccn1
E3 Binder	CHEMBL3693799	ChEMBL	7.44	—	—	CCOC(c1ccccc1)(c1ccccc1)c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693794	ChEMBL	7.89	—	—	CCOC(c1ccccc1)(c1ccccc1)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3892427	ChEMBL	8.4	—	—	CCON1CCC(Nc2ncc(C(=O)NO)cn2)(C(C)C)CC1
E3 Binder	CHEMBL3901374	ChEMBL	8.54	—	—	CCON1CCC(Nc2ncc(C(=O)NO)cn2)(c2ccccc2)CC1
E3 Binder	CHEMBL4174805	ChEMBL	7.76	—	—	CCOc1cc(C(C)(C)C)ccc1C1=NC(c2ccc(Cl)cc2)C(c2ccc(Cl)cc2)N1C(=O)N1CCN(CCCCCCC(=O)NO)CC1
E3 Binder	CHEMBL3984639	ChEMBL	7.1	—	—	CCOc1ccc(-c2ccc(C(=O)NO)cn2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3956031	ChEMBL	6.07	—	—	CCOc1ccc(-c2ccc(C(=O)NO)nc2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3799246	ChEMBL	6.22	—	—	CCOc1ccc(C(=O)NO)cc1NC(=O)c1ccc(-c2ccccc2)cc1
E3 Binder	CHEMBL3798892	ChEMBL	6.0	—	—	CCOc1ccc(C(=O)Nc2cc(C(=O)NO)ccc2OC)cc1
E3 Binder	CHEMBL3901988	ChEMBL	6.89	—	—	CCOc1ccc(C2CC(C(=O)NO)C2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3900593	ChEMBL	7.04	—	—	CCOc1ccc(CC2CC(C(=O)NO)C2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3944571	ChEMBL	6.38	—	—	CCOc1ccc(CC2CCC(C(=O)NO)C2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3976546	ChEMBL	6.46	—	—	CCOc1ccc(CC2CCC(CC(=O)NO)CC2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3914813	ChEMBL	6.4	—	—	CCOc1ccc(CC2CCN(c3ccc(C(=O)NO)cn3)CC2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3427656	ChEMBL	7.16	—	—	CCOc1ccc(CCn2cccc(/C=C/C(=O)NO)c2=O)cc1
E3 Binder	CHEMBL3923840	ChEMBL	6.42	—	—	CCOc1ccc(CN2CCN(c3ncc(C(=O)NO)cn3)CC2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3940720	ChEMBL	7.24	—	—	CCOc1ccc(C[C@H]2CC[C@@H](C(=O)NO)CC2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3970271	ChEMBL	6.29	—	—	CCOc1ccc(C[C@H]2CC[C@H](C(=O)NO)CC2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3955253	ChEMBL	6.84	—	—	CCOc1ccc(C[C@H]2C[C@@H](C(=O)NO)C2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3982024	ChEMBL	6.9	—	—	CCOc1ccc(C[C@H]2C[C@H](C(=O)NO)C2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3936651	ChEMBL	6.43	—	—	CCOc1ccc(OC2CCN(c3ncc(C(=O)NO)cn3)CC2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL3974954	ChEMBL	6.71	—	—	CCOc1ccc(Oc2ccc(C(=O)NO)cc2)cc1-c1nc2c(CC)nn(C)c2c(=O)[nH]1
E3 Binder	CHEMBL4203874	ChEMBL	7.47	—	—	CCOc1cccc(-c2ccc3c(NC(=O)c4ccc(C(=O)NO)cc4)n[nH]c3c2)c1
E3 Binder	CHEMBL3427655	ChEMBL	6.92	—	—	CCOc1cccc(CCn2cccc(/C=C/C(=O)NO)c2=O)c1
E3 Binder	CHEMBL3427666	ChEMBL	7.3	—	—	CCOc1ccccc1CCCn1cccc(/C=C/C(=O)NO)c1=O
E3 Binder	CHEMBL3427654	ChEMBL	6.5	—	—	CCOc1ccccc1CCn1cccc(/C=C/C(=O)NO)c1=O
E3 Binder	CHEMBL242895	ChEMBL	7.3	—	—	CCSC(=S)SCC(=O)CCCCCCC(=O)Nc1ccccc1
E3 Binder	CHEMBL481703	ChEMBL	8.1	—	—	CCSC(=S)SCC(=O)c1ccc(-c2ccc(CNc3cnc4ccccc4c3)cn2)s1
E3 Binder	CHEMBL481878	ChEMBL	7.37	—	—	CCSC(=S)SCC(=O)c1ccc(-c2ccc(N)cn2)s1
E3 Binder	CHEMBL480973	ChEMBL	7.5	—	—	CCSC(=S)SCC(=O)c1ccc(C(=O)NCCOc2ccccc2)cc1
E3 Binder	CHEMBL479786	ChEMBL	7.82	—	—	CCSC(=S)SCC(=O)c1ccc(C(=O)NCc2cc(C)cc(C)c2)s1
E3 Binder	CHEMBL482270	ChEMBL	7.05	—	—	CCSC(=S)SCC(=O)c1ccc(C(=O)NCc2ccccc2)cc1
E3 Binder	CHEMBL482137	ChEMBL	7.72	—	—	CCSC(=S)SCC(=O)c1ccc(C(=O)NCc2ccccc2)s1
E3 Binder	CHEMBL517997	ChEMBL	7.31	—	—	CCSC(=S)SCC(=O)c1ccc(C(=O)N[C@@H](C)c2ccccc2)s1
E3 Binder	CHEMBL480005	ChEMBL	7.1	—	—	CCSC(=S)SCC(=O)c1ccc(C(=O)Nc2ccc(Cl)cc2)cc1
E3 Binder	CHEMBL517076	ChEMBL	7.13	—	—	CCSC(=S)SCC(=O)c1ccc(C(=O)Nc2ccccc2)cc1
E3 Binder	CHEMBL479970	ChEMBL	7.2	—	—	CCSC(=S)SCC(=O)c1ccc(C(=O)Nc2ccccc2)s1
E3 Binder	CHEMBL388710	ChEMBL	6.43	—	—	CCSC(=S)SCC(=O)c1ccc(C)cc1
E3 Binder	CHEMBL479602	ChEMBL	7.75	—	—	CCSC(=S)SCC(=O)c1ccc(CC(=O)NCCOc2ccccc2)s1
E3 Binder	CHEMBL516915	ChEMBL	7.58	—	—	CCSC(=S)SCC(=O)c1ccc(CC(=O)NCc2ccc(OC)cc2)s1
E3 Binder	CHEMBL479971	ChEMBL	7.42	—	—	CCSC(=S)SCC(=O)c1ccc(CC(=O)NCc2ccccc2)s1
E3 Binder	CHEMBL479601	ChEMBL	8.0	—	—	CCSC(=S)SCC(=O)c1ccc(CC(=O)Nc2ccc(OC)cc2)s1
E3 Binder	CHEMBL490067	ChEMBL	6.99	—	—	CCSC(=S)SCC(=O)c1ccc(CCNC(C)=O)cc1
E3 Binder	CHEMBL482287	ChEMBL	6.59	—	—	CCSC(=S)SCC(=O)c1ccc(CN(C)C(C)=O)cc1
E3 Binder	CHEMBL242896	ChEMBL	7.4	—	—	CCSC(=S)SCC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1
E3 Binder	CHEMBL482271	ChEMBL	7.34	—	—	CCSC(=S)SCC(=O)c1ccc(CNC(=O)c2ccccc2)cc1
E3 Binder	CHEMBL480884	ChEMBL	6.46	—	—	CCSC(=S)SCC(=O)c1ccc(CNC(C)=O)cc1
E3 Binder	CHEMBL242683	ChEMBL	7.1	—	—	CCSC(=S)SCC(=O)c1ccc(Cl)c(Cl)c1
E3 Binder	CHEMBL242038	ChEMBL	6.0	—	—	CCSC(=S)SCC(=O)c1ccc(Cl)cc1
E3 Binder	CHEMBL481131	ChEMBL	7.4	—	—	CCSC(=S)SCC(=O)c1ccc(NC(=O)Nc2ccccc2)cc1
E3 Binder	CHEMBL482280	ChEMBL	7.13	—	—	CCSC(=S)SCC(=O)c1ccc(NC(=O)c2ccccc2)cc1
E3 Binder	CHEMBL482095	ChEMBL	6.76	—	—	CCSC(=S)SCC(=O)c1ccc(NC(=O)c2cccnc2)cc1
E3 Binder	CHEMBL482075	ChEMBL	7.18	—	—	CCSC(=S)SCC(=O)c1ccc(NC(=O)c2cnc3ccccc3c2)cc1
E3 Binder	CHEMBL244199	ChEMBL	6.75	—	—	CCSC(=S)SCC(=O)c1ccc(NC(C)=O)cc1
E3 Binder	CHEMBL450723	ChEMBL	7.6	—	—	CCSC(=S)SCC(=O)c1ccc(NS(=O)(=O)c2ccc(Cl)cc2)cc1
E3 Binder	CHEMBL520781	ChEMBL	7.38	—	—	CCSC(=S)SCC(=O)c1ccc(NS(=O)(=O)c2ccccc2)cc1
E3 Binder	CHEMBL482094	ChEMBL	6.42	—	—	CCSC(=S)SCC(=O)c1ccc(Nc2ncnc3ccccc23)cc1
E3 Binder	CHEMBL243996	ChEMBL	6.1	—	—	CCSC(=S)SCC(=O)c1ccc(OC(F)F)cc1
E3 Binder	CHEMBL242039	ChEMBL	6.43	—	—	CCSC(=S)SCC(=O)c1ccc(OC)cc1
E3 Binder	CHEMBL517384	ChEMBL	8.1	—	—	CCSC(=S)SCC(=O)c1ccc(S(=O)(=O)Nc2ccc(Cl)cc2)cc1
E3 Binder	CHEMBL518961	ChEMBL	7.8	—	—	CCSC(=S)SCC(=O)c1ccc(S(=O)(=O)Nc2ccc(OC)cc2)cc1
E3 Binder	CHEMBL243998	ChEMBL	6.2	—	—	CCSC(=S)SCC(=O)c1ccc(S(N)(=O)=O)cc1
E3 Binder	CHEMBL242261	ChEMBL	6.3	—	—	CCSC(=S)SCC(=O)c1ccc2c(c1)OCCO2
E3 Binder	CHEMBL242472	ChEMBL	6.3	—	—	CCSC(=S)SCC(=O)c1ccc2c(c1)OCO2
E3 Binder	CHEMBL482272	ChEMBL	7.57	—	—	CCSC(=S)SCC(=O)c1cccc(C(=O)NCCOc2ccccc2)c1
E3 Binder	CHEMBL451289	ChEMBL	7.31	—	—	CCSC(=S)SCC(=O)c1cccc(C(=O)NCc2ccccc2)c1
E3 Binder	CHEMBL481922	ChEMBL	6.91	—	—	CCSC(=S)SCC(=O)c1cccc(C(=O)Nc2ccccc2)c1
E3 Binder	CHEMBL439842	ChEMBL	6.09	—	—	CCSC(=S)SCC(=O)c1cccc(CNC(C)=O)c1
E3 Binder	CHEMBL479611	ChEMBL	7.19	—	—	CCSC(=S)SCC(=O)c1cccc(NC(=O)c2ccccc2)c1
E3 Binder	CHEMBL519134	ChEMBL	7.42	—	—	CCSC(=S)SCC(=O)c1cccc(NC(=O)c2cccnc2)c1
E3 Binder	CHEMBL482096	ChEMBL	7.44	—	—	CCSC(=S)SCC(=O)c1cccc(NC(=O)c2cnc3ccccc3c2)c1
E3 Binder	CHEMBL242473	ChEMBL	6.48	—	—	CCSC(=S)SCC(=O)c1cccc(NC(C)=O)c1
E3 Binder	CHEMBL481955	ChEMBL	7.32	—	—	CCSC(=S)SCC(=O)c1cccc(NS(=O)(=O)c2ccc(Cl)cc2)c1
E3 Binder	CHEMBL482281	ChEMBL	6.98	—	—	CCSC(=S)SCC(=O)c1cccc(NS(=O)(=O)c2ccccc2)c1
E3 Binder	CHEMBL481311	ChEMBL	6.96	—	—	CCSC(=S)SCC(=O)c1cccc(S(=O)(=O)N(C)c2ccc(OC)cc2)c1
E3 Binder	CHEMBL481148	ChEMBL	7.82	—	—	CCSC(=S)SCC(=O)c1cccc(S(=O)(=O)Nc2ccc(OC)cc2)c1
E3 Binder	CHEMBL482136	ChEMBL	7.85	—	—	CCSC(=S)SCC(=O)c1cccc(S(=O)(=O)Nc2ccc3c(c2)OCO3)c1
E3 Binder	CHEMBL481319	ChEMBL	7.01	—	—	CCSC(=S)SCC(=O)c1cccc(S(=O)(=O)Nc2cccc(C(N)=O)c2)c1
E3 Binder	CHEMBL520279	ChEMBL	6.85	—	—	CCSC(=S)SCC(=O)c1ccn(S(=O)(=O)c2ccccc2)c1
E3 Binder	CHEMBL4551531	ChEMBL	7.51	—	—	CCSc1ccc2c(c1)N(Cc1ccc(C(=O)NO)cc1)c1ccccc1S2
E3 Binder	CHEMBL189497	ChEMBL	7.17	—	—	CC[C@@H](C(=O)Nc1ccc(C(=O)NO)cc1)c1ccccc1
E3 Binder	CHEMBL1790587	ChEMBL	8.48	—	—	CC[C@@H](C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCCN2C1=O
E3 Binder	CHEMBL4299384	ChEMBL	7.48	—	—	CC[C@@H]1OC(=O)[C@@H](C)[C@H](O[C@@H]2C[C@](C)(OC)[C@@](O)(CN(C)C)[C@@H](C)O2)[C@H](C)[C@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@@](C)(OC)C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299407	ChEMBL	7.5	—	—	CC[C@@H]1OC(=O)[C@@H](C)[C@H](O[C@@H]2C[C@](C)(OC)[C@@](O)(CN(C)C)[C@@H](C)O2)[C@H](C)[C@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@@](C)(OC)C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299469	ChEMBL	7.61	—	—	CC[C@@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@@H](C)[C@H](O[C@H]2O[C@@H](C)C[C@@H](N(C)C)[C@@H]2O)[C@](C)(O)C[C@H](C)CN(Cc2ccc(-c3cn(CCCCC(=O)NO)nn3)cc2)[C@H](C)[C@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299447	ChEMBL	8.33	—	—	CC[C@@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@@H](C)[C@H](O[C@H]2O[C@@H](C)C[C@@H](N(C)C)[C@@H]2O)[C@](C)(O)C[C@H](C)CN(Cc2ccc(-c3cn(CCCCCCC(=O)NO)nn3)cc2)[C@H](C)[C@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299429	ChEMBL	6.04	—	—	CC[C@@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCC(=O)NO)nn4)cc3)[C@H]2O)[C@@](C)(OC)C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299380	ChEMBL	6.92	—	—	CC[C@@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@@](C)(OC)C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299491	ChEMBL	8.18	—	—	CC[C@@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@@](C)(OC)C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299448	ChEMBL	6.57	—	—	CC[C@@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@](O)(CN(C)Cc3ccc(-c4cn(CCCCC(=O)NO)nn4)cc3)[C@H](C)O2)[C@H](C)[C@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C)[C@H]2O)[C@@](C)(OC)C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299370	ChEMBL	8.54	—	—	CC[C@@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@](O)(CN(C)Cc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc3)[C@H](C)O2)[C@H](C)[C@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C)[C@H]2O)[C@@](C)(OC)C[C@H](C)C(=O)[C@@H](C)[C@@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299362	ChEMBL	6.74	—	—	CC[C@@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@@](O)(CN(C)Cc3ccc(-c4cn(CCCC(=O)NO)nn4)cc3)[C@@H](C)O2)[C@@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299428	ChEMBL	7.5	—	—	CC[C@@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@@](O)(CN(C)Cc3ccc(-c4cn(CCCCCC(=O)NO)nn4)cc3)[C@@H](C)O2)[C@@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299445	ChEMBL	6.84	—	—	CC[C@@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@H](O)[C@@H](C)O2)[C@@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299411	ChEMBL	7.36	—	—	CC[C@@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@H](O)[C@@H](C)O2)[C@@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3cccc(-c4cn(CCCCCC(=O)NO)nn4)c3)[C@H]2O)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299419	ChEMBL	7.39	—	—	CC[C@@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@H](O)[C@@H](C)O2)[C@@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3cccc(-c4cn(CCCCCCC(=O)NO)nn4)c3)[C@H]2O)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299427	ChEMBL	6.75	—	—	CC[C@@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@H](O)[C@@H](C)O2)[C@@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccccc3-c3cn(CCCCCC(=O)NO)nn3)[C@H]2O)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299472	ChEMBL	7.51	—	—	CC[C@@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@H](O)[C@@H](C)O2)[C@@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccccc3-c3cn(CCCCCCC(=O)NO)nn3)[C@H]2O)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299468	ChEMBL	7.83	—	—	CC[C@@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@](O)(CN(C)C)[C@H](C)O2)[C@@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL4290191	ChEMBL	6.15	—	—	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2c-1nc1ccccc1c2/C=N/OCCCCCC(=O)NCCSSCCNC(=O)/C(Cc1ccc(O)c(Br)c1)=N\O
E3 Binder	CHEMBL2386910	ChEMBL	6.84	—	—	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3cc(OCc4cn(CCCCC(=O)NO)nn4)ccc3nc2-1
E3 Binder	CHEMBL2386911	ChEMBL	6.95	—	—	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3cc(OCc4cn(CCCCCC(=O)NO)nn4)ccc3nc2-1
E3 Binder	CHEMBL2386912	ChEMBL	7.25	—	—	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3cc(OCc4cn(CCCCCCC(=O)NO)nn4)ccc3nc2-1
E3 Binder	CHEMBL65	ChEMBL	7.3	EHD	—	CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1
E3 Binder	CHEMBL188270	ChEMBL	7.47	—	—	CC[C@H](C(=O)Nc1ccc(C(=O)NO)cc1)c1ccccc1
E3 Binder	CHEMBL2347006	ChEMBL	7.29	—	—	CC[C@H](C)C(=O)O[C@H]1C[C@@H](C)C=C2C=C[C@H](C)[C@H](CC[C@@H](O)C[C@@H](O)CC(=O)NO)[C@H]21
E3 Binder	CHEMBL5170036	ChEMBL	9.52	—	—	CC[C@H](C)C1NC(=O)C(Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCC(=O)C(C)O)NC(=O)[C@H]2CCCCN2C1=O
E3 Binder	CHEMBL1798008	ChEMBL	6.8	—	—	CC[C@H](C)[C@@H](CN1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1)NC(=O)CC(C)(C)C
E3 Binder	CHEMBL1798007	ChEMBL	7.03	—	—	CC[C@H](C)[C@@H](CN1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1)NC(=O)OC(C)(C)C
E3 Binder	CHEMBL253308	ChEMBL	6.51	—	—	CC[C@H](C)[C@@H]1NC(=O)C(C)(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
E3 Binder	CHEMBL2371803	ChEMBL	6.75	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@@H](Cc2ccc(OC)cc2)NC(=O)[C@H](CCCCSCC(=O)C(F)(F)F)NC(=O)[C@H]2CCCN2C1=O
E3 Binder	CHEMBL1793828	ChEMBL	6.55	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCC(=O)O)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL2371005	ChEMBL	7.13	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCC(=O)OC)NC(=O)[C@H]2CCCCN2C1=O
E3 Binder	CHEMBL1793936	ChEMBL	7.13	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCC(=O)OC)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL1793824	ChEMBL	7.52	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)C(C)=O)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL1793946	ChEMBL	6.63	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)C(C)C)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL2371003	ChEMBL	9.0	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)C(C)F)NC(=O)[C@H]2CCCCN2C1=O
E3 Binder	CHEMBL1793823	ChEMBL	9.0	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)C(C)F)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL2370998	ChEMBL	9.52	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)C(C)O)NC(=O)[C@H]2CCCCN2C1=O
E3 Binder	CHEMBL1793822	ChEMBL	9.52	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)C(C)O)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL2371007	ChEMBL	9.7	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCCCN2C1=O
E3 Binder	CHEMBL1793811	ChEMBL	9.7	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL2370999	ChEMBL	7.82	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)O)NC(=O)[C@H]2CCCCN2C1=O
E3 Binder	CHEMBL1793827	ChEMBL	7.82	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)O)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL2371000	ChEMBL	9.4	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)OC)NC(=O)[C@H]2CCCCN2C1=O
E3 Binder	CHEMBL1793816	ChEMBL	9.4	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)OC)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL1793942	ChEMBL	6.16	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(=O)c2ccccc2)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL1793938	ChEMBL	8.7	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC(C)=O)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL1793813	ChEMBL	7.22	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC2(CC)CO2)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL1793937	ChEMBL	8.22	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCC=O)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL1793821	ChEMBL	6.07	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCCC(=O)O)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL2371004	ChEMBL	8.15	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCCC(=O)OC)NC(=O)[C@H]2CCCCN2C1=O
E3 Binder	CHEMBL1793819	ChEMBL	8.15	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCCC(=O)OC)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL1793809	ChEMBL	6.35	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCP(=O)(OC)OC)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL1793818	ChEMBL	6.75	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCP(=O)([O-])O)NC(=O)[C@H]2CCCCN2CC1=O.[K+]
E3 Binder	CHEMBL1793945	ChEMBL	8.52	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCSC(C)=O)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL1793940	ChEMBL	6.49	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCCSC)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL1793939	ChEMBL	6.96	—	—	CC[C@H](C)[C@@H]1NC(=O)[C@H](Cc2cn(OC)c3ccccc23)NC(=O)[C@H](CCCCSC(C)=O)NC(=O)[C@H]2CCCCN2CC1=O
E3 Binder	CHEMBL1798003	ChEMBL	6.79	—	—	CC[C@H](C)[C@H](NC(=O)C1CCN(C(=O)OC(C)(C)C)CC1)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1
E3 Binder	CHEMBL1798006	ChEMBL	7.15	—	—	CC[C@H](C)[C@H](NC(=O)C1CCNCC1)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1.Cl
E3 Binder	CHEMBL1828920	ChEMBL	7.28	—	—	CC[C@H](C)[C@H](NC(=O)CC(C)(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1
E3 Binder	CHEMBL1797983	ChEMBL	7.33	—	—	CC[C@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1
E3 Binder	CHEMBL2336048	ChEMBL	6.42	—	—	CC[C@H](C)[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](COc1ccc(/C=C/C(=O)NO)cc1OC)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL1798005	ChEMBL	7.14	—	—	CC[C@H](C)[C@H](NC(=O)[C@@H](N)C(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1.Cl
E3 Binder	CHEMBL1798002	ChEMBL	6.94	—	—	CC[C@H](C)[C@H](NC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1
E3 Binder	CHEMBL1798004	ChEMBL	6.97	—	—	CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1.Cl
E3 Binder	CHEMBL1798001	ChEMBL	7.19	—	—	CC[C@H](C)[C@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(=O)N1Cc2cc(OCC(=O)NO)ccc2C[C@H]1C(=O)Nc1ccc(OC)cc1
E3 Binder	CHEMBL1164599	ChEMBL	6.52	—	—	CC[C@H](C)[C@H]1CC(=O)NCC(=O)N[C@@H](CCCCCC(=O)O)C(=O)N[C@@H](Cc2cc3ccccc3[nH]2)C(=O)N1
E3 Binder	CHEMBL1836144	ChEMBL	6.42	—	—	CC[C@H](C)[C@H]1NC(=O)[C@@H](CS)NC(=O)[C@@H](CCSC)NC(=O)C[C@@H](/C=C/CCS)OC(=O)C[C@@H]1O
E3 Binder	CHEMBL1836142	ChEMBL	6.08	—	—	CC[C@H](C)[C@H]1NC(=O)[C@H]2CSSCC/C=C/[C@H](CC(=O)N[C@H](CCSC)C(=O)N2)OC(=O)C[C@@H]1O
E3 Binder	CHEMBL4459679	ChEMBL	8.4	—	—	CC[C@H](Nc1cc(C)nc(N)n1)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4439481	ChEMBL	7.85	—	—	CC[C@H](Nc1nc(C)nc(N)c1C#N)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4450191	ChEMBL	7.28	—	—	CC[C@H](Nc1nc(N)nc(C(F)(F)F)c1C#N)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4435002	ChEMBL	7.57	—	—	CC[C@H](Nc1nc(N)nc(C(F)F)c1C#N)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4443378	ChEMBL	7.55	—	—	CC[C@H](Nc1nc(N)nc(C)c1C#N)c1nc2cccc(CCCCCC(=O)NO)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4455923	ChEMBL	7.92	—	—	CC[C@H](Nc1nc(N)nc(C)c1C#N)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4449301	ChEMBL	7.66	—	—	CC[C@H](Nc1nc(N)nc(C)c1Cl)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4452989	ChEMBL	7.33	—	—	CC[C@H](Nc1nc(N)nc(C2CC2)c1C#N)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4550648	ChEMBL	7.16	—	—	CC[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(CCCCCC(=O)NO)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4450613	ChEMBL	7.11	—	—	CC[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(CCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL5220776	ChEMBL	7.35	—	—	CC[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(C(=O)NO)s1
E3 Binder	CHEMBL4464812	ChEMBL	8.4	—	—	CC[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4448226	ChEMBL	8.05	—	—	CC[C@H](Nc1nc(N)nc(N)c1Cl)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4525968	ChEMBL	7.35	—	—	CC[C@H](Nc1nc(N)ncc1C)c1nc2cccc(CCCCCC(=O)NO)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4578757	ChEMBL	8.4	—	—	CC[C@H](Nc1ncnc(N)c1C#N)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4467927	ChEMBL	8.4	—	—	CC[C@H](Nc1ncnc(N)c1Cl)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4456827	ChEMBL	8.52	—	—	CC[C@H](Nc1ncnc(N)c1Cl)c1nc2cccc(NCc3ccc(C(=O)NO)cn3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4539040	ChEMBL	7.41	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc(CCCCCC(=O)NO)c2ccccc2n1
E3 Binder	CHEMBL4439820	ChEMBL	6.37	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc(NCCCC(=O)NO)c2ccccc2n1
E3 Binder	CHEMBL4563838	ChEMBL	6.44	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(-c3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4445342	ChEMBL	7.44	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CCCCC(=O)NO)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4451623	ChEMBL	8.3	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CCCCCC(=O)NO)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4555432	ChEMBL	6.05	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4464003	ChEMBL	8.0	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CNC(=O)c3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4581057	ChEMBL	8.22	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(CNc3ncc(C(=O)NO)cn3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL5221043	ChEMBL	6.92	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(F)c2c(=O)n1CCCCCC(=O)NO
E3 Binder	CHEMBL5218549	ChEMBL	7.35	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(F)c2c(=O)n1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4588261	ChEMBL	7.43	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(NCCCC(=O)NO)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4516095	ChEMBL	8.3	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4443548	ChEMBL	8.05	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(NCc3ccc(C(=O)NO)cn3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4445210	ChEMBL	6.77	—	—	CC[C@H](Nc1ncnc2[nH]cnc12)c1nc2cccc(NCc3ccc(C(=O)NO)nc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4299391	ChEMBL	6.97	—	—	CC[C@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@H](O[C@H]2O[C@@H](C)C[C@@H](N(C)Cc3ccc(-c4cn(CCCC(=O)NO)nn4)cc3)[C@@H]2O)[C@@](C)(O)C[C@H](C)CN(C)[C@@H](C)[C@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299470	ChEMBL	7.84	—	—	CC[C@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@H](O[C@H]2O[C@@H](C)C[C@@H](N(C)Cc3ccc(-c4cn(CCCCCC(=O)NO)nn4)cc3)[C@@H]2O)[C@@](C)(O)C[C@H](C)CN(C)[C@@H](C)[C@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299417	ChEMBL	8.14	—	—	CC[C@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@H](O[C@H]2O[C@@H](C)C[C@@H](N(C)Cc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc3)[C@@H]2O)[C@@](C)(O)C[C@H](C)CN(C)[C@@H](C)[C@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299467	ChEMBL	7.72	—	—	CC[C@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@](O)(CN(C)C)[C@H](C)O2)[C@H](C)[C@H](O[C@H]2O[C@@H](C)C[C@@H](N(C)Cc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc3)[C@@H]2O)[C@@](C)(O)C[C@H](C)CN(C)[C@@H](C)[C@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299456	ChEMBL	7.02	—	—	CC[C@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@](O)(CN(C)Cc3ccc(-c4cn(CCCCC(=O)NO)nn4)cc3)[C@H](C)O2)[C@H](C)[C@H](O[C@H]2O[C@@H](C)C[C@@H](N(C)C)[C@@H]2O)[C@@](C)(O)C[C@H](C)CN(C)[C@@H](C)[C@H](O)[C@@]1(C)O
E3 Binder	CHEMBL4299488	ChEMBL	7.5	—	—	CC[C@H]1OC(=O)[C@@H](C)[C@H](O[C@H]2C[C@@](C)(OC)[C@](O)(CN(C)Cc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc3)[C@H](C)O2)[C@H](C)[C@H](O[C@H]2O[C@@H](C)C[C@@H](N(C)C)[C@@H]2O)[C@@](C)(O)C[C@H](C)CN(C)[C@@H](C)[C@H](O)[C@@]1(C)O
E3 Binder	CHEMBL3735456	ChEMBL	6.71	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCC(=O)NO)nn4)cc3)[C@H]2O)[C@@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL3734952	ChEMBL	7.11	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL3735736	ChEMBL	8.05	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL1214759	ChEMBL	8.11	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL3736342	ChEMBL	8.16	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL1214760	ChEMBL	8.99	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL1214761	ChEMBL	6.98	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL1214762	ChEMBL	6.79	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL1214763	ChEMBL	6.68	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL3735212	ChEMBL	7.76	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3cccc(-c4cn(CCCCCC(=O)NO)nn4)c3)[C@H]2O)[C@@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL3736314	ChEMBL	8.43	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3cccc(-c4cn(CCCCCCC(=O)NO)nn4)c3)[C@H]2O)[C@@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL3734946	ChEMBL	6.61	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccccc3-c3cn(CCCCCC(=O)NO)nn3)[C@H]2O)[C@@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL3736170	ChEMBL	7.12	—	—	CC[C@H]1OC(=O)[C@H](C)C(=O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccccc3-c3cn(CCCCCCC(=O)NO)nn3)[C@H]2O)[C@@](C)(OC)C[C@@H](C)C2=NCCN3C(=O)O[C@@]1(C)[C@H]3[C@H]2C
E3 Binder	CHEMBL504040	ChEMBL	6.93	—	—	CC[C@H]1OC(=O)[C@H](C)[C@@H](O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL472250	ChEMBL	6.83	—	—	CC[C@H]1OC(=O)[C@H](C)[C@@H](O)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@](C)(OC)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299368	ChEMBL	6.44	—	—	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@@](O)(CN(C)Cc3ccc(-c4cn(CCCC(=O)NO)nn4)cc3)[C@@H](C)O2)[C@@H](C)[C@@H](O[C@H]2O[C@@H](C)C[C@@H](N(C)C)[C@@H]2O)[C@](C)(OC)C[C@@H](C)C(=O)[C@H](C)[C@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299426	ChEMBL	8.23	—	—	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@@](O)(CN(C)Cc3ccc(-c4cn(CCCCCC(=O)NO)nn4)cc3)[C@@H](C)O2)[C@@H](C)[C@@H](O[C@H]2O[C@@H](C)C[C@@H](N(C)C)[C@@H]2O)[C@](C)(OC)C[C@@H](C)C(=O)[C@H](C)[C@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299406	ChEMBL	7.15	—	—	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@H](O)[C@@H](C)O2)[C@@H](C)[C@@H](O[C@H]2O[C@@H](C)C[C@@H](N(C)Cc3ccc(-c4cn(CCCC(=O)NO)nn4)cc3)[C@@H]2O)[C@](C)(OC)C[C@@H](C)C(=O)[C@H](C)[C@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299435	ChEMBL	8.44	—	—	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@H](O)[C@@H](C)O2)[C@@H](C)[C@@H](O[C@H]2O[C@@H](C)C[C@@H](N(C)Cc3ccc(-c4cn(CCCCCC(=O)NO)nn4)cc3)[C@@H]2O)[C@](C)(OC)C[C@@H](C)C(=O)[C@H](C)[C@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299403	ChEMBL	6.21	—	—	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@H](O)[C@@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C)[C@H]2O)[C@@](C)(O)C[C@@H](C)CN(Cc2ccc(-c3cn(CCCC(=O)NO)nn3)cc2)[C@@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL4299449	ChEMBL	7.99	—	—	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@@H]2C[C@](C)(OC)[C@H](O)[C@@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C)[C@H]2O)[C@@](C)(O)C[C@@H](C)CN(Cc2ccc(-c3cn(CCCCCC(=O)NO)nn3)cc2)[C@@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL506834	ChEMBL	7.11	—	—	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL455735	ChEMBL	7.05	—	—	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)Cc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc3)[C@H]2O)[C@](C)(OC)C[C@@H](C)C(=O)[C@H](C)[C@@H](O)[C@]1(C)O
E3 Binder	CHEMBL472574	ChEMBL	7.66	—	—	CC[C@]1(C)NC(=O)[C@H](CCCCCC(=O)[C@@H](C)O)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O
E3 Binder	CHEMBL513595	ChEMBL	7.77	—	—	CC[C@]1(C)NC(=O)[C@H](CCCCCC(=O)[C@@H](C)O)NC(=O)[C@H]2C[C@H](C)CN2C(=O)[C@H](Cc2ccccc2)NC1=O
E3 Binder	CHEMBL4761829	ChEMBL	6.72	—	—	CC[N+]1=C(/C=C/C2=C3Oc4cc(O)cc(OCCCCCCCC(=O)NO)c4C=C3CCC2)C(C)(C)c2ccccc21.[I-]
E3 Binder	CHEMBL5275736	ChEMBL	8.02	—	—	CC[N+]1=C(/C=C/C=C/C=C2/N(CCCCC(=O)N(CCc3c(C)[nH]c4ccccc34)Cc3ccc(/C=C/C(=O)NO)cc3)c3ccc4c(S(=O)(=O)O)cc(S(=O)(=O)O)cc4c3C2(C)C)C(C)(C)c2c1ccc1c(S(=O)(=O)[O-])cc(S(=O)(=O)O)cc21
E3 Binder	CHEMBL5079915	ChEMBL	7.1	—	—	CCc1c(C(=O)Nc2cc(/C=C/C(=O)NO)ccc2O)[nH]c(C)c1C(C)=O
E3 Binder	CHEMBL5077168	ChEMBL	7.38	—	—	CCc1c(C(=O)Nc2cc(/C=C/C(=O)NO)ccc2OC)[nH]c(C)c1C(C)=O
E3 Binder	CHEMBL5092849	ChEMBL	7.14	—	—	CCc1c(C(=O)Nc2cc(S(=O)(=O)Nc3cccc(/C=C/C(=O)NO)c3)ccc2OC)[nH]c(C)c1C(C)=O
E3 Binder	CHEMBL5094795	ChEMBL	7.35	—	—	CCc1c(C(=O)Nc2cccc(/C=C/C(=O)NO)c2)[nH]c(C)c1C(C)=O
E3 Binder	CHEMBL5094765	ChEMBL	6.18	S7T	—	CCc1c(C(=O)Nc2cccc(CCC(=O)NO)c2)[nH]c(C)c1C(C)=O
E3 Binder	CHEMBL4237494	ChEMBL	6.66	—	—	CCc1c2c(nc3ccc(O)cc13)-c1cc3c(c(=O)n1C2)COC(=O)[C@@]3(CC)OC(=O)CCCCCC(=O)NO
E3 Binder	CHEMBL4241658	ChEMBL	6.6	—	—	CCc1c2c(nc3ccc(O)cc13)-c1cc3c(c(=O)n1C2)COC(=O)[C@@]3(CC)OC(=O)CCCCCCC(=O)NO
E3 Binder	CHEMBL4248849	ChEMBL	6.68	—	—	CCc1c2c(nc3ccc(O)cc13)-c1cc3c(c(=O)n1C2)COC(=O)[C@@]3(CC)OC(=O)CCCCCCCC(=O)NO
E3 Binder	CHEMBL4237816	ChEMBL	6.5	—	—	CCc1c2c(nc3ccc(O)cc13)-c1cc3c(c(=O)n1C2)COC(=O)[C@@]3(CC)OC(=O)CCCCCCCCC(=O)NO
E3 Binder	CHEMBL4242465	ChEMBL	6.21	—	—	CCc1c2c(nc3ccc(O)cc13)-c1cc3c(c(=O)n1C2)COC(=O)[C@@]3(CC)OC(=O)CCCCCCCCCC(=O)NO
E3 Binder	CHEMBL4248785	ChEMBL	6.07	—	—	CCc1c2c(nc3ccc(O)cc13)-c1cc3c(c(=O)n1C2)COC(=O)[C@@]3(CC)OC(=O)CNC(=O)CCCCCCC(=O)NO
E3 Binder	CHEMBL2386905	ChEMBL	7.07	—	—	CCc1c2c(nc3ccc(OCc4cn(CCCC(=O)NO)nn4)cc13)-c1cc3c(c(=O)n1C2)COC(=O)[C@]3(O)CC
E3 Binder	CHEMBL2386906	ChEMBL	6.81	—	—	CCc1c2c(nc3ccc(OCc4cn(CCCCC(=O)NO)nn4)cc13)-c1cc3c(c(=O)n1C2)COC(=O)[C@]3(O)CC
E3 Binder	CHEMBL2386907	ChEMBL	7.38	—	—	CCc1c2c(nc3ccc(OCc4cn(CCCCCC(=O)NO)nn4)cc13)-c1cc3c(c(=O)n1C2)COC(=O)[C@]3(O)CC
E3 Binder	CHEMBL2386908	ChEMBL	7.44	—	—	CCc1c2c(nc3ccc(OCc4cn(CCCCCCC(=O)NO)nn4)cc13)-c1cc3c(c(=O)n1C2)COC(=O)[C@]3(O)CC
E3 Binder	CHEMBL2386909	ChEMBL	7.12	—	—	CCc1c2c(nc3ccc(OCc4cn(CCCCCCCC(=O)NO)nn4)cc13)-c1cc3c(c(=O)n1C2)COC(=O)[C@]3(O)CC
E3 Binder	CHEMBL4226024	ChEMBL	7.16	—	—	CCc1cc(-c2ccc(F)cc2)n(Cc2ccc(C(=O)NO)cc2)n1
E3 Binder	CHEMBL4224911	ChEMBL	7.46	—	—	CCc1cc(-c2ccc(F)cc2)nn1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3427662	ChEMBL	6.51	—	—	CCc1ccc(CCCn2cccc(/C=C/C(=O)NO)c2=O)cc1
E3 Binder	CHEMBL3427651	ChEMBL	7.16	—	—	CCc1ccc(CCn2cccc(/C=C/C(=O)NO)c2=O)cc1
E3 Binder	CHEMBL3427641	ChEMBL	7.0	—	—	CCc1ccc(Cn2cccc(/C=C/C(=O)NO)c2=O)cc1
E3 Binder	CHEMBL1093042	ChEMBL	7.58	—	—	CCc1ccc(NC(=O)CCCCC(=O)NO)cc1
E3 Binder	CHEMBL4062908	ChEMBL	7.01	—	—	CCc1ccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)cc1
E3 Binder	CHEMBL1093041	ChEMBL	7.68	—	—	CCc1cccc(NC(=O)CCCCC(=O)NO)c1
E3 Binder	CHEMBL4089922	ChEMBL	7.23	—	—	CCc1cccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c1
E3 Binder	CHEMBL3427640	ChEMBL	6.64	—	—	CCc1ccccc1Cn1cccc(/C=C/C(=O)NO)c1=O
E3 Binder	CHEMBL1093040	ChEMBL	6.67	—	—	CCc1ccccc1NC(=O)CCCCC(=O)NO
E3 Binder	CHEMBL4634096	ChEMBL	7.14	—	—	CCc1nc(N)nc(N)c1-c1ccc(-c2ccc(/C=C/C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4649487	ChEMBL	7.34	—	—	CCc1nc(N)nc(N)c1-c1ccc(-c2cn(CCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL4635479	ChEMBL	7.77	—	—	CCc1nc(N)nc(N)c1-c1ccc(-c2cn(CCCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL4636452	ChEMBL	7.68	—	—	CCc1nc(N)nc(N)c1-c1ccc(-c2cn(CCCCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL4633409	ChEMBL	6.4	—	—	CCc1nc(N)nc(N)c1-c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL2425952	ChEMBL	7.1	—	—	CCc1nc2c(Cc3ccc(C(=O)NO)cc3)cccc2c(=O)n1CCc1ccccc1
E3 Binder	CHEMBL2425967	ChEMBL	7.85	—	—	CCc1nc2cc(/C=C/C(=O)NO)c(F)cc2c(=O)n1CCc1ccccc1
E3 Binder	CHEMBL2425962	ChEMBL	7.48	—	—	CCc1nc2cc(/C=C/C(=O)NO)ccc2c(=O)n1CCCc1ccccc1
E3 Binder	CHEMBL2425966	ChEMBL	7.37	—	—	CCc1nc2cc(/C=C/C(=O)NO)ccc2c(=O)n1CCc1ccc(F)cc1
E3 Binder	CHEMBL2425965	ChEMBL	7.39	—	—	CCc1nc2cc(/C=C/C(=O)NO)ccc2c(=O)n1CCc1ccc(OC)cc1
E3 Binder	CHEMBL2425961	ChEMBL	7.96	—	—	CCc1nc2cc(/C=C/C(=O)NO)ccc2c(=O)n1CCc1ccccc1
E3 Binder	CHEMBL2425971	ChEMBL	8.05	—	—	CCc1nc2cc(Cc3ccc(C(=O)NO)cc3)ccc2c(=O)n1CCc1ccccc1
E3 Binder	CHEMBL2425969	ChEMBL	6.13	—	—	CCc1nc2cc(Cl)c(/C=C/C(=O)NO)cc2c(=O)n1CCc1ccccc1
E3 Binder	CHEMBL2425968	ChEMBL	8.1	—	—	CCc1nc2cc(F)c(/C=C/C(=O)NO)cc2c(=O)n1CCc1ccccc1
E3 Binder	CHEMBL2425970	ChEMBL	7.96	—	—	CCc1nc2ccc(Cc3ccc(C(=O)NO)cc3)cc2c(=O)n1CCc1ccccc1
E3 Binder	CHEMBL3287252	ChEMBL	6.03	—	—	CCc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO
E3 Binder	CHEMBL3329992	ChEMBL	8.47	—	—	CCn1c(C)c(CCNS(=O)(=O)c2ccc(/C=C/C(=O)NO)cc2)c2ccccc21
E3 Binder	CHEMBL5287701	ChEMBL	8.48	—	—	CCn1c(C)c(CCNS(=O)(=O)c2ccc(/C=C/C=C/C(=O)NO)cc2)c2ccccc21
E3 Binder	CHEMBL4438671	ChEMBL	7.44	—	—	CCn1cnc(-c2ccc(OC)cc2)c1-c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4562156	ChEMBL	6.97	—	—	CCn1cnc(-c2ccccc2)c1-c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL3763388	ChEMBL	7.57	—	—	CN(/N=C/c1ccc(C(=O)NO)cc1)C(=O)c1ccc(N(C)C)cc1
E3 Binder	CHEMBL190359	ChEMBL	6.28	—	—	CN(C(=O)CCCc1ccccc1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4464527	ChEMBL	6.93	—	—	CN(C(=O)CN(C)S(=O)(=O)c1ccc(F)cc1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4565392	ChEMBL	7.7	—	—	CN(C(=O)CN(Cc1c(F)c(F)c(F)c(F)c1F)S(=O)(=O)c1ccc(F)cc1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3972758	ChEMBL	8.66	—	—	CN(C(=O)N1CCC(Nc2ncc(C(=O)NO)cn2)(c2ccccc2)CC1)c1ccccc1
E3 Binder	CHEMBL3640673	ChEMBL	8.4	—	—	CN(C)C(=O)c1ccc(C(O)(c2ccccc2)c2ccc(C(=O)NCCCCCCC(=O)NO)cc2)cc1
E3 Binder	CHEMBL3640674	ChEMBL	8.52	—	—	CN(C)C(=O)c1cccc(C(O)(c2ccccc2)c2ccc(C(=O)NCCCCCCC(=O)NO)cc2)c1
E3 Binder	CHEMBL4086671	ChEMBL	8.07	—	—	CN(C)C(=O)c1cn(Cc2ccc(/C=C/C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL4096845	ChEMBL	8.1	—	—	CN(C)C(=O)c1cn(Cc2ccc(C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL4104572	ChEMBL	7.97	—	—	CN(C)C(=O)c1cn(S(=O)(=O)c2ccc(/C=C/C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL4078822	ChEMBL	6.7	—	—	CN(C)C(=O)c1cn(S(=O)(=O)c2cccc(/C=C/C(=O)NO)c2)c2ccccc12
E3 Binder	CHEMBL5270464	ChEMBL	6.07	—	—	CN(C)C1=NC2C(Br)=C(Br)C(Br)=C(Br)C2N1CCCCCC(=O)NO
E3 Binder	CHEMBL1830397	ChEMBL	7.03	—	—	CN(C)CC(C)(C)Cn1c(CC(C)(C)C)nc2cc(/C=C/C(=O)NO)ccc21
E3 Binder	CHEMBL460963	ChEMBL	7.64	—	—	CN(C)CC(C)(C)Cn1c(CCc2ccccc2)nc2cc(/C=C/C(=O)NO)ccc21
E3 Binder	CHEMBL5192285	ChEMBL	6.19	—	—	CN(C)CCCNC(=O)c1ccc(/C=C2\CCn3c2nc2cc(N4CCN(CCCCCCCC(=O)NO)CC4)c(F)cc2c3=O)cc1.Cl
E3 Binder	CHEMBL5194009	ChEMBL	7.16	—	—	CN(C)CCCNC(=O)c1ccc(/C=C2\CCn3c2nc2cc(NCCCCCCC(=O)NO)c(F)cc2c3=O)cc1.Cl
E3 Binder	CHEMBL5177837	ChEMBL	7.22	—	—	CN(C)CCCNC(=O)c1ccc(/C=C2\CCn3c2nc2ccc(OCCCCCCC(=O)NO)cc2c3=O)cc1.Cl
E3 Binder	CHEMBL18786	ChEMBL	6.09	—	—	CN(C)CCCSc1ccccc1NC(=O)/C=C/c1ccccc1
E3 Binder	CHEMBL4763662	ChEMBL	6.89	—	—	CN(C)CCNC(=O)c1ccc([C@H]2C[C@@H]2NCC2CCN(CCCc3ccc(C(=O)NO)cc3)CC2)cc1
E3 Binder	CHEMBL285802	ChEMBL	6.22	ZOT	—	CN(C)CCOC1=Cc2ccccc2Sc2ccc(Cl)cc21
E3 Binder	CHEMBL4798571	ChEMBL	7.59	—	—	CN(C)CCOc1ccc(-c2cc(=O)c3c(O)cc(OCCCCCC(=O)NO)cc3o2)cc1.Cl
E3 Binder	CHEMBL494526	ChEMBL	6.75	—	—	CN(C)CCOc1ccc(-c2nc([C@H](CCCCNS(N)(=O)=O)NC(=O)OCc3ccccc3)cs2)cc1
E3 Binder	CHEMBL3907295	ChEMBL	7.9	TWV	—	CN(C)CCc1cn(Cc2ccc(C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL3952983	ChEMBL	6.9	—	—	CN(C)CCc1nc2ccccc2n1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL1095710	ChEMBL	7.1	—	—	CN(C)CCn1c(-c2cccc(/C=C/C(=O)NO)c2)nc2ccccc21
E3 Binder	CHEMBL2103863	ChEMBL	7.92	—	—	CN(C)Cc1c(C(=O)NCCOc2ccc(C(=O)NO)cc2)oc2ccccc12
E3 Binder	CHEMBL4296717	ChEMBL	7.31	P7D	—	CN(C)Cc1ccc(S(=O)(=O)n2ccc(/C=C/C(=O)NO)c2)cc1
E3 Binder	CHEMBL4102147	ChEMBL	7.37	—	—	CN(C)Cc1cn(Cc2ccc(/C=C/C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL4066920	ChEMBL	7.66	TWM	—	CN(C)Cc1cn(Cc2ccc(C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL4077893	ChEMBL	7.78	—	—	CN(C)Cc1cn(S(=O)(=O)c2ccc(/C=C/C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL4094410	ChEMBL	7.05	—	—	CN(C)Cc1cn(S(=O)(=O)c2cccc(/C=C/C(=O)NO)c2)c2ccccc12
E3 Binder	CHEMBL4470067	ChEMBL	6.9	—	—	CN(C)Cc1nn(Cc2ccc(C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL4637992	ChEMBL	7.39	—	—	CN(C)S(=O)(=O)c1ccc(NCCCCCC(=O)NO)c2nonc12
E3 Binder	CHEMBL4647479	ChEMBL	7.96	—	—	CN(C)S(=O)(=O)c1ccc(NCCCCCCC(=O)NO)c2nonc12
E3 Binder	CHEMBL3640701	ChEMBL	7.48	—	—	CN(C)[C@@H]1CCN(c2ncc(C(=O)NCCCCCCC(=O)NO)cn2)C1
E3 Binder	CHEMBL3958552	ChEMBL	7.92	—	—	CN(C)c1ccc(-c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL478115	ChEMBL	8.37	—	—	CN(C)c1ccc(-c2cn(CCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL478116	ChEMBL	6.97	—	—	CN(C)c1ccc(-c2cn(CCCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL590567	ChEMBL	7.8	—	—	CN(C)c1ccc(-c2cn(CCCCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL590566	ChEMBL	6.22	—	—	CN(C)c1ccc(-c2cn(CCCCCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL3110282	ChEMBL	6.0	—	—	CN(C)c1ccc(-c2cn(CCCCCn3cccc(O)c3=S)nn2)cc1
E3 Binder	CHEMBL5278415	ChEMBL	8.12	—	—	CN(C)c1ccc(-c2nc(C(=O)NCc3ccc(/C=C/C(=O)NO)cc3)cc3c2[nH]c2ccccc23)cc1
E3 Binder	CHEMBL328710	ChEMBL	6.2	—	—	CN(C)c1ccc(/C=C2\C(=O)Nc3ccccc32)cc1
E3 Binder	CHEMBL459265	ChEMBL	6.02	CVI	—	CN(C)c1ccc(C(=C2C=CC(=[N+](C)C)C=C2)c2ccc(N(C)C)cc2)cc1
E3 Binder	CHEMBL5209024	ChEMBL	7.7	—	—	CN(C)c1ccc(C(=O)N(CC(=O)NC(C)(C)C)Cc2ccc(C(=O)NO)cc2F)cc1
E3 Binder	CHEMBL4063658	ChEMBL	8.8	—	—	CN(C)c1ccc(C(=O)N(CC(=O)NC2CCCCC2)Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL5199849	ChEMBL	7.8	—	—	CN(C)c1ccc(C(=O)N(CC(=O)NC2CCCCC2)Cc2ccc(C(=O)NO)cc2F)cc1
E3 Binder	CHEMBL4170198	ChEMBL	7.96	HB7	—	CN(C)c1ccc(C(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL5187433	ChEMBL	8.0	M0I	—	CN(C)c1ccc(C(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(C(=O)NO)cc2F)cc1
E3 Binder	CHEMBL4553076	ChEMBL	6.07	—	—	CN(C)c1ccc(C(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(C(=O)Nc3cc(-c4ccccc4)ccc3N)cc2)cc1
E3 Binder	CHEMBL4474656	ChEMBL	6.96	—	—	CN(C)c1ccc(C(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(C(=O)Nc3ccccc3N)cc2)cc1
E3 Binder	CHEMBL4583725	ChEMBL	8.0	—	—	CN(C)c1ccc(C(=O)N(CCC(=O)NCc2ccc(Cl)cc2)Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4476049	ChEMBL	7.83	—	—	CN(C)c1ccc(C(=O)N(CCC(=O)NCc2ccccc2)Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4069631	ChEMBL	6.57	—	—	CN(C)c1ccc(C(=O)N(CCCCCC(=O)NO)CC(=O)NCc2ccccc2)cc1
E3 Binder	CHEMBL4866446	ChEMBL	7.16	—	—	CN(C)c1ccc(C(=O)N(Cc2ccc(C(=O)NO)cc2)C(C)(C)C(=O)NCc2ccccc2)cc1
E3 Binder	CHEMBL3764525	ChEMBL	7.82	—	—	CN(C)c1ccc(C(=O)N/N=C/c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL3765502	ChEMBL	6.41	—	—	CN(C)c1ccc(C(=O)N/N=C/c2cccc(C(=O)NO)c2)cc1
E3 Binder	CHEMBL46942	ChEMBL	6.96	—	—	CN(C)c1ccc(C(=O)NCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL140000	ChEMBL	7.56	B3N	—	CN(C)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL143047	ChEMBL	6.84	—	—	CN(C)c1ccc(C(=O)NCCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL440018	ChEMBL	6.32	—	—	CN(C)c1ccc(C(=O)NCCCCCCNC(=O)CS)cc1
E3 Binder	CHEMBL324126	ChEMBL	6.21	—	—	CN(C)c1ccc(C(=O)NCCCCCCS)cc1
E3 Binder	CHEMBL180911	ChEMBL	6.94	—	—	CN(C)c1ccc(C(=O)NCCCCCNC(=O)CS)cc1
E3 Binder	CHEMBL427510	ChEMBL	6.21	—	—	CN(C)c1ccc(C(=O)NCCCCNC(=O)CS)cc1
E3 Binder	CHEMBL180064	ChEMBL	6.67	—	—	CN(C)c1ccc(C(=O)NCCCNC(=O)CS)cc1
E3 Binder	CHEMBL152133	ChEMBL	6.76	—	—	CN(C)c1ccc(C(=O)NCc2ccc(/C=C/C(=O)NO)cc2)cc1
E3 Binder	CHEMBL221654	ChEMBL	6.03	—	—	CN(C)c1ccc(C(=O)N[C@@H](CCCCCC(=O)NO)C(=O)Nc2cccc3cccnc23)cc1
E3 Binder	CHEMBL2047704	ChEMBL	6.16	—	—	CN(C)c1ccc(C/C(=N\O)C(=O)NCCS)cc1Br
E3 Binder	CHEMBL3966405	ChEMBL	6.52	—	—	CN(C)c1ccc(CCCOCCN(C)c2ccc(NC(=O)CCCCCCC(=O)NO)cc2)cc1
E3 Binder	CHEMBL5078295	ChEMBL	7.54	—	—	CN(C)c1ccc(CN(Cc2ccc(C(=O)NO)cc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL227119	ChEMBL	7.34	—	—	CN(C)c1ccc(CNC(=O)NCCC(=O)NO)cc1
E3 Binder	CHEMBL270333	ChEMBL	6.1	—	—	CN(C)c1ccc(CNC(=O)NCCCCC(=O)NO)cc1
E3 Binder	CHEMBL405586	ChEMBL	6.1	—	—	CN(C)c1ccc(CNC(=O)NCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL271115	ChEMBL	6.0	—	—	CN(C)c1ccc(CNC(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL271320	ChEMBL	6.16	—	—	CN(C)c1ccc(CNC(=O)NCCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3984046	ChEMBL	7.92	—	—	CN(C)c1ccc(Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL596660	ChEMBL	6.52	—	—	CN(C)c1ccc(NC(=O)CCCCC/C=C(\F)CS)cc1
E3 Binder	CHEMBL227120	ChEMBL	7.46	—	—	CN(C)c1ccc(NC(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL5280773	ChEMBL	6.17	—	—	CN(C)c1ccc(NC(=O)NCCCCNC(=O)CS)cc1
E3 Binder	CHEMBL3339029	ChEMBL	8.57	—	—	CN(C)c1ccc(Nc2ncnc3sc(NC(=O)CCCCCCC(=O)NO)cc23)cc1F
E3 Binder	CHEMBL201710	ChEMBL	6.75	—	—	CN(C)c1ccc([S+]([O-])CCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3910885	ChEMBL	7.15	—	—	CN(C)c1cccc(Cc2ccc(C(=O)NO)cc2)c1
E3 Binder	CHEMBL4457698	ChEMBL	6.88	—	—	CN(C)c1cccc2c(S(=O)(=O)N(CC(=O)NCc3ccccc3)Cc3ccc(C(=O)NO)cc3)cccc12
E3 Binder	CHEMBL4437165	ChEMBL	7.34	—	—	CN(C)c1cccc2c(S(=O)(=O)N(CCCCCC(=O)NO)CC(=O)NCc3ccccc3)cccc12
E3 Binder	CHEMBL4759256	ChEMBL	6.89	—	—	CN(C)c1cccc2c(S(=O)(=O)NCCCCCC(=O)NO)cccc12
E3 Binder	CHEMBL5283088	ChEMBL	8.01	—	—	CN(C)c1cccc2c(S(=O)(=O)N[C@H](C(=O)Nc3ccc(C(=O)NO)cc3)c3ccccc3)cccc12
E3 Binder	CHEMBL5271192	ChEMBL	7.1	—	—	CN(C)c1cccc2c(SNCCCCCC(=O)NO)cccc12
E3 Binder	CHEMBL1616372	ChEMBL	6.05	—	—	CN(C)c1nc(N)c(C(=O)Nc2cccnc2)nc1Cl
E3 Binder	CHEMBL5220745	ChEMBL	6.07	—	—	CN(C)c1nc2c(Br)c(Br)c(Br)c(Br)c2n1CCCCCC(=O)NO
E3 Binder	CHEMBL2385397	ChEMBL	6.8	—	—	CN(C)c1nc2c(s1)Cc1cc(/C=C/C(=O)NO)ccc1-2
E3 Binder	CHEMBL4576056	ChEMBL	7.26	—	—	CN(CC(=O)N(Cc1ccc(C(C)(C)C)cc1)c1ccc(C(=O)NO)cc1)S(=O)(=O)c1ccc(F)cc1
E3 Binder	CHEMBL3916309	ChEMBL	7.0	—	—	CN(CCC(=O)NO)CC[C@H](CSc1ccccc1)Nc1ccc(S(=O)(=O)NC(=O)c2ccc(N3CCN(Cc4ccccc4-c4ccc(Cl)cc4)CC3)cc2)cc1[N+](=O)[O-]
E3 Binder	CHEMBL3913571	ChEMBL	7.0	—	—	CN(CCCC(=O)NO)CC[C@H](CSc1ccccc1)Nc1ccc(S(=O)(=O)NC(=O)c2ccc(N3CCN(Cc4ccccc4-c4ccc(Cl)cc4)CC3)cc2)cc1[N+](=O)[O-]
E3 Binder	CHEMBL3969644	ChEMBL	7.0	—	—	CN(CCCCC(=O)NO)CC[C@H](CSc1ccccc1)Nc1ccc(S(=O)(=O)NC(=O)c2ccc(N3CCN(Cc4ccccc4-c4ccc(Cl)cc4)CC3)cc2)cc1[N+](=O)[O-]
E3 Binder	CHEMBL349646	ChEMBL	6.35	—	—	CN(CCCCCC(=O)NO)C(=O)c1ccc(N(C)C)cc1
E3 Binder	CHEMBL3953980	ChEMBL	7.0	—	—	CN(CCCCCC(=O)NO)CC[C@H](CSc1ccccc1)Nc1ccc(S(=O)(=O)NC(=O)c2ccc(N3CCN(Cc4ccccc4-c4ccc(Cl)cc4)CC3)cc2)cc1[N+](=O)[O-]
E3 Binder	CHEMBL3693805	ChEMBL	7.64	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(C(C)(O)c2ccc(F)cc2)cc1
E3 Binder	CHEMBL3693809	ChEMBL	7.44	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(C(C)(O)c2ccccn2)cc1
E3 Binder	CHEMBL3640655	ChEMBL	7.82	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(C(O)(c2cc(F)cc(F)c2)c2cc(F)cc(F)c2)cc1
E3 Binder	CHEMBL3640661	ChEMBL	7.62	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(C(O)(c2ccc(F)cc2)c2ccccn2)cc1
E3 Binder	CHEMBL3640651	ChEMBL	7.89	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(C(O)(c2ccc(F)cc2F)c2ccc(F)cc2F)cc1
E3 Binder	CHEMBL3693796	ChEMBL	8.0	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(C(O)(c2cccc(F)c2)c2cccc(F)c2)cc1
E3 Binder	CHEMBL3693790	ChEMBL	7.75	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(C(O)(c2ccccc2)c2ccncc2)cc1
E3 Binder	CHEMBL3640647	ChEMBL	8.05	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(C(O)(c2ccccc2F)c2ccccc2F)cc1
E3 Binder	CHEMBL3693784	ChEMBL	7.44	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(C(O)(c2ccccn2)c2ccccn2)cc1
E3 Binder	CHEMBL3693792	ChEMBL	7.33	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(C(c2ccccc2)c2ccccc2)cc1
E3 Binder	CHEMBL3693776	ChEMBL	7.57	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(N(C(=O)c2ccccc2)c2ccccc2)cc1
E3 Binder	CHEMBL3693744	ChEMBL	7.46	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(N(C)c2ccccc2C#N)cc1
E3 Binder	CHEMBL3693738	ChEMBL	6.97	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(N(C)c2nc3ccccc3o2)cc1
E3 Binder	CHEMBL3693713	ChEMBL	7.09	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(N(c2ccccc2)c2ccccc2)cc1
E3 Binder	CHEMBL3693753	ChEMBL	7.82	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(N(c2ccccc2)c2ccccn2)cc1
E3 Binder	CHEMBL3693743	ChEMBL	7.19	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(N(c2ccccc2)c2cccnc2)cc1
E3 Binder	CHEMBL3693766	ChEMBL	7.75	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(N(c2ccccc2)c2ncccn2)cc1
E3 Binder	CHEMBL3693714	ChEMBL	6.7	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(N(c2ncccn2)c2ncccn2)cc1
E3 Binder	CHEMBL3693748	ChEMBL	7.96	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(Nc2ccccc2)cc1
E3 Binder	CHEMBL3693756	ChEMBL	7.7	—	—	CN(CCCCCCC(=O)NO)C(=O)c1ccc(Nc2nc3ccccc3s2)cc1
E3 Binder	CHEMBL3640666	ChEMBL	7.14	—	—	CN(CCCCCCC(=O)NO)C(=O)c1cccc(C(O)(c2ccc(F)cc2)c2ccc(F)cc2)c1
E3 Binder	CHEMBL5090769	ChEMBL	7.75	—	—	CN(CCOc1ccc(C(=O)NO)cc1)c1nc(N)n2nc(-c3ccco3)nc2n1
E3 Binder	CHEMBL5219361	ChEMBL	6.8	—	—	CN(CCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1)C(=O)c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL3943273	ChEMBL	6.0	—	—	CN(CC[C@H](CSc1ccccc1)Nc1ccc(S(=O)(=O)NC(=O)c2ccc(N3CCN(Cc4ccccc4-c4ccc(Cl)cc4)CC3)cc2)cc1[N+](=O)[O-])CC(=O)NO
E3 Binder	CHEMBL5080630	ChEMBL	7.76	—	—	CN(CCc1ccc(C(=O)NO)cc1)c1nc(N)n2nc(-c3ccco3)nc2n1
E3 Binder	CHEMBL5274004	ChEMBL	8.3	—	—	CN(CCc1ccccc1)S(=O)(=O)c1cccc(/C=C/C(=O)NO)c1
E3 Binder	CHEMBL5219048	ChEMBL	7.96	—	—	CN(Cc1ccc(C(=O)NO)cc1)C(=O)O[C@@H]1C[C@@H](c2nc3cccc(Cl)c3c(=O)n2C)N(c2nc(N)nc(N)c2C#N)C1
E3 Binder	CHEMBL4744157	ChEMBL	7.76	—	—	CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1c(F)c(F)c(F)c(F)c1F
E3 Binder	CHEMBL5188138	ChEMBL	7.51	—	—	CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1ccccc1
E3 Binder	CHEMBL5198759	ChEMBL	8.7	—	—	CN(Cc1ccc(C(=O)NO)cc1)S(=O)(=O)c1c(F)c(F)c(F)c(F)c1F
E3 Binder	CHEMBL4165724	ChEMBL	7.22	—	—	CN(Cc1ccc(C(=O)NO)cc1F)CC12CC3CC(CC(C3)C1)C2
E3 Binder	CHEMBL5171822	ChEMBL	7.22	—	—	CN(Cc1ccc(C(=O)NO)cc1[18F])CC12CC3CC(CC(C3)C1)C2
E3 Binder	CHEMBL4848432	ChEMBL	6.08	—	—	CN(Cc1ccc(C(=O)NO)cn1)C12CC3C[C@@](C)(C1)C[C@](C)(C3)C2
E3 Binder	CHEMBL497332	ChEMBL	7.05	—	—	CN(Cc1ccc2nccnc2c1)C(=O)c1ccc(C(=O)C(F)(F)F)s1
E3 Binder	CHEMBL493782	ChEMBL	6.19	—	—	CN(Cc1ccccc1)C(=O)c1cc(C(=O)C(F)(F)F)cs1
E3 Binder	CHEMBL462209	ChEMBL	6.64	—	—	CN(Cc1ccccc1)C(=O)c1ccc(C(=O)C(F)(F)F)s1
E3 Binder	CHEMBL496511	ChEMBL	6.31	—	—	CN(Cc1ccccc1)Cc1ccc(C(=O)C(F)(F)F)s1
E3 Binder	CHEMBL494813	ChEMBL	6.14	—	—	CN(Cc1ccccc1)S(=O)(=O)c1ccc(C(=O)C(F)(F)F)s1
E3 Binder	CHEMBL4567832	ChEMBL	8.01	—	—	CN(Cc1ccccc1)c1ccc2c3c(cccc13)C(=O)N(CCCCCC(=O)NO)C2=O
E3 Binder	CHEMBL3827814	ChEMBL	8.49	—	—	CN(Cc1nc2c(N3CCOCC3)nc(-c3ccc(N)cc3)nc2n1C)c1ncc(C(=O)NO)cn1
E3 Binder	CHEMBL3827517	ChEMBL	8.57	—	—	CN(Cc1nc2c(N3CCOCC3)nc(-c3ccncc3)nc2n1C)c1ncc(C(=O)NO)cn1
E3 Binder	CHEMBL3827894	ChEMBL	8.48	—	—	CN(Cc1nc2c(N3CCOCC3)nc(-c3cnc(N)nc3)nc2n1C)c1ncc(C(=O)NO)cn1
E3 Binder	CHEMBL1801251	ChEMBL	7.64	—	—	CN([C@H]1[C@@H]2CN(c3ncc(C(=O)NO)cn3)C[C@@H]21)S(=O)(=O)c1ccc2ccccc2c1
E3 Binder	CHEMBL3693704	ChEMBL	8.52	—	—	CN(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1c(Cl)cccc1Cl
E3 Binder	CHEMBL3693720	ChEMBL	8.7	—	—	CN(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1c(F)cccc1F
E3 Binder	CHEMBL3693740	ChEMBL	8.4	—	—	CN(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1ccccc1C#N
E3 Binder	CHEMBL3693706	ChEMBL	8.52	—	—	CN(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1ccccc1C(F)(F)F
E3 Binder	CHEMBL3693725	ChEMBL	7.68	—	—	CN(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1cnccn1
E3 Binder	CHEMBL3693739	ChEMBL	7.96	—	—	CN(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1nc2ccccc2o1
E3 Binder	CHEMBL3652232	ChEMBL	7.42	—	—	CN(c1ccc(Cl)c(Cl)c1)c1ncc(C(=O)NO)cn1
E3 Binder	CHEMBL3774793	ChEMBL	7.85	—	—	CN(c1ccc(OCC(=O)NO)cc1)c1ncnc2ccccc12
E3 Binder	CHEMBL3775209	ChEMBL	7.47	—	—	CN(c1ccc(OCCCC(=O)NO)cc1)c1ncnc2ccccc12
E3 Binder	CHEMBL3774858	ChEMBL	7.31	—	—	CN(c1ccc(OCCCCC(=O)NO)cc1)c1ncnc2ccccc12
E3 Binder	CHEMBL3774993	ChEMBL	7.72	—	—	CN(c1ccc(OCCCCCC(=O)NO)cc1)c1ncnc2ccccc12
E3 Binder	CHEMBL1162969	ChEMBL	6.32	—	—	CN(c1ccccc1)S(=O)(=O)c1cccc(/C=C/C(=O)NO)c1
E3 Binder	CHEMBL3693708	ChEMBL	8.22	—	—	CN(c1ccccc1)c1ncc(C(=O)NCCCCCCC(=O)NO)cn1
E3 Binder	CHEMBL2408819	ChEMBL	6.42	—	—	CN1C(=O)C(NC(=O)CCCCC(=O)NO)N=C(c2ccccc2)c2ccccc21
E3 Binder	CHEMBL2408820	ChEMBL	6.75	—	—	CN1C(=O)C(NC(=O)CCCCCC(=O)NO)N=C(c2ccccc2)c2ccccc21
E3 Binder	CHEMBL2408818	ChEMBL	6.22	—	—	CN1C(=O)C(NC(=O)CCCCCCCC(=O)NO)N=C(c2ccccc2)c2ccccc21
E3 Binder	CHEMBL4092802	ChEMBL	9.38	—	—	CN1C(=O)C2CN(Cc3c2c2cc(O)ccc2n3Cc2ccc(C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL4072045	ChEMBL	9.32	—	—	CN1C(=O)C2CN(Cc3c2c2cc(OCCN4CCOCC4)ccc2n3Cc2ccc(C(=O)NO)cc2)C1=O.Cl
E3 Binder	CHEMBL4082520	ChEMBL	10.1	—	—	CN1C(=O)C2CN(Cc3c2c2cc(OCc4ccccc4)ccc2n3Cc2ccc(C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL4100615	ChEMBL	8.75	—	—	CN1C(=O)C2CN(Cc3c2c2ccc4ccccc4c2n3Cc2ccc(C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL4065219	ChEMBL	8.38	—	—	CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2ccc(/C=C/C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL4087616	ChEMBL	9.15	—	—	CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2ccc(C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL4065283	ChEMBL	9.35	—	—	CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2ccc(C(=O)NO)cc2)C1=S
E3 Binder	CHEMBL4085143	ChEMBL	7.14	—	—	CN1C(=O)C2CN(Cc3c2c2ccccc2n3Cc2cccc(/C=C/C(=O)NO)c2)C1=O
E3 Binder	CHEMBL4291041	ChEMBL	8.62	—	—	CN1C(=O)C2Cc3c(n(Cc4ccc(C(=O)NO)cc4)c4ccccc34)CN2C1=O
E3 Binder	CHEMBL4073813	ChEMBL	8.73	—	—	CN1C(=O)C2c3c(n(Cc4ccc(C(=O)NO)cc4)c4ccccc34)CCN2C1=O
E3 Binder	CHEMBL3309286	ChEMBL	6.89	—	—	CN1C(=O)CC(C)(C)c2cc(C(=O)NCCCCCCC(=O)NO)ccc21
E3 Binder	CHEMBL3356526	ChEMBL	8.52	—	—	CN1C(=O)CCC[C@H]1C(=O)N[C@@H](CCCCCS)C(=O)Nc1ccccc1
E3 Binder	CHEMBL3356921	ChEMBL	8.3	—	—	CN1C(=O)CC[C@@H]1C(=O)N[C@@H](CCCCCS)C(=O)Nc1ccccc1
E3 Binder	CHEMBL5272650	ChEMBL	7.78	—	—	CN1C(=O)CN(Cc2ccc(C(=O)NO)cc2)C(=O)C1Cc1ccccc1
E3 Binder	CHEMBL2408692	ChEMBL	6.8	—	—	CN1C(=O)CN=C(c2ccccc2)c2cc(C#C/C=C/C(=O)NO)ccc21
E3 Binder	CHEMBL4873563	ChEMBL	6.97	—	—	CN1C(=O)N(Cc2ccc(C(=O)NO)cc2)C(=O)C1Cc1ccccc1
E3 Binder	CHEMBL4525288	ChEMBL	7.93	—	—	CN1C(=O)N(c2ccc(Cl)cc2)C(=O)C1CCC(=O)NCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4475603	ChEMBL	8.15	—	—	CN1C(=O)N(c2ccc(Cl)cc2)C(=O)C1CCC(=O)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4083713	ChEMBL	9.06	—	—	CN1C(=O)N2Cc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)C(C2)C1=S
E3 Binder	CHEMBL2408696	ChEMBL	6.92	—	—	CN1C(=O)[C@@H](NC(=O)CCCCCCC(=O)NO)N=C(c2ccccc2)c2ccccc21
E3 Binder	CHEMBL4092880	ChEMBL	9.15	—	—	CN1C(=O)[C@@H]2CN(Cc3c2c2ccccc2n3Cc2ccc(C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL2408695	ChEMBL	6.51	—	—	CN1C(=O)[C@H](NC(=O)CCCCCCC(=O)NO)N=C(c2ccccc2)c2ccccc21
E3 Binder	CHEMBL2408689	ChEMBL	6.44	—	—	CN1C(=O)[C@H](O)N=C(c2ccccc2)c2cc(C#CCCCC(=O)NO)ccc21
E3 Binder	CHEMBL4066262	ChEMBL	8.7	—	—	CN1C(=O)[C@H]2CN(Cc3c2c2ccccc2n3Cc2ccc(C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL2391006	ChEMBL	6.59	—	—	CN1C(=O)c2cc(/C=C/C(=O)NO)ccc2OC12CCN(CCc1ccccc1)CC2
E3 Binder	CHEMBL2391005	ChEMBL	6.86	—	—	CN1C(=O)c2cc(/C=C/C(=O)NO)ccc2OC12CCN(Cc1ccc(F)cc1)CC2
E3 Binder	CHEMBL2391004	ChEMBL	6.87	—	—	CN1C(=O)c2cc(/C=C/C(=O)NO)ccc2OC12CCN(Cc1ccccc1)CC2
E3 Binder	CHEMBL2391002	ChEMBL	6.69	—	—	CN1C(=O)c2cc(/C=C/C(=O)NO)ccc2OC12CCNCC2
E3 Binder	CHEMBL4864178	ChEMBL	6.93	—	—	CN1CC(=O)N(Cc2ccc(C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL4292944	ChEMBL	7.87	—	—	CN1CC(=O)N2Cc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)CC2C1=O
E3 Binder	CHEMBL239800	ChEMBL	6.17	—	—	CN1CC(=O)N=C1NC(=O)Nc1cccc(Cl)c1
E3 Binder	CHEMBL3758204	ChEMBL	6.78	—	—	CN1CC2(CC(=O)c3cc(/C=C/C(=O)NO)ccc3O2)C1
E3 Binder	CHEMBL4846606	ChEMBL	9.0	—	—	CN1CC2(CCCCC2)CC[C@H]1Cc1cc(F)cc(C(=O)NO)c1
E3 Binder	CHEMBL4790744	ChEMBL	6.58	QQG	—	CN1CC2(CCN(Cc3ccc(C(=O)NO)cc3)CC2)c2ccccc21
E3 Binder	CHEMBL4075722	ChEMBL	9.29	—	—	CN1CC2CN(Cc3c2c2ccccc2n3Cc2ccc(C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL4456269	ChEMBL	6.72	—	—	CN1CCC(CNC(=O)c2cccc(C(=O)NO)c2)(c2nc(-c3ccccc3)cs2)CC1
E3 Binder	CHEMBL3759365	ChEMBL	6.92	—	—	CN1CCC2(CC(=O)c3cc(/C=C/C(=O)NO)ccc3O2)C1
E3 Binder	CHEMBL1938430	ChEMBL	6.54	—	—	CN1CCC2(CC1)CC(=O)c1cc(/C=C/C(=O)NO)ccc1O2
E3 Binder	CHEMBL4287273	ChEMBL	6.69	—	—	CN1CCC2(CC1)CN(Cc1ccc(C(=O)NO)cc1)c1ccccc12
E3 Binder	CHEMBL2390998	ChEMBL	7.0	—	—	CN1CCC2(CC1)NC(=O)c1cc(/C=C/C(=O)NO)ccc1O2
E3 Binder	CHEMBL2391003	ChEMBL	6.28	—	—	CN1CCC2(CC1)Oc1ccc(/C=C/C(=O)NO)cc1C(=O)N2C
E3 Binder	CHEMBL2390991	ChEMBL	6.76	—	—	CN1CCC2(CC1)Oc1ccc(/C=C/C(=O)NO)cc1C(=O)N2Cc1ccccc1
E3 Binder	CHEMBL1938442	ChEMBL	6.27	—	—	CN1CCC2(CC1)Oc1ccc(/C=C/C(=O)NO)cc1C2=O
E3 Binder	CHEMBL5291414	ChEMBL	6.78	—	—	CN1CCC2(CC1)c1ccccc1N(Cc1ccc(C(=O)NO)cc1)C2c1ccc(Cl)cc1
E3 Binder	CHEMBL5280477	ChEMBL	6.85	—	—	CN1CCC2(CC1)c1ccccc1N(Cc1ccc(C(=O)NO)cc1)C2c1ccc(F)cc1
E3 Binder	CHEMBL5276825	ChEMBL	6.96	—	—	CN1CCC2(CC1)c1ccccc1N(Cc1ccc(C(=O)NO)cc1)C2c1cccc(Cl)c1
E3 Binder	CHEMBL5282958	ChEMBL	7.13	—	—	CN1CCC2(CC1)c1ccccc1N(Cc1ccc(C(=O)NO)cc1)C2c1ccccc1
E3 Binder	CHEMBL5269954	ChEMBL	7.54	—	—	CN1CCC2(CC1)c1ccccc1N(Cc1ccc(C(=O)NO)cc1)C2c1ccccc1F
E3 Binder	CHEMBL5290574	ChEMBL	6.95	—	—	CN1CCC2(CC1)c1ccccc1N(Cc1ccc(C(=O)NO)cc1)C2c1cccnc1
E3 Binder	CHEMBL4436806	ChEMBL	7.5	—	—	CN1CCC2=C(C1)N(Cc1ccc(C(=O)NO)cc1)c1ccccc1S2
E3 Binder	CHEMBL1094158	ChEMBL	7.1	—	—	CN1CCCC(n2c(-c3cccc(/C=C/C(=O)NO)c3)nc3ccccc32)C1
E3 Binder	CHEMBL4532181	ChEMBL	6.9	—	—	CN1CCCC1c1cn(Cc2ccc(C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL3758219	ChEMBL	6.62	—	—	CN1CCCC2(CC(=O)c3cc(/C=C/C(=O)NO)ccc3O2)C1
E3 Binder	CHEMBL3759339	ChEMBL	6.94	—	—	CN1CCCC2(CC1)CC(=O)c1cc(/C=C/C(=O)NO)ccc1O2
E3 Binder	CHEMBL1094159	ChEMBL	7.0	—	—	CN1CCC[C@@H](n2c(-c3cccc(/C=C/C(=O)NO)c3)nc3ccccc32)C1
E3 Binder	CHEMBL1095449	ChEMBL	7.3	—	—	CN1CCC[C@H](n2c(-c3cccc(/C=C/C(=O)NO)c3)nc3ccccc32)C1
E3 Binder	CHEMBL593858	ChEMBL	8.16	—	—	CN1CCN(CC(/C=C/c2ccccc2)N2CCN(c3ncc(C(=O)NO)cn3)CC2)CC1
E3 Binder	CHEMBL4283513	ChEMBL	8.21	—	—	CN1CCN(CC(=O)Nc2ccc(-c3ccnc(Nc4ccc(OCCCCCCC(=O)NO)cc4)n3)cc2)CC1
E3 Binder	CHEMBL4294092	ChEMBL	8.17	—	—	CN1CCN(CC(=O)Nc2ccc(-c3ccnc(Nc4cccc(OCCCCCCC(=O)NO)c4)n3)cc2)CC1
E3 Binder	CHEMBL3927240	ChEMBL	8.53	—	—	CN1CCN(CCc2cn(CC3=CCC(C(=O)NO)C=C3)c3ccccc23)CC1
E3 Binder	CHEMBL569753	ChEMBL	6.74	—	—	CN1CCN(Cc2ccc(C(=O)/C=C/c3ccc(/C=C/C(=O)NO)cc3)cc2)CC1
E3 Binder	CHEMBL570214	ChEMBL	7.57	—	—	CN1CCN(Cc2ccc(C(=O)/C=C/c3ccc(/C=C/C(=O)NO)nc3)cc2)CC1
E3 Binder	CHEMBL569546	ChEMBL	7.77	—	—	CN1CCN(Cc2ccc(C(=O)/C=C/c3cccc(/C=C/C(=O)NO)c3)cc2)CC1
E3 Binder	CHEMBL568872	ChEMBL	7.39	—	—	CN1CCN(Cc2ccc(C(=O)/C=C/c3cccc(/C=C/C(=O)NO)n3)cc2)CC1
E3 Binder	CHEMBL5203383	ChEMBL	6.55	L8C	—	CN1CCN(Cc2ccc(C(=O)NO)cc2)CC1
E3 Binder	CHEMBL570213	ChEMBL	6.65	—	—	CN1CCN(Cc2cccc(C(=O)/C=C/c3ccc(/C=C/C(=O)NO)cc3)c2)CC1
E3 Binder	CHEMBL569748	ChEMBL	7.28	—	—	CN1CCN(Cc2cccc(C(=O)/C=C/c3ccc(/C=C/C(=O)NO)nc3)c2)CC1
E3 Binder	CHEMBL569959	ChEMBL	7.62	—	—	CN1CCN(Cc2cccc(C(=O)/C=C/c3cccc(/C=C/C(=O)NO)c3)c2)CC1
E3 Binder	CHEMBL569730	ChEMBL	7.25	—	—	CN1CCN(Cc2cccc(C(=O)/C=C/c3cccc(/C=C/C(=O)NO)n3)c2)CC1
E3 Binder	CHEMBL583028	ChEMBL	6.46	—	—	CN1CCN(Cc2ccccc2C(=O)/C=C/c2ccc(/C=C/C(=O)NO)cc2)CC1
E3 Binder	CHEMBL569327	ChEMBL	7.92	—	—	CN1CCN(Cc2ccccc2C(=O)/C=C/c2ccc(/C=C/C(=O)NO)nc2)CC1
E3 Binder	CHEMBL577946	ChEMBL	7.13	—	—	CN1CCN(Cc2ccccc2C(=O)/C=C/c2cccc(/C=C/C(=O)NO)c2)CC1
E3 Binder	CHEMBL584733	ChEMBL	7.28	—	—	CN1CCN(Cc2ccccc2C(=O)/C=C/c2cccc(/C=C/C(=O)NO)n2)CC1
E3 Binder	CHEMBL569749	ChEMBL	6.76	—	—	CN1CCN(c2ccc(C(=O)/C=C/c3ccc(/C=C/C(=O)NO)nc3)cc2)CC1
E3 Binder	CHEMBL583545	ChEMBL	7.57	—	—	CN1CCN(c2ccc(C(=O)/C=C/c3cccc(/C=C/C(=O)NO)c3)cc2)CC1
E3 Binder	CHEMBL569731	ChEMBL	7.82	—	—	CN1CCN(c2ccc(C(=O)/C=C/c3cccc(/C=C/C(=O)NO)n3)cc2)CC1
E3 Binder	CHEMBL4292408	ChEMBL	8.51	—	—	CN1CCN(c2ccc(Nc3nccc(-c4ccc(NC(=O)CCCCCCC(=O)NO)cc4)n3)cc2)CC1
E3 Binder	CHEMBL569984	ChEMBL	6.55	—	—	CN1CCN(c2cccc(C(=O)/C=C/c3ccc(/C=C/C(=O)NO)cc3)c2)CC1
E3 Binder	CHEMBL571103	ChEMBL	7.52	—	—	CN1CCN(c2cccc(C(=O)/C=C/c3ccc(/C=C/C(=O)NO)nc3)c2)CC1
E3 Binder	CHEMBL571993	ChEMBL	7.7	—	—	CN1CCN(c2cccc(C(=O)/C=C/c3cccc(/C=C/C(=O)NO)c3)c2)CC1
E3 Binder	CHEMBL571104	ChEMBL	7.5	—	—	CN1CCN(c2cccc(C(=O)/C=C/c3cccc(/C=C/C(=O)NO)n3)c2)CC1
E3 Binder	CHEMBL569716	ChEMBL	6.73	—	—	CN1CCN(c2ccccc2C(=O)/C=C/c2ccc(/C=C/C(=O)NO)cc2)CC1
E3 Binder	CHEMBL578606	ChEMBL	6.85	—	—	CN1CCN(c2ccccc2C(=O)/C=C/c2ccc(/C=C/C(=O)NO)nc2)CC1
E3 Binder	CHEMBL570215	ChEMBL	7.06	—	—	CN1CCN(c2ccccc2C(=O)/C=C/c2cccc(/C=C/C(=O)NO)c2)CC1
E3 Binder	CHEMBL577513	ChEMBL	7.48	—	—	CN1CCN(c2ccccc2C(=O)/C=C/c2cccc(/C=C/C(=O)NO)n2)CC1
E3 Binder	CHEMBL4873811	ChEMBL	7.25	—	—	CN1CCN(c2nc(-c3ccc(C(=O)NO)cc3)nc3cc(Cl)ccc23)CC1
E3 Binder	CHEMBL5201448	ChEMBL	8.38	—	—	CN1CCN(c2nc(-c3cnc(N)nc3)cn(Cc3ccc(C(=O)NO)cc3)c2=O)CC1
E3 Binder	CHEMBL3640703	ChEMBL	8.3	—	—	CN1CCN(c2ncc(C(=O)NCCCCCCC(=O)NO)cn2)C(c2ccccc2)C1
E3 Binder	CHEMBL3640707	ChEMBL	7.75	—	—	CN1CCN(c2ncc(C(=O)NCCCCCCC(=O)NO)cn2)CC1
E3 Binder	CHEMBL2018301	ChEMBL	9.15	—	—	CN1CCc2c(c3cc(Br)ccc3n2Cc2ccc(C(=O)NO)cc2)C1
E3 Binder	CHEMBL2018298	ChEMBL	7.65	—	—	CN1CCc2c(c3cc(C(C)(C)C)ccc3n2Cc2ccc(C(=O)NO)cc2)C1
E3 Binder	CHEMBL2018300	ChEMBL	8.99	—	—	CN1CCc2c(c3cc(Cl)ccc3n2Cc2ccc(C(=O)NO)cc2)C1
E3 Binder	CHEMBL3675749	ChEMBL	6.67	—	—	CN1CCc2c(c3ccccc3n2CCCCCC(=O)NO)C1
E3 Binder	CHEMBL4084222	ChEMBL	7.38	—	—	CN1CCc2c(c3ccccc3n2Cc2ccc(/C=C/C(=O)NO)cc2)C1
E3 Binder	CHEMBL2018302	ChEMBL	8.72	N9W	—	CN1CCc2c(c3ccccc3n2Cc2ccc(C(=O)NO)cc2)C1
E3 Binder	CHEMBL3770936	ChEMBL	7.82	—	—	CN1CCc2c(c3ccccc3n2Cc2ccc(C(=O)NO)cc2)C1.Cl
E3 Binder	CHEMBL4062520	ChEMBL	6.72	—	—	CN1CCc2c(c3ccccc3n2S(=O)(=O)c2cccc(/C=C/C(=O)NO)c2)C1
E3 Binder	CHEMBL3675748	ChEMBL	8.85	—	—	CN1CCc2c(n(CCCCCC(=O)NO)c3ccccc23)C1
E3 Binder	CHEMBL2018451	ChEMBL	9.0	—	—	CN1CCc2c(n(Cc3ccc(C(=O)NO)cc3)c3ccccc23)C1
E3 Binder	CHEMBL4074800	ChEMBL	9.64	—	—	CN1CN2Cc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)C(C2)C1=O
E3 Binder	CHEMBL4856445	ChEMBL	9.0	—	—	CN1Cc2cc(C(=O)NO)ccc2CN1Cc1ccccc1
E3 Binder	CHEMBL5073322	ChEMBL	7.05	—	—	CN1c2ccc(F)cc2C(=O)N2CCc3c([nH]c4ccc(OCc5ccc(/C=C/C(=O)NO)cc5)cc34)C21
E3 Binder	CHEMBL3577694	ChEMBL	7.89	—	—	CN1c2ccc(NCc3ccc(-c4noc(CCCCCCC(=O)NO)n4)cc3)cc2C(=O)N2CCc3c([nH]c4ccc(O)cc34)C21
E3 Binder	CHEMBL595909	ChEMBL	8.48	—	—	CNC(=O)C(/C=C/c1ccccc1)N1CCN(c2ncc(C(=O)NO)cn2)CC1
E3 Binder	CHEMBL112446	ChEMBL	8.43	—	—	CNC(=O)C(=O)CCCCCCC(=O)Nc1cccc(-c2ccccc2)c1
E3 Binder	CHEMBL112211	ChEMBL	6.47	—	—	CNC(=O)C(=O)CCCCCCC(=O)Nc1ccccc1
E3 Binder	CHEMBL113033	ChEMBL	8.51	—	—	CNC(=O)C(=O)CCCCCCC(=O)Nc1nc(-c2ccc(CCN(C)C)cc2)cs1
E3 Binder	CHEMBL324429	ChEMBL	8.04	—	—	CNC(=O)C(=O)CCCCCCC(=O)Nc1nc(-c2ccc(OC)cc2)cs1
E3 Binder	CHEMBL271800	ChEMBL	8.37	—	—	CNC(=O)C(=O)CCCCCCC(=O)Nc1nc(-c2cccnc2)cs1
E3 Binder	CHEMBL113303	ChEMBL	6.96	—	—	CNC(=O)C(=O)CCCCCCOc1ccc(-c2ccccc2)cc1
E3 Binder	CHEMBL4870348	ChEMBL	8.17	—	—	CNC(=O)CCCCCCCn1nc(-c2ccc3oc(N)nc3c2)c2c(N)ncnc21
E3 Binder	CHEMBL4849568	ChEMBL	7.22	—	—	CNC(=O)CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1ccc(C(C)C)cc1
E3 Binder	CHEMBL3951862	ChEMBL	8.77	—	—	CNC(=O)N1CCC(Nc2ncc(C(=O)NO)cn2)(c2ccccc2)CC1
E3 Binder	CHEMBL2333343	ChEMBL	7.55	—	—	CNC(=O)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4160296	ChEMBL	6.7	—	—	CNC(=O)c1ccc(Nc2c[nH]c3ccccc23)cc1
E3 Binder	CHEMBL4168213	ChEMBL	7.85	—	—	CNC(=O)c1ccc(Nc2csc3ccccc23)cc1
E3 Binder	CHEMBL1289926	ChEMBL	6.39	AXI	—	CNC(=O)c1ccccc1Sc1ccc2c(/C=C/c3ccccn3)n[nH]c2c1
E3 Binder	CHEMBL99661	ChEMBL	8.85	—	—	CNCC(=O)[C@@H](Cc1ccccc1)NC(=O)CCCCCCC(=O)NO
E3 Binder	CHEMBL4472676	ChEMBL	6.8	—	—	CNCCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1
E3 Binder	CHEMBL5172950	ChEMBL	6.06	—	—	CNNC(=O)c1ccc(CNC(=O)c2ccccc2)cc1
E3 Binder	CHEMBL4575735	ChEMBL	6.98	—	—	CNc1nc(Nc2cnn(CCCCCC(=O)NO)c2)ncc1Cl
E3 Binder	CHEMBL4439450	ChEMBL	7.43	—	—	CNc1nc(Nc2cnn(CCCCCCC(=O)NO)c2)ncc1C(F)(F)F
E3 Binder	CHEMBL4451298	ChEMBL	7.82	—	—	CNc1nc(Nc2cnn(CCCCCCC(=O)NO)c2)ncc1Cl
E3 Binder	CHEMBL2385379	ChEMBL	6.6	—	—	CNc1nc2c(s1)Cc1cc(/C=C/C(=O)NO)ccc1-2
E3 Binder	CHEMBL5202725	ChEMBL	8.04	—	—	CNc1ncc(-c2cn(Cc3ccc(C(=O)NO)cc3)c(=O)c(N3CCOCC3)n2)cn1
E3 Binder	CHEMBL2047669	ChEMBL	6.66	—	—	CO/N=C(\Cc1ccc(O)c(Br)c1)C(=O)NCCS
E3 Binder	CHEMBL5281979	ChEMBL	7.89	—	—	COC(=O)/C=C/c1ccc(OCCCNc2cc3c([nH]c4ccccc43)c(-c3ccc(OC)cc3)n2)c(OC)c1
E3 Binder	CHEMBL5266011	ChEMBL	7.77	—	—	COC(=O)/C=C/c1ccc(OCCNc2cc3c([nH]c4ccccc43)c(-c3ccc(OC)cc3)n2)c(OC)c1
E3 Binder	CHEMBL432243	ChEMBL	6.96	—	—	COC(=O)C(=O)CCCCCCCOc1ccc(-c2ccccc2)cc1
E3 Binder	CHEMBL432618	ChEMBL	7.21	—	—	COC(=O)C(=O)CCCCCCOc1ccc(-c2ccccc2)cc1
E3 Binder	CHEMBL321689	ChEMBL	7.09	—	—	COC(=O)C(=O)CCCCCOc1ccc(-c2ccccc2)cc1
E3 Binder	CHEMBL210858	ChEMBL	6.01	—	—	COC(=O)CC1CC(c2ccc(O)cc2)=NO1
E3 Binder	CHEMBL3979648	ChEMBL	6.77	—	—	COC(=O)CCCCCCCc1ccc(N2C(=S)N(c3ccc(C#N)c(C(F)(F)F)c3)C(=O)C2(C)C)cc1F
E3 Binder	CHEMBL3885174	ChEMBL	8.0	—	—	COC(=O)Cc1c(C)n(Cc2ccc(-c3cn(CCCCCCC(=O)NO)nn3)cc2)c2ccc(OC)cc12
E3 Binder	CHEMBL3885011	ChEMBL	8.3	—	—	COC(=O)Cc1c(C)n(Cc2ccc(-c3cn(CCCCCCCC(=O)NO)nn3)cc2)c2ccc(OC)cc12
E3 Binder	CHEMBL343476	ChEMBL	7.36	—	—	COC(=O)NCCSSCCNC(=O)/C(Cc1ccc(O)c(Br)c1)=N/O
E3 Binder	CHEMBL388195	ChEMBL	7.86	—	—	COC(=O)[C@@H]1Cc2cccc(c2)C[C@H](NC(C)=O)C(=O)N[C@@H](CCCCCC(=O)NO)C(=O)N1
E3 Binder	CHEMBL259517	ChEMBL	6.16	—	—	COC(=O)[C@H](Cc1ccc(-c2ccc(-c3ccccc3)cc2)cc1)NC(=O)CCCCCCC(=O)NO
E3 Binder	CHEMBL227663	ChEMBL	6.78	—	—	COC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H](C)NC(C)=O
E3 Binder	CHEMBL4455730	ChEMBL	6.67	—	—	COC(=O)c1c(CCCCCCCC(=O)NO)cccc1OC
E3 Binder	CHEMBL471043	ChEMBL	7.03	—	—	COC(=O)c1ccc(CO/N=C/c2ccc(/C=C/C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4563988	ChEMBL	7.02	—	—	COC(=O)c1ccc2ccccc2c1OCCCCCCCC(=O)NO
E3 Binder	CHEMBL3693811	ChEMBL	7.38	—	—	COC(C)(c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1)c1ccccn1
E3 Binder	CHEMBL3693810	ChEMBL	8.4	—	—	COC(C)(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1ccccn1
E3 Binder	CHEMBL3693807	ChEMBL	7.77	—	—	COC(C)(c1ccc(F)cc1)c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693806	ChEMBL	8.52	—	—	COC(C)(c1ccc(F)cc1)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL4752855	ChEMBL	6.54	—	—	COC(c1c(F)cccc1Cl)c1c[nH]c2ncc(-c3c(C)noc3C)cc12
E3 Binder	CHEMBL3640657	ChEMBL	7.77	—	—	COC(c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1)(c1cc(F)cc(F)c1)c1cc(F)cc(F)c1
E3 Binder	CHEMBL3640653	ChEMBL	7.58	—	—	COC(c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1)(c1ccc(F)cc1F)c1ccc(F)cc1F
E3 Binder	CHEMBL3693802	ChEMBL	7.33	—	—	COC(c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1)(c1cccc(F)c1)c1cccc(F)c1
E3 Binder	CHEMBL3640649	ChEMBL	7.77	—	—	COC(c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1)(c1ccccc1F)c1ccccc1F
E3 Binder	CHEMBL3640656	ChEMBL	7.7	—	—	COC(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)(c1cc(F)cc(F)c1)c1cc(F)cc(F)c1
E3 Binder	CHEMBL3640659	ChEMBL	6.9	—	—	COC(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)(c1ccc(F)cc1C)c1ccc(F)cc1C
E3 Binder	CHEMBL3640652	ChEMBL	7.7	—	—	COC(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)(c1ccc(F)cc1F)c1ccc(F)cc1F
E3 Binder	CHEMBL3693797	ChEMBL	7.82	—	—	COC(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)(c1cccc(F)c1)c1cccc(F)c1
E3 Binder	CHEMBL3640648	ChEMBL	8.22	—	—	COC(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)(c1ccccc1F)c1ccccc1F
E3 Binder	CHEMBL3640663	ChEMBL	7.64	—	—	COC(c1ccc(F)cc1)(c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1)c1ccccn1
E3 Binder	CHEMBL3640668	ChEMBL	8.0	—	—	COC(c1ccc(F)cc1)(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)C(F)(F)F
E3 Binder	CHEMBL3640662	ChEMBL	8.52	—	—	COC(c1ccc(F)cc1)(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1ccccn1
E3 Binder	CHEMBL3693779	ChEMBL	7.89	—	—	COC(c1ccc(F)cc1)(c1ccc(F)cc1)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3640672	ChEMBL	7.7	—	—	COC(c1cccc(C(=O)NCCCCCCC(=O)NO)c1)(c1ccccn1)c1ccccn1
E3 Binder	CHEMBL3693781	ChEMBL	7.72	—	—	COC(c1ccccc1)(c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1)c1cccnc1
E3 Binder	CHEMBL3640677	ChEMBL	8.4	—	—	COC(c1ccccc1)(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1ccc(C(=O)N(C)C)cc1
E3 Binder	CHEMBL3640678	ChEMBL	8.52	—	—	COC(c1ccccc1)(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1cccc(C(=O)N(C)C)c1
E3 Binder	CHEMBL3693782	ChEMBL	8.52	—	—	COC(c1ccccc1)(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1ccccn1
E3 Binder	CHEMBL3693780	ChEMBL	8.52	—	—	COC(c1ccccc1)(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1cccnc1
E3 Binder	CHEMBL3693789	ChEMBL	8.52	—	—	COC(c1ccccc1)(c1ccncc1)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL5206736	ChEMBL	7.0	—	—	COC1=CC(OCc2cccc(-c3ccc4c(c3)OCCO4)c2C)=CC(OC)C1CNCCCCCCC(=O)NO
E3 Binder	CHEMBL5190763	ChEMBL	8.13	—	—	COC1CCN(c2nc(-c3cnc(N)nc3)cn(Cc3ccc(C(=O)NO)cc3)c2=O)CC1
E3 Binder	CHEMBL593846	ChEMBL	8.82	—	—	COCC(/C=C/c1ccccc1)N1CCN(c2ncc(C(=O)NO)cn2)CC1
E3 Binder	CHEMBL2179245	ChEMBL	7.22	—	—	COCCCN(C(=O)NCc1ccc(C(=O)NO)cc1)c1ccccc1
E3 Binder	CHEMBL2179616	ChEMBL	7.93	—	—	COCCCN(Cc1ccc(C(=O)NO)cc1)C(=O)Nc1ccccc1
E3 Binder	CHEMBL3601342	ChEMBL	7.87	—	—	COCCCNc1nccc2ccc(NC(=O)CCCCCCC(=O)NO)cc12
E3 Binder	CHEMBL518907	ChEMBL	6.92	—	—	COCCCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)CSC(C)=O)cn2)cc1
E3 Binder	CHEMBL3601339	ChEMBL	6.83	—	—	COCCN(CCOC)c1nccc2ccc(NC(=O)CCCCCCC(=O)NO)cc12
E3 Binder	CHEMBL2179617	ChEMBL	8.03	—	—	COCCN(Cc1ccc(C(=O)NO)cc1)C(=O)Nc1ccccc1
E3 Binder	CHEMBL5191960	ChEMBL	7.56	—	—	COCCN(Cc1ccc(C(=O)NO)cc1)S(=O)(=O)c1cc(F)c(F)c(F)c1F
E3 Binder	CHEMBL3640695	ChEMBL	7.89	—	—	COCCN1CCN(c2ncc(C(=O)NCCCCCCC(=O)NO)cn2)CC1
E3 Binder	CHEMBL2385393	ChEMBL	6.85	—	—	COCCNc1nc2c(s1)Cc1cc(/C=C/C(=O)NO)ccc1-2
E3 Binder	CHEMBL4593341	ChEMBL	7.54	—	—	COCCOCC(=O)SCCCCCC(NC(=O)OCc1ccccc1)C(=O)Nc1cccc2cccnc12
E3 Binder	CHEMBL4793958	ChEMBL	6.25	—	—	COCCOc1cc2ncnc(Nc3ccc(/C=C/C(=O)NO)cc3)c2cc1OCCOC
E3 Binder	CHEMBL3944171	ChEMBL	6.0	—	—	COCCOc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)CCCC(=O)NO
E3 Binder	CHEMBL3946801	ChEMBL	7.0	—	—	COCCOc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)CCCCC(=O)NO
E3 Binder	CHEMBL597569	ChEMBL	8.08	—	—	COCCOc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL443241	ChEMBL	6.53	—	—	COCCSC(=S)SCC(=O)c1ccc(OC)cc1
E3 Binder	CHEMBL4445881	ChEMBL	7.2	—	—	COCCc1cn(Cc2ccc(C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL4250891	ChEMBL	8.68	—	—	COCCn1cc(-c2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc3[nH]ccc23)cn1
E3 Binder	CHEMBL3940062	ChEMBL	6.82	—	—	COC[C@@H]1CCCC1c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3938052	ChEMBL	6.82	—	—	COC[C@@H]1CCCN1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4777726	ChEMBL	7.21	—	—	COc1c(-c2ccccc2)c2ccccc2n(Cc2ccc(C(=O)NO)cc2)c1=O
E3 Binder	CHEMBL5170300	ChEMBL	7.21	—	—	COc1c(OCCCCCC(=O)NO)ccc2c1N=C(NC(=O)c1ccccc1)N1CCN=C21
E3 Binder	CHEMBL3759998	ChEMBL	7.08	—	—	COc1cc(-c2cc(C(=O)NCCCCCCS)[nH]n2)cc(OC)c1OC
E3 Binder	CHEMBL5192364	ChEMBL	8.14	—	—	COc1cc(-c2nc(-c3nnc(CCCCC(=O)NO)o3)cc3c2[nH]c2ccccc23)cc(OC)c1OC
E3 Binder	CHEMBL4534004	ChEMBL	8.14	—	—	COc1cc(-c2nc(NCc3ccc(/C=C/C(=O)NO)cc3)cc3c2[nH]c2ccccc23)cc(OC)c1OC
E3 Binder	CHEMBL4278715	ChEMBL	9.03	—	—	COc1cc(-c2nc(NCc3ccc(C(=O)NO)cc3)cc3c2[nH]c2ccccc23)cc(OC)c1OC
E3 Binder	CHEMBL4461441	ChEMBL	8.51	—	—	COc1cc(-c2nc(NCc3cccc(/C=C/C(=O)NO)c3)cc3c2[nH]c2ccccc23)cc(OC)c1OC
E3 Binder	CHEMBL5079482	ChEMBL	7.0	—	—	COc1cc(-c2ncc(/C=C/C(=O)NO)s2)cc(OC)c1OC
E3 Binder	CHEMBL5070026	ChEMBL	7.1	—	—	COc1cc(-c2ncc(/C=C/C(=O)Nc3ccccc3N)s2)cc(OC)c1OC
E3 Binder	CHEMBL5075320	ChEMBL	6.17	—	—	COc1cc(-c2ncc(C(=O)NCCCCCCC(=O)NO)s2)cc(OC)c1OC
E3 Binder	CHEMBL1076939	ChEMBL	8.41	—	—	COc1cc(-n2cc(-c3cccc(NC(=O)CCCCCCC(=O)NO)c3)nn2)ccc1F
E3 Binder	CHEMBL116438	ChEMBL	6.27	—	—	COc1cc(/C=C/C(=O)/C=C(O)/C=C/c2ccc(O)c(OC)c2)ccc1O
E3 Binder	CHEMBL5280065	ChEMBL	7.7	—	—	COc1cc(/C=C/C(=O)NO)ccc1C(=O)NCC1CCN(Cc2ccccc2)CC1
E3 Binder	CHEMBL4581044	ChEMBL	6.42	—	—	COc1cc(/C=C/C(=O)NO)ccc1OCCCCN(C)C(=O)c1ccccc1O
E3 Binder	CHEMBL4543731	ChEMBL	6.44	—	—	COc1cc(/C=C/C(=O)NO)ccc1OCCCCNC(=O)c1ccccc1O
E3 Binder	CHEMBL4467212	ChEMBL	6.46	—	—	COc1cc(/C=C/C(=O)NO)ccc1OCCCN(C)C(=O)c1ccccc1O
E3 Binder	CHEMBL4468821	ChEMBL	6.26	—	—	COc1cc(/C=C/C(=O)NO)ccc1OCCCNC(=O)c1ccccc1O
E3 Binder	CHEMBL4465947	ChEMBL	6.37	—	—	COc1cc(/C=C/C(=O)NO)ccc1OCCN(C)C(=O)c1ccccc1O
E3 Binder	CHEMBL2336045	ChEMBL	6.77	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC(=O)OC(C)(C)C
E3 Binder	CHEMBL2335646	ChEMBL	6.21	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C
E3 Binder	CHEMBL2335638	ChEMBL	6.37	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C
E3 Binder	CHEMBL2335635	ChEMBL	6.75	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](NC(=O)OC(C)(C)C)[C@@H](C)O
E3 Binder	CHEMBL2335639	ChEMBL	6.1	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H]1CC2(CN1C(=O)OC(C)(C)C)SCCS2
E3 Binder	CHEMBL2335634	ChEMBL	6.37	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C
E3 Binder	CHEMBL2331640	ChEMBL	6.8	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](C)NC(=O)OC(C)(C)C
E3 Binder	CHEMBL2336047	ChEMBL	6.24	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C
E3 Binder	CHEMBL2331641	ChEMBL	6.75	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCSC)NC(=O)OC(C)(C)C
E3 Binder	CHEMBL2335636	ChEMBL	6.85	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CO)NC(=O)OC(C)(C)C
E3 Binder	CHEMBL2336044	ChEMBL	6.31	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C
E3 Binder	CHEMBL2335637	ChEMBL	6.5	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C
E3 Binder	CHEMBL2336046	ChEMBL	6.21	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C
E3 Binder	CHEMBL2335641	ChEMBL	6.14	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NC(=O)c1ccc(NC(=O)OC(C)(C)C)cc1
E3 Binder	CHEMBL2335645	ChEMBL	6.15	—	—	COc1cc(/C=C/C(=O)NO)ccc1OC[C@H](Cc1c[nH]c2ccccc12)NS(=O)(=O)c1ccc(NC(C)=O)cc1
E3 Binder	CHEMBL83527	ChEMBL	6.26	—	—	COc1cc(/C=C/c2ccc(O)cc2)cc(OC)c1
E3 Binder	CHEMBL5175648	ChEMBL	7.63	—	—	COc1cc(/C=C/c2ccc(OCCCCCCC(=O)NO)cc2)cc(OC)c1
E3 Binder	CHEMBL5274737	ChEMBL	7.05	—	—	COc1cc(/C=C2\N=C(c3ccccc3)N(n3c(SCC(=O)NO)nnc3-c3ccccc3)C2=O)ccc1O
E3 Binder	CHEMBL5281824	ChEMBL	6.32	—	—	COc1cc(/C=C2\SC(=O)N(CCNC(=O)Nc3c(C)n(C)n(-c4ccccc4)c3=O)C2=O)cc(OC)c1OC
E3 Binder	CHEMBL4102654	ChEMBL	7.97	—	—	COc1cc(C(=O)NCCc2ccc(/C=C/C(=O)NO)cc2)ccc1O
E3 Binder	CHEMBL4643795	ChEMBL	7.22	—	—	COc1cc(C(=O)NOCCCCCC(=O)NO)cc(OC)c1OC
E3 Binder	CHEMBL1164564	ChEMBL	6.7	—	—	COc1cc(C(=O)OCCCCCCCOC(=O)c2ccc(O)c(OC)c2)ccc1O
E3 Binder	CHEMBL395976	ChEMBL	6.0	—	—	COc1cc(C(=O)c2cc3cc(/C=C/C(=O)NO)ccc3o2)cc(OC)c1OC
E3 Binder	CHEMBL4215029	ChEMBL	6.84	—	—	COc1cc(C(=O)c2ccc3c(ccn3Cc3ccc(/C=C/C(=O)NO)cc3)c2)cc(OC)c1OC
E3 Binder	CHEMBL4202838	ChEMBL	6.01	—	—	COc1cc(C(=O)c2ccc3c(ccn3S(=O)(=O)c3ccc(/C=C/C(=O)NO)cc3)c2)cc(OC)c1OC
E3 Binder	CHEMBL4218915	ChEMBL	6.25	—	—	COc1cc(C(=O)c2ccc3c(ccn3S(=O)(=O)c3cccc(/C=C/C(=O)NO)c3)c2)cc(OC)c1OC
E3 Binder	CHEMBL4098353	ChEMBL	6.86	—	—	COc1cc(C(=O)c2cn(Cc3ccc(/C=C/C(=O)NO)cc3)c3ccccc23)cc(OC)c1OC
E3 Binder	CHEMBL4072479	ChEMBL	6.1	—	—	COc1cc(C(=O)c2cn(S(=O)(=O)c3cccc(/C=C/C(=O)NO)c3)c3ccccc23)cc(OC)c1OC
E3 Binder	CHEMBL2047696	ChEMBL	6.29	—	—	COc1cc(C/C(=N\O)C(=O)NCCS)cc(Br)c1OC
E3 Binder	CHEMBL2047695	ChEMBL	6.57	—	—	COc1cc(C/C(=N\O)C(=O)NCCS)cc(I)c1OC
E3 Binder	CHEMBL4437259	ChEMBL	7.4	—	—	COc1cc(C/C(=N\O)C(=O)NCCSSCCNC(=O)/C(Cc2ccc(O)c(OC)c2)=N/O)ccc1O
E3 Binder	CHEMBL5288040	ChEMBL	6.77	—	—	COc1cc(CCC(=O)NO)ccc1C(=O)NCC1CCN(Cc2ccccc2)CC1
E3 Binder	CHEMBL4440734	ChEMBL	7.01	—	—	COc1cc(CCc2nc(CCC(=O)NO)cs2)cc(OC)c1OC
E3 Binder	CHEMBL3655932	ChEMBL	8.7	—	—	COc1cc(F)ccc1CNc1ncc(C(=O)NO)cn1
E3 Binder	CHEMBL429090	ChEMBL	7.22	—	—	COc1cc(NC(=O)CCCCCCC(=O)NO)ccc1-c1cnco1
E3 Binder	CHEMBL5191956	ChEMBL	7.07	—	—	COc1cc(NC(=O)CCCCCCC(=O)NO)ccc1Nc1nccc(-c2cn(C)c3ccccc23)n1
E3 Binder	CHEMBL4870955	ChEMBL	7.07	—	—	COc1cc(NC(=O)CCCCCCCCCCC(=O)NO)ccc1Nc1nccc(-c2cn(C)c3ccccc23)n1
E3 Binder	CHEMBL515295	ChEMBL	6.36	—	—	COc1cc(NC(=O)CCCCCNS(N)(=O)=O)c2ncccc2c1
E3 Binder	CHEMBL4067006	ChEMBL	8.55	—	—	COc1cc(NC(=O)NOCCCCCC(=O)NO)c2nc(OC)cc(C)c2c1
E3 Binder	CHEMBL4088276	ChEMBL	7.61	—	—	COc1cc(NC(=O)NOCCCCCC(=O)NO)c2nccc(C)c2c1
E3 Binder	CHEMBL4070745	ChEMBL	8.21	—	—	COc1cc(NC(=O)NOCCCCCC(=O)NO)c2ncccc2c1
E3 Binder	CHEMBL473082	ChEMBL	7.22	—	—	COc1cc(NC(=O)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc2ccccc2)c2ncccc2c1
E3 Binder	CHEMBL562551	ChEMBL	6.39	—	—	COc1cc(NC(=O)c2ccccn2)ccc1Cl
E3 Binder	CHEMBL3652241	ChEMBL	8.3	—	—	COc1cc(Nc2ncc(C(=O)NO)cn2)cc(C(F)(F)F)c1
E3 Binder	CHEMBL3652243	ChEMBL	8.52	—	—	COc1cc(Nc2ncc(C(=O)NO)cn2)cc(OC)c1
E3 Binder	CHEMBL3921816	ChEMBL	7.73	—	—	COc1cc(Nc2ncnc3ccc(-c4cn(CCCCCC(=O)NO)nn4)cc23)ccc1Oc1ccccc1
E3 Binder	CHEMBL3982710	ChEMBL	7.8	—	—	COc1cc(Nc2ncnc3ccc(-c4cn(CCCCCCC(=O)NO)nn4)cc23)ccc1Oc1ccccc1
E3 Binder	CHEMBL4096161	ChEMBL	6.54	—	—	COc1cc(OC)c2c(=O)[nH]c(-c3cc(C)c(OCCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4785540	ChEMBL	6.54	—	—	COc1cc(OC)c2c(=O)[nH]c(-c3ccc(OC/C=C/C(=O)NO)cc3)nc2c1
E3 Binder	CHEMBL4799694	ChEMBL	7.5	—	—	COc1cc(OC)c2c(=O)[nH]c(-c3ccc(OCCCC(=O)NO)cc3)nc2c1
E3 Binder	CHEMBL4064918	ChEMBL	6.54	—	—	COc1cc(OC)c2c(=O)[nH]c(-c3ccc(OCCCCC(=O)NO)cc3)nc2c1
E3 Binder	CHEMBL4091545	ChEMBL	6.54	—	—	COc1cc(OC)c2c(=O)[nH]c(-c3ccc(OCCCCCC(=O)NO)cc3)nc2c1
E3 Binder	CHEMBL4792138	ChEMBL	6.54	—	—	COc1cc(OC)c2c(=O)[nH]c(-c3ccc(OCCCCCCC(=O)NO)cc3)nc2c1
E3 Binder	CHEMBL4779876	ChEMBL	6.54	—	—	COc1cc(OC)c2c(=O)[nH]c(-c3ccc(OCCCCCCCC(=O)NO)cc3)nc2c1
E3 Binder	CHEMBL4782913	ChEMBL	6.54	—	—	COc1cc(OC)c2c(=O)[nH]c(-c3ccc(OCc4cc(C)c(/C=C/C(=O)NO)c(C)c4)cc3)nc2c1
E3 Binder	CHEMBL4091222	ChEMBL	6.54	—	—	COc1cc(OC)c2c(=O)[nH]c(-c3ccc(OCc4ccc(/C=C/C(=O)NO)cc4)cc3)nc2c1
E3 Binder	CHEMBL4748700	ChEMBL	6.54	—	—	COc1cc(OC)c2c(=O)[nH]c(-c3ccc(Oc4ccc(C(=O)NO)cn4)cc3)nc2c1
E3 Binder	CHEMBL4798807	ChEMBL	6.14	—	—	COc1cc(OC)c2c(N3CCC(F)(F)CC3)nc(-c3cc(C)c(OCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4784047	ChEMBL	6.47	—	—	COc1cc(OC)c2c(N3CCC(F)(F)CC3)nc(-c3cc(C)c(OCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4796983	ChEMBL	6.73	—	—	COc1cc(OC)c2c(N3CCC(F)(F)CC3)nc(-c3cc(C)c(OCCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4796311	ChEMBL	6.41	—	—	COc1cc(OC)c2c(N3CCCC3)nc(-c3cc(C)c(OCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4781332	ChEMBL	6.51	—	—	COc1cc(OC)c2c(N3CCCC3)nc(-c3cc(C)c(OCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4799432	ChEMBL	6.99	—	—	COc1cc(OC)c2c(N3CCCC3)nc(-c3cc(C)c(OCCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4790422	ChEMBL	6.32	—	—	COc1cc(OC)c2c(N3CCCCC3)nc(-c3cc(C)c(OCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4785179	ChEMBL	6.69	—	—	COc1cc(OC)c2c(N3CCCCC3)nc(-c3cc(C)c(OCCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4798124	ChEMBL	6.19	—	—	COc1cc(OC)c2c(N3CCN(C)CC3)nc(-c3cc(C)c(OCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4800256	ChEMBL	6.96	—	—	COc1cc(OC)c2c(N3CCN(C)CC3)nc(-c3cc(C)c(OCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4781177	ChEMBL	7.93	—	—	COc1cc(OC)c2c(N3CCN(C)CC3)nc(-c3cc(C)c(OCCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4783090	ChEMBL	6.46	—	—	COc1cc(OC)c2c(N3CCOCC3)nc(-c3cc(C)c(OCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4799485	ChEMBL	6.68	—	—	COc1cc(OC)c2c(N3CCOCC3)nc(-c3cc(C)c(OCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4782504	ChEMBL	6.92	—	—	COc1cc(OC)c2c(N3CCOCC3)nc(-c3cc(C)c(OCCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4790567	ChEMBL	6.44	—	—	COc1cc(OC)c2c(N3CCOC[C@@H]3C)nc(-c3cc(C)c(OCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4784467	ChEMBL	6.72	—	—	COc1cc(OC)c2c(N3CCOC[C@@H]3C)nc(-c3cc(C)c(OCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4784631	ChEMBL	7.01	—	—	COc1cc(OC)c2c(N3CCOC[C@@H]3C)nc(-c3cc(C)c(OCCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4787879	ChEMBL	6.48	—	—	COc1cc(OC)c2c(N3CCOC[C@H]3C)nc(-c3cc(C)c(OCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4778309	ChEMBL	6.66	—	—	COc1cc(OC)c2c(N3CCOC[C@H]3C)nc(-c3cc(C)c(OCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4779480	ChEMBL	6.99	—	—	COc1cc(OC)c2c(N3CCOC[C@H]3C)nc(-c3cc(C)c(OCCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4793662	ChEMBL	6.07	—	—	COc1cc(OC)c2c(N3CCS(=O)(=O)CC3)nc(-c3cc(C)c(OCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4784493	ChEMBL	6.89	—	—	COc1cc(OC)c2c(N3CCS(=O)(=O)CC3)nc(-c3cc(C)c(OCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4790998	ChEMBL	7.26	—	—	COc1cc(OC)c2c(N3CCS(=O)(=O)CC3)nc(-c3cc(C)c(OCCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4779947	ChEMBL	6.38	—	—	COc1cc(OC)c2c(N3CCSCC3)nc(-c3cc(C)c(OCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4777336	ChEMBL	6.54	—	—	COc1cc(OC)c2c(N3CCSCC3)nc(-c3cc(C)c(OCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL4793037	ChEMBL	6.89	—	—	COc1cc(OC)c2c(N3CCSCC3)nc(-c3cc(C)c(OCCCCCC(=O)NO)c(C)c3)nc2c1
E3 Binder	CHEMBL294194	ChEMBL	8.51	—	—	COc1cc(OC)c2cc(C(=O)NCCCCCCC(=O)NO)[nH]c2c1
E3 Binder	CHEMBL4210899	ChEMBL	6.62	—	—	COc1cc(OC)cc(-c2ccc3c(NC(=O)c4ccc(C(=O)NO)cc4)n[nH]c3c2)c1
E3 Binder	CHEMBL5093312	ChEMBL	6.14	—	—	COc1cc(OC)cc(-c2ncc(/C=C/C(=O)NO)s2)c1
E3 Binder	CHEMBL5085919	ChEMBL	6.12	—	—	COc1cc(OC)cc(-c2ncc(C(=O)NCCCCCCC(=O)NO)s2)c1
E3 Binder	CHEMBL4562808	ChEMBL	7.58	—	—	COc1cc(OC)cc(C(=O)N(CCC(=O)NCc2ccccc2)Cc2ccc(C(=O)NO)cc2)c1
E3 Binder	CHEMBL4645688	ChEMBL	7.52	—	—	COc1cc(OC)cc(C(=O)NOCCCCCC(=O)NO)c1
E3 Binder	CHEMBL3655998	ChEMBL	8.52	—	—	COc1cc(OC)cc(C2(Nc3ncc(C(=O)NO)cn3)CC2)c1
E3 Binder	CHEMBL5186206	ChEMBL	6.97	—	—	COc1cc(OC)cc(N(CCCCC(=O)NO)c2ccc3ncc(-c4cnn(C)c4)nc3c2)c1
E3 Binder	CHEMBL5179582	ChEMBL	8.2	—	—	COc1cc(OC)cc(N(CCCCCC(=O)NO)c2ccc3ncc(-c4cnn(C)c4)nc3c2)c1
E3 Binder	CHEMBL5191916	ChEMBL	7.89	—	—	COc1cc(OC)cc(N(CCCCCCC(=O)NO)c2ccc3ncc(-c4cnn(C)c4)nc3c2)c1
E3 Binder	CHEMBL5177696	ChEMBL	8.59	—	—	COc1cc(OC)cc(N(CCNC(C)C)c2ccc3ncc(-c4cnn(CCCCCCC(=O)NO)c4)nc3c2)c1
E3 Binder	CHEMBL5181688	ChEMBL	8.47	—	—	COc1cc(OC)cc(N(CCNC(C)C)c2ccc3ncc(-c4cnn(CCOc5ccc(C(=O)NO)cc5)c4)nc3c2)c1
E3 Binder	CHEMBL5175835	ChEMBL	6.85	—	—	COc1cc(OCc2cccc(-c3ccc4c(c3)OCCO4)c2C)cc(OC)c1CNCCCCCC(=O)NO
E3 Binder	CHEMBL5208995	ChEMBL	6.19	—	—	COc1cc(OCc2cccc(-c3ccccc3)c2C)cc(OC)c1CN(C)CCCCC(=O)NO
E3 Binder	CHEMBL5198026	ChEMBL	6.37	—	—	COc1cc(OCc2cccc(-c3ccccc3)c2C)cc(OC)c1CNCCCCCC(=O)NO
E3 Binder	CHEMBL5185866	ChEMBL	7.64	—	—	COc1cc(OCc2cccc(-c3ccccc3)c2C)cc(OC)c1CNCCCCCCC(=O)NO
E3 Binder	CHEMBL4644775	ChEMBL	7.58	—	—	COc1cc(Oc2ccc3nc(/C=C/C(=O)NO)ccc3c2)cc(OC)c1OC
E3 Binder	CHEMBL2442697	ChEMBL	6.89	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3ccc(NC(=O)CCCCCC(=O)NO)cc3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442698	ChEMBL	7.05	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442791	ChEMBL	6.67	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3ccc(OCCCC(=O)NO)cc3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442794	ChEMBL	7.06	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3ccc(OCCCCC(=O)NO)cc3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442797	ChEMBL	7.58	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3ccc(OCCCCCC(=O)NO)cc3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442800	ChEMBL	7.8	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3ccc(OCCCCCCC(=O)NO)cc3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442691	ChEMBL	7.28	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3ccc(OCCCCCCCC(=O)NO)cc3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442699	ChEMBL	6.28	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3cccc(NC(=O)CCCCC(=O)NO)c3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442789	ChEMBL	6.8	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3cccc(NC(=O)CCCCCC(=O)NO)c3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442790	ChEMBL	7.4	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3cccc(NC(=O)CCCCCCC(=O)NO)c3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442792	ChEMBL	6.39	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3cccc(OCCCC(=O)NO)c3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442795	ChEMBL	7.38	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3cccc(OCCCCC(=O)NO)c3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442798	ChEMBL	7.82	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3cccc(OCCCCCC(=O)NO)c3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442801	ChEMBL	8.25	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3cccc(OCCCCCCC(=O)NO)c3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442692	ChEMBL	7.16	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3cccc(OCCCCCCCC(=O)NO)c3)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442793	ChEMBL	6.45	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3ccccc3OCCCC(=O)NO)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442796	ChEMBL	7.08	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3ccccc3OCCCCC(=O)NO)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442799	ChEMBL	7.7	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3ccccc3OCCCCCC(=O)NO)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL2442802	ChEMBL	7.57	—	—	COc1cc([C@@H]2c3cc4c(cc3[C@@H](Nc3ccccc3OCCCCCCC(=O)NO)[C@H]3COC(=O)[C@H]23)OCO4)cc(OC)c1O
E3 Binder	CHEMBL513024	ChEMBL	6.17	—	—	COc1cc2c(=O)c(-c3ccc(O)cc3)coc2cc1O
E3 Binder	CHEMBL4854447	ChEMBL	7.41	—	—	COc1cc2c(NC3CCN(Cc4ccc(C(=O)NO)cc4)CC3)cc(-c3ccc(C)o3)nc2cc1OCCCN1CCCC1
E3 Binder	CHEMBL4855710	ChEMBL	6.88	—	—	COc1cc2c(NC3CCN(c4ccc(C(=O)NO)cc4)CC3)cc(-c3ccc(C)o3)nc2cc1OCCCN1CCCC1
E3 Binder	CHEMBL4863011	ChEMBL	6.93	—	—	COc1cc2c(NC3CCN(c4ncc(C(=O)NO)cn4)CC3)cc(C)nc2cc1OCCCN1CCCC1
E3 Binder	CHEMBL4850606	ChEMBL	7.47	—	—	COc1cc2c(NCC3CCC(C(=O)NO)CC3)cc(-c3ccc(C)o3)nc2cc1OCCCN1CCCC1
E3 Binder	CHEMBL4849689	ChEMBL	6.91	—	—	COc1cc2c(NCC3CCC(c4ccc(C(=O)NO)cc4)CC3)cc(-c3ccc(C)o3)nc2cc1OCCCN1CCCC1
E3 Binder	CHEMBL4856184	ChEMBL	7.28	—	—	COc1cc2c(NCC3CCN(Cc4ccc(C(=O)NO)cc4)CC3)cc(-c3ccc(C)o3)nc2cc1OCCCN1CCCC1
E3 Binder	CHEMBL4873711	ChEMBL	7.17	—	—	COc1cc2c(NCC3CCN(c4ccc(C(=O)NO)cc4)CC3)cc(-c3ccc(C)o3)nc2cc1OCCCN1CCCC1
E3 Binder	CHEMBL4876993	ChEMBL	6.46	—	—	COc1cc2c(NCC3CCN(c4ncc(C(=O)NO)cn4)CC3)cc(-c3ccc(C)o3)nc2cc1OCC1CCNCC1
E3 Binder	CHEMBL4852593	ChEMBL	6.82	—	—	COc1cc2c(NCC3CCN(c4ncc(C(=O)NO)cn4)CC3)cc(-c3ccc(C)o3)nc2cc1OCCCN1CCCC1
E3 Binder	CHEMBL4865830	ChEMBL	6.46	—	—	COc1cc2c(NCC3CCN(c4ncc(C(=O)NO)cn4)CC3)cc(C)nc2cc1OCCCN1CCCC1
E3 Binder	CHEMBL4866673	ChEMBL	6.9	—	—	COc1cc2c(NCc3ccc(-c4ccc(C(=O)NO)cc4)cc3)cc(-c3ccc(C)o3)nc2cc1OCCCN1CCCC1
E3 Binder	CHEMBL4872188	ChEMBL	7.96	—	—	COc1cc2c(NCc3ccc(C(=O)NO)cc3)cc(-c3ccc(C)o3)nc2cc1OCCCN1CCCC1
E3 Binder	CHEMBL4850038	ChEMBL	6.46	—	—	COc1cc2c(NCc3ccc([C@H]4CC[C@@H](C(=O)NO)CC4)cc3)cc(-c3ccc(C)o3)nc2cc1OCCCN1CCCC1
E3 Binder	CHEMBL598610	ChEMBL	7.18	—	—	COc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL3892687	ChEMBL	7.0	—	—	COc1cc2c(Nc3ccc4[nH]c(C)cc4c3F)ncnc2cc1OCCCCC(=O)NO
E3 Binder	CHEMBL5290012	ChEMBL	6.25	—	—	COc1cc2c(Nc3cccc(/C=C/C(=O)NO)c3)ncnc2cc1OCCCN1CCOCC1
E3 Binder	CHEMBL3981567	ChEMBL	6.62	—	—	COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCC(=O)NO
E3 Binder	CHEMBL3911566	ChEMBL	8.08	—	—	COc1cc2c(Oc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL2385954	ChEMBL	6.36	—	—	COc1cc2c(c(OC)c1OC)-c1ccc(OC)c(=O)cc1[C@@H](NC(=O)CCCCC(=O)NO)CC2
E3 Binder	CHEMBL2385955	ChEMBL	6.12	—	—	COc1cc2c(c(OC)c1OC)-c1ccc(OC)c(=O)cc1[C@@H](NC(=O)CCCCCC(=O)NO)CC2
E3 Binder	CHEMBL3640691	ChEMBL	8.7	—	—	COc1cc2c(cc1OC)CN(c1ncc(C(=O)NCCCCCCC(=O)NO)cn1)CC2
E3 Binder	CHEMBL4860396	ChEMBL	7.85	—	—	COc1cc2c(cc1OC)N(Cc1ccc(C(=O)NO)cc1)CCCC2
E3 Binder	CHEMBL1631913	ChEMBL	8.71	—	—	COc1cc2cc(c1)COc1ccccc1NC(=O)C(CCCCCC(=O)NO)OC/C=C\2
E3 Binder	CHEMBL1631916	ChEMBL	8.07	—	—	COc1cc2cc(c1)COc1ccccc1NC(=O)C(CCCCCC(=O)NO)OCCC2
E3 Binder	CHEMBL1631915	ChEMBL	7.99	—	—	COc1cc2cc(c1)COc1ccccc1NC(=O)[C@@H](CCCCCC(=O)NO)OC/C=C\2
E3 Binder	CHEMBL1631918	ChEMBL	8.41	—	—	COc1cc2cc(c1)COc1ccccc1NC(=O)[C@@H](CCCCCC(=O)NO)OCCC2
E3 Binder	CHEMBL1631914	ChEMBL	9.08	—	—	COc1cc2cc(c1)COc1ccccc1NC(=O)[C@H](CCCCCC(=O)NO)OC/C=C\2
E3 Binder	CHEMBL1631917	ChEMBL	8.46	—	—	COc1cc2cc(c1)COc1ccccc1NC(=O)[C@H](CCCCCC(=O)NO)OCCC2
E3 Binder	CHEMBL4172420	ChEMBL	8.07	—	—	COc1cc2ccn(CCCCOc3cccc(NC(=O)CCCCCCC(=O)NO)c3)c2c(OC)c1OC
E3 Binder	CHEMBL4176214	ChEMBL	8.15	—	—	COc1cc2ccn(CCOc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)c2cc1OC
E3 Binder	CHEMBL4162183	ChEMBL	8.02	—	—	COc1cc2ccn(CCOc3cccc(NC(=O)CCCCCCC(=O)NO)c3)c2c(OC)c1OC
E3 Binder	CHEMBL4850570	ChEMBL	6.9	—	—	COc1cc2nc(-c3cc(C)oc3C)cc(NCC3CCN(c4ncc(C(=O)NO)cn4)CC3)c2cc1OC
E3 Binder	CHEMBL4862662	ChEMBL	6.46	—	—	COc1cc2nc(-c3ccc(C)o3)cc(NC3CCN(c4ncc(C(=O)NO)cn4)CC3)c2cc1OC
E3 Binder	CHEMBL4876823	ChEMBL	6.62	—	—	COc1cc2nc(-c3ccc(C)o3)cc(NCC3C4CCC3CN(c3ncc(C(=O)NO)cn3)C4)c2cc1OC
E3 Binder	CHEMBL4862781	ChEMBL	7.39	—	—	COc1cc2nc(-c3ccc(C)o3)cc(NCC3CCC(C(=O)NO)CC3)c2cc1OC
E3 Binder	CHEMBL4870578	ChEMBL	7.08	—	—	COc1cc2nc(-c3ccc(C)o3)cc(NCC3CCN(Cc4ccc(C(=O)NO)cc4)CC3)c2cc1OC
E3 Binder	CHEMBL4869419	ChEMBL	7.18	—	—	COc1cc2nc(-c3ccc(C)o3)cc(NCC3CCN(Cc4ccc(C(=O)NO)s4)CC3)c2cc1OC
E3 Binder	CHEMBL4854659	ChEMBL	6.33	—	—	COc1cc2nc(-c3ccc(C)o3)cc(NCC3CCN(c4ccc(C(=O)NO)cn4)CC3)c2cc1OC
E3 Binder	CHEMBL4856110	ChEMBL	6.28	—	—	COc1cc2nc(-c3ccc(C)o3)cc(NCC3CCN(c4ncc(C(=O)NO)cn4)CC3)c2cc1OC
E3 Binder	CHEMBL4863394	ChEMBL	7.66	—	—	COc1cc2nc(-c3ccc(C)o3)cc(NCc3ccc(C(=O)NO)cc3)c2cc1OC
E3 Binder	CHEMBL4855823	ChEMBL	6.69	—	—	COc1cc2nc(-c3ccc(C)o3)cc(NCc3ccc(C(=O)NO)cn3)c2cc1OC
E3 Binder	CHEMBL4854765	ChEMBL	6.3	—	—	COc1cc2nc(-c3ccc(C)o3)nc(NCC3CCN(c4ncc(C(=O)NO)cn4)CC3)c2cc1OC
E3 Binder	CHEMBL4847870	ChEMBL	6.64	—	—	COc1cc2nc(-c3ccccc3)cc(NCC3CCN(c4ncc(C(=O)NO)cn4)CC3)c2cc1OC
E3 Binder	CHEMBL4848955	ChEMBL	6.6	—	—	COc1cc2nc(C)cc(NCC3CCN(c4ncc(C(=O)NO)cn4)CC3)c2cc1OC
E3 Binder	CHEMBL4845706	ChEMBL	6.96	—	—	COc1cc2nc(C3CCCCC3)cc(NCC3CCN(c4ncc(C(=O)NO)cn4)CC3)c2cc1OC
E3 Binder	CHEMBL4858828	ChEMBL	6.63	—	—	COc1cc2nc(N3CCCCC3)cc(NCC3CCN(c4ncc(C(=O)NO)cn4)CC3)c2cc1OC
E3 Binder	CHEMBL4572459	ChEMBL	7.45	—	—	COc1cc2nc(N3CCN(C(=O)CCCCCCC(=O)NO)CC3)nc(NC3CCN(Cc4ccccc4)CC3)c2cc1OC
E3 Binder	CHEMBL5171820	ChEMBL	7.62	—	—	COc1cc2nc(N3CCN(CCCCCC(=O)NO)CC3)nc(NC3CCN(C(C)C)CC3)c2cc1OC
E3 Binder	CHEMBL5191361	ChEMBL	7.89	—	—	COc1cc2nc(N3CCN(CCCCCC(=O)NO)CC3)nc(NC3CCN(Cc4ccccc4)CC3)c2cc1OC
E3 Binder	CHEMBL5206158	ChEMBL	7.3	—	—	COc1cc2nc(N3CCN(Cc4ccc(/C=C/C(=O)NO)cc4)CC3)nc(NC3CCN(Cc4ccccc4)CC3)c2cc1OC
E3 Binder	CHEMBL5171881	ChEMBL	6.88	—	—	COc1cc2nc(NCCCCCC(=O)NO)nc(NC3CCN(C(C)C)CC3)c2cc1OC
E3 Binder	CHEMBL5182385	ChEMBL	7.29	—	—	COc1cc2nc(NCCCCCC(=O)NO)nc(NC3CCN(C)CC3)c2cc1OC
E3 Binder	CHEMBL5201140	ChEMBL	7.77	—	—	COc1cc2nc(NCCCCCC(=O)NO)nc(NC3CCN(Cc4ccccc4)CC3)c2cc1OC
E3 Binder	CHEMBL5204152	ChEMBL	7.92	—	—	COc1cc2nc(NCCCCCCC(=O)NO)nc(NC3CCN(C(C)C)CC3)c2cc1OC
E3 Binder	CHEMBL5187697	ChEMBL	7.8	—	—	COc1cc2nc(NCCCCCCC(=O)NO)nc(NC3CCN(C)CC3)c2cc1OC
E3 Binder	CHEMBL4551593	ChEMBL	8.1	—	—	COc1cc2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc(NC3CCN(Cc4ccc(F)cc4)CC3)c2cc1OC
E3 Binder	CHEMBL4461884	ChEMBL	8.04	—	—	COc1cc2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc(NC3CCN(Cc4ccccc4Cl)CC3)c2cc1OC
E3 Binder	CHEMBL4753795	ChEMBL	6.8	—	—	COc1cc2nc3ccccc3c(Nc3ccc(C(=O)NO)cc3)c2c(OC)c1OC
E3 Binder	CHEMBL71191	ChEMBL	6.41	—	—	COc1cc2ncc(-c3ccccc3)nc2cc1OC
E3 Binder	CHEMBL5283086	ChEMBL	6.43	—	—	COc1cc2ncn(Cc3ccc(C(=O)NO)cc3)c(=O)c2cc1OC
E3 Binder	CHEMBL596957	ChEMBL	7.95	—	—	COc1cc2ncnc(NCc3ccc(Cl)c(F)c3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL596964	ChEMBL	8.25	—	—	COc1cc2ncnc(NCc3ccc(F)cc3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL596761	ChEMBL	8.38	—	—	COc1cc2ncnc(NCc3ccccc3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL598407	ChEMBL	6.73	—	—	COc1cc2ncnc(N[C@@H](C)c3ccc(Cl)cc3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL598406	ChEMBL	6.78	—	—	COc1cc2ncnc(N[C@@H](C)c3ccc(F)cc3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL599218	ChEMBL	7.59	—	—	COc1cc2ncnc(N[C@@H](C)c3ccccc3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL2309507	ChEMBL	7.0	—	—	COc1cc2ncnc(N[C@H](C)c3ccc(Cl)cc3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL2309506	ChEMBL	7.0	—	—	COc1cc2ncnc(N[C@H](C)c3ccc(F)cc3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL605976	ChEMBL	7.01	—	—	COc1cc2ncnc(N[C@H](C)c3ccccc3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL3633770	ChEMBL	6.46	—	—	COc1cc2ncnc(Nc3cc(Cl)ccc3Cl)c2cc1OCCC(=O)NO
E3 Binder	CHEMBL3633771	ChEMBL	7.24	—	—	COc1cc2ncnc(Nc3cc(Cl)ccc3Cl)c2cc1OCCCC(=O)NO
E3 Binder	CHEMBL3633772	ChEMBL	7.68	—	—	COc1cc2ncnc(Nc3cc(Cl)ccc3Cl)c2cc1OCCCCC(=O)NO
E3 Binder	CHEMBL3633773	ChEMBL	8.08	—	—	COc1cc2ncnc(Nc3cc(Cl)ccc3Cl)c2cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL3759232	ChEMBL	6.26	—	—	COc1cc2ncnc(Nc3ccc(Br)cc3)c2cc1OCCCC(=O)NO
E3 Binder	CHEMBL3758940	ChEMBL	7.17	—	—	COc1cc2ncnc(Nc3ccc(Br)cc3)c2cc1OCCCCC(=O)NO
E3 Binder	CHEMBL3758697	ChEMBL	8.66	—	—	COc1cc2ncnc(Nc3ccc(Br)cc3)c2cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL3759186	ChEMBL	8.66	—	—	COc1cc2ncnc(Nc3ccc(Br)cc3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL3758229	ChEMBL	6.16	—	—	COc1cc2ncnc(Nc3ccc(Cl)cc3)c2cc1OCCCC(=O)NO
E3 Binder	CHEMBL3758489	ChEMBL	6.88	—	—	COc1cc2ncnc(Nc3ccc(Cl)cc3)c2cc1OCCCCC(=O)NO
E3 Binder	CHEMBL3759261	ChEMBL	7.96	—	—	COc1cc2ncnc(Nc3ccc(Cl)cc3)c2cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL3758839	ChEMBL	8.49	—	—	COc1cc2ncnc(Nc3ccc(Cl)cc3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL3633766	ChEMBL	6.67	—	—	COc1cc2ncnc(Nc3ccc(Cl)cc3Cl)c2cc1OCCC(=O)NO
E3 Binder	CHEMBL3633767	ChEMBL	7.07	—	—	COc1cc2ncnc(Nc3ccc(Cl)cc3Cl)c2cc1OCCCC(=O)NO
E3 Binder	CHEMBL3633768	ChEMBL	7.85	—	—	COc1cc2ncnc(Nc3ccc(Cl)cc3Cl)c2cc1OCCCCC(=O)NO
E3 Binder	CHEMBL3633769	ChEMBL	8.55	—	—	COc1cc2ncnc(Nc3ccc(Cl)cc3Cl)c2cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL5220848	ChEMBL	8.55	—	—	COc1cc2ncnc(Nc3ccc(Cl)cc3Cl)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL3899973	ChEMBL	7.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1-c1ccc(C#CCCCC(=O)NO)o1
E3 Binder	CHEMBL3915573	ChEMBL	6.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1C#CCCC(=O)NO
E3 Binder	CHEMBL3923619	ChEMBL	6.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1C#CCCCC(=O)NO
E3 Binder	CHEMBL3946860	ChEMBL	7.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1CCCCC(=O)NO
E3 Binder	CHEMBL3890344	ChEMBL	6.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)CCCC(=O)NO
E3 Binder	CHEMBL597773	ChEMBL	7.82	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)CCCCCCC(=O)NO
E3 Binder	CHEMBL596736	ChEMBL	7.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCC(=O)NO
E3 Binder	CHEMBL598163	ChEMBL	7.51	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL598377	ChEMBL	8.19	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL3913614	ChEMBL	7.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCOc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3982861	ChEMBL	7.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCOc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3947615	ChEMBL	6.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCN(CCO)CCCC(=O)NO
E3 Binder	CHEMBL3952020	ChEMBL	7.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCNCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3943805	ChEMBL	7.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL3951191	ChEMBL	7.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3916142	ChEMBL	6.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOc1ccc(CC(=O)NO)cc1
E3 Binder	CHEMBL3966861	ChEMBL	6.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1Oc1ccc(C#CCCC(=O)NO)cc1
E3 Binder	CHEMBL3974474	ChEMBL	6.0	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1Oc1ccc(C#CCCCC(=O)NO)cc1
E3 Binder	CHEMBL596755	ChEMBL	6.92	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1S(=O)(=O)CCCCCCC(=O)NO
E3 Binder	CHEMBL596754	ChEMBL	7.4	—	—	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1SCCCCCCC(=O)NO
E3 Binder	CHEMBL3759041	ChEMBL	6.86	—	—	COc1cc2ncnc(Nc3ccc(F)cc3)c2cc1OCCCCC(=O)NO
E3 Binder	CHEMBL3759565	ChEMBL	7.54	—	—	COc1cc2ncnc(Nc3ccc(F)cc3)c2cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL3758380	ChEMBL	8.07	—	—	COc1cc2ncnc(Nc3ccc(F)cc3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL598799	ChEMBL	7.24	—	—	COc1cc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL5204164	ChEMBL	6.25	—	—	COc1cc2ncnc(Nc3cccc(/C=C/C(=O)NO)c3)c2cc1OCCCN1CCOCC1
E3 Binder	CHEMBL3633762	ChEMBL	6.28	—	—	COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1OCCC(=O)NO
E3 Binder	CHEMBL3633763	ChEMBL	7.01	—	—	COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1OCCCC(=O)NO
E3 Binder	CHEMBL3633764	ChEMBL	7.82	—	—	COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1OCCCCC(=O)NO
E3 Binder	CHEMBL3633765	ChEMBL	8.35	—	—	COc1cc2ncnc(Nc3cccc(Br)c3)c2cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL3633758	ChEMBL	6.19	—	—	COc1cc2ncnc(Nc3cccc(Cl)c3)c2cc1OCCC(=O)NO
E3 Binder	CHEMBL3633759	ChEMBL	6.92	—	—	COc1cc2ncnc(Nc3cccc(Cl)c3)c2cc1OCCCC(=O)NO
E3 Binder	CHEMBL3633760	ChEMBL	7.77	—	—	COc1cc2ncnc(Nc3cccc(Cl)c3)c2cc1OCCCCC(=O)NO
E3 Binder	CHEMBL3633761	ChEMBL	8.27	—	—	COc1cc2ncnc(Nc3cccc(Cl)c3)c2cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL3759327	ChEMBL	6.08	—	—	COc1cc2ncnc(Nc3ccccc3Br)c2cc1OCCCC(=O)NO
E3 Binder	CHEMBL3759868	ChEMBL	7.13	—	—	COc1cc2ncnc(Nc3ccccc3Br)c2cc1OCCCCC(=O)NO
E3 Binder	CHEMBL3758725	ChEMBL	7.51	—	—	COc1cc2ncnc(Nc3ccccc3Br)c2cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL3759591	ChEMBL	8.06	—	—	COc1cc2ncnc(Nc3ccccc3Br)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL3759853	ChEMBL	6.89	—	—	COc1cc2ncnc(Nc3ccccc3Cl)c2cc1OCCCCC(=O)NO
E3 Binder	CHEMBL3759149	ChEMBL	7.54	—	—	COc1cc2ncnc(Nc3ccccc3Cl)c2cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL3759279	ChEMBL	7.75	—	—	COc1cc2ncnc(Nc3ccccc3Cl)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL3760069	ChEMBL	6.17	—	—	COc1cc2ncnc(Nc3ccccc3F)c2cc1OCCCC(=O)NO
E3 Binder	CHEMBL3758922	ChEMBL	6.26	—	—	COc1cc2ncnc(Nc3ccccc3F)c2cc1OCCCCC(=O)NO
E3 Binder	CHEMBL3759111	ChEMBL	6.84	—	—	COc1cc2ncnc(Nc3ccccc3F)c2cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL3759313	ChEMBL	7.5	—	—	COc1cc2ncnc(Nc3ccccc3F)c2cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL3906273	ChEMBL	7.0	—	—	COc1ccc(-c2c(C(=O)NCCC(=O)NO)noc2-c2cc(Cl)c(O)cc2O)cc1
E3 Binder	CHEMBL3670668	ChEMBL	9.36	—	—	COc1ccc(-c2cc(-c3ccccc3)[nH]c2C(=O)NCc2ccc(C(=O)NCCS)cc2)cc1
E3 Binder	CHEMBL3670666	ChEMBL	7.37	—	—	COc1ccc(-c2cc(-c3ccccc3)[nH]c2C(=O)NCc2ccc(C(=O)Nc3ccccc3N)cc2)cc1
E3 Binder	CHEMBL3670667	ChEMBL	8.18	—	—	COc1ccc(-c2cc(-c3ccccc3)[nH]c2C(=O)NCc2ccc(C(=O)Nc3ccccc3S)cc2)cc1
E3 Binder	CHEMBL3670669	ChEMBL	9.15	—	—	COc1ccc(-c2cc(-c3ccccc3)[nH]c2C(=O)NCc2ccc(C(=O)Nc3ccccn3)cc2)cc1
E3 Binder	CHEMBL3670664	ChEMBL	8.17	—	—	COc1ccc(-c2cc(-c3ccccc3)[nH]c2C(=O)Nc2cccc(CC(=O)NO)c2)cc1
E3 Binder	CHEMBL4087897	ChEMBL	8.7	—	—	COc1ccc(-c2cc(-c3ccoc3)c(C(=O)NCc3ccc(C(=O)NO)cc3)[nH]2)cc1
E3 Binder	CHEMBL5075694	ChEMBL	6.96	—	—	COc1ccc(-c2cc(/C=C/c3ccc(C(=O)NO)cc3)ccn2)cc1
E3 Binder	CHEMBL90568	ChEMBL	6.28	—	—	COc1ccc(-c2cc(=O)c3c(O)cc(O)cc3o2)cc1O
E3 Binder	CHEMBL3760046	ChEMBL	6.82	—	—	COc1ccc(-c2cc(C(=O)NCCCCCCS)[nH]n2)cc1
E3 Binder	CHEMBL3760115	ChEMBL	7.25	—	—	COc1ccc(-c2cc(C(=O)NCCCCCCS)[nH]n2)cc1OC
E3 Binder	CHEMBL4462577	ChEMBL	7.77	—	—	COc1ccc(-c2cc(OCCN(C)c3ncc(C(=O)NO)cn3)c3ncnc(C)c3c2)cn1
E3 Binder	CHEMBL561209	ChEMBL	7.43	—	—	COc1ccc(-c2ccc(/C=C/C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4217830	ChEMBL	7.39	—	—	COc1ccc(-c2ccc3c(NC(=O)c4ccc(C(=O)NO)cc4)n[nH]c3c2)cc1
E3 Binder	CHEMBL4211463	ChEMBL	7.48	—	—	COc1ccc(-c2ccc3c(NC(=O)c4ccc(C(=O)NO)cc4)n[nH]c3c2)cc1OC
E3 Binder	CHEMBL4636226	ChEMBL	7.31	—	—	COc1ccc(-c2ccc3nc(/C=C/C(=O)NO)ccc3c2)cc1
E3 Binder	CHEMBL4849225	ChEMBL	6.3	—	—	COc1ccc(-c2ccccc2)c2c1CCN(Cc1ccc(C(=O)NO)cc1)CC2
E3 Binder	CHEMBL476902	ChEMBL	8.68	—	—	COc1ccc(-c2cn(CCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL4450360	ChEMBL	8.62	—	—	COc1ccc(-c2cnc(-c3nc(C(=O)N[C@@H](C)c4ccc(C(=O)NO)cc4)c(C4CC4)s3)s2)cc1
E3 Binder	CHEMBL123626	ChEMBL	8.68	—	—	COc1ccc(-c2cnc(CCCCCCC(=O)NO)o2)cc1
E3 Binder	CHEMBL242341	ChEMBL	6.54	—	—	COc1ccc(-c2coc3cc(O)ccc3c2=O)cc1
E3 Binder	CHEMBL124282	ChEMBL	8.6	—	—	COc1ccc(-c2csc(CCCCCCC(=O)NO)n2)cc1
E3 Binder	CHEMBL127953	ChEMBL	7.52	—	—	COc1ccc(-c2csc(NC(=O)CCCCCCC(=O)c3ncco3)n2)cc1
E3 Binder	CHEMBL514478	ChEMBL	6.7	—	—	COc1ccc(-c2csc(NC(=O)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc3ccccc3)n2)cc1
E3 Binder	CHEMBL4533956	ChEMBL	7.04	—	—	COc1ccc(-c2nc(C(=O)N(CCN(C)C)Cc3ccc(C(=O)NO)cc3)cc3c2[nH]c2ccccc23)cc1
E3 Binder	CHEMBL3745788	ChEMBL	7.21	—	—	COc1ccc(-c2nc(C(=O)NCCCC(=O)NO)cc3c2[nH]c2ccccc23)cc1
E3 Binder	CHEMBL3745844	ChEMBL	6.09	—	—	COc1ccc(-c2nc(C(=O)NCCCCC(=O)NO)cc3c2[nH]c2ccccc23)cc1
E3 Binder	CHEMBL3769415	ChEMBL	6.71	—	—	COc1ccc(-c2nc(C(=O)NO)co2)cc1
E3 Binder	CHEMBL4865197	ChEMBL	6.79	—	—	COc1ccc(-c2nc(CNc3ccc(C(=O)NO)cc3)n(-c3ccccc3)n2)cc1
E3 Binder	CHEMBL3828518	ChEMBL	8.47	—	—	COc1ccc(-c2nc(N3CCOCC3)c3nc(CN(C)c4ncc(C(=O)NO)cn4)n(C)c3n2)cc1
E3 Binder	CHEMBL3827281	ChEMBL	8.21	—	—	COc1ccc(-c2nc(N3CCOCC3)c3nc(CN(C)c4ncc(C(=O)NO)cn4)n(C)c3n2)cn1
E3 Binder	CHEMBL5278968	ChEMBL	7.57	—	—	COc1ccc(-c2nc(N3CCOCC3)c3sc(CN(C)c4ccc(C(=O)NO)cc4)cc3n2)cn1
E3 Binder	CHEMBL3622533	ChEMBL	8.17	—	—	COc1ccc(-c2nc(N3CCOCC3)c3sc(CN(C)c4ncc(C(=O)NO)cn4)cc3n2)cn1
E3 Binder	CHEMBL3746015	ChEMBL	6.44	—	—	COc1ccc(-c2nc(NC(=O)NCCC(=O)NO)cc3c2[nH]c2ccccc23)cc1
E3 Binder	CHEMBL3747043	ChEMBL	7.47	—	—	COc1ccc(-c2nc(NC(=O)NCCCC(=O)NO)cc3c2[nH]c2ccccc23)cc1
E3 Binder	CHEMBL3747076	ChEMBL	6.82	—	—	COc1ccc(-c2nc(NC(=O)NCCCC(=O)NO)cc3c4ccccc4n(C)c23)cc1
E3 Binder	CHEMBL3745758	ChEMBL	7.03	—	—	COc1ccc(-c2nc(NC(=O)NCCCCC(=O)NO)cc3c2[nH]c2ccccc23)cc1
E3 Binder	CHEMBL3746446	ChEMBL	6.07	—	—	COc1ccc(-c2nc(NC(=O)NCCCCC(=O)NO)cc3c4ccccc4n(C)c23)cc1
E3 Binder	CHEMBL3745848	ChEMBL	6.09	—	—	COc1ccc(-c2nc(NC(=O)NCCCCCC(=O)NO)cc3c2[nH]c2ccccc23)cc1
E3 Binder	CHEMBL4442355	ChEMBL	7.89	—	—	COc1ccc(-c2nc(NCCCOc3ccc(/C=C/C(=O)NO)cc3OC)cc3c2[nH]c2ccccc23)cc1
E3 Binder	CHEMBL4555936	ChEMBL	7.77	—	—	COc1ccc(-c2nc(NCCOc3ccc(/C=C/C(=O)NO)cc3OC)cc3c2[nH]c2ccccc23)cc1
E3 Binder	CHEMBL523033	ChEMBL	6.32	—	—	COc1ccc(-c2nc([C@H](CCCCNS(N)(=O)=O)NC(=O)OCc3ccccc3)cs2)cc1
E3 Binder	CHEMBL270129	ChEMBL	6.4	—	—	COc1ccc(-c2nc3cc(-c4ccccc4)ccc3o2)cc1NC(=O)NCCCCCC(=O)NO
E3 Binder	CHEMBL409286	ChEMBL	6.89	—	—	COc1ccc(-c2nc3cc(Cl)cc(Cl)c3o2)cc1NC(=O)NCCCCCC(=O)NO
E3 Binder	CHEMBL270519	ChEMBL	6.84	—	—	COc1ccc(-c2nc3cc(Cl)ccc3o2)cc1NC(=O)NCCCCCC(=O)NO
E3 Binder	CHEMBL258606	ChEMBL	7.82	—	—	COc1ccc(-c2nc3cc(F)ccc3o2)cc1NC(=O)NCCCCCC(=O)NO
E3 Binder	CHEMBL428960	ChEMBL	7.75	—	—	COc1ccc(-c2nc3ccc(F)cc3o2)cc1NC(=O)NCCCCCC(=O)NO
E3 Binder	CHEMBL410434	ChEMBL	7.92	—	—	COc1ccc(-c2nc3ccccc3o2)cc1NC(=O)NCCCCCC(=O)NO
E3 Binder	CHEMBL5069541	ChEMBL	6.96	—	—	COc1ccc(-c2ncc(/C=C/C(=O)NO)s2)c(OC)c1OC
E3 Binder	CHEMBL5076163	ChEMBL	6.89	—	—	COc1ccc(-c2ncc(/C=C/C(=O)NO)s2)cc1
E3 Binder	CHEMBL5081121	ChEMBL	6.2	—	—	COc1ccc(-c2ncc(/C=C/C(=O)Nc3ccccc3N)s2)c(OC)c1OC
E3 Binder	CHEMBL5078614	ChEMBL	6.15	—	—	COc1ccc(-c2ncc(/C=C/C(=O)Nc3ccccc3N)s2)cc1
E3 Binder	CHEMBL5077674	ChEMBL	6.28	—	—	COc1ccc(-c2ncc(/C=C/C(=O)Nc3ccccc3N)s2)cc1OC
E3 Binder	CHEMBL5086366	ChEMBL	6.14	—	—	COc1ccc(-c2ncc(C(=O)NCCCC(=O)NO)s2)c(OC)c1
E3 Binder	CHEMBL5083767	ChEMBL	6.21	—	—	COc1ccc(-c2ncc(C(=O)NCCCCC(=O)NO)s2)c(OC)c1
E3 Binder	CHEMBL5085871	ChEMBL	7.12	—	—	COc1ccc(-c2ncc(C(=O)NCCCCCC(=O)NO)s2)c(OC)c1
E3 Binder	CHEMBL5092352	ChEMBL	7.32	—	—	COc1ccc(-c2ncc(C(=O)NCCCCCCC(=O)NO)[nH]2)c(OC)c1
E3 Binder	CHEMBL5093832	ChEMBL	7.51	—	—	COc1ccc(-c2ncc(C(=O)NCCCCCCC(=O)NO)s2)c(OC)c1
E3 Binder	CHEMBL5094432	ChEMBL	6.21	—	—	COc1ccc(-c2ncc(C(=O)NCCCCCCC(=O)NO)s2)cc1
E3 Binder	CHEMBL1099095	ChEMBL	7.2	—	—	COc1ccc(-n2c(-c3cccc(/C=C/C(=O)NO)c3)nc3ccccc32)cc1
E3 Binder	CHEMBL4855642	ChEMBL	6.99	—	—	COc1ccc(-n2nc(-c3ccc(O)cc3)nc2CNc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4856212	ChEMBL	6.9	—	—	COc1ccc(-n2nc(-c3ccccc3)nc2CNc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4530175	ChEMBL	6.33	—	—	COc1ccc(/C=C(\C)C(=O)c2cc(OC)c(OC)c(OC)c2)cc1OCCCC(=O)NO
E3 Binder	CHEMBL4468802	ChEMBL	7.87	—	—	COc1ccc(/C=C(\C)C(=O)c2cc(OC)c(OC)c(OC)c2)cc1OCCCCCCCC(=O)NO
E3 Binder	CHEMBL3260007	ChEMBL	6.14	—	—	COc1ccc(/C=C/C(=O)NO)cc1OCC(=O)Nc1ccc(Br)cc1
E3 Binder	CHEMBL3260008	ChEMBL	6.24	—	—	COc1ccc(/C=C/C(=O)NO)cc1OCC(=O)Nc1ccccc1F
E3 Binder	CHEMBL2046609	ChEMBL	6.35	—	—	COc1ccc(/C=C/C(=O)Nc2ccc(C(=O)N3CCc4nc(C(=O)NO)sc4C3)cc2)cc1
E3 Binder	CHEMBL4568168	ChEMBL	8.34	—	—	COc1ccc(/C=C/C(=O)c2cc(OC)c(OC)c(OC)c2)cc1OCCCCCCC(=O)NO
E3 Binder	CHEMBL595479	ChEMBL	9.02	—	—	COc1ccc(/C=C/C(CO)N2CCN(c3ncc(C(=O)NO)cn3)CC2)cc1
E3 Binder	CHEMBL5271493	ChEMBL	6.59	—	—	COc1ccc(/C=C2\SC(=O)N(CCNC(=O)Nc3c(C)n(C)n(-c4ccccc4)c3=O)C2=O)cc1
E3 Binder	CHEMBL4874942	ChEMBL	6.37	—	—	COc1ccc(/C=C\c2cc(OC)c(OC)c(OC)c2)cc1/C=C/C(=O)Nc1ccccc1N
E3 Binder	CHEMBL4865690	ChEMBL	6.41	—	—	COc1ccc(/C=C\c2cc(OC)c(OC)c(OC)c2)cc1OCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5269123	ChEMBL	7.45	—	—	COc1ccc(/C=N/NC(=O)CCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL4854716	ChEMBL	6.96	—	—	COc1ccc(Br)c2c1CCN(Cc1ccc(C(=O)NO)cc1)CC2
E3 Binder	CHEMBL389368	ChEMBL	6.9	—	—	COc1ccc(C(=O)CS)cc1
E3 Binder	CHEMBL493872	ChEMBL	6.33	—	—	COc1ccc(C(=O)CSC(=S)SCCNC(C)=O)cc1
E3 Binder	CHEMBL493871	ChEMBL	6.89	—	—	COc1ccc(C(=O)CSC(=S)SCCOc2ccccc2)cc1
E3 Binder	CHEMBL242271	ChEMBL	6.3	—	—	COc1ccc(C(=O)CSC(C)=O)cc1
E3 Binder	CHEMBL4549502	ChEMBL	7.6	—	—	COc1ccc(C(=O)N(CCC(=O)NCc2ccccc2)Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL3353057	ChEMBL	7.37	—	—	COc1ccc(C(=O)N2CCn3cc(C(=O)NO)cc3C2)cc1
E3 Binder	CHEMBL3353064	ChEMBL	6.09	—	—	COc1ccc(C(=O)N2CCn3nc(C(=O)NO)cc3C2)cc1
E3 Binder	CHEMBL4789607	ChEMBL	6.15	—	—	COc1ccc(C(=O)NO)cc1C(=O)Nc1ccc2c(c1)cc(C)c(=O)n2C
E3 Binder	CHEMBL3800394	ChEMBL	6.41	GQN	—	COc1ccc(C(=O)NO)cc1NC(=O)c1ccc(-c2ccccc2)cc1
E3 Binder	CHEMBL3798503	ChEMBL	6.05	—	—	COc1ccc(C(=O)NO)cc1NC(=O)c1ccc(Cl)cc1
E3 Binder	CHEMBL3233705	ChEMBL	8.32	—	—	COc1ccc(C(=O)N[C@H](COc2ccc(/C=C/C(=O)NO)cc2)Cc2c[nH]c3ccccc23)cc1
E3 Binder	CHEMBL4070891	ChEMBL	7.06	—	—	COc1ccc(C(=O)N[C@H](COc2ccc(/C=C/C(=O)NO)cc2OC)Cc2c[nH]c3ccccc23)cc1
E3 Binder	CHEMBL3354913	ChEMBL	7.03	—	—	COc1ccc(C(=O)N[C@H](COc2cccc(/C=C/C(=O)NO)c2)Cc2c[nH]c3ccccc23)cc1
E3 Binder	CHEMBL235210	ChEMBL	6.82	—	—	COc1ccc(C(=O)Nc2cc(-c3cccs3)ccc2N)cc1
E3 Binder	CHEMBL3797455	ChEMBL	6.89	—	—	COc1ccc(C(=O)Nc2cc(C(=O)NO)ccc2Cl)cc1
E3 Binder	CHEMBL3799297	ChEMBL	6.4	—	—	COc1ccc(C(=O)Nc2cc(C(=O)NO)ccc2OC)cc1
E3 Binder	CHEMBL4854066	ChEMBL	6.6	—	—	COc1ccc(C(=O)c2cc(OC)c(OC)c(OC)c2)cc1OCC(=O)NO
E3 Binder	CHEMBL4210107	ChEMBL	6.97	—	—	COc1ccc(C(=O)c2ccc3c(ccn3Cc3ccc(/C=C/C(=O)NO)cc3)c2)cc1
E3 Binder	CHEMBL4218266	ChEMBL	8.41	—	—	COc1ccc(C(=O)c2ccc3c(ccn3Cc3ccc(C(=O)NO)cc3)c2)cc1
E3 Binder	CHEMBL4206021	ChEMBL	7.81	—	—	COc1ccc(C(=O)c2ccc3c(ccn3Cc3ccc(C(=O)NO)cc3)c2)cc1OC
E3 Binder	CHEMBL4214502	ChEMBL	6.07	—	—	COc1ccc(C(=O)c2ccc3c(ccn3S(=O)(=O)c3ccc(/C=C/C(=O)NO)cc3)c2)cc1
E3 Binder	CHEMBL4213856	ChEMBL	6.12	—	—	COc1ccc(C(=O)c2ccc3c(ccn3S(=O)(=O)c3cccc(/C=C/C(=O)NO)c3)c2)cc1
E3 Binder	CHEMBL4066975	ChEMBL	6.96	—	—	COc1ccc(C(=O)c2cn(Cc3ccc(C(=O)NO)cc3)c3cc(OC)ccc23)cc1
E3 Binder	CHEMBL2047681	ChEMBL	6.5	—	—	COc1ccc(C/C(=N\N)C(=O)NCCS)cc1Br
E3 Binder	CHEMBL2047691	ChEMBL	6.62	—	—	COc1ccc(C/C(=N\O)C(=O)NCCS)cc1I
E3 Binder	CHEMBL4589593	ChEMBL	7.52	—	—	COc1ccc(C/C(=N\O)C(=O)NCCSSCCNC(=O)/C(Cc2ccc(OC)c(O)c2)=N/O)cc1O
E3 Binder	CHEMBL4545761	ChEMBL	6.92	—	—	COc1ccc(C/C(=N\O)C(=O)NCCSSCCNC(=O)/C(Cc2ccc(OC)cc2)=N/O)cc1
E3 Binder	CHEMBL3656007	ChEMBL	8.1	—	—	COc1ccc(C2(Nc3ncc(C(=O)NO)cn3)CC2)cc1OC
E3 Binder	CHEMBL3656021	ChEMBL	8.4	—	—	COc1ccc(C2(Nc3ncc(C(=O)NO)cn3)CCCC2)cc1
E3 Binder	CHEMBL3655991	ChEMBL	7.7	—	—	COc1ccc(C2(Nc3ncc(C(=O)NO)cn3)CCCCC2)cc1
E3 Binder	CHEMBL4871812	ChEMBL	7.66	—	—	COc1ccc(C2CC2)c2c1CCN(Cc1ccc(C(=O)NO)cc1)CC2
E3 Binder	CHEMBL2046456	ChEMBL	6.6	—	—	COc1ccc(CC(=O)C(=O)NCCS)cc1Br
E3 Binder	CHEMBL4434656	ChEMBL	8.3	—	—	COc1ccc(CC(=O)N[C@@H](Cc2cscn2)C(=O)Nc2ccc(C(=O)NO)cc2)cc1OC
E3 Binder	CHEMBL4863335	ChEMBL	7.14	—	—	COc1ccc(CC2(c3ccccc3)NC(=O)N(Cc3ccc(C(=O)NO)cc3)C2=O)cc1
E3 Binder	CHEMBL3427665	ChEMBL	6.85	—	—	COc1ccc(CCCn2cccc(/C=C/C(=O)NO)c2=O)cc1
E3 Binder	CHEMBL4547600	ChEMBL	7.29	—	—	COc1ccc(CCc2nc(CCC(=O)NO)cs2)cc1
E3 Binder	CHEMBL4449062	ChEMBL	7.21	—	—	COc1ccc(CCc2nc(CCC(=O)NO)cs2)cc1OC
E3 Binder	CHEMBL4437282	ChEMBL	7.7	—	—	COc1ccc(CCn2c(=O)c3ccccc3n(Cc3ccc(C(=O)NO)cc3)c2=O)cc1
E3 Binder	CHEMBL4862983	ChEMBL	6.99	—	—	COc1ccc(CN2C(=O)N(Cc3ccc(C(=O)NO)cc3)C(=O)C2Cc2ccccc2)cc1
E3 Binder	CHEMBL4872084	ChEMBL	7.55	—	—	COc1ccc(CN2CC(=O)N(Cc3ccc(C(=O)NO)cc3)C2=O)cc1
E3 Binder	CHEMBL4554522	ChEMBL	8.59	—	—	COc1ccc(CN2CCC(Nc3nc(Nc4ccc(NC(=O)CCCCCCC(=O)NO)cc4)nc4cc(OC)c(OC)cc34)CC2)cc1
E3 Binder	CHEMBL211802	ChEMBL	6.3	—	—	COc1ccc(CN2CCC=C(CCC(=O)NO)C2=O)c(OC)c1
E3 Binder	CHEMBL250476	ChEMBL	6.36	—	—	COc1ccc(CN2CCC=C(CCC(=O)NO)C2=O)cc1
E3 Binder	CHEMBL2018445	ChEMBL	8.52	—	—	COc1ccc(CN2CCc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)C2)cc1
E3 Binder	CHEMBL1270034	ChEMBL	7.02	—	—	COc1ccc(CN2C[C@@H]3CN(c4ncc(C(=O)NO)cn4)C[C@@H]3C2)cc1
E3 Binder	CHEMBL5202479	ChEMBL	6.17	—	—	COc1ccc(CNC(=O)c2cc(C(=O)Nc3ccccc3N)ccc2N2CCOCC2)cc1O
E3 Binder	CHEMBL5191492	ChEMBL	6.86	—	—	COc1ccc(CNC(=O)c2cc(F)ccc2N2CCOCC2)cc1/C=C/C(=O)NO
E3 Binder	CHEMBL497123	ChEMBL	6.62	—	—	COc1ccc(CNC(=O)c2ccc(C(=O)C(F)(F)F)s2)cc1
E3 Binder	CHEMBL384961	ChEMBL	7.89	—	—	COc1ccc(CNCCn2ccc(-c3ccc(C(=O)NO)s3)n2)cc1
E3 Binder	CHEMBL217604	ChEMBL	6.97	—	—	COc1ccc(CNCCn2ccc(-c3ccc(C(=O)NO)s3)n2)cc1OC
E3 Binder	CHEMBL1801244	ChEMBL	7.7	—	—	COc1ccc(CN[C@H]2[C@@H]3CN(c4ncc(C(=O)NO)cn4)C[C@@H]32)cc1
E3 Binder	CHEMBL251011	ChEMBL	7.7	—	—	COc1ccc(COC(CCCCCC(=O)NO)C(=O)Nc2ccccc2)cc1
E3 Binder	CHEMBL496512	ChEMBL	6.39	—	—	COc1ccc(COCc2ccc(C(=O)C(F)(F)F)s2)cc1
E3 Binder	CHEMBL5274050	ChEMBL	6.9	—	—	COc1ccc(COc2cccc3ccc(C(=O)NCCCCCC(=O)NO)nc23)cc1
E3 Binder	CHEMBL5267546	ChEMBL	7.39	—	—	COc1ccc(COc2cccc3ccc(C(=O)NCc4ccc(C(=O)NO)cc4)nc23)cc1
E3 Binder	CHEMBL4068870	ChEMBL	7.92	—	—	COc1ccc(Cl)cc1C(=O)NCCc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4089964	ChEMBL	7.38	—	—	COc1ccc(Cl)cc1C(=O)NCCc1ccc(CCC(=O)NO)cc1
E3 Binder	CHEMBL4087230	ChEMBL	7.4	—	—	COc1ccc(Cl)cc1C(=O)NCCc1cccc(/C=C/C(=O)NO)c1
E3 Binder	CHEMBL3656008	ChEMBL	8.4	—	—	COc1ccc(Cl)cc1C1(Nc2ncc(C(=O)NO)cn2)CC1
E3 Binder	CHEMBL521355	ChEMBL	6.76	—	—	COc1ccc(Cl)cc1N1CCN(C(=O)c2ccc(C(=O)C(F)(F)F)s2)CC1
E3 Binder	CHEMBL3601775	ChEMBL	7.0	—	—	COc1ccc(Cn2ccc3ccc(NC(=O)CCCCCCC(=O)NO)cc3c2=O)c(OC)c1
E3 Binder	CHEMBL3427644	ChEMBL	6.42	—	—	COc1ccc(Cn2cccc(/C=C/C(=O)NO)c2=O)cc1
E3 Binder	CHEMBL4212669	ChEMBL	7.19	—	—	COc1ccc(F)cc1-c1ccc2c(NC(=O)c3ccc(C(=O)NO)cc3)n[nH]c2c1
E3 Binder	CHEMBL5081983	ChEMBL	7.03	—	—	COc1ccc(F)cc1-c1cncc(/C=C/c2ccc(C(=O)NO)cc2)c1
E3 Binder	CHEMBL5183440	ChEMBL	6.0	—	—	COc1ccc(N(C)c2cc(C#N)nc3ccccc23)cc1/C=C/C(=O)NO
E3 Binder	CHEMBL3774414	ChEMBL	7.77	—	—	COc1ccc(N(C)c2nc(C)nc3ccccc23)cc1OCCCC(=O)NO
E3 Binder	CHEMBL3775654	ChEMBL	6.96	—	—	COc1ccc(N(C)c2nc(C)nc3ccccc23)cc1OCCCCC(=O)NO
E3 Binder	CHEMBL3774890	ChEMBL	7.64	—	—	COc1ccc(N(C)c2nc(C)nc3ccccc23)cc1OCCCCCC(=O)NO
E3 Binder	CHEMBL3675763	ChEMBL	7.89	—	—	COc1ccc(N(CCCCCCC(=O)NO)c2ccccn2)nc1
E3 Binder	CHEMBL3693703	ChEMBL	6.7	—	—	COc1ccc(N(c2ccc(OC)cc2)c2ccc(C(=O)NCCCCCCC(=O)NO)cc2)cc1
E3 Binder	CHEMBL1958431	ChEMBL	6.97	—	—	COc1ccc(N2CCN(S(=O)(=O)c3cccc(/C=C/C(=O)NO)c3)CC2)cc1
E3 Binder	CHEMBL3640694	ChEMBL	8.4	—	—	COc1ccc(N2CCN(c3ncc(C(=O)NCCCCCCC(=O)NO)cn3)CC2)cc1
E3 Binder	CHEMBL4535357	ChEMBL	7.05	—	—	COc1ccc(NC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)c2ccc(/C=C/C(=O)NO)cc2)cc1
E3 Binder	CHEMBL1091487	ChEMBL	7.5	—	—	COc1ccc(NC(=O)CCCCC(=O)NO)cc1
E3 Binder	CHEMBL349015	ChEMBL	6.55	—	—	COc1ccc(NC(=O)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3260006	ChEMBL	6.03	—	—	COc1ccc(NC(=O)COc2cc(/C=C/C(=O)NO)ccc2OC)cc1
E3 Binder	CHEMBL3916257	ChEMBL	8.82	—	—	COc1ccc(NC(=O)N2CCC(Nc3ncc(C(=O)NO)cn3)(c3ccccc3)CC2)cc1
E3 Binder	CHEMBL3909006	ChEMBL	8.08	—	—	COc1ccc(NC(=O)NCc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4535463	ChEMBL	6.92	—	—	COc1ccc(NC(=O)NOCc2ccc(/C=C/C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4227702	ChEMBL	7.45	—	—	COc1ccc(NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)/C=C/c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL1808378	ChEMBL	6.05	—	—	COc1ccc(NC(=O)[C@H](Cc2ccc(OCC(=O)NO)cc2)NC(=O)CCc2ccccc2)cc1
E3 Binder	CHEMBL1808272	ChEMBL	6.45	—	—	COc1ccc(NC(=O)[C@H](Cc2ccc(OCC(=O)NO)cc2)NC(=O)c2ccccc2)cc1
E3 Binder	CHEMBL1958439	ChEMBL	7.89	—	—	COc1ccc(NS(=O)(=O)c2cccc(/C=C/C(=O)NO)c2)cc1
E3 Binder	CHEMBL272847	ChEMBL	7.64	—	—	COc1ccc(NS(=O)(=O)c2cccc(/C=C/C(=O)NO)c2)cc1OC
E3 Binder	CHEMBL4237803	ChEMBL	7.64	—	—	COc1ccc(Nc2c(NCCCCCC(=O)NO)c(=O)c2=O)cc1
E3 Binder	CHEMBL4070705	ChEMBL	6.32	—	—	COc1ccc(Nc2ccn(-c3ccccc3)n2)cc1
E3 Binder	CHEMBL4457617	ChEMBL	8.52	—	—	COc1ccc(Nc2nc(Nc3cnn(CCCCCCC(=O)NO)c3)ncc2Cl)cc1
E3 Binder	CHEMBL3652229	ChEMBL	7.82	—	—	COc1ccc(Nc2ncc(C(=O)NO)cn2)cc1
E3 Binder	CHEMBL4064767	ChEMBL	6.96	—	—	COc1ccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c(C)c1
E3 Binder	CHEMBL4082243	ChEMBL	7.15	—	—	COc1ccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)cc1
E3 Binder	CHEMBL4632668	ChEMBL	7.68	—	—	COc1ccc(Oc2ccc3nc(/C=C/C(=O)NO)ccc3c2)cc1
E3 Binder	CHEMBL1909955	ChEMBL	6.5	—	—	COc1ccc(S(=O)(=O)N2CCC(CCCC(=O)NO)CC2)cc1OC
E3 Binder	CHEMBL399467	ChEMBL	6.8	—	—	COc1ccc(S(=O)(=O)N2CCN(c3ncc(/C=C/C(=O)NO)s3)CC2)cc1OC
E3 Binder	CHEMBL251183	ChEMBL	7.16	—	—	COc1ccc(S(=O)(=O)N2CCN(c3ncc(C(=O)NO)s3)CC2)cc1OC
E3 Binder	CHEMBL4459443	ChEMBL	6.5	—	—	COc1ccc(S(=O)(=O)N2CCc3cccc(NCc4ccc(C(=O)Nc5ccccc5N)cc4)c32)cc1
E3 Binder	CHEMBL82931	ChEMBL	7.13	—	—	COc1ccc(S(=O)(=O)Nc2ccc(/C=C(C)/C=C/C(=O)NO)cc2)cc1
E3 Binder	CHEMBL480931	ChEMBL	7.3	—	—	COc1ccc(S(=O)(=O)Nc2ccc(C(=O)CSC(C)=O)cc2)cc1
E3 Binder	CHEMBL473426	ChEMBL	6.55	—	—	COc1ccc(S(=O)(=O)Nc2ccc(C(=O)CSC(C)=O)cc2)cc1OC
E3 Binder	CHEMBL488168	ChEMBL	7.54	—	—	COc1ccc(S(=O)(=O)Nc2ccc(C(=O)CSC(C)=O)cn2)cc1
E3 Binder	CHEMBL270354	ChEMBL	6.86	—	—	COc1ccc(S(=O)(=O)Nc2cccc(/C=C/C(=O)NO)c2)cc1OC
E3 Binder	CHEMBL5080049	ChEMBL	7.34	—	—	COc1ccc(S(=O)(=O)n2ccc(/C=C/C(=O)NO)c2)cc1NC(=O)c1[nH]c(C)c2c1CCCCC2=O
E3 Binder	CHEMBL2048749	ChEMBL	8.48	—	—	COc1ccc(S(=O)(=O)n2ccc3cc(/C=C/C(=O)NO)ccc32)cc1
E3 Binder	CHEMBL2048750	ChEMBL	8.01	—	—	COc1ccc(S(=O)(=O)n2ccc3cc(/C=C/C(=O)NO)ccc32)cc1OC
E3 Binder	CHEMBL399121	ChEMBL	6.0	6JP	—	COc1ccc([C@@H]2CC(=O)c3c(O)cc(O)cc3O2)cc1O
E3 Binder	CHEMBL4741936	ChEMBL	7.42	—	—	COc1ccc([C@H]2C[C@@H]2NCC2CCN(CCCc3ccc(C(=O)NO)cc3)CC2)cc1
E3 Binder	CHEMBL4745394	ChEMBL	7.55	—	—	COc1ccc([C@H]2C[C@@H]2NCc2cn3c(n2)CN(CCCc2ccc(C(=O)NO)cc2)CC3)cc1
E3 Binder	CHEMBL293812	ChEMBL	8.19	—	—	COc1ccc2[nH]c(C(=O)NCCCCCCC(=O)NO)cc2c1
E3 Binder	CHEMBL396559	ChEMBL	6.55	—	—	COc1ccc2[nH]c(C(=O)c3ccc(/C=C/C(=O)NO)cc3)cc2c1
E3 Binder	CHEMBL140220	ChEMBL	6.11	D3L	—	COc1ccc2[nH]c(C(=O)c3ccccc3)cc2c1
E3 Binder	CHEMBL216641	ChEMBL	7.35	—	—	COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCCC(=O)NO)C(=O)NCCc3c(-c4ccccc4)[nH]c4ccccc34)c2c1
E3 Binder	CHEMBL406927	ChEMBL	6.01	—	—	COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCCC(C)=O)c3nc4ccc(Cl)cc4[nH]3)c2c1
E3 Binder	CHEMBL407959	ChEMBL	6.47	—	—	COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCCC(C)=O)c3ncc(-c4ccccc4)[nH]3)c2c1
E3 Binder	CHEMBL466215	ChEMBL	6.92	—	—	COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCCC(N)=O)c3ncc(-c4ccc5ccccc5c4)[nH]3)c2c1
E3 Binder	CHEMBL494124	ChEMBL	6.23	—	—	COc1ccc2[nH]c(C)c(CC(=O)N[C@@H](CCCCNS(N)(=O)=O)C(=O)Nc3nc(-c4ccccc4)cs3)c2c1
E3 Binder	CHEMBL5087002	ChEMBL	6.45	—	—	COc1ccc2[nH]cc(CCN(CCCCCC(=O)NO)C(=O)/C=C/c3ccc(O)c(OC)c3)c2c1
E3 Binder	CHEMBL5080111	ChEMBL	7.59	—	—	COc1ccc2[nH]cc(CCN(Cc3ccc(/C=C/C(=O)NO)cc3)C(=O)/C=C/c3ccc(O)c(OC)c3)c2c1
E3 Binder	CHEMBL5072502	ChEMBL	7.51	—	—	COc1ccc2[nH]cc(CCN(Cc3ccc(C(=O)NO)cc3)C(=O)/C=C/c3ccc(O)c(OC)c3)c2c1
E3 Binder	CHEMBL5070312	ChEMBL	7.47	—	—	COc1ccc2[nH]cc(CCNC(=O)/C=C/c3ccc(C(=O)NO)cc3)c2c1
E3 Binder	CHEMBL5092694	ChEMBL	7.24	—	—	COc1ccc2[nH]cc(CCNC(=O)CN(CCCCCC(=O)NO)C(=O)/C=C/c3ccc(O)c(OC)c3)c2c1
E3 Binder	CHEMBL5092272	ChEMBL	7.27	—	—	COc1ccc2[nH]cc(CCNC(=O)CN(Cc3ccc(/C=C/C(=O)NO)cc3)C(=O)/C=C/c3ccc(O)c(OC)c3)c2c1
E3 Binder	CHEMBL5090786	ChEMBL	7.72	—	—	COc1ccc2[nH]cc(CCNC(=O)c3ccc(/C=C/C(=O)NO)cc3)c2c1
E3 Binder	CHEMBL141502	ChEMBL	7.85	—	—	COc1ccc2[nH]cc(CCNCc3ccc(/C=C/C(=O)NO)cc3)c2c1
E3 Binder	CHEMBL4207448	ChEMBL	6.54	—	—	COc1ccc2[nH]cc(Cn3cc(COc4ccc(/C=C/C(=O)NO)cc4OC)nn3)c2c1
E3 Binder	CHEMBL4538745	ChEMBL	6.08	—	—	COc1ccc2c(=O)n(-c3ccccc3Cl)c(SCc3ccc(C(=O)Nc4ccccc4N)cc3)nc2c1
E3 Binder	CHEMBL4474354	ChEMBL	6.0	—	—	COc1ccc2c(=O)n(C)c(SCc3ccc(C(=O)Nc4ccccc4N)cc3)nc2c1
E3 Binder	CHEMBL4537684	ChEMBL	7.29	—	—	COc1ccc2c(=O)n(CCc3ccccc3)c(=O)n(Cc3ccc(C(=O)NO)cc3)c2c1
E3 Binder	CHEMBL4070232	ChEMBL	7.15	—	—	COc1ccc2c(C(=O)c3cc(OC)c(OC)c(OC)c3)cn(Cc3ccc(/C=C/C(=O)NO)cc3)c2c1
E3 Binder	CHEMBL4093691	ChEMBL	7.19	—	—	COc1ccc2c(C(=O)c3cc(OC)c(OC)c(OC)c3)cn(Cc3ccc(C(=O)NO)cc3)c2c1
E3 Binder	CHEMBL4081822	ChEMBL	6.56	—	—	COc1ccc2c(C(=O)c3cc(OC)c(OC)c(OC)c3)cn(S(=O)(=O)c3cccc(/C=C/C(=O)NO)c3)c2c1
E3 Binder	CHEMBL4783280	ChEMBL	7.68	—	—	COc1ccc2c(c1)/C(=C1/Nc3ccccc3/C1=N\O)C(=O)N2CCCCCCC(=O)NO
E3 Binder	CHEMBL4791243	ChEMBL	8.3	—	—	COc1ccc2c(c1)/C(=C1/Nc3ccccc3/C1=N\O)C(=O)N2Cc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4751879	ChEMBL	7.6	—	—	COc1ccc2c(c1)/C(=C1/Nc3ccccc3/C1=N\O)C(=O)N2Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5280583	ChEMBL	7.17	—	—	COc1ccc2c(c1)C(C)(C)C(c1cccnc1)N2Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4854123	ChEMBL	8.25	—	—	COc1ccc2c(c1)CCCCN2Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4858918	ChEMBL	7.54	—	—	COc1ccc2c(c1)CCN(Cc1ccc(C(=O)NO)cc1)CC2
E3 Binder	CHEMBL1688190	ChEMBL	6.55	—	—	COc1ccc2c(c1)N(CCCCCC(=O)NO)C(=O)c1ccccc1N2
E3 Binder	CHEMBL1688185	ChEMBL	6.7	—	—	COc1ccc2c(c1)N(CCCCCC(=O)NO)C(=O)c1ccccc1O2
E3 Binder	CHEMBL1688186	ChEMBL	6.82	—	—	COc1ccc2c(c1)N(CCCCCC(=O)NO)C(=O)c1ccccc1S2
E3 Binder	CHEMBL1688183	ChEMBL	7.52	—	—	COc1ccc2c(c1)N(CCCCCC(=O)NO)C(=O)c1ccccc1S2(=O)=O
E3 Binder	CHEMBL4875748	ChEMBL	8.09	—	—	COc1ccc2c(c1)N(Cc1ccc(C(=O)NO)cc1)CCCC2
E3 Binder	CHEMBL4545246	ChEMBL	8.0	—	—	COc1ccc2c(c1)N(Cc1ccc(C(=O)NO)cc1)c1ccccc1S2
E3 Binder	CHEMBL4858210	ChEMBL	7.5	—	—	COc1ccc2c(c1)N(Cc1ccc(C(=O)NO)cc1)c1ccccc1[S+]2[O-]
E3 Binder	CHEMBL3884118	ChEMBL	7.31	—	—	COc1ccc2c(c1)c(CC(=O)NCCCCCC(=O)NO)c(C)n2C(=O)c1ccc(Cl)cc1
E3 Binder	CHEMBL3885367	ChEMBL	7.31	—	—	COc1ccc2c(c1)c(CC(=O)NCCCCCCC(=O)NO)c(C)n2C(=O)c1ccc(Cl)cc1
E3 Binder	CHEMBL3885245	ChEMBL	7.3	—	—	COc1ccc2c(c1)c(CC(=O)NCCCCCCCC(=O)NO)c(C)n2C(=O)c1ccc(Cl)cc1
E3 Binder	CHEMBL3884506	ChEMBL	7.66	—	—	COc1ccc2c(c1)c(CC(=O)O)c(C)n2Cc1ccc(-c2cn(CCCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL5081920	ChEMBL	7.28	—	—	COc1ccc2c(c1)c(CCNC(C)=O)cn2CCCCCC(=O)NO
E3 Binder	CHEMBL5078976	ChEMBL	7.16	—	—	COc1ccc2c(c1)c(CCNC(C)=O)cn2Cc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL5076794	ChEMBL	7.95	—	—	COc1ccc2c(c1)c(CCNC(C)=O)cn2Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL2018299	ChEMBL	8.51	—	—	COc1ccc2c(c1)c1c(n2Cc2ccc(C(=O)NO)cc2)CCN(C)C1
E3 Binder	CHEMBL4101480	ChEMBL	9.8	—	—	COc1ccc2c(c1)c1c(n2Cc2ccc(C(=O)NO)cc2)CN2CC1C(=O)N(C)C2
E3 Binder	CHEMBL4100534	ChEMBL	9.82	—	—	COc1ccc2c(c1)c1c(n2Cc2ccc(C(=O)NO)cc2)CN2CC1C(=O)N(C)C2=O
E3 Binder	CHEMBL4857648	ChEMBL	7.28	—	—	COc1ccc2c(c1)c1c(n2Cc2ccc(C(=O)NO)cn2)CCN(C)C1
E3 Binder	CHEMBL5175796	ChEMBL	8.64	—	—	COc1ccc2c(c1)cc(C(=O)NC1C3CC4CC(C3)CC1C4)n2CCCCCCC(=O)NO
E3 Binder	CHEMBL244040	ChEMBL	6.58	—	—	COc1ccc2c(c1)cc(C(=O)c1ccc(/C=C/C(=O)NO)cc1)n2S(=O)(=O)c1ccccc1
E3 Binder	CHEMBL4159460	ChEMBL	8.23	—	—	COc1ccc2c(ccn2CCOc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c1
E3 Binder	CHEMBL1269925	ChEMBL	7.52	—	—	COc1ccc2c(ccn2N2C[C@H]3CN(c4ncc(C(=O)NO)cn4)C[C@H]3C2)c1
E3 Binder	CHEMBL5195946	ChEMBL	10.0	—	—	COc1ccc2c3c(cccc13)C(=O)N(Cc1ccc(C(=O)NO)cc1)C2=O
E3 Binder	CHEMBL4062190	ChEMBL	9.49	—	—	COc1ccc2c3c(n(Cc4ccc(C(=O)NO)cc4)c2c1)CN1CC3C(=O)N(C)C1=O
E3 Binder	CHEMBL478727	ChEMBL	8.74	—	—	COc1ccc2cc(-c3cn(CCCCCC(=O)NO)nn3)ccc2c1
E3 Binder	CHEMBL477501	ChEMBL	7.82	—	—	COc1ccc2cc(-c3cn(CCCCCCC(=O)NO)nn3)ccc2c1
E3 Binder	CHEMBL590872	ChEMBL	6.65	—	—	COc1ccc2cc(-c3cn(CCCCCCCC(=O)NO)nn3)ccc2c1
E3 Binder	CHEMBL3770029	ChEMBL	6.74	—	—	COc1ccc2cc(-c3nc(C(=O)NO)co3)ccc2c1
E3 Binder	CHEMBL3309288	ChEMBL	7.4	—	—	COc1ccc2cc(C(=O)NCCCCCCC(=O)NO)ccc2n1
E3 Binder	CHEMBL1958430	ChEMBL	7.55	—	—	COc1ccc2nc(/C=C/C(=O)NO)ccc2c1
E3 Binder	CHEMBL128988	ChEMBL	6.23	—	—	COc1ccc2nc(NC(=O)Nc3ccccc3)sc2c1
E3 Binder	CHEMBL4244887	ChEMBL	7.54	—	—	COc1ccc2nc3cc(Cl)ccc3c(Nc3ccc(-c4cn(CCCCCC(=O)NO)nn4)cc3)c2c1
E3 Binder	CHEMBL4750838	ChEMBL	6.47	—	—	COc1ccc2nc3cc(Cl)ccc3c(Nc3ccc(C(=O)NO)cc3)c2n1
E3 Binder	CHEMBL4248226	ChEMBL	7.09	—	—	COc1ccc2nc3cc(Cl)ccc3c(Nc3ccc(CCC(=O)NO)cc3)c2c1
E3 Binder	CHEMBL4244419	ChEMBL	7.88	—	—	COc1ccc2nc3cc(Cl)ccc3c(Nc3cccc(-c4cn(CCCCCC(=O)NO)nn4)c3)c2c1
E3 Binder	CHEMBL410433	ChEMBL	7.92	—	—	COc1ccc2oc(-c3cccc(NC(=O)NCCCCCC(=O)NO)c3)nc2c1
E3 Binder	CHEMBL56344	ChEMBL	7.82	—	—	COc1ccc2oc(C(=O)NCCCCCCC(=O)NO)cc2c1
E3 Binder	CHEMBL4214652	ChEMBL	6.88	—	—	COc1cccc(-c2ccc3c(NC(=O)c4ccc(C(=O)NO)cc4)n[nH]c3c2)c1
E3 Binder	CHEMBL4205573	ChEMBL	7.24	—	—	COc1cccc(-c2ccc3c(NC(=O)c4ccc(C(=O)NO)cc4)n[nH]c3c2)c1F
E3 Binder	CHEMBL518268	ChEMBL	7.86	—	—	COc1cccc(-c2cn(CCCCCC(=O)NO)nn2)c1
E3 Binder	CHEMBL474051	ChEMBL	6.38	—	—	COc1cccc(-c2csc(NC(=O)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc3ccccc3)n2)c1
E3 Binder	CHEMBL4456371	ChEMBL	8.55	—	—	COc1cccc(-c2nc(NCc3ccc(/C=C/C(=O)NO)cc3)cc3c2[nH]c2ccccc23)c1
E3 Binder	CHEMBL4285608	ChEMBL	8.74	—	—	COc1cccc(-c2nc(NCc3ccc(C(=O)NO)cc3)cc3c2[nH]c2ccccc23)c1
E3 Binder	CHEMBL4453484	ChEMBL	8.35	—	—	COc1cccc(-c2nc(NCc3cccc(/C=C/C(=O)NO)c3)cc3c2[nH]c2ccccc23)c1
E3 Binder	CHEMBL5080369	ChEMBL	6.18	—	—	COc1cccc(-c2ncc(/C=C/C(=O)NO)s2)c1
E3 Binder	CHEMBL5079646	ChEMBL	6.24	—	—	COc1cccc(-c2ncc(/C=C/C(=O)Nc3ccccc3N)s2)c1
E3 Binder	CHEMBL5080669	ChEMBL	6.36	—	—	COc1cccc(-c2ncc(C(=O)NCCCCCCC(=O)NO)s2)c1
E3 Binder	CHEMBL5286013	ChEMBL	7.94	—	—	COc1cccc(-c2ncn(Cc3ccc(C(=O)NO)cc3)n2)c1
E3 Binder	CHEMBL4174925	ChEMBL	6.54	—	—	COc1cccc(-n2nc(C(=O)NCC(=O)NO)nc2-c2cc(OC)c(OC)c(OC)c2)c1
E3 Binder	CHEMBL4168150	ChEMBL	6.56	—	—	COc1cccc(-n2nc(C(=O)NCCCCCC(=O)NO)nc2-c2cc(OC)c(OC)c(OC)c2)c1
E3 Binder	CHEMBL5308487	ChEMBL	7.31	—	—	COc1cccc(/C=N/C=N/c2cccc(OC)c2)c1
E3 Binder	CHEMBL3354919	ChEMBL	7.17	—	—	COc1cccc(C(=O)N[C@H](COc2cccc(/C=C/C(=O)NO)c2)Cc2c[nH]c3ccccc23)c1
E3 Binder	CHEMBL244885	ChEMBL	6.48	—	—	COc1cccc(C(=O)c2cc3cc(/C=C/C(=O)NO)ccc3[nH]2)c1
E3 Binder	CHEMBL390910	ChEMBL	6.92	—	—	COc1cccc(C(=O)c2cc3cc(/C=C/C(=O)NO)ccc3n2S(=O)(=O)c2ccccc2)c1
E3 Binder	CHEMBL244887	ChEMBL	6.19	—	—	COc1cccc(C(=O)c2cc3cc(/C=C/C(=O)NO)ccc3o2)c1
E3 Binder	CHEMBL4210907	ChEMBL	7.79	—	—	COc1cccc(C(=O)c2ccc3c(ccn3Cc3ccc(C(=O)NO)cc3)c2)c1
E3 Binder	CHEMBL3655989	ChEMBL	8.4	—	—	COc1cccc(C2(Nc3ncc(C(=O)NO)cn3)CC2)c1
E3 Binder	CHEMBL4463058	ChEMBL	6.72	—	—	COc1cccc(CCCCCCCC(=O)NO)c1
E3 Binder	CHEMBL3427664	ChEMBL	7.52	—	—	COc1cccc(CCCn2cccc(/C=C/C(=O)NO)c2=O)c1
E3 Binder	CHEMBL3427653	ChEMBL	7.16	—	—	COc1cccc(CCn2cccc(/C=C/C(=O)NO)c2=O)c1
E3 Binder	CHEMBL5282117	ChEMBL	7.86	—	—	COc1cccc(CN2C(=O)CN(Cc3ccc(C(=O)NO)cc3)C(=O)[C@H]2Cc2ccccc2)c1
E3 Binder	CHEMBL2018444	ChEMBL	8.53	—	—	COc1cccc(CN2CCc3c(c4ccccc4n3Cc3ccc(C(=O)NO)cc3)C2)c1
E3 Binder	CHEMBL5091030	ChEMBL	7.42	—	—	COc1cccc(Cn2ccc3cnc(Nc4cnn(CCCCCC(=O)NO)c4)nc32)c1
E3 Binder	CHEMBL5077078	ChEMBL	7.54	—	—	COc1cccc(Cn2ccc3cnc(Nc4cnn(CCCCCCC(=O)NO)c4)nc32)c1
E3 Binder	CHEMBL3427643	ChEMBL	6.82	—	—	COc1cccc(Cn2cccc(/C=C/C(=O)NO)c2=O)c1
E3 Binder	CHEMBL487370	ChEMBL	6.77	—	—	COc1cccc(N2CCN(C(=O)c3ccc(C(=O)C(F)(F)F)s3)CC2)c1
E3 Binder	CHEMBL122413	ChEMBL	6.54	—	—	COc1cccc(NC(=O)/C=C/c2ccc(Cl)cc2)c1
E3 Binder	CHEMBL1958434	ChEMBL	7.66	—	—	COc1cccc(NS(=O)(=O)c2cccc(/C=C/C(=O)NO)c2)c1
E3 Binder	CHEMBL4098561	ChEMBL	7.68	—	—	COc1cccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c1
E3 Binder	CHEMBL476904	ChEMBL	6.5	—	—	COc1cccc(OC)c1-c1cn(CCCCCC(=O)NO)nn1
E3 Binder	CHEMBL435415	ChEMBL	8.37	—	—	COc1cccc(OC)c1-c1csc(CCCCCCC(=O)NO)n1
E3 Binder	CHEMBL520109	ChEMBL	6.77	—	—	COc1cccc(S(=O)(=O)Nc2ccc(C(=O)CSC(C)=O)cc2)c1
E3 Binder	CHEMBL519087	ChEMBL	6.72	—	—	COc1cccc(S(=O)(=O)Nc2ccc(C(=O)CSC(C)=O)cn2)c1
E3 Binder	CHEMBL57792	ChEMBL	8.51	—	—	COc1cccc2[nH]c(C(=O)NCCCCCCC(=O)NO)cc12
E3 Binder	CHEMBL561483	ChEMBL	8.59	—	—	COc1cccc2c(C(CCCCCC(=O)NO)c3c[nH]c4c(OC)cccc34)c[nH]c12
E3 Binder	CHEMBL178	ChEMBL	7.7	DM1	—	COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@@](O)(C(C)=O)C[C@@H]3O[C@H]1C[C@H](N)[C@H](O)[C@H](C)O1
E3 Binder	CHEMBL2023527	ChEMBL	6.26	—	—	COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@@](O)(C(C)=O)C[C@@H]3O[C@H]1C[C@H](NCc2ccc(-c3cn(CCCCC(=O)NO)nn3)cc2)[C@H](O)[C@H](C)O1
E3 Binder	CHEMBL2023528	ChEMBL	7.52	—	—	COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@@](O)(C(C)=O)C[C@@H]3O[C@H]1C[C@H](NCc2ccc(-c3cn(CCCCCC(=O)NO)nn3)cc2)[C@H](O)[C@H](C)O1
E3 Binder	CHEMBL2023529	ChEMBL	7.7	—	—	COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@@](O)(C(C)=O)C[C@@H]3O[C@H]1C[C@H](NCc2ccc(-c3cn(CCCCCCC(=O)NO)nn3)cc2)[C@H](O)[C@H](C)O1
E3 Binder	CHEMBL2023530	ChEMBL	7.72	—	—	COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@@](O)(C(C)=O)C[C@@H]3O[C@H]1C[C@H](NCc2ccc(-c3cn(CCCCCCCC(=O)NO)nn3)cc2)[C@H](O)[C@H](C)O1
E3 Binder	CHEMBL2023526	ChEMBL	7.7	—	—	COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)C[C@@](O)(C(C)=O)C[C@@H]3O[C@H]1C[C@H](NCc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)[C@H](O)[C@H](C)O1
E3 Binder	CHEMBL4858810	ChEMBL	8.19	—	—	COc1cccc2c1CCCCN2Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4849884	ChEMBL	6.5	—	—	COc1cccc2c1CCN(Cc1ccc(C(=O)NO)cc1)CC2
E3 Binder	CHEMBL5270568	ChEMBL	7.3	—	—	COc1cccc2ccc(C(=O)NCc3ccc(C(=O)NO)cc3)nc12
E3 Binder	CHEMBL5081128	ChEMBL	7.55	—	—	COc1ccccc1-c1cc(/C=C/c2ccc(C(=O)NO)cc2)ccn1
E3 Binder	CHEMBL4204972	ChEMBL	7.4	—	—	COc1ccccc1-c1ccc2c(NC(=O)c3ccc(C(=O)NO)cc3)n[nH]c2c1
E3 Binder	CHEMBL476903	ChEMBL	7.12	—	—	COc1ccccc1-c1cn(CCCCCC(=O)NO)nn1
E3 Binder	CHEMBL4294431	ChEMBL	6.02	—	—	COc1ccccc1-c1nc(C(=O)N(C)Cc2ccc(C(=O)NO)cc2)cc2c1[nH]c1ccccc12
E3 Binder	CHEMBL5082644	ChEMBL	6.57	—	—	COc1ccccc1-c1ncc(C(=O)NCCCCCCC(=O)NO)s1
E3 Binder	CHEMBL4468198	ChEMBL	6.48	—	—	COc1ccccc1-n1nc(-c2cccs2)nc1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5188237	ChEMBL	7.42	—	—	COc1ccccc1C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5201168	ChEMBL	7.77	—	—	COc1ccccc1C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(C(=O)NO)cc1F
E3 Binder	CHEMBL5183285	ChEMBL	7.7	—	—	COc1ccccc1C(=O)N(CC(=O)NC1CCCCC1)Cc1ccc(C(=O)NO)cc1F
E3 Binder	CHEMBL3354920	ChEMBL	7.62	—	—	COc1ccccc1C(=O)N[C@H](COc1cccc(/C=C/C(=O)NO)c1)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL3656002	ChEMBL	8.52	—	—	COc1ccccc1C1(Nc2ncc(C(=O)NO)cn2)CC1
E3 Binder	CHEMBL4554270	ChEMBL	8.68	—	—	COc1ccccc1CCn1c(=O)c2ccccc2n(Cc2ccc(C(=O)NO)cc2)c1=O
E3 Binder	CHEMBL249223	ChEMBL	6.07	—	—	COc1ccccc1CN1CCC=C(CCC(=O)NO)C1=O
E3 Binder	CHEMBL3655928	ChEMBL	8.4	—	—	COc1ccccc1CNc1ncc(C(=O)NO)cn1
E3 Binder	CHEMBL3943331	ChEMBL	7.13	—	—	COc1ccccc1N1C(=O)N(Cc2ccc(C(=O)NO)cc2)C(C)(C)C1=O
E3 Binder	CHEMBL1958433	ChEMBL	7.66	—	—	COc1ccccc1N1CCN(S(=O)(=O)c2cccc(/C=C/C(=O)NO)c2)CC1
E3 Binder	CHEMBL426343	ChEMBL	8.1	—	—	COc1ccccc1NC(=O)Cn1ccc(-c2ccc(C(=O)NO)s2)n1
E3 Binder	CHEMBL2179248	ChEMBL	6.34	—	—	COc1ccccc1NC(=O)N(CCCN(C)C)Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL2179249	ChEMBL	8.62	—	—	COc1ccccc1NC(=O)N(CCCO)Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL2179250	ChEMBL	6.33	—	—	COc1ccccc1NC(=O)N(CCc1c[nH]c2ccccc12)Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL2179615	ChEMBL	8.24	—	—	COc1ccccc1NC(=O)N(CCc1ccc(O)cc1)Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL2179247	ChEMBL	6.86	—	—	COc1ccccc1NC(=O)NCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5284956	ChEMBL	6.53	—	—	COc1ccccc1NC(=O)N[C@H](C(=O)Nc1ccc(C(=O)NO)cc1)c1ccccc1
E3 Binder	CHEMBL140505	ChEMBL	6.96	—	—	COc1ccccc1NCCNCc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4536105	ChEMBL	8.18	—	—	COc1ncc(-c2cc(OCCCCCCC(=O)NO)c3ncnc(C)c3c2)cc1F
E3 Binder	CHEMBL4237600	ChEMBL	8.64	—	—	CS(=O)(=O)CCn1cc(-c2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc3[nH]ccc23)cn1
E3 Binder	CHEMBL512516	ChEMBL	6.64	—	—	CS(=O)(=O)Cc1noc(-c2ccc(C(=O)C(F)(F)F)s2)n1
E3 Binder	CHEMBL3912061	ChEMBL	9.77	—	—	CS(=O)(=O)NCCc1cn(Cc2ccc(C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL4159366	ChEMBL	7.13	—	—	CS(=O)(=O)Nc1ccc(-c2ccnc(Nc3ccc(N4CCC(C(=O)NCCCCCCCC(=O)NO)CC4)cc3)n2)cc1
E3 Binder	CHEMBL4175555	ChEMBL	7.34	—	—	CS(=O)(=O)Nc1ccc(-c2ccnc(Nc3ccc(N4CCC(C(=O)Nc5ccc(/C=C/C(=O)NO)cc5)CC4)cc3)n2)cc1
E3 Binder	CHEMBL5272716	ChEMBL	7.34	—	—	CS(=O)(=O)Nc1ccc(-c2ccnc(Nc3ccc(N4CCC(CCc5ccc(/C=C/CC(=O)NO)cc5)CC4)cc3)n2)cc1
E3 Binder	CHEMBL2105534	ChEMBL	6.11	—	—	CS(=O)(=O)c1ccc(-c2cn3ccccc3n2)cc1
E3 Binder	CHEMBL5093377	ChEMBL	7.97	—	—	CS(=O)(=O)c1ccc(-n2ccc3cnc(Nc4cnn(CCCCCC(=O)NO)c4)nc32)cc1
E3 Binder	CHEMBL5079785	ChEMBL	8.23	—	—	CS(=O)(=O)c1ccc(-n2ccc3cnc(Nc4cnn(CCCCCCC(=O)NO)c4)nc32)cc1
E3 Binder	CHEMBL3415620	ChEMBL	6.85	—	—	CS(=O)(=O)c1ccc(N2CCC(Nc3ccc(C(=O)NO)cc3)C2=O)cc1
E3 Binder	CHEMBL243327	ChEMBL	6.4	—	—	CSC(=S)SCC(=O)c1ccc(C)cc1
E3 Binder	CHEMBL244812	ChEMBL	7.0	—	—	CSC(=S)SCC(=O)c1ccc(Cl)c(Cl)c1
E3 Binder	CHEMBL3233684	ChEMBL	6.59	—	—	CSCC[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](COc1ccc(/C=C/C(=O)NO)cc1)Cc1c[nH]c2ccccc12
E3 Binder	CHEMBL5268495	ChEMBL	6.35	—	—	CSCC[C@H](NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCSC)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCNC(=N)N)NC(C)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CC(C)C)C(=O)NCCCCCC(=O)NO
E3 Binder	CHEMBL3126833	ChEMBL	6.11	—	—	CSCC[C@H]1NC(=O)C[C@H]2/C=C/CCSSC[C@@H](NC1=O)C(=O)N[C@H](C(C)C)[C@@H](O)CC(=O)O2
E3 Binder	CHEMBL2047694	ChEMBL	6.72	—	—	CSc1ccc(C/C(=N\O)C(=O)NCCS)cc1Br
E3 Binder	CHEMBL4877300	ChEMBL	8.03	—	—	CSc1ccc2c(c1)N(Cc1ccc(C(=O)NO)cc1)c1ccccc1S2
E3 Binder	CHEMBL4872697	ChEMBL	7.45	—	—	CSc1ccc2c(c1)N(Cc1ccc(C(=O)NO)cc1)c1ccccc1[S+]2[O-]
E3 Binder	CHEMBL4113424	ChEMBL	7.92	—	—	C[C@@H](C(=O)N1CCC(C)(Nc2ncc(C(=O)NO)cn2)CC1)c1ccccc1
E3 Binder	CHEMBL3956211	ChEMBL	6.0	—	—	C[C@@H](NC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)C(=O)NO
E3 Binder	CHEMBL507716	ChEMBL	6.44	—	—	C[C@@H](NC(=O)c1ccc(C(=O)C(F)(F)F)s1)c1ccccc1
E3 Binder	CHEMBL4548247	ChEMBL	6.68	—	—	C[C@@H](NC(=O)c1nc(-c2nccs2)sc1C1CC1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL494645	ChEMBL	6.08	—	—	C[C@@H](NCc1ccc(C(=O)C(F)(F)F)s1)c1ccccc1
E3 Binder	CHEMBL3655944	ChEMBL	9.0	—	—	C[C@@H](Nc1ncc(C(=O)NO)cn1)c1ccccc1
E3 Binder	CHEMBL3905131	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(C(=O)NCCNCCCCCC(=O)NO)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3984055	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(C(=O)NO)cc3)cc12)c1ccc(F)cc1
E3 Binder	CHEMBL3917670	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(C(=O)NO)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3928746	ChEMBL	6.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CN4CCC(NCCCCCC(=O)NO)CC4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3924396	ChEMBL	6.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CN4CCC(NCCCCCCC(=O)NO)CC4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3968380	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CN4CCC(NCCCCCCCC(=O)NO)CC4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3903506	ChEMBL	6.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CN4CCN(CCCC(=O)NO)CC4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3972249	ChEMBL	6.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CN4CCN(CCCCC(=O)NO)CC4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3938265	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CN4CCN(CCCCCC(=O)NO)CC4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3916600	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CN4CCN(CCCCCCC(=O)NO)CC4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3890703	ChEMBL	6.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CN4CCN(CCOCCCCC(=O)NO)CC4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3910297	ChEMBL	6.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CNCC(=O)NO)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3936547	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CNCCCCCC(=O)NO)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3898480	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CNCCCCCCCC(=O)NO)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3968968	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CNCc4ccc(C(=O)NO)cc4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3921652	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(NC(=O)CCCC(=O)NO)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3909969	ChEMBL	6.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(NC(=O)Nc4ccc(/C=C/C(=O)NO)cc4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3953109	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(NC(=O)Nc4ccc(C(=O)NO)cc4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3929290	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(NCc4ccc(/C=C/C(=O)NO)cc4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3932057	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(NCc4ccc(C(=O)NO)cc4)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3977186	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(OCCCC(=O)NO)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3899385	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(OCCCCC(=O)NO)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3904673	ChEMBL	6.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(OCCCNCCCCCC(=O)NO)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3914310	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(OCCNCCCCCC(=O)NO)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3956995	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(OCCNCCCCCCC(=O)NO)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3954393	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(OCCNCCCCCCCC(=O)NO)cc3)cc12)c1ccccc1
E3 Binder	CHEMBL3917093	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2c1cc(-c1ccc(C(=O)NCCNCCCCCCC(=O)NO)cc1)n2C)c1ccccc1
E3 Binder	CHEMBL3943474	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2c1cc(-c1ccc(CNCCN)cc1)n2CCCCCC(=O)NO)c1ccccc1
E3 Binder	CHEMBL3895707	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2c1cc(-c1ccc(N)cc1)n2CCCCCC(=O)NO)c1ccccc1
E3 Binder	CHEMBL3924787	ChEMBL	7.0	—	—	C[C@@H](Nc1ncnc2ccc(OCCCCCC(=O)NO)cc12)c1ccccc1
E3 Binder	CHEMBL198556	ChEMBL	6.6	—	—	C[C@@H](c1ccccc1)N1C(=O)c2ccc(/C=C/C(=O)NO)cc2C1=O
E3 Binder	CHEMBL1094793	ChEMBL	7.2	—	—	C[C@@H](c1ccccc1)n1c(-c2cccc(/C=C/C(=O)NO)c2)nc2ccccc21
E3 Binder	CHEMBL4532398	ChEMBL	8.74	—	—	C[C@@H]1CN(C(=O)Nc2ccc(-c3nc(N4CCOCC4)c4cnn(CCCCCCC(=O)NO)c4n3)cc2)CCO1
E3 Binder	CHEMBL5193563	ChEMBL	7.39	—	—	C[C@@H]1CN(Cc2ccc(C(=O)NO)cc2)C[C@H](C)N1Cc1cccc(Cl)c1
E3 Binder	CHEMBL5205841	ChEMBL	7.4	—	—	C[C@@H]1CN(Cc2ccc(C(=O)NO)cc2)C[C@H]1c1nc2c(cnn2C2CCCC2)c(=O)[nH]1
E3 Binder	CHEMBL3640687	ChEMBL	8.15	—	—	C[C@@H]1CN(c2ncc(C(=O)NCCCCCCC(=O)NO)cn2)C[C@H](C)O1
E3 Binder	CHEMBL2408693	ChEMBL	6.47	—	—	C[C@@H]1N=C(c2ccccc2)c2cc(C#CCCCC(=O)NO)ccc2NC1=O
E3 Binder	CHEMBL238596	ChEMBL	6.37	—	—	C[C@@H]1NC(=O)C(C)(C)NC(=O)[C@H](CCCCCSSc2ccccn2)NC(=O)[C@H]2CCCN2C1=O
E3 Binder	CHEMBL370056	ChEMBL	7.52	—	—	C[C@@H]1NC(=O)[C@@H](C)NC(=O)[C@H](CCCCCC(=O)[C@@H]2CO2)NC(=O)[C@H]2CCCN2C1=O
E3 Binder	CHEMBL3315350	ChEMBL	8.19	—	—	C[C@@H]1NC(=O)[C@H](CCCCCC(=O)[C@@H]2CO2)NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC1=O
E3 Binder	CHEMBL279636	ChEMBL	6.37	—	—	C[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@H](CCCCCC(=O)[C@@H]2CO2)NC(=O)[C@@H](C)NC1=O
E3 Binder	CHEMBL3693804	ChEMBL	8.52	—	—	C[C@@](O)(c1ccc(F)cc1)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3415630	ChEMBL	6.58	—	—	C[C@@]1(Nc2ccc(C(=O)NO)cc2)CCN(c2ccc(Cl)cc2)C1=O
E3 Binder	CHEMBL3526395	ChEMBL	7.21	—	—	C[C@@]12Nc3ccccc3[C@]1(O)CCN2Cc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL55974	ChEMBL	6.45	—	—	C[C@H](CCCCC(=O)NO)NC(=O)c1ccc(N(C)C)cc1
E3 Binder	CHEMBL4761969	ChEMBL	6.57	—	—	C[C@H](NC(=O)[C@H](CC(=O)NC(C)(C)C)NC(=O)c1ccc(C(=O)NO)cc1)C(=O)NCc1ccccc1
E3 Binder	CHEMBL4167623	ChEMBL	6.57	FGY	—	C[C@H](NC(=O)[C@H](CC(=O)NCC(C)(C)C)NC(=O)c1ccc(C(=O)NO)cc1)C(=O)NCc1ccccc1
E3 Binder	CHEMBL462208	ChEMBL	6.82	—	—	C[C@H](NC(=O)c1ccc(C(=O)C(F)(F)F)s1)c1ccccc1
E3 Binder	CHEMBL4584020	ChEMBL	7.74	—	—	C[C@H](NC(=O)c1nc(-c2nc3c(s2)CCCC3)sc1C1CC1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4443998	ChEMBL	8.7	—	—	C[C@H](NC(=O)c1nc(-c2ncc(-c3ccc(F)cc3)s2)sc1C1CC1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4460552	ChEMBL	8.8	—	—	C[C@H](NC(=O)c1nc(-c2ncc(-c3ccccc3)s2)sc1C1CC1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4476497	ChEMBL	7.85	—	—	C[C@H](NC(=O)c1nc(-c2nccs2)sc1C1CC1)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4522666	ChEMBL	7.8	—	—	C[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(CNC(=O)c3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL4583074	ChEMBL	8.52	—	—	C[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(CNc3ncc(C(=O)NO)cn3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL5221123	ChEMBL	7.18	—	—	C[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(C(=O)NO)s1
E3 Binder	CHEMBL4460447	ChEMBL	8.22	—	—	C[C@H](Nc1nc(N)nc(N)c1C#N)c1nc2cccc(NCc3ccc(C(=O)NO)cc3)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL3655943	ChEMBL	7.72	—	—	C[C@H](Nc1ncc(C(=O)NO)cn1)c1ccccc1
E3 Binder	CHEMBL1096981	ChEMBL	6.88	—	—	C[C@H](O)C(=O)CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O
E3 Binder	CHEMBL194509	ChEMBL	6.54	—	—	C[C@H](c1ccccc1)N1C(=O)c2ccc(/C=C/C(=O)NO)cc2C1=O
E3 Binder	CHEMBL1094792	ChEMBL	7.4	—	—	C[C@H](c1ccccc1)n1c(-c2cccc(/C=C/C(=O)NO)c2)nc2ccccc21
E3 Binder	CHEMBL2347005	ChEMBL	6.86	—	—	C[C@H]1C=C2C=C[C@H](C)[C@H](CC[C@@H]3C[C@@H](O[Si](C)(C)C(C)(C)C)CC(=O)O3)[C@H]2[C@@H](OC(=O)NCCCCCCC(=O)NO)C1
E3 Binder	CHEMBL2347011	ChEMBL	7.47	—	—	C[C@H]1C=C2C=C[C@H](C)[C@H](CC[C@@H]3C[C@@H](O[Si](C)(C)C(C)(C)C)CC(=O)O3)[C@H]2[C@@H](OC(=O)NCc2ccc(-c3cn(CCCCCCC(=O)NO)nn3)cc2)C1
E3 Binder	CHEMBL2347010	ChEMBL	6.89	—	—	C[C@H]1C=C2C=C[C@H](C)[C@H](CC[C@@H]3C[C@@H](O[Si](C)(C)C(C)(C)C)CC(=O)O3)[C@H]2[C@@H](OC(=O)Nc2ccc(-c3cn(CCCCCCC(=O)NO)nn3)cc2)C1
E3 Binder	CHEMBL5172893	ChEMBL	6.29	—	—	C[C@H]1CN(Cc2ccc(/C=C/C(=O)NO)cc2)C[C@@H]1c1nc2c(cnn2C2CCOCC2)c(=O)[nH]1
E3 Binder	CHEMBL5205968	ChEMBL	7.4	—	—	C[C@H]1CN(Cc2ccc(C(=O)NO)cc2)C[C@@H]1c1nc2c(cnn2C2CCCC2)c(=O)[nH]1
E3 Binder	CHEMBL5199795	ChEMBL	7.68	—	—	C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c(=O)c(C(=O)NCC4CN(CC(=O)NO)N=N4)cn1c23
E3 Binder	CHEMBL4636049	ChEMBL	7.68	—	—	C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c(=O)c(C(=O)NCc4cn(CCCCCC(=O)NO)nn4)cn1c23
E3 Binder	CHEMBL4649154	ChEMBL	7.68	—	—	C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c(=O)c(C(=O)NCc4cn(CCCCCCC(=O)NO)nn4)cn1c23
E3 Binder	CHEMBL4644409	ChEMBL	7.68	—	—	C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c(=O)c(C(=O)NCc4cn(CCCCCCCC(=O)NO)nn4)cn1c23
E3 Binder	CHEMBL4645270	ChEMBL	7.68	—	—	C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c(=O)c(C(=O)OCc4cn(CCCCCC(=O)NO)nn4)cn1c23
E3 Binder	CHEMBL4643070	ChEMBL	7.68	—	—	C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c(=O)c(C(=O)OCc4cn(CCCCCCC(=O)NO)nn4)cn1c23
E3 Binder	CHEMBL4638706	ChEMBL	7.68	—	—	C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c(=O)c(C(=O)OCc4cn(CCCCCCCC(=O)NO)nn4)cn1c23
E3 Binder	CHEMBL3693803	ChEMBL	8.52	—	—	C[C@](O)(c1ccc(F)cc1)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3415629	ChEMBL	7.77	—	—	C[C@]1(Nc2ccc(C(=O)NO)cc2)CCN(c2ccc(Cl)cc2)C1=O
E3 Binder	CHEMBL4852393	ChEMBL	6.27	—	—	C[C@]12CC3CC(NCc4ccc(C(=O)NO)cn4)(C1)C[C@@](C)(C3)C2
E3 Binder	CHEMBL2401843	ChEMBL	8.1	—	—	C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC[C@@]2(O)c1cn(CCCC(=O)NO)nn1
E3 Binder	CHEMBL2401844	ChEMBL	8.1	—	—	C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC[C@@]2(O)c1cn(CCCCC(=O)NO)nn1
E3 Binder	CHEMBL2401845	ChEMBL	7.5	—	—	C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC[C@@]2(O)c1cn(CCCCCC(=O)NO)nn1
E3 Binder	CHEMBL2401846	ChEMBL	7.89	—	—	C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC[C@@]2(O)c1cn(CCCCCCC(=O)NO)nn1
E3 Binder	CHEMBL2401847	ChEMBL	7.89	—	—	C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC[C@@]2(O)c1cn(CCCCCCCC(=O)NO)nn1
E3 Binder	CHEMBL3980861	ChEMBL	7.0	—	—	Cc1[nH]c(/C=C2\C(=O)Nc3ccc(F)cc32)c(C)c1C(=O)NCCC(=O)NO
E3 Binder	CHEMBL3940740	ChEMBL	6.0	—	—	Cc1[nH]c(/C=C2\C(=O)Nc3ccc(F)cc32)c(C)c1C(=O)NCCCC(=O)NO
E3 Binder	CHEMBL3943406	ChEMBL	7.0	—	—	Cc1[nH]c(/C=C2\C(=O)Nc3ccc(F)cc32)c(C)c1C(=O)NCCCCCC(=O)NO
E3 Binder	CHEMBL3947208	ChEMBL	7.0	—	—	Cc1[nH]c(/C=C2\C(=O)Nc3ccc(F)cc32)c(C)c1C(=O)NCCOc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL3919147	ChEMBL	7.0	—	—	Cc1[nH]c(/C=C2\C(=O)Nc3ccc(F)cc32)c(C)c1C(=O)NCCOc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5083849	ChEMBL	7.17	—	—	Cc1[nH]c(C(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2OCCCCCCCC(=O)NO)c2c1C(=O)CCCC2
E3 Binder	CHEMBL3793310	ChEMBL	6.0	—	—	Cc1[nH]c2ccccc2c1/C=C/c1ccccc1-c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL5185310	ChEMBL	7.89	—	—	Cc1[nH]c2ccccc2c1C1=CCC(NCc2ccc(OCC(=O)NO)cc2F)CC1
E3 Binder	CHEMBL3329997	ChEMBL	8.04	—	—	Cc1[nH]c2ccccc2c1CCN(C(C)C)S(=O)(=O)c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL3329995	ChEMBL	7.32	—	—	Cc1[nH]c2ccccc2c1CCN(C)S(=O)(=O)c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL483254	ChEMBL	9.15	LBH	—	Cc1[nH]c2ccccc2c1CCNCc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL3330002	ChEMBL	8.12	—	—	Cc1[nH]c2ccccc2c1CCNCc1ccc(/C=C/CNO)cc1.Cl
E3 Binder	CHEMBL4080164	ChEMBL	7.84	—	—	Cc1[nH]c2ccccc2c1CCNCc1cccc(/C=C/C(=O)NO)c1.Cl
E3 Binder	CHEMBL3329991	ChEMBL	8.55	—	—	Cc1[nH]c2ccccc2c1CCNS(=O)(=O)c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL3330001	ChEMBL	6.11	—	—	Cc1[nH]c2ccccc2c1CCNS(=O)(=O)c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3329993	ChEMBL	8.1	—	—	Cc1[nH]c2ccccc2c1CCNS(=O)(=O)c1cccc(/C=C/C(=O)NO)c1
E3 Binder	CHEMBL1095450	ChEMBL	7.2	—	—	Cc1c(-c2ccccc2)nc(-c2cccc(/C=C/C(=O)NO)c2)n1CCN1CCOCC1
E3 Binder	CHEMBL1095451	ChEMBL	7.2	—	—	Cc1c(-c2ccccc2)nc(-c2cccc(/C=C/C(=O)NO)c2)n1CCc1ccccc1
E3 Binder	CHEMBL1096093	ChEMBL	7.1	—	—	Cc1c(-c2ccccc2)nc(-c2cccc(/C=C/C(=O)NO)c2)n1[C@@H]1CCCN(C(C)C)C1
E3 Binder	CHEMBL1094648	ChEMBL	7.2	—	—	Cc1c(-c2ccccc2)nc(-c2cccc(/C=C/C(=O)NO)c2)n1[C@@H]1CCCN(C)C1
E3 Binder	CHEMBL3971436	ChEMBL	8.39	—	—	Cc1c(C)n(Cc2ccc(C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL3329990	ChEMBL	8.48	—	—	Cc1c(CCNS(=O)(=O)c2ccc(/C=C/C(=O)NO)cc2)c2ccccc2n1C
E3 Binder	CHEMBL5283979	ChEMBL	8.47	—	—	Cc1c(CCNS(=O)(=O)c2ccc(/C=C/C=C/C(=O)NO)cc2)c2ccccc2n1C
E3 Binder	CHEMBL4441675	ChEMBL	8.9	—	—	Cc1c(CN(C)C)c2ccccc2n1-c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4079799	ChEMBL	7.02	—	—	Cc1c(CN(C)C)c2ccccc2n1Cc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4100664	ChEMBL	8.21	—	—	Cc1c(CN(C)C)c2ccccc2n1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4104052	ChEMBL	7.2	—	—	Cc1c(CN(C)C)c2ccccc2n1S(=O)(=O)c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4073888	ChEMBL	7.07	—	—	Cc1c(CN(C)C)c2ccccc2n1S(=O)(=O)c1cccc(/C=C/C(=O)NO)c1
E3 Binder	CHEMBL4562547	ChEMBL	8.84	—	—	Cc1c(CN)c2ccccc2n1-c1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3960564	ChEMBL	8.84	—	—	Cc1c(CN)c2ccccc2n1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5173964	ChEMBL	6.03	—	—	Cc1c(COc2ccc(CN(C)CCCCC(=O)NO)c(F)c2)cccc1-c1ccccc1
E3 Binder	CHEMBL5199949	ChEMBL	6.33	—	—	Cc1c(COc2ccc(CNCCCCCC(=O)NO)c(F)c2)cccc1-c1ccc2c(c1)OCCO2
E3 Binder	CHEMBL5186043	ChEMBL	6.44	—	—	Cc1c(COc2ccc(CNCCCCCC(=O)NO)c(F)c2)cccc1-c1ccccc1
E3 Binder	CHEMBL5206651	ChEMBL	6.37	—	—	Cc1c(COc2ccc(CNCCCCCCC(=O)NO)c(F)c2)cccc1-c1ccc2c(c1)OCCO2
E3 Binder	CHEMBL5172459	ChEMBL	7.32	—	—	Cc1c(COc2ccc(CNCCCCCCC(=O)NO)c(F)c2)cccc1-c1ccccc1
E3 Binder	CHEMBL5191149	ChEMBL	6.48	—	—	Cc1c(COc2ccc(CNCCCCCCC(=O)NO)c(OCc3cccc(C#N)c3)c2)cccc1-c1ccccc1
E3 Binder	CHEMBL1095437	ChEMBL	7.1	—	—	Cc1c(Cc2ccccc2)nc(-c2cccc(/C=C/C(=O)NO)c2)n1CCN1CCOCC1
E3 Binder	CHEMBL1099048	ChEMBL	7.2	—	—	Cc1c(Cc2ccccc2)nc(-c2cccc(/C=C/C(=O)NO)c2)n1CCc1ccccc1
E3 Binder	CHEMBL1099049	ChEMBL	7.2	—	—	Cc1c(Cc2ccccc2)nc(-c2cccc(/C=C/C(=O)NO)c2)n1[C@@H]1CCCN(C)C1
E3 Binder	CHEMBL4863455	ChEMBL	7.57	—	—	Cc1c(F)cc(C(=O)NO)cc1F
E3 Binder	CHEMBL5287581	ChEMBL	6.84	—	—	Cc1c(NC(=O)NCCN2C(=O)S/C(=C\c3ccc([N+](=O)[O-])cc3)C2=O)c(=O)n(-c2ccccc2)n1C
E3 Binder	CHEMBL1617398	ChEMBL	6.1	JBO	—	Cc1c(Nc2ncccc2C(=O)O)cccc1C(F)(F)F
E3 Binder	CHEMBL5088769	ChEMBL	6.5	—	—	Cc1c2c(c(C(=O)Nc3cc(S(=O)(=O)N4CCOCC4)ccc3OCCCCCCCC(=O)NO)n1C)CCCCC2=O
E3 Binder	CHEMBL4215609	ChEMBL	6.17	—	—	Cc1c2ccc(N(C)c3ccnc(Nc4ccc(C(=O)NCCCCC(=O)NO)cc4)n3)cc2nn1C
E3 Binder	CHEMBL4217092	ChEMBL	7.77	—	—	Cc1c2ccc(N(C)c3ccnc(Nc4ccc(C(=O)NCCCCCC(=O)NO)cc4)n3)cc2nn1C
E3 Binder	CHEMBL4212117	ChEMBL	8.48	—	—	Cc1c2ccc(N(C)c3ccnc(Nc4ccc(C(=O)NCCCCCCC(=O)NO)cc4)n3)cc2nn1C
E3 Binder	CHEMBL4212674	ChEMBL	7.6	—	—	Cc1c2ccc(N(C)c3ccnc(Nc4ccc(C(=O)NCCCCCCCC(=O)NO)cc4)n3)cc2nn1C
E3 Binder	CHEMBL4207767	ChEMBL	6.75	—	—	Cc1c2ccc(N(C)c3ccnc(Nc4cccc(C(=O)NCCCCCC(=O)NO)c4)n3)cc2nn1C
E3 Binder	CHEMBL4225230	ChEMBL	7.7	—	—	Cc1cc(-c2ccc(F)cc2)n(Cc2ccc(C(=O)NO)cc2)n1
E3 Binder	CHEMBL4225171	ChEMBL	8.1	—	—	Cc1cc(-c2ccc(F)cc2)nn1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4225495	ChEMBL	7.8	—	—	Cc1cc(-c2ccc3c(c2)OCO3)n(Cc2ccc(C(=O)NO)cc2)n1
E3 Binder	CHEMBL4228987	ChEMBL	8.3	—	—	Cc1cc(-c2ccc3c(c2)OCO3)nn1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4551888	ChEMBL	6.6	—	—	Cc1cc(-c2nc3sc4c(c3c(=O)[nH]2)CCN(C)C4)cc(C)c1OCCCC(=O)NO
E3 Binder	CHEMBL4514808	ChEMBL	7.14	—	—	Cc1cc(-c2nc3sc4c(c3c(=O)[nH]2)CCN(C)C4)cc(C)c1OCCCCCC(=O)NO
E3 Binder	CHEMBL4465878	ChEMBL	6.8	—	—	Cc1cc(-c2nc3sc4c(c3c(=O)[nH]2)CCN(C)C4)cc(C)c1OCCOCc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4548155	ChEMBL	6.7	—	—	Cc1cc(-c2nc3sc4c(c3c(=O)[nH]2)CCN(C)C4)cc(C)c1OCc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4592260	ChEMBL	6.73	—	—	Cc1cc(-c2nc3sc4c(c3c(=O)[nH]2)CCN(C)C4)cc(C)c1OCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4443980	ChEMBL	6.11	—	—	Cc1cc(-c2nc3sc4c(c3c(=O)[nH]2)CCN(C)C4)cc(C)c1OCc1cccc(C(=O)NO)c1
E3 Binder	CHEMBL4548542	ChEMBL	6.89	—	—	Cc1cc(-c2nc3sc4c(c3c(=O)[nH]2)CCN(CCCCCC(=O)NO)C4)cc(C)c1O
E3 Binder	CHEMBL4461219	ChEMBL	8.22	—	—	Cc1cc(-c2nnc(Sc3c(F)cc(C(=O)NO)cc3F)n2C)nn1C
E3 Binder	CHEMBL4475365	ChEMBL	8.3	—	—	Cc1cc(-c2nnc(Sc3ccc(C(=O)NO)cc3)n2C)nn1C
E3 Binder	CHEMBL3589010	ChEMBL	6.29	—	—	Cc1cc(/C=C2\SC(=O)N(c3ccccc3)C2=O)c(C)n1-c1cccnc1
E3 Binder	CHEMBL3758409	ChEMBL	6.15	—	—	Cc1cc(C(=O)NCCCCCCS)[nH]n1
E3 Binder	CHEMBL3655955	ChEMBL	8.4	—	—	Cc1cc(C(C)(C)Nc2ncc(C(=O)NO)cn2)ccc1F
E3 Binder	CHEMBL3656016	ChEMBL	8.52	—	—	Cc1cc(C(F)(F)F)cc(C2(Nc3ncc(C(=O)NO)cn3)CC2)c1
E3 Binder	CHEMBL3621295	ChEMBL	6.35	—	—	Cc1cc(C)c(/C=C2\C(=O)Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc32)[nH]1
E3 Binder	CHEMBL5193584	ChEMBL	6.82	—	—	Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(N4CCN(C(=O)CCCCCC(=O)NO)CC4)nc3)cc3c2cnn3C(C)C)c(=O)[nH]1
E3 Binder	CHEMBL5192423	ChEMBL	7.09	—	—	Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(N4CCN(C(=O)CCCCCCC(=O)NO)CC4)nc3)cc3c2cnn3C(C)C)c(=O)[nH]1
E3 Binder	CHEMBL5184172	ChEMBL	6.15	—	—	Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(N4CCN(CCCCCCC(=O)NO)CC4)nc3)cc3c2cnn3C(C)C)c(=O)[nH]1
E3 Binder	CHEMBL5191470	ChEMBL	6.39	—	—	Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(N4CCN(CCCCCCCC(=O)NO)CC4)nc3)cc3c2cnn3C(C)C)c(=O)[nH]1
E3 Binder	CHEMBL5173660	ChEMBL	6.41	—	—	Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(N4CCN(CCCCCCCCC(=O)NO)CC4)nc3)cc3c2cnn3C(C)C)c(=O)[nH]1
E3 Binder	CHEMBL5187019	ChEMBL	6.16	—	—	Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(N4CCN(Cc5ccc(NC(=O)CCCCCCC(=O)NO)cc5)CC4)nc3)cc3c2cnn3C(C)C)c(=O)[nH]1
E3 Binder	CHEMBL5189365	ChEMBL	6.16	—	—	Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(N4CCN(c5ncc(C(=O)NO)cn5)CC4)nc3)cc3c2cnn3C(C)C)c(=O)[nH]1
E3 Binder	CHEMBL5192032	ChEMBL	6.6	—	—	Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(NC(=O)CCCCCC(=O)NO)cc3)cc3c2cnn3C(C)C)c(=O)[nH]1
E3 Binder	CHEMBL5182624	ChEMBL	6.75	—	—	Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(NC(=O)CCCCCCC(=O)NO)cc3)cc3c2cnn3C(C)C)c(=O)[nH]1
E3 Binder	CHEMBL4633299	ChEMBL	8.3	—	—	Cc1cc(C)c(CNC(=O)c2cc(C)n(-c3cccc(NC(=O)CCCCCCC(=O)NO)c3)c2C)c(=O)[nH]1
E3 Binder	CHEMBL4639495	ChEMBL	8.0	—	—	Cc1cc(C)c(CNC(=O)c2cnn(-c3cccc(NC(=O)CCCCCCC(=O)NO)c3)c2C)c(=O)[nH]1
E3 Binder	CHEMBL4513524	ChEMBL	7.34	—	—	Cc1cc(C)c(NC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)c2ccc(/C=C/C(=O)NO)cc2)c(C)c1
E3 Binder	CHEMBL4228336	ChEMBL	7.65	—	—	Cc1cc(C)c(NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)/C=C/c2ccc(C(=O)NO)cc2)c(C)c1
E3 Binder	CHEMBL3639926	ChEMBL	7.46	—	—	Cc1cc(C)c(Nc2ccc(C(=O)N(C)CCCCCCC(=O)NO)cc2)c(C)c1
E3 Binder	CHEMBL3693769	ChEMBL	7.42	—	—	Cc1cc(C)c(Nc2ncc(C(=O)N(C)CCCCCCC(=O)NO)cn2)c(C)c1
E3 Binder	CHEMBL2018297	ChEMBL	7.42	—	—	Cc1cc(C)c2c3c(n(Cc4ccc(C(=O)NO)cc4)c2c1)CCN(C)C3
E3 Binder	CHEMBL4210578	ChEMBL	6.6	—	—	Cc1cc(C)cc(-c2ccc3c(NC(=O)c4ccc(C(=O)NO)cc4)n[nH]c3c2)c1
E3 Binder	CHEMBL4868592	ChEMBL	6.64	—	—	Cc1cc(C)cc(C(=O)N(CC(=O)N(C)C)Cc2ccc(C(=O)NO)cc2)c1
E3 Binder	CHEMBL4878538	ChEMBL	6.89	—	—	Cc1cc(C)cc(C(=O)N(CC(=O)N2CCCCC2)Cc2ccc(C(=O)NO)cc2)c1
E3 Binder	CHEMBL5194945	ChEMBL	7.62	—	—	Cc1cc(C)cc(C(=O)N(CC(=O)NC(C)(C)C)Cc2ccc(C(=O)NO)cc2F)c1
E3 Binder	CHEMBL4173361	ChEMBL	7.96	HBG	—	Cc1cc(C)cc(C(=O)N(CC(=O)NC2CCCCC2)Cc2ccc(C(=O)NO)cc2)c1
E3 Binder	CHEMBL5180418	ChEMBL	7.7	—	—	Cc1cc(C)cc(C(=O)N(CC(=O)NC2CCCCC2)Cc2ccc(C(=O)NO)cc2F)c1
E3 Binder	CHEMBL5189808	ChEMBL	7.89	—	—	Cc1cc(C)cc(C(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(C(=O)NO)cc2F)c1
E3 Binder	CHEMBL4587363	ChEMBL	6.2	—	—	Cc1cc(C)cc(C(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(C(=O)Nc3cc(-c4ccccc4)ccc3N)cc2)c1
E3 Binder	CHEMBL4541820	ChEMBL	6.33	—	—	Cc1cc(C)cc(C(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(C(=O)Nc3cc(F)ccc3N)cc2)c1
E3 Binder	CHEMBL4459617	ChEMBL	6.75	—	—	Cc1cc(C)cc(C(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(C(=O)Nc3ccccc3N)cc2)c1
E3 Binder	CHEMBL4461005	ChEMBL	7.69	—	—	Cc1cc(C)cc(C(=O)N(CCC(=O)NCc2ccccc2)Cc2ccc(C(=O)NO)cc2)c1
E3 Binder	CHEMBL4095934	ChEMBL	6.67	—	—	Cc1cc(C)cc(C(=O)N(CCCCCC(=O)NO)CC(=O)NC2CCCCC2)c1
E3 Binder	CHEMBL4090647	ChEMBL	6.87	—	—	Cc1cc(C)cc(C(=O)N(CCCCCC(=O)NO)CC(=O)NCc2ccccc2)c1
E3 Binder	CHEMBL4564332	ChEMBL	6.33	—	—	Cc1cc(C)cc(C(=O)N(CCCCCC(=O)Nc2cc(-c3ccccc3)ccc2N)CC(=O)NCc2ccccc2)c1
E3 Binder	CHEMBL4740787	ChEMBL	7.1	—	—	Cc1cc(C)cc(C(=O)N(Cc2ccc(C(=O)NO)cc2)Cc2nnnn2Cc2ccccc2)c1
E3 Binder	CHEMBL4643138	ChEMBL	6.38	—	—	Cc1cc(C)cc(C(=O)NOCCCCC(=O)NO)c1
E3 Binder	CHEMBL2312168	ChEMBL	7.92	—	—	Cc1cc(C)cc(C(=O)NOCCCCCC(=O)NO)c1
E3 Binder	CHEMBL4434784	ChEMBL	6.05	—	—	Cc1cc(C)cc(C(=O)NOCc2ccc(/C=C/C(=O)NO)cc2)c1
E3 Binder	CHEMBL1093713	ChEMBL	7.46	—	—	Cc1cc(C)cc(NC(=O)CCCCC(=O)NO)c1
E3 Binder	CHEMBL3652239	ChEMBL	8.4	—	—	Cc1cc(C)cc(Nc2ncc(C(=O)NO)cn2)c1
E3 Binder	CHEMBL3656011	ChEMBL	8.22	—	—	Cc1cc(C2(Nc3ncc(C(=O)NO)cn3)CC2)ccc1F
E3 Binder	CHEMBL3655935	ChEMBL	8.52	—	—	Cc1cc(Cl)ccc1CNc1ncc(C(=O)NO)cn1
E3 Binder	CHEMBL4794499	ChEMBL	7.76	—	—	Cc1cc(F)cc(C)c1Oc1ccc(C(C)(C)O)cc1-c1cn(C)c(=O)c2[nH]c(C(=O)NCCCCCCC(=O)NO)cc12
E3 Binder	CHEMBL4753842	ChEMBL	7.41	—	—	Cc1cc(F)cc(C)c1Oc1ccc(C(C)(C)O)cc1-c1cn(C)c(=O)c2[nH]c(C(=O)NCc3ccc(C(=O)NO)cc3)cc12
E3 Binder	CHEMBL3655907	ChEMBL	8.3	—	—	Cc1cc(F)cc(Nc2ncc(C(=O)NO)cn2)c1
E3 Binder	CHEMBL3655949	ChEMBL	7.72	—	—	Cc1cc(F)ccc1C(C)(C)Nc1ncc(C(=O)NO)cn1
E3 Binder	CHEMBL3640658	ChEMBL	7.23	—	—	Cc1cc(F)ccc1C(O)(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1ccc(F)cc1C
E3 Binder	CHEMBL4083750	ChEMBL	6.92	—	—	Cc1cc(F)ccc1Nc1ncnc2cc(NC(=O)CCCCCCC(=O)NO)sc12
E3 Binder	CHEMBL3890261	ChEMBL	8.16	—	—	Cc1cc(NC(=O)NCc2ccc(C(=O)NO)cc2)no1
E3 Binder	CHEMBL3655914	ChEMBL	8.0	—	—	Cc1cc(Nc2ncc(C(=O)NO)cn2)ccn1
E3 Binder	CHEMBL1910047	ChEMBL	6.91	—	—	Cc1cc(S(=O)(=O)N2CCC(CCCC(=O)NO)CC2)cc2ccccc12
E3 Binder	CHEMBL4788940	ChEMBL	6.82	—	—	Cc1cc2cc(NS(=O)(=O)Cc3ccc(C(=O)NO)cc3)ccc2n(C)c1=O
E3 Binder	CHEMBL4789481	ChEMBL	6.46	—	—	Cc1cc2cc(NS(=O)(=O)c3ccc(C(=O)NO)cc3)ccc2n(C)c1=O
E3 Binder	CHEMBL3893799	ChEMBL	8.6	—	—	Cc1cc2ccccc2n1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL2403451	ChEMBL	6.0	—	—	Cc1cc2sc(C(=O)NO)cc2cc1O
E3 Binder	CHEMBL5093633	ChEMBL	7.82	—	—	Cc1ccc(-c2cc(/C=C/c3ccc(C(=O)NO)cc3)ccn2)c(F)c1
E3 Binder	CHEMBL5081200	ChEMBL	6.82	—	—	Cc1ccc(-c2cc(/C=C/c3ccc(C(=O)NO)cc3)ccn2)cc1
E3 Binder	CHEMBL3883667	ChEMBL	7.04	—	—	Cc1ccc(-c2cc(C(=O)NCCCCCC(=O)NO)nn2-c2ccc(S(N)(=O)=O)cc2)cc1
E3 Binder	CHEMBL3884141	ChEMBL	7.3	—	—	Cc1ccc(-c2cc(C(=O)NCCCCCCC(=O)NO)nn2-c2ccc(S(C)(=O)=O)cc2)cc1
E3 Binder	CHEMBL3884279	ChEMBL	7.08	—	—	Cc1ccc(-c2cc(C(=O)NCCCCCCC(=O)NO)nn2-c2ccc(S(N)(=O)=O)cc2)cc1
E3 Binder	CHEMBL3883560	ChEMBL	6.74	—	—	Cc1ccc(-c2cc(C(=O)NCCCCCCCC(=O)NO)nn2-c2ccc(S(N)(=O)=O)cc2)cc1
E3 Binder	CHEMBL4229123	ChEMBL	7.11	—	—	Cc1ccc(-c2cc(C(F)(F)F)n(CCc3ccc(C(=O)NO)cc3)n2)cc1
E3 Binder	CHEMBL4225331	ChEMBL	7.8	—	—	Cc1ccc(-c2cc(C(F)(F)F)n(Cc3ccc(C(=O)NO)cc3)n2)cc1
E3 Binder	CHEMBL4228699	ChEMBL	6.45	—	—	Cc1ccc(-c2cc(C(F)(F)F)nn2-c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL3884044	ChEMBL	7.12	—	—	Cc1ccc(-c2cc(C(F)(F)F)nn2-c2ccc(S(=O)(=O)NCCCCCC(=O)NO)cc2)cc1
E3 Binder	CHEMBL3885496	ChEMBL	7.18	—	—	Cc1ccc(-c2cc(C(F)(F)F)nn2-c2ccc(S(=O)(=O)NCCCCCCC(=O)NO)cc2)cc1
E3 Binder	CHEMBL3883830	ChEMBL	7.21	—	—	Cc1ccc(-c2cc(C(F)(F)F)nn2-c2ccc(S(=O)(=O)NCCCCCCCC(=O)NO)cc2)cc1
E3 Binder	CHEMBL118	ChEMBL	6.19	CEL	—	Cc1ccc(-c2cc(C(F)(F)F)nn2-c2ccc(S(N)(=O)=O)cc2)cc1
E3 Binder	CHEMBL4227717	ChEMBL	6.27	—	—	Cc1ccc(-c2cc(C(F)(F)F)nn2CCc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4227770	ChEMBL	7.57	—	—	Cc1ccc(-c2cc(C(F)(F)F)nn2Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4229248	ChEMBL	8.15	—	—	Cc1ccc(-c2cc(C)n(Cc3ccc(C(=O)NO)cc3)n2)cc1
E3 Binder	CHEMBL4228291	ChEMBL	7.66	—	—	Cc1ccc(-c2cc(C)nn2Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL2337869	ChEMBL	6.34	—	—	Cc1ccc(-c2ccc(Cn3cccc(O)c3=S)cc2)cc1
E3 Binder	CHEMBL507682	ChEMBL	7.36	—	—	Cc1ccc(-c2cn(CCCCCC(=O)NO)nn2)cc1
E3 Binder	CHEMBL3110277	ChEMBL	6.09	—	—	Cc1ccc(-c2cn(CCCCCn3cccc(O)c3=S)nn2)cc1
E3 Binder	CHEMBL5089538	ChEMBL	6.82	—	—	Cc1ccc(-c2cncc(/C=C/c3ccc(C(=O)NO)cc3)c2)c(F)c1
E3 Binder	CHEMBL3771174	ChEMBL	6.5	—	—	Cc1ccc(-c2nc(C(=O)NO)co2)cc1
E3 Binder	CHEMBL4866529	ChEMBL	6.65	—	—	Cc1ccc(-c2nc(CNc3ccc(C(=O)NO)cc3)n(-c3ccccc3)n2)cc1
E3 Binder	CHEMBL4871247	ChEMBL	8.15	—	—	Cc1ccc(-c2nc(CNc3ccc(C(=O)NO)cc3)n(-c3ccccc3)n2)s1
E3 Binder	CHEMBL4288953	ChEMBL	8.96	—	—	Cc1ccc(-c2nc(NCc3ccc(C(=O)NO)cc3)cc3c2[nH]c2ccccc23)cc1
E3 Binder	CHEMBL5078008	ChEMBL	6.18	—	—	Cc1ccc(-c2ncc(/C=C/C(=O)Nc3ccccc3N)s2)cc1
E3 Binder	CHEMBL509207	ChEMBL	6.22	—	—	Cc1ccc(-c2nnc(-c3ccc(C(=O)C(F)(F)F)s3)o2)cc1
E3 Binder	CHEMBL453953	ChEMBL	6.07	—	—	Cc1ccc(-c2noc(-c3ccc(C(=O)C(F)(F)F)s3)n2)cc1
E3 Binder	CHEMBL4862349	ChEMBL	6.51	—	—	Cc1ccc(-n2nc(-c3ccccc3)nc2CNc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL595711	ChEMBL	9.0	—	—	Cc1ccc(/C=C/C(CO)N2CCN(c3ncc(C(=O)NO)cn3)CC2)cc1
E3 Binder	CHEMBL243760	ChEMBL	6.6	—	—	Cc1ccc(C(=O)CSC(=S)SC(C)(C)C)cc1
E3 Binder	CHEMBL446711	ChEMBL	6.5	—	—	Cc1ccc(C(=O)CSC(=S)SCCc2ccccc2)cc1
E3 Binder	CHEMBL244602	ChEMBL	6.6	—	—	Cc1ccc(C(=O)CSC(=S)SCc2ccccc2)cc1
E3 Binder	CHEMBL4853947	ChEMBL	7.4	—	—	Cc1ccc(C(=O)N(CC(=O)NC2CCCCC2)Cc2ccc(C(=O)NO)cc2)c(C)c1
E3 Binder	CHEMBL4868526	ChEMBL	7.22	—	—	Cc1ccc(C(=O)N(CC(=O)NCc2ccccc2)Cc2ccc(C(=O)NO)cc2)c(C)c1
E3 Binder	CHEMBL4539004	ChEMBL	7.78	—	—	Cc1ccc(C(=O)N(CCC(=O)NCc2ccccc2)Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL154302	ChEMBL	6.85	—	—	Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4873055	ChEMBL	7.31	—	—	Cc1ccc(C(=O)NO)cc1F
E3 Binder	CHEMBL3798183	ChEMBL	7.05	—	—	Cc1ccc(C(=O)NO)cc1NC(=O)c1ccc2ccccc2n1
E3 Binder	CHEMBL3797597	ChEMBL	6.05	GOW	—	Cc1ccc(C(=O)NO)cc1NC(=O)c1ccccc1
E3 Binder	CHEMBL4877419	ChEMBL	7.16	—	—	Cc1ccc(C(=O)NO)cn1
E3 Binder	CHEMBL2312167	ChEMBL	7.74	—	—	Cc1ccc(C(=O)NOCCCCCC(=O)NO)cc1C
E3 Binder	CHEMBL3354914	ChEMBL	6.66	—	—	Cc1ccc(C(=O)N[C@H](COc2cccc(/C=C/C(=O)NO)c2)Cc2c[nH]c3ccccc23)cc1
E3 Binder	CHEMBL4757957	ChEMBL	8.8	—	—	Cc1ccc(C(=O)Nc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4209463	ChEMBL	7.92	—	—	Cc1ccc(C(=O)c2ccc3c(ccn3Cc3ccc(C(=O)NO)cc3)c2)cc1
E3 Binder	CHEMBL1093357	ChEMBL	6.85	—	—	Cc1ccc(C)c(NC(=O)CCCCC(=O)NO)c1
E3 Binder	CHEMBL4548656	ChEMBL	6.58	—	—	Cc1ccc(C/C(=N\O)C(=O)NCCSSCCNC(=O)/C(Cc2ccc(C)cc2)=N/O)cc1
E3 Binder	CHEMBL3655970	ChEMBL	8.52	—	—	Cc1ccc(C2(Nc3ncc(C(=O)NO)cn3)CC2)cc1
E3 Binder	CHEMBL4878639	ChEMBL	7.08	—	—	Cc1ccc(CC2(c3ccccc3)NC(=O)N(Cc3ccc(C(=O)NO)cc3)C2=O)cc1
E3 Binder	CHEMBL5075515	ChEMBL	8.22	—	—	Cc1ccc(CN(Cc2ccc(C(=O)NO)cc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL4562382	ChEMBL	7.77	—	—	Cc1ccc(CN2C(=O)N(C3CCCCC3)C(=O)C2CCC(=O)NCc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4532064	ChEMBL	7.99	—	—	Cc1ccc(CN2C(=O)N(C3CCCCC3)C(=O)C2CCC(=O)Nc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4850829	ChEMBL	7.42	—	—	Cc1ccc(CN2C(=O)N(Cc3ccc(C(=O)NO)cc3)C(=O)C2Cc2ccccc2)cc1
E3 Binder	CHEMBL4442442	ChEMBL	7.72	—	—	Cc1ccc(CN2C(=O)N(c3ccc(Cl)cc3)C(=O)C2CCC(=O)NCc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4445862	ChEMBL	8.36	—	—	Cc1ccc(CN2C(=O)N(c3ccc(Cl)cc3)C(=O)C2CCC(=O)Nc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL197949	ChEMBL	6.32	—	—	Cc1ccc(CN2C(=O)c3ccc(/C=C/C(=O)NO)cc3C2=O)cc1
E3 Binder	CHEMBL4859429	ChEMBL	7.75	—	—	Cc1ccc(CN2CC(=O)N(Cc3ccc(C(=O)NO)cc3)C2=O)cc1
E3 Binder	CHEMBL4517151	ChEMBL	7.25	—	—	Cc1ccc(CN2CCC(c3noc(CN(C)c4ncc(C(=O)NO)cn4)n3)CC2)cc1
E3 Binder	CHEMBL4580143	ChEMBL	7.84	—	—	Cc1ccc(CNC(=O)CCN(Cc2ccc(C(=O)NO)cc2)C(=O)c2ccc(N(C)C)cc2)cc1
E3 Binder	CHEMBL5274591	ChEMBL	7.34	—	—	Cc1ccc(COc2cccc3ccc(C(=O)NCc4ccc(C(=O)NO)cc4)nc23)cc1
E3 Binder	CHEMBL4760813	ChEMBL	6.54	—	—	Cc1ccc(Cc2cn(CCCCCC(=O)NO)c3ccc(-c4c(C)noc4C)cc23)cc1
E3 Binder	CHEMBL4741281	ChEMBL	6.54	—	—	Cc1ccc(Cc2cn(CCCCCCC(=O)NO)c3ccc(-c4c(C)noc4C)cc23)cc1
E3 Binder	CHEMBL4063718	ChEMBL	7.53	—	—	Cc1ccc(F)c(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c1
E3 Binder	CHEMBL3675761	ChEMBL	7.51	—	—	Cc1ccc(N(CCCCCCC(=O)NO)c2ccccn2)nc1
E3 Binder	CHEMBL4549490	ChEMBL	6.77	—	—	Cc1ccc(NC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)c2ccc(/C=C/C(=O)NO)cc2)cc1
E3 Binder	CHEMBL1092032	ChEMBL	6.77	—	—	Cc1ccc(NC(=O)CCCCC(=O)NO)c(C)c1
E3 Binder	CHEMBL1092762	ChEMBL	7.52	—	—	Cc1ccc(NC(=O)CCCCC(=O)NO)cc1
E3 Binder	CHEMBL1093359	ChEMBL	7.7	—	—	Cc1ccc(NC(=O)CCCCC(=O)NO)cc1C
E3 Binder	CHEMBL3098605	ChEMBL	7.92	—	—	Cc1ccc(NC(=O)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL4458544	ChEMBL	7.51	—	—	Cc1ccc(NC(=O)CCN(Cc2ccc(C(=O)NO)cc2)C(=O)c2cc(C)cc(C)c2)cc1
E3 Binder	CHEMBL4522149	ChEMBL	7.71	—	—	Cc1ccc(NC(=O)CCN(Cc2ccc(C(=O)NO)cc2)C(=O)c2ccc(N(C)C)cc2)cc1
E3 Binder	CHEMBL4455083	ChEMBL	7.97	—	—	Cc1ccc(NC(=O)CCN(Cc2ccc(C(=O)NO)cc2)C(=O)c2ccccc2)cc1
E3 Binder	CHEMBL4098365	ChEMBL	6.1	—	—	Cc1ccc(NC(=O)CN(CCCCCC(=O)NO)C(=O)c2cc(C)cc(C)c2)cc1
E3 Binder	CHEMBL4080343	ChEMBL	6.97	—	—	Cc1ccc(NC(=O)CN(CCCCCC(=O)NO)C(=O)c2ccc(N(C)C)cc2)cc1
E3 Binder	CHEMBL4162282	ChEMBL	8.52	HBJ	—	Cc1ccc(NC(=O)CN(Cc2ccc(C(=O)NO)cc2)C(=O)c2ccc(N(C)C)cc2)cc1
E3 Binder	CHEMBL3923499	ChEMBL	8.7	—	—	Cc1ccc(NC(=O)N2CCC(Nc3ncc(C(=O)NO)cn3)(c3ccccc3)CC2)cc1
E3 Binder	CHEMBL3098606	ChEMBL	8.4	—	—	Cc1ccc(NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCC(=O)N2)cc1
E3 Binder	CHEMBL3356917	ChEMBL	8.7	—	—	Cc1ccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCCC(=O)N2)cc1
E3 Binder	CHEMBL4225611	ChEMBL	7.65	—	—	Cc1ccc(NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)/C=C/c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL4202863	ChEMBL	7.13	—	—	Cc1ccc(NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL1080580	ChEMBL	7.39	—	—	Cc1ccc(NC(=O)c2ccc(/C=C/C(=O)NO)cc2)cc1Nc1nc(-c2cccnc2)cs1
E3 Binder	CHEMBL493315	ChEMBL	7.41	—	—	Cc1ccc(NC(=O)c2ccc(/C=C/C(=O)NO)s2)cc1Nc1ncc(-c2cccnc2)s1
E3 Binder	CHEMBL521652	ChEMBL	7.05	—	—	Cc1ccc(NC(=O)c2ccc(C(=O)NO)cc2)cc1Nc1ncc(-c2cccnc2)s1
E3 Binder	CHEMBL515109	ChEMBL	6.34	—	—	Cc1ccc(NC(=O)c2ccc(C(=O)Nc3ccccc3N)s2)cc1Nc1ncc(-c2cccnc2)s1
E3 Binder	CHEMBL4861336	ChEMBL	7.1	—	—	Cc1ccc(NC(=O)c2ccc3c(c2)N(Cc2ccc(C(=O)NO)cc2)c2ccccc2S3)nc1
E3 Binder	CHEMBL4303329	ChEMBL	6.08	—	—	Cc1ccc(NCCCc2ccccc2)c(N)c1
E3 Binder	CHEMBL514351	ChEMBL	7.44	—	—	Cc1ccc(NCc2ccc(/C=C/C(=O)NO)cc2)cc1Nc1nccc(-c2cccnc2)n1
E3 Binder	CHEMBL3692642	ChEMBL	6.13	—	—	Cc1ccc(NS(=O)(=O)c2ccc(-c3noc(C(F)(F)F)n3)cc2)cc1
E3 Binder	CHEMBL404604	ChEMBL	7.75	—	—	Cc1ccc(NS(=O)(=O)c2cccc(/C=C/C(=O)NO)c2)cc1
E3 Binder	CHEMBL5204931	ChEMBL	7.82	—	—	Cc1ccc(Nc2nc(Cl)nc3c2ncn3CCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3652228	ChEMBL	8.05	—	—	Cc1ccc(Nc2ncc(C(=O)NO)cn2)cc1
E3 Binder	CHEMBL4209243	ChEMBL	6.09	—	—	Cc1ccc(Nc2nccc(N(C)c3ccc4c(C)n(C)nc4c3)n2)cc1C(=O)NCCCCCC(=O)NO
E3 Binder	CHEMBL3601337	ChEMBL	8.2	—	—	Cc1ccc(Nc2nccc3ccc(NC(=O)CCCCCCC(=O)NO)cc23)c(Br)c1
E3 Binder	CHEMBL3601336	ChEMBL	7.52	—	—	Cc1ccc(Nc2nccc3ccc(NC(=O)CCCCCCC(=O)NO)cc23)c(Cl)c1
E3 Binder	CHEMBL3601335	ChEMBL	7.39	—	—	Cc1ccc(Nc2nccc3ccc(NC(=O)CCCCCCC(=O)NO)cc23)c(F)c1
E3 Binder	CHEMBL3601333	ChEMBL	8.42	—	—	Cc1ccc(Nc2nccc3ccc(NC(=O)CCCCCCC(=O)NO)cc23)cc1
E3 Binder	CHEMBL3601780	ChEMBL	6.52	—	—	Cc1ccc(Nc2nccc3ccc(NCc4ccc(/C=C/C(=O)NO)cc4)cc23)c(Br)c1
E3 Binder	CHEMBL3601779	ChEMBL	6.54	—	—	Cc1ccc(Nc2nccc3ccc(NCc4ccc(/C=C/C(=O)NO)cc4)cc23)c(Cl)c1
E3 Binder	CHEMBL3601778	ChEMBL	7.23	—	—	Cc1ccc(Nc2nccc3ccc(NCc4ccc(/C=C/C(=O)NO)cc4)cc23)cc1
E3 Binder	CHEMBL3601777	ChEMBL	6.45	—	—	Cc1ccc(Nc2nccc3ccc(NCc4ccc(C(=O)NO)cc4)cc23)cc1
E3 Binder	CHEMBL3339023	ChEMBL	7.71	—	—	Cc1ccc(Nc2ncnc3sc(NC(=O)CCCCCC(=O)NO)cc23)cc1
E3 Binder	CHEMBL3339025	ChEMBL	7.77	—	—	Cc1ccc(Nc2ncnc3sc(NC(=O)CCCCCC(=O)NO)cc23)cc1C
E3 Binder	CHEMBL3339024	ChEMBL	8.27	—	—	Cc1ccc(Nc2ncnc3sc(NC(=O)CCCCCCC(=O)NO)cc23)cc1
E3 Binder	CHEMBL3339026	ChEMBL	7.94	—	—	Cc1ccc(Nc2ncnc3sc(NC(=O)CCCCCCC(=O)NO)cc23)cc1C
E3 Binder	CHEMBL88553	ChEMBL	6.66	—	—	Cc1ccc(O)c(/N=N/c2ccccc2)n1
E3 Binder	CHEMBL2413298	ChEMBL	6.26	—	—	Cc1ccc(OCCCCN(Cc2ccccc2)Cc2ccc(/C=C/C(=O)NO)o2)cc1
E3 Binder	CHEMBL2413296	ChEMBL	6.03	—	—	Cc1ccc(OCCCN(Cc2ccccc2)Cc2ccc(/C=C/C(=O)NO)o2)cc1
E3 Binder	CHEMBL2413289	ChEMBL	6.08	—	—	Cc1ccc(OCCN(CCc2ccc3c(c2)OCO3)Cc2ccc(/C=C/C(=O)NO)o2)cc1
E3 Binder	CHEMBL4303623	ChEMBL	6.32	—	—	Cc1ccc(OCCSc2ncccn2)c(Br)c1
E3 Binder	CHEMBL3930762	ChEMBL	7.89	—	—	Cc1ccc(Oc2ccc(Nc3ncnc4ccc(-c5cn(CCCCCC(=O)NO)nn5)cc34)cc2C)cn1
E3 Binder	CHEMBL3893822	ChEMBL	7.86	—	—	Cc1ccc(Oc2ccc(Nc3ncnc4ccc(-c5cn(CCCCCCC(=O)NO)nn5)cc34)cc2C)cn1
E3 Binder	CHEMBL3938587	ChEMBL	8.35	—	—	Cc1ccc(S(=O)(=O)N2CCC(Nc3ncc(C(=O)NO)cn3)(c3ccccc3)CC2)cc1
E3 Binder	CHEMBL438522	ChEMBL	6.26	—	—	Cc1ccc(S(=O)(=O)N2CCN(c3ncc(/C=C/C(=O)NO)s3)CC2)cc1
E3 Binder	CHEMBL250790	ChEMBL	7.05	—	—	Cc1ccc(S(=O)(=O)N2CCN(c3ncc(C(=O)NO)s3)CC2)cc1
E3 Binder	CHEMBL3233688	ChEMBL	6.2	—	—	Cc1ccc(S(=O)(=O)N[C@H](COc2ccc(/C=C/C(=O)NO)cc2)Cc2c[nH]c3ccccc23)cc1
E3 Binder	CHEMBL250398	ChEMBL	6.23	—	—	Cc1ccc(S(=O)(=O)Nc2ccc(CN3CCC=C(CCC(=O)NO)C3=O)cc2)cc1
E3 Binder	CHEMBL406161	ChEMBL	6.91	—	—	Cc1ccc(S(=O)(=O)Nc2cccc(/C=C/C(=O)NO)c2)cc1
E3 Binder	CHEMBL4517827	ChEMBL	6.77	—	—	Cc1ccc2c(=O)n(CCc3ccccc3)c(=O)n(Cc3ccc(C(=O)NO)cc3)c2c1
E3 Binder	CHEMBL5289831	ChEMBL	6.77	—	—	Cc1ccc2c(=O)n(Cc3ccc(/C=C/C(=O)NO)cc3)cnc2c1
E3 Binder	CHEMBL4745319	ChEMBL	7.75	—	—	Cc1ccc2c(c1)/C(=C1/Nc3ccccc3/C1=N\O)C(=O)N2CCCCCCC(=O)NO
E3 Binder	CHEMBL4793145	ChEMBL	7.7	—	—	Cc1ccc2c(c1)/C(=C1/Nc3ccccc3/C1=N\O)C(=O)N2Cc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL4781628	ChEMBL	8.3	—	—	Cc1ccc2c(c1)/C(=C1/Nc3ccccc3/C1=N\O)C(=O)N2Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4854768	ChEMBL	7.92	—	—	Cc1ccc2c(c1)N(Cc1ccc(C(=O)NO)cc1)CCCC2
E3 Binder	CHEMBL2018296	ChEMBL	8.31	—	—	Cc1ccc2c(c1)c1c(n2Cc2ccc(C(=O)NO)cc2)CCN(C)C1
E3 Binder	CHEMBL4850396	ChEMBL	7.08	—	—	Cc1ccc2c(c1)c1c(n2Cc2ccc(C(=O)NO)cn2)CCN(C)C1
E3 Binder	CHEMBL2018295	ChEMBL	7.94	—	—	Cc1ccc2c3c(n(Cc4ccc(C(=O)NO)cc4)c2c1)CCN(C)C3
E3 Binder	CHEMBL2403445	ChEMBL	6.34	—	—	Cc1ccc2cc(C(=O)NO)sc2c1F
E3 Binder	CHEMBL4064437	ChEMBL	7.94	—	—	Cc1ccc2cccc(NCc3ccc(C(=O)NO)cc3)c2n1
E3 Binder	CHEMBL4849102	ChEMBL	7.88	—	—	Cc1ccc2ccccc2c1N1CC(=O)N(Cc2ccc(C(=O)NO)cc2)C1=O
E3 Binder	CHEMBL5091856	ChEMBL	7.48	—	—	Cc1ccc2nc3c4ccccc4c(NCCCCCCC(=O)NO)nn3c(=O)c2c1
E3 Binder	CHEMBL5092046	ChEMBL	7.43	—	—	Cc1ccc2nc3c4ccccc4c(NCCCCCCCC(=O)NO)nn3c(=O)c2c1
E3 Binder	CHEMBL2337868	ChEMBL	6.09	—	—	Cc1cccc(-c2ccc(Cn3cccc(O)c3=S)cc2)c1
E3 Binder	CHEMBL516732	ChEMBL	7.5	—	—	Cc1cccc(-c2cn(CCCCCC(=O)NO)nn2)c1
E3 Binder	CHEMBL4857331	ChEMBL	6.55	—	—	Cc1cccc(-c2nc(CNc3ccc(C(=O)NO)cc3)n(-c3ccccc3)n2)c1
E3 Binder	CHEMBL5075815	ChEMBL	6.09	—	—	Cc1cccc(-c2ncc(/C=C/C(=O)Nc3ccccc3N)s2)c1
E3 Binder	CHEMBL5274632	ChEMBL	7.83	—	—	Cc1cccc(-c2ncn(Cc3ccc(C(=O)NO)cc3)n2)c1
E3 Binder	CHEMBL509445	ChEMBL	6.17	—	—	Cc1cccc(-c2noc(-c3ccc(C(=O)C(F)(F)F)s3)n2)c1
E3 Binder	CHEMBL4871029	ChEMBL	6.41	—	—	Cc1cccc(-n2nc(-c3ccccc3)nc2CNc2ccc(C(=O)NO)cc2)c1
E3 Binder	CHEMBL88612	ChEMBL	6.46	—	—	Cc1cccc(/C=C/c2ccccc2)n1
E3 Binder	CHEMBL66654	ChEMBL	6.32	—	—	Cc1cccc(C#Cc2ccccc2)n1
E3 Binder	CHEMBL2381522	ChEMBL	6.19	—	—	Cc1cccc(C(=O)NO)c1
E3 Binder	CHEMBL2312164	ChEMBL	7.57	—	—	Cc1cccc(C(=O)NOCCCCCC(=O)NO)c1
E3 Binder	CHEMBL3655937	ChEMBL	7.68	—	—	Cc1cccc(C)c1CNc1ncc(C(=O)NO)cn1
E3 Binder	CHEMBL3693754	ChEMBL	7.43	—	—	Cc1cccc(C)c1N(C(=O)C(C)C)c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693757	ChEMBL	7.18	—	—	Cc1cccc(C)c1N(C(=O)CC(C)C)c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693749	ChEMBL	8.05	—	—	Cc1cccc(C)c1N(C)c1ccc(C(=O)N(C)CCCCCCC(=O)NO)c(F)c1
E3 Binder	CHEMBL3693747	ChEMBL	8.3	—	—	Cc1cccc(C)c1N(C)c1ccc(C(=O)NCCCCCCC(=O)NO)c(F)c1
E3 Binder	CHEMBL3693770	ChEMBL	7.62	—	—	Cc1cccc(C)c1N(c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1)c1ncccn1
E3 Binder	CHEMBL3693765	ChEMBL	8.4	—	—	Cc1cccc(C)c1N(c1ccc(C(=O)NCCCCCCC(=O)NO)cc1)c1ncccn1
E3 Binder	CHEMBL3693787	ChEMBL	8.3	—	—	Cc1cccc(C)c1N(c1ccccc1)c1ncc(C(=O)NCCCCCCC(=O)NO)cn1
E3 Binder	CHEMBL1093358	ChEMBL	6.21	—	—	Cc1cccc(C)c1NC(=O)CCCCC(=O)NO
E3 Binder	CHEMBL3693772	ChEMBL	6.44	—	—	Cc1cccc(C)c1Nc1ccc(C(=O)N(C)CCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693767	ChEMBL	7.34	—	—	Cc1cccc(C)c1Nc1ccc(C(=O)N(C)CCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693726	ChEMBL	8.15	—	—	Cc1cccc(C)c1Nc1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693758	ChEMBL	7.92	—	—	Cc1cccc(C)c1Nc1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1F
E3 Binder	CHEMBL3693746	ChEMBL	8.52	—	—	Cc1cccc(C)c1Nc1ccc(C(=O)NCCCCCCC(=O)NO)c(F)c1
E3 Binder	CHEMBL3693711	ChEMBL	8.52	—	—	Cc1cccc(C)c1Nc1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693755	ChEMBL	8.4	—	—	Cc1cccc(C)c1Nc1ccc(C(=O)NCCCCCCC(=O)NO)cc1F
E3 Binder	CHEMBL3693788	ChEMBL	8.52	—	—	Cc1cccc(C)c1Nc1ccc2c(c1)CN(CCCCCCC(=O)NO)C2=O
E3 Binder	CHEMBL3693760	ChEMBL	7.57	—	—	Cc1cccc(C)c1Nc1cccc(C(=O)N(C)CCCCCCC(=O)NO)c1
E3 Binder	CHEMBL3693759	ChEMBL	8.0	—	—	Cc1cccc(C)c1Nc1cccc(C(=O)NCCCCCCC(=O)NO)c1
E3 Binder	CHEMBL3693763	ChEMBL	7.32	—	—	Cc1cccc(C)c1Nc1ccccc1C(=O)N(C)CCCCCCC(=O)NO
E3 Binder	CHEMBL3693733	ChEMBL	7.48	—	—	Cc1cccc(C)c1Nc1ncc(C(=O)N(C)CCCCCCC(=O)NO)cn1
E3 Binder	CHEMBL3693724	ChEMBL	7.48	—	—	Cc1cccc(C)c1Nc1ncc(C(=O)NCCCCCCC(=O)NO)cn1
E3 Binder	CHEMBL3656003	ChEMBL	8.52	—	—	Cc1cccc(C2(Nc3ncc(C(=O)NO)cn3)CC2)c1
E3 Binder	CHEMBL5196979	ChEMBL	6.4	—	—	Cc1cccc(C2CC(=O)N2C2CCN(C(=O)NCc3ccc(C(=O)NO)cc3)CC2)c1
E3 Binder	CHEMBL3356937	ChEMBL	7.82	—	—	Cc1cccc(CCNC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCCC(=O)N2)c1
E3 Binder	CHEMBL4744442	ChEMBL	6.54	—	—	Cc1cccc(Cc2cn(CCCCCC(=O)NO)c3ccc(-c4c(C)noc4C)cc23)c1
E3 Binder	CHEMBL4752047	ChEMBL	6.54	—	—	Cc1cccc(Cc2cn(CCCCCCC(=O)NO)c3ccc(-c4c(C)noc4C)cc23)c1
E3 Binder	CHEMBL3693719	ChEMBL	8.4	—	—	Cc1cccc(Cl)c1N(C)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693764	ChEMBL	7.96	—	—	Cc1cccc(Cl)c1Nc1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL1089339	ChEMBL	7.52	—	—	Cc1cccc(NC(=O)CCCCC(=O)NO)c1
E3 Binder	CHEMBL1093043	ChEMBL	6.69	—	—	Cc1cccc(NC(=O)CCCCC(=O)NO)c1C
E3 Binder	CHEMBL3098603	ChEMBL	7.66	—	—	Cc1cccc(NC(=O)CCCCCCC(=O)NO)c1
E3 Binder	CHEMBL3098604	ChEMBL	8.52	—	—	Cc1cccc(NC(=O)[C@H](CCCCCC(=O)NO)NC(=O)[C@H]2CCC(=O)N2)c1
E3 Binder	CHEMBL3356922	ChEMBL	9.0	—	—	Cc1cccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCC(=O)N2)c1
E3 Binder	CHEMBL3356916	ChEMBL	9.0	—	—	Cc1cccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@@H]2CCCC(=O)N2)c1
E3 Binder	CHEMBL3356923	ChEMBL	8.7	—	—	Cc1cccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@H]2CCC(=O)N2)c1
E3 Binder	CHEMBL3356924	ChEMBL	9.0	—	—	Cc1cccc(NC(=O)[C@H](CCCCCS)NC(=O)[C@H]2CCC(=O)N2C)c1
E3 Binder	CHEMBL3692639	ChEMBL	6.33	—	—	Cc1cccc(NS(=O)(=O)c2ccc(-c3noc(C(F)(F)F)n3)cc2)c1
E3 Binder	CHEMBL3233694	ChEMBL	6.17	—	—	Cc1cccc(Nc2ccccc2C(=O)N[C@H](COc2ccc(/C=C/C(=O)NO)cc2)Cc2c[nH]c3ccccc23)c1C
E3 Binder	CHEMBL565269	ChEMBL	6.69	—	—	Cc1cccc(Nc2nc(-c3ccncc3)cs2)c1
E3 Binder	CHEMBL5283177	ChEMBL	7.87	—	—	Cc1cccc2c(C(=O)N3CCN(Cc4ccc(C(=O)NO)cc4)CC3)c[nH]c12
E3 Binder	CHEMBL2018294	ChEMBL	7.46	—	—	Cc1cccc2c3c(n(Cc4ccc(C(=O)NO)cc4)c12)CCN(C)C3
E3 Binder	CHEMBL2337867	ChEMBL	6.51	—	—	Cc1ccccc1-c1ccc(Cn2cccc(O)c2=S)cc1
E3 Binder	CHEMBL478310	ChEMBL	7.76	—	—	Cc1ccccc1-c1cn(CCCCCC(=O)NO)nn1
E3 Binder	CHEMBL601044	ChEMBL	8.55	—	—	Cc1ccccc1-c1cn(CCCCCCC(=O)NO)nn1
E3 Binder	CHEMBL3110279	ChEMBL	6.2	—	—	Cc1ccccc1-c1cn(CCCCCn2cccc(O)c2=S)nn1
E3 Binder	CHEMBL5187265	ChEMBL	7.29	—	—	Cc1ccccc1C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5188109	ChEMBL	7.57	—	—	Cc1ccccc1C(=O)N(CC(=O)NC(C)(C)C)Cc1ccc(C(=O)NO)cc1F
E3 Binder	CHEMBL4854335	ChEMBL	7.52	—	—	Cc1ccccc1C(=O)N(CC(=O)NC12CC3CC(CC(C3)C1)C2)Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5190554	ChEMBL	7.75	—	—	Cc1ccccc1C(=O)N(CC(=O)NC1CCCCC1)Cc1ccc(C(=O)NO)cc1F
E3 Binder	CHEMBL4847978	ChEMBL	7.52	—	—	Cc1ccccc1C(=O)N(CC(=O)NCc1ccccc1)Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4781216	ChEMBL	7.22	—	—	Cc1ccccc1C(=O)N(Cc1ccc(C(=O)NO)cc1)Cc1nnnn1C1CCCCC1
E3 Binder	CHEMBL3655996	ChEMBL	8.7	—	—	Cc1ccccc1C1(Nc2ncc(C(=O)NO)cn2)CC1
E3 Binder	CHEMBL4740417	ChEMBL	6.54	—	—	Cc1ccccc1Cc1cn(CCCCCC(=O)NO)c2ccc(-c3c(C)noc3C)cc12
E3 Binder	CHEMBL4781636	ChEMBL	6.54	—	—	Cc1ccccc1Cc1cn(CCCCCCC(=O)NO)c2ccc(-c3c(C)noc3C)cc12
E3 Binder	CHEMBL3693768	ChEMBL	8.05	—	—	Cc1ccccc1N(c1ccccc1)c1ncc(C(=O)NCCCCCCC(=O)NO)cn1
E3 Binder	CHEMBL3693785	ChEMBL	8.05	—	—	Cc1ccccc1N(c1ncc(C(=O)NCCCCCCC(=O)NO)cn1)c1ccccc1C
E3 Binder	CHEMBL4577052	ChEMBL	6.64	—	—	Cc1ccccc1NC(=O)C(Cc1c[nH]c2ccccc12)NC(=O)c1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL1076794	ChEMBL	6.6	—	—	Cc1ccccc1NC(=O)CCCCC(=O)NO
E3 Binder	CHEMBL3692637	ChEMBL	6.16	—	—	Cc1ccccc1NS(=O)(=O)c1ccc(-c2noc(C(F)(F)F)n2)cc1
E3 Binder	CHEMBL4082812	ChEMBL	7.06	—	—	Cc1ccccc1Nc1ncnc2cc(NC(=O)CCCCCCC(=O)NO)sc12
E3 Binder	CHEMBL3967312	ChEMBL	8.35	—	—	Cc1ccccc1S(=O)(=O)N1CCC(Nc2ncc(C(=O)NO)cn2)(c2ccccc2)CC1
E3 Binder	CHEMBL3693762	ChEMBL	7.57	—	—	Cc1cccnc1N(c1ccccc1)c1ccc(C(=O)N(C)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3693737	ChEMBL	7.7	—	—	Cc1cccnc1N(c1ccccc1)c1ccc(C(=O)NCCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3914736	ChEMBL	8.66	—	—	Cc1ccnc(NC(=O)NCc2ccc(C(=O)NO)cc2)c1
E3 Binder	CHEMBL4856928	ChEMBL	7.51	—	—	Cc1ccsc1-c1nc(CNc2ccc(C(=O)NO)cc2)n(-c2ccccc2)n1
E3 Binder	CHEMBL3979548	ChEMBL	8.29	—	—	Cc1cn(Cc2ccc(C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL3770555	ChEMBL	7.63	—	—	Cc1cnc(-c2nc(C(=O)NCCCCC(=O)C(F)(F)F)c(C3CC3)s2)s1
E3 Binder	CHEMBL4435503	ChEMBL	7.73	—	—	Cc1cnc(-c2nc(C(=O)N[C@@H](C)c3ccc(C(=O)NO)cc3)c(C3CC3)s2)s1
E3 Binder	CHEMBL4289006	ChEMBL	8.68	—	—	Cc1cnc(Nc2ccc(N3CCN(C)CC3)cc2)nc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL4281785	ChEMBL	8.43	—	—	Cc1cnc(Nc2ccc(N3CCOCC3)cc2)nc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3948298	ChEMBL	7.04	—	—	Cc1csc(-c2nc(C(=O)NCCCCC(=O)NO)c(C3CC3)s2)n1
E3 Binder	CHEMBL4577858	ChEMBL	7.72	—	—	Cc1csc(-c2nc(C(=O)N[C@@H](C)c3ccc(C(=O)NO)cc3)c(C3CC3)s2)n1
E3 Binder	CHEMBL4560818	ChEMBL	6.86	—	—	Cc1csc(Nc2ccc(C(=O)NO)cc2)n1
E3 Binder	CHEMBL1164729	ChEMBL	7.26	TEI	—	Cc1nc(-c2ccc(OCC(C)C)c(C#N)c2)sc1C(=O)O
E3 Binder	CHEMBL1096432	ChEMBL	6.92	—	—	Cc1nc(-c2cccc(/C=C/C(=O)NO)c2)n(CCN2CCOCC2)c1-c1ccccc1
E3 Binder	CHEMBL1095718	ChEMBL	6.8	—	—	Cc1nc(-c2cccc(/C=C/C(=O)NO)c2)n(CCN2CCOCC2)c1C
E3 Binder	CHEMBL1095972	ChEMBL	7.1	—	—	Cc1nc(-c2cccc(/C=C/C(=O)NO)c2)n(CCN2CCOCC2)c1Cc1ccccc1
E3 Binder	CHEMBL1096433	ChEMBL	7.1	—	—	Cc1nc(-c2cccc(/C=C/C(=O)NO)c2)n(CCc2ccccc2)c1-c1ccccc1
E3 Binder	CHEMBL1095719	ChEMBL	7.2	—	—	Cc1nc(-c2cccc(/C=C/C(=O)NO)c2)n(CCc2ccccc2)c1C
E3 Binder	CHEMBL1096705	ChEMBL	7.3	—	—	Cc1nc(-c2cccc(/C=C/C(=O)NO)c2)n(CCc2ccccc2)c1Cc1ccccc1
E3 Binder	CHEMBL1095120	ChEMBL	7.0	—	—	Cc1nc(-c2cccc(/C=C/C(=O)NO)c2)n([C@@H]2CCCN(C(C)C)C2)c1-c1ccccc1
E3 Binder	CHEMBL1095118	ChEMBL	7.1	—	—	Cc1nc(-c2cccc(/C=C/C(=O)NO)c2)n([C@@H]2CCCN(C)C2)c1-c1ccccc1
E3 Binder	CHEMBL1095400	ChEMBL	7.1	—	—	Cc1nc(-c2ccccc2)n(CCc2ccccc2)c1-c1cccc(/C=C/C(=O)NO)c1
E3 Binder	CHEMBL3925099	ChEMBL	6.25	—	—	Cc1nc(-c2nc(C(=O)NCCCCC(=O)NO)c(C3CC3)s2)sc1C
E3 Binder	CHEMBL1096034	ChEMBL	6.92	—	—	Cc1nc(C)n(CCc2ccccc2)c1-c1cccc(/C=C/C(=O)NO)c1
E3 Binder	CHEMBL1094094	ChEMBL	7.2	—	—	Cc1nc(Cc2ccccc2)n(CCc2ccccc2)c1-c1cccc(/C=C/C(=O)NO)c1
E3 Binder	CHEMBL3775521	ChEMBL	8.07	—	—	Cc1nc(N(C)c2ccc(OCC(=O)NO)cc2)c2ccccc2n1
E3 Binder	CHEMBL3775662	ChEMBL	6.71	—	—	Cc1nc(N(C)c2ccc(OCCCC(=O)NO)cc2)c2ccccc2n1
E3 Binder	CHEMBL3775817	ChEMBL	7.24	—	—	Cc1nc(N(C)c2ccc(OCCCCC(=O)NO)cc2)c2ccccc2n1
E3 Binder	CHEMBL3775409	ChEMBL	7.47	—	—	Cc1nc(N(C)c2ccc(OCCCCCC(=O)NO)cc2)c2ccccc2n1
E3 Binder	CHEMBL4526673	ChEMBL	8.1	—	—	Cc1nc(N)nc(N[C@@H](C)c2nc3cccc(NCc4ccc(C(=O)NO)cc4)c3c(=O)n2-c2ccccc2)c1C#N
E3 Binder	CHEMBL3945209	ChEMBL	6.0	—	—	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CC(=O)NO)CC2)n1
E3 Binder	CHEMBL3947855	ChEMBL	6.0	—	—	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCC(=O)NO)CC2)n1
E3 Binder	CHEMBL3964750	ChEMBL	6.0	—	—	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCC(=O)NO)CC2)n1
E3 Binder	CHEMBL3907624	ChEMBL	7.0	—	—	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCC(=O)NO)CC2)n1
E3 Binder	CHEMBL3904339	ChEMBL	7.0	—	—	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCC(=O)NO)CC2)n1
E3 Binder	CHEMBL2425956	ChEMBL	6.16	—	—	Cc1nc2c(/C=C/C(=O)NO)cccc2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL5220945	ChEMBL	8.23	—	—	Cc1nc2c(F)cc(-c3nc(Nc4ccc(CNC(=O)CC(=O)NO)cc4)ncc3F)cc2n1C(C)C
E3 Binder	CHEMBL5190225	ChEMBL	8.23	—	—	Cc1nc2c(F)cc(-c3nc(Nc4ccc(CNC(=O)CCCCCCC(=O)NO)cc4)ncc3F)cc2n1C(C)C
E3 Binder	CHEMBL47529	ChEMBL	6.45	8WX	—	Cc1nc2c(OCc3ccccc3)cccn2c1CC#N
E3 Binder	CHEMBL3775581	ChEMBL	7.77	—	—	Cc1nc2c(c(N(C)c3ccc(OCC(=O)NO)cc3)n1)CCC2
E3 Binder	CHEMBL3775269	ChEMBL	7.4	—	—	Cc1nc2c(c(N(C)c3ccc(OCCCC(=O)NO)cc3)n1)CCC2
E3 Binder	CHEMBL3774691	ChEMBL	7.2	—	—	Cc1nc2c(c(N(C)c3ccc(OCCCCC(=O)NO)cc3)n1)CCC2
E3 Binder	CHEMBL3775072	ChEMBL	7.7	—	—	Cc1nc2c(c(N(C)c3ccc(OCCCCCC(=O)NO)cc3)n1)CCC2
E3 Binder	CHEMBL4442157	ChEMBL	7.43	—	—	Cc1nc2c(s1)Sc1ccccc1N2Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL2425955	ChEMBL	7.06	—	—	Cc1nc2cc(/C=C/C(=O)NO)ccc2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL2425959	ChEMBL	7.82	—	—	Cc1nc2cc(/C=C/C(=O)NO)ccc2c(=O)n1CCc1c[nH]c2ccccc12
E3 Binder	CHEMBL2425958	ChEMBL	7.54	—	—	Cc1nc2cc(/C=C/C(=O)NO)ccc2c(=O)n1CCc1ccccc1
E3 Binder	CHEMBL2425957	ChEMBL	7.62	—	—	Cc1nc2cc(/C=C/C(=O)NO)ccc2c(=O)n1Cc1ccccc1
E3 Binder	CHEMBL3907479	ChEMBL	7.08	LWJ	—	Cc1nc2ccc(-n3ncc(C(=O)c4cc5ccccc5[nH]4)c3N)cc2[nH]1
E3 Binder	CHEMBL2425954	ChEMBL	7.5	—	—	Cc1nc2ccc(/C=C/C(=O)NO)cc2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL5267835	ChEMBL	6.12	—	—	Cc1nc2ccc(Cl)cc2c(=O)n1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL142931	ChEMBL	7.42	—	—	Cc1nc2ccccc2n1CCNCc1ccc(/C=C/C(=O)NO)cc1
E3 Binder	CHEMBL3918660	ChEMBL	8.04	—	—	Cc1nc2ccccc2n1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4080014	ChEMBL	9.1	—	—	Cc1nc2ccccc2n1Cc1ccc(C(=O)NO)cc1F
E3 Binder	CHEMBL4469978	ChEMBL	6.45	—	—	Cc1nnc(-c2ccc(C(=O)NO)cc2)[nH]1
E3 Binder	CHEMBL471344	ChEMBL	6.19	—	—	Cc1noc(-c2ccc(C(=O)C(F)(F)F)s2)n1
E3 Binder	CHEMBL4780262	ChEMBL	7.24	—	—	Cc1noc(C)c1-c1ccc([C@H]2C[C@@H]2NCC2CCN(CCCc3ccc(C(=O)NO)cc3)CC2)cc1
E3 Binder	CHEMBL4740945	ChEMBL	6.54	—	—	Cc1noc(C)c1-c1ccc2c(c1)c(CCc1ccc(F)cc1)cn2CCCCCC(=O)NO
E3 Binder	CHEMBL4788948	ChEMBL	6.54	—	—	Cc1noc(C)c1-c1ccc2c(c1)c(CCc1ccc(F)cc1)cn2CCCCCCC(=O)NO
E3 Binder	CHEMBL4751464	ChEMBL	6.54	—	—	Cc1noc(C)c1-c1ccc2c(c1)c(CCc1ccccc1)cn2CCCCCC(=O)NO
E3 Binder	CHEMBL4761763	ChEMBL	6.54	—	—	Cc1noc(C)c1-c1ccc2c(c1)c(CCc1ccccc1)cn2CCCCCCC(=O)NO
E3 Binder	CHEMBL4749697	ChEMBL	6.54	—	—	Cc1noc(C)c1-c1ccc2c(c1)c(Cc1ccc(F)cc1)cn2CCCCCC(=O)NO
E3 Binder	CHEMBL4788583	ChEMBL	6.54	—	—	Cc1noc(C)c1-c1ccc2c(c1)c(Cc1cccc(C(F)(F)F)c1)cn2CCCCCC(=O)NO
E3 Binder	CHEMBL4784085	ChEMBL	6.54	—	—	Cc1noc(C)c1-c1ccc2c(c1)c(Cc1ccccc1)cn2CCCCCC(=O)NO
E3 Binder	CHEMBL4779677	ChEMBL	6.54	—	—	Cc1noc(C)c1-c1ccc2c(c1)c(Cc1ccccc1)cn2CCCCCCC(=O)NO
E3 Binder	CHEMBL5171575	ChEMBL	7.5	—	—	Cc1noc(C)c1-c1cn(Cc2ccc(C(=O)NO)cc2)c(=O)c(N2CCOCC2)n1
E3 Binder	CHEMBL4553337	ChEMBL	6.34	—	—	Cc1noc(C)c1-c1nc2sc3c(c2c(=O)[nH]1)CCN(CC(=O)NO)C3
E3 Binder	CHEMBL4581033	ChEMBL	6.41	—	—	Cc1noc(C)c1-c1nc2sc3c(c2c(=O)[nH]1)CCN(CC(=O)Nc1ccccc1N)C3
E3 Binder	CHEMBL4436262	ChEMBL	6.33	—	—	Cc1noc(C)c1-c1nc2sc3c(c2c(=O)[nH]1)CCN(CCCC(=O)NO)C3
E3 Binder	CHEMBL4530039	ChEMBL	6.81	—	—	Cc1noc(C)c1-c1nc2sc3c(c2c(=O)[nH]1)CCN(CCCCCC(=O)NO)C3
E3 Binder	CHEMBL4438753	ChEMBL	6.71	—	—	Cc1noc(C)c1-c1nc2sc3c(c2c(=O)[nH]1)CCN(CCCCCC(=O)Nc1ccccc1N)C3
E3 Binder	CHEMBL2417783	ChEMBL	6.58	—	—	Cc1onc(-c2ccccc2)c1C(=O)NCCCCCNC(=O)CS
E3 Binder	CHEMBL2417784	ChEMBL	6.55	—	—	Cc1onc(-c2ccccc2)c1C(=O)NCCCCCNC(=O)[C@@H](C)S
E3 Binder	CHEMBL5288844	ChEMBL	6.07	—	—	Cc1onc(-c2ccccc2)c1COCCCCCNC(=O)C(C)S
E3 Binder	CHEMBL5280419	ChEMBL	6.08	—	—	Cc1onc(-c2ccccc2)c1COCCCCCNC(=O)[C@@H](C)S
E3 Binder	CHEMBL5198491	ChEMBL	7.5	—	—	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)NCCCC(=O)Nc1ccccc1N)c1nnc(C)n1-2
E3 Binder	CHEMBL4850926	ChEMBL	7.68	—	—	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)Nc1ccc(C(=O)NO)cc1)c1nnc(C)n1-2
E3 Binder	CHEMBL1957266	ChEMBL	6.54	—	—	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)OC(C)(C)C)c1nnc(C)n1-2
E3 Binder	CHEMBL5093798	ChEMBL	7.07	—	—	Cl.Cn1cc(CN2CC3(CCN(c4ncc(C(=O)NO)cn4)C3)C2)c2ccc(C#N)cc21
E3 Binder	CHEMBL4167599	ChEMBL	7.3	—	—	Cl.NCCCCNCCCCNCCCN1C(=O)c2ccc3c4c(ccc(c24)C1=O)C(=O)N(CCCCCC(=O)NO)C3=O
E3 Binder	CHEMBL4175475	ChEMBL	6.28	—	—	Cl.NCCCNCCCCNCCCN1C(=O)c2ccc3c4c(ccc(c24)C1=O)C(=O)N(CCCCCC(=O)NO)C3=O
E3 Binder	CHEMBL4160757	ChEMBL	6.39	—	—	Cl.NCCCNCCCN1C(=O)c2ccc3c4c(ccc(c24)C1=O)C(=O)N(CCCCCC(=O)NO)C3=O
E3 Binder	CHEMBL4171407	ChEMBL	6.43	—	—	Cl.NCCCNCCCNCCCN1C(=O)c2ccc3c4c(ccc(c24)C1=O)C(=O)N(CCCCCC(=O)NO)C3=O
E3 Binder	CHEMBL4172024	ChEMBL	6.26	—	—	Cl.NCCCNCCNCCCN1C(=O)c2ccc3c4c(ccc(c24)C1=O)C(=O)N(CCCCCC(=O)NO)C3=O
E3 Binder	CHEMBL1630844	ChEMBL	8.12	—	—	Cl.Nc1cccc(-c2csc(NC(=O)CCCCCCC(=O)NO)n2)c1
E3 Binder	CHEMBL470843	ChEMBL	6.76	—	—	Cl.O=C(/C=C/c1ccc(-c2cc(CN3CCOCC3)on2)cc1)NO
E3 Binder	CHEMBL3233708	ChEMBL	6.8	—	—	Cl.O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NCc2ccc(Cl)cc2)cc1)NO
E3 Binder	CHEMBL3233707	ChEMBL	6.83	—	—	Cl.O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NCc2ccc(F)cc2)cc1)NO
E3 Binder	CHEMBL3233706	ChEMBL	6.7	—	—	Cl.O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NCc2ccccc2)cc1)NO
E3 Binder	CHEMBL5195044	ChEMBL	7.3	—	—	Cl.O=C(CCCCCCNC(=O)c1ccc(/C=C2\CCn3c2nc2cc(NCCCN4CCCC4)c(F)cc2c3=O)cc1)NO
E3 Binder	CHEMBL4859948	ChEMBL	8.6	—	—	Cl.O=C(NO)c1ccc(CN2c3ccccc3Sc3ccccc32)nc1
E3 Binder	CHEMBL1098379	ChEMBL	7.1	—	—	Cn1c(-c2cccc(/C=C/C(=O)NO)c2)nc2ccccc21
E3 Binder	CHEMBL3426805	ChEMBL	6.12	—	—	Cn1c(/C=C/C(=O)NO)ccc1/C=C/C(=O)c1cccc(F)c1
E3 Binder	CHEMBL1213458	ChEMBL	7.52	—	—	Cn1c(/C=C/C(=O)NO)ccc1C(=O)Cc1ccccc1
E3 Binder	CHEMBL4795944	ChEMBL	6.29	—	—	Cn1c(=O)c(OCc2ccc(C(=O)NO)cc2)c(-c2ccccc2)c2ccccc21
E3 Binder	CHEMBL4787955	ChEMBL	7.34	—	—	Cn1c(=O)c(OCc2ccc(C(=O)NO)cc2)c(-c2cccnc2)c2ccccc21
E3 Binder	CHEMBL4752147	ChEMBL	7.48	—	—	Cn1c(=O)c(OCc2ccc(C(=O)NO)cc2)c(C2CCCCC2)c2ccccc21
E3 Binder	CHEMBL3309284	ChEMBL	7.07	—	—	Cn1c(=O)ccc2cc(C(=O)NCCCCCCC(=O)NO)ccc21
E3 Binder	CHEMBL1879463	ChEMBL	8.7	—	—	Cn1c(=O)n(-c2ccc(C(C)(C)C#N)cc2)c2c3cc(-c4cnc5ccccc5c4)ccc3ncc21
E3 Binder	CHEMBL3353054	ChEMBL	7.48	—	—	Cn1c(C(=O)N2CCn3cc(C(=O)NO)cc3C2)cc(Cl)c1Cl
E3 Binder	CHEMBL3353065	ChEMBL	7.12	—	—	Cn1c(C(=O)N2CCn3nc(C(=O)NO)cc3C2)cc2ccccc21
E3 Binder	CHEMBL487253	ChEMBL	8.22	—	—	Cn1c(CCCC(=O)O)nc2cc(N(CCCl)CCCl)ccc21
E3 Binder	CHEMBL216625	ChEMBL	8.22	—	—	Cn1c(CNCCn2ccc(-c3ccc(C(=O)NO)s3)n2)cc2ccccc21
E3 Binder	CHEMBL4438267	ChEMBL	7.77	—	—	Cn1c(Cc2ccc(C(=O)NO)cc2)nnc1-c1ccccc1
E3 Binder	CHEMBL3693728	ChEMBL	8.05	—	—	Cn1c(Nc2ccc(C(=O)NCCCCCCC(=O)NO)cc2)nc2ccccc21
E3 Binder	CHEMBL4516856	ChEMBL	8.3	—	—	Cn1c(Sc2c(F)cc(C(=O)NO)cc2F)nnc1-c1ccc(CN2CCCCC2)cc1
E3 Binder	CHEMBL4583522	ChEMBL	8.0	—	—	Cn1c(Sc2c(F)cc(C(=O)NO)cc2F)nnc1-c1cccc(CN2CCCCCC2)c1
E3 Binder	CHEMBL4556171	ChEMBL	7.89	—	—	Cn1c(Sc2c(F)cc(C(=O)NO)cc2F)nnc1-c1cccnn1
E3 Binder	CHEMBL4445138	ChEMBL	8.05	—	—	Cn1c(Sc2c(F)cc(C(=O)NO)cc2F)nnc1-c1cccs1
E3 Binder	CHEMBL4470302	ChEMBL	8.22	—	—	Cn1c(Sc2c(F)cc(C(=O)NO)cc2F)nnc1-c1ncccc1F
E3 Binder	CHEMBL4537736	ChEMBL	8.1	—	—	Cn1c(Sc2ccc(C(=O)NO)cc2)nnc1-c1cccs1
E3 Binder	CHEMBL5219657	ChEMBL	7.44	—	—	Cn1c([C@@H]2C[C@@H](OC(=O)NCCc3ccc(C(=O)NO)cc3)CN2c2nc(N)nc(N)c2C#N)nc2cccc(Cl)c2c1=O
E3 Binder	CHEMBL5219798	ChEMBL	7.57	—	—	Cn1c([C@@H]2C[C@@H](OC(=O)NCc3ccc(C(=O)NO)cc3)CN2c2nc(N)nc(N)c2C#N)nc2cccc(Cl)c2c1=O
E3 Binder	CHEMBL5220310	ChEMBL	7.37	—	—	Cn1c([C@@H]2C[C@@H](OC(=O)NCc3ccc(C(=O)NO)s3)CN2c2nc(N)nc(N)c2C#N)nc2cccc(Cl)c2c1=O
E3 Binder	CHEMBL5218525	ChEMBL	7.89	—	—	Cn1c([C@@H]2C[C@@H](OCc3ccc(C(=O)NO)cc3)CN2c2nc(N)nc(N)c2C#N)nc2cccc(Cl)c2c1=O
E3 Binder	CHEMBL5220434	ChEMBL	7.89	—	—	Cn1c([C@@H]2C[C@@H](OCc3ccc(C(=O)NO)s3)CN2c2nc(N)nc(N)c2C#N)nc2cccc(Cl)c2c1=O
E3 Binder	CHEMBL4854340	ChEMBL	9.0	—	—	Cn1c2c(c3ccccc31)CCN(Cc1ccc(C(=O)NO)cc1F)C2
E3 Binder	CHEMBL4784336	ChEMBL	8.26	—	—	Cn1cc(-c2cc(C(C)(C)O)ccc2OC2CC2)c2cc(C(=O)NCCCCCCC(=O)NO)[nH]c2c1=O
E3 Binder	CHEMBL4781215	ChEMBL	8.1	—	—	Cn1cc(-c2cc(C(C)(C)O)ccc2OC2CC2)c2cc(C(=O)NCc3ccc(C(=O)NO)cc3)[nH]c2c1=O
E3 Binder	CHEMBL4749756	ChEMBL	8.06	—	—	Cn1cc(-c2cc(C(C)(C)O)ccc2Oc2ccc(F)cc2F)c2cc(C(=O)NCCCCCCC(=O)NO)[nH]c2c1=O
E3 Binder	CHEMBL4788497	ChEMBL	7.81	—	—	Cn1cc(-c2cc(C(C)(C)O)ccc2Oc2ccc(F)cc2F)c2cc(C(=O)NCc3ccc(C(=O)NO)cc3)[nH]c2c1=O
E3 Binder	CHEMBL4777609	ChEMBL	7.18	—	—	Cn1cc(-c2ccc([C@H]3C[C@@H]3NCC3CCN(CCCc4ccc(C(=O)NO)cc4)CC3)cc2)cn1
E3 Binder	CHEMBL4778531	ChEMBL	6.84	—	—	Cn1cc(-c2ccccc2Oc2ccccc2)c2cc(C(=O)NCCCC(=O)NO)[nH]c2c1=O
E3 Binder	CHEMBL4800001	ChEMBL	8.4	—	—	Cn1cc(-c2ccccc2Oc2ccccc2)c2cc(C(=O)NCCCCC(=O)NO)[nH]c2c1=O
E3 Binder	CHEMBL4777392	ChEMBL	8.47	—	—	Cn1cc(-c2ccccc2Oc2ccccc2)c2cc(C(=O)NCCCCCC(=O)NO)[nH]c2c1=O
E3 Binder	CHEMBL4798212	ChEMBL	8.33	—	—	Cn1cc(-c2ccccc2Oc2ccccc2)c2cc(C(=O)NCCCCCCC(=O)NO)[nH]c2c1=O
E3 Binder	CHEMBL4793324	ChEMBL	7.82	—	—	Cn1cc(-c2ccccc2Oc2ccccc2)c2cc(C(=O)NCc3ccc(C(=O)NO)cc3)[nH]c2c1=O
E3 Binder	CHEMBL4746995	ChEMBL	6.98	—	—	Cn1cc(-c2ccnc(Nc3ccc(C(=O)NCCCCCCC(=O)NO)cc3)n2)c2ccccc21
E3 Binder	CHEMBL5182660	ChEMBL	7.68	—	—	Cn1cc(-c2cn(Cc3ccc(C(=O)NO)cc3)c(=O)c(N3CCOCC3)n2)cn1
E3 Binder	CHEMBL5308477	ChEMBL	6.27	—	—	Cn1cc(/C=C2/C(=O)Nc3cccnc32)c2ccccc21
E3 Binder	CHEMBL411020	ChEMBL	6.0	—	—	Cn1cc(C(=O)/C=C/c2ccccc2)cc1/C=C/C(=O)NO
E3 Binder	CHEMBL12760	ChEMBL	7.0	AGE	—	Cn1cc(C(=O)Cc2ccccc2)cc1/C=C/C(=O)NO
E3 Binder	CHEMBL5273721	ChEMBL	7.26	—	—	Cn1cc(C(=O)N2CCN(Cc3ccc(C(=O)NO)cc3)CC2)c2ccccc21
E3 Binder	CHEMBL3353060	ChEMBL	6.72	—	—	Cn1cc(C(=O)N2CCn3cc(C(=O)NO)cc3C2)c2ccccc21
E3 Binder	CHEMBL343557	ChEMBL	7.64	—	—	Cn1cc(CCNCc2ccc(/C=C/C(=O)NO)cc2)c2ccccc21
E3 Binder	CHEMBL3329999	ChEMBL	8.24	—	—	Cn1cc(CCNS(=O)(=O)c2ccc(/C=C/C(=O)NO)cc2)c2ccccc21
E3 Binder	CHEMBL3760098	ChEMBL	7.21	—	—	Cn1cc(CN2CC3(CC(=O)c4cc(/C=C/C(=O)NO)ccc4O3)C2)c2ccccc21
E3 Binder	CHEMBL3759353	ChEMBL	7.07	—	—	Cn1cc(CN2CCC3(CC(=O)c4cc(/C=C/C(=O)NO)ccc4O3)C2)c2ccccc21
E3 Binder	CHEMBL3758341	ChEMBL	6.74	—	—	Cn1cc(CN2CCCC3(CC(=O)c4cc(/C=C/C(=O)NO)ccc4O3)C2)c2ccccc21
E3 Binder	CHEMBL3758352	ChEMBL	6.94	—	—	Cn1cc(CN2CCCC3(CC2)CC(=O)c2cc(/C=C/C(=O)NO)ccc2O3)c2ccccc21
E3 Binder	CHEMBL2105763	ChEMBL	7.77	GOK	—	Cn1cc(CNCC2CCN(c3ncc(C(=O)NO)cn3)CC2)c2ccccc21
E3 Binder	CHEMBL3233682	ChEMBL	6.22	—	—	Cn1cc(C[C@@H](COc2ccc(/C=C/C(=O)NO)cc2)NC(=O)OC(C)(C)C)c2ccccc21
E3 Binder	CHEMBL4797928	ChEMBL	7.34	—	—	Cn1ccc(-c2ccc([C@H]3C[C@@H]3NCC3CCN(CCCc4ccc(C(=O)NO)cc4)CC3)cc2)cc1=O
E3 Binder	CHEMBL4065026	ChEMBL	8.17	—	—	Cn1ccc2c(CCNS(=O)(=O)c3ccc(/C=C/C(=O)NO)cc3)cccc21
E3 Binder	CHEMBL3353061	ChEMBL	7.07	—	—	Cn1ccc2cc(C(=O)N3CCn4cc(C(=O)NO)cc4C3)ccc21
E3 Binder	CHEMBL297784	ChEMBL	6.37	—	—	Cn1ccc2cc3c(cc21)CCN3C(=O)Nc1cccnc1
E3 Binder	CHEMBL2431912	ChEMBL	6.58	—	—	Cn1cccc1C(=O)N1CCCc2cc(C(=O)NO)ccc2C1
E3 Binder	CHEMBL2431901	ChEMBL	7.44	—	—	Cn1cccc1C(=O)N1CCc2cc(C(=O)NO)ccc2C1
E3 Binder	CHEMBL2431916	ChEMBL	8.3	—	—	Cn1cccc1C(=O)N1CCc2cc(C(=O)NO)sc2C1
E3 Binder	CHEMBL2431908	ChEMBL	6.89	—	—	Cn1cccc1C(=O)N1CCc2ccc(C(=O)NO)cc2CC1
E3 Binder	CHEMBL2431919	ChEMBL	7.75	—	—	Cn1cccc1C(=O)N1CCc2sc(C(=O)NO)cc2C1
E3 Binder	CHEMBL3353053	ChEMBL	7.48	—	—	Cn1cccc1C(=O)N1CCn2cc(C(=O)NO)cc2C1
E3 Binder	CHEMBL3353066	ChEMBL	6.89	—	—	Cn1cccc1C(=O)N1CCn2cc(C(=O)NO)nc2C1
E3 Binder	CHEMBL3353063	ChEMBL	6.46	—	—	Cn1cccc1C(=O)N1CCn2nc(C(=O)NO)cc2C1
E3 Binder	CHEMBL2431906	ChEMBL	7.4	—	—	Cn1cccc1C(=O)N1Cc2ccc(C(=O)NO)cc2C1
E3 Binder	CHEMBL2431862	ChEMBL	7.72	—	—	Cn1cccc1C(=O)NCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL2431865	ChEMBL	7.72	—	—	Cn1cccc1C(=O)NCc1ccc(C(=O)NO)s1
E3 Binder	CHEMBL2431866	ChEMBL	7.28	—	—	Cn1cccc1C(=O)NCc1ncc(C(=O)NO)s1
E3 Binder	CHEMBL5075423	ChEMBL	6.21	—	—	Cn1cccc1C(=O)Nc1cccc(CCC(=O)NO)c1
E3 Binder	CHEMBL4541796	ChEMBL	7.1	—	—	Cn1cncc1-c1cn(Cc2ccc(C(=O)NO)cc2)c2ccccc12
E3 Binder	CHEMBL216885	ChEMBL	6.12	—	—	Cn1nc(C(F)(F)F)cc1-c1ccc(C(=O)NO)s1
E3 Binder	CHEMBL4242626	ChEMBL	9.07	—	—	N#CCCn1cc(-c2nc(Nc3ccc(NC(=O)CCCCCCC(=O)NO)cc3)nc3[nH]ccc23)cn1
E3 Binder	CHEMBL1789941	ChEMBL	7.82	RXT	—	N#CC[C@H](C1CCCC1)n1cc(-c2ncnc3[nH]ccc23)cn1
E3 Binder	CHEMBL3235790	ChEMBL	6.39	—	—	N#CCc1ccc(-c2ccc(/C=C/C(=O)NO)cc2Cl)cc1C12CC3CC(CC(C3)C1)C2
E3 Binder	CHEMBL1077183	ChEMBL	8.05	—	—	N#C[Se]CCCCCC(=O)Nc1ccccc1
E3 Binder	CHEMBL5219246	ChEMBL	6.66	—	—	N#Cc1c(N)nc(N)nc1N1CC2(CC2)C[C@H]1c1nc(NCCc2ccc(C(=O)NO)cc2)c2c(Cl)cccc2n1
E3 Binder	CHEMBL5220325	ChEMBL	6.4	—	—	N#Cc1c(N)nc(N)nc1N1CC2(CC2)C[C@H]1c1nc(NCc2ccc(C(=O)NO)cc2)c2c(Cl)cccc2n1
E3 Binder	CHEMBL5220243	ChEMBL	6.22	—	—	N#Cc1c(N)nc(N)nc1N1CC2(CC2)C[C@H]1c1nc2cccc(Cl)c2c(=O)n1Cc1cc(C(=O)NO)no1
E3 Binder	CHEMBL5218681	ChEMBL	6.48	—	—	N#Cc1c(N)nc(N)nc1N1CC2(CC2)C[C@H]1c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5218472	ChEMBL	7.89	—	—	N#Cc1c(N)nc(N)nc1N1CC2(CC2)C[C@H]1c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(C(=O)NO)s1
E3 Binder	CHEMBL5218764	ChEMBL	7.57	—	—	N#Cc1c(N)nc(N)nc1N1CC2(CC2)C[C@H]1c1nc2cccc(F)c2c(=O)n1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5218454	ChEMBL	7.5	—	—	N#Cc1c(N)nc(N)nc1N1CC2(CC2)C[C@H]1c1nc2cccc(F)c2c(=O)n1Cc1ccc(C(=O)NO)s1
E3 Binder	CHEMBL5219356	ChEMBL	6.57	—	—	N#Cc1c(N)nc(N)nc1N1CCC[C@H]1c1nc(NCc2ccc(C(=O)NO)cc2)c2c(Cl)cccc2n1
E3 Binder	CHEMBL5218504	ChEMBL	6.55	—	—	N#Cc1c(N)nc(N)nc1N1CCC[C@H]1c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL5219941	ChEMBL	7.17	—	—	N#Cc1c(N)nc(N)nc1N1CCC[C@H]1c1nc2cccc(Cl)c2c(=O)n1Cc1ccc(C(=O)NO)s1
E3 Binder	CHEMBL5219509	ChEMBL	6.78	—	—	N#Cc1c(N)nc(N)nc1N1C[C@@H](OC(=O)NCc2ccc(C(=O)NO)cc2)C[C@H]1c1nc2cccc(Cl)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL5218671	ChEMBL	7.06	—	—	N#Cc1c(N)nc(N)nc1N1C[C@H](OC(=O)NCc2ccc(C(=O)NO)cc2)C[C@H]1c1nc2cccc(Cl)c2c(=O)n1-c1ccccc1
E3 Binder	CHEMBL2337870	ChEMBL	6.43	—	—	N#Cc1cc(-c2ccccc2)ccc1Cn1cccc(O)c1=S
E3 Binder	CHEMBL568955	ChEMBL	7.39	—	—	N#Cc1ccc(-c2ccc(C(=O)C(F)(F)F)s2)cc1
E3 Binder	CHEMBL2337872	ChEMBL	6.02	—	—	N#Cc1ccc(-c2ccc(Cn3cccc(O)c3=S)cc2)cc1
E3 Binder	CHEMBL4746111	ChEMBL	6.69	—	—	N#Cc1ccc(-c2ccc([C@H]3C[C@@H]3NCC3CCN(CCCc4ccc(C(=O)NO)cc4)CC3)cc2)cc1
E3 Binder	CHEMBL3110280	ChEMBL	6.04	—	—	N#Cc1ccc(-c2cn(CCCCCn3cccc(O)c3=S)nn2)cc1
E3 Binder	CHEMBL3110283	ChEMBL	6.18	—	—	N#Cc1ccc(-c2cn(CCCCCn3cccc(O)c3=S)nn2)cc1C(F)(F)F
E3 Binder	CHEMBL4518594	ChEMBL	6.96	—	—	N#Cc1ccc(CCc2nc(CCC(=O)NO)cs2)cc1
E3 Binder	CHEMBL1801242	ChEMBL	7.52	—	—	N#Cc1ccc(CN[C@H]2[C@@H]3CN(c4ncc(C(=O)NO)cn4)C[C@@H]32)cc1
E3 Binder	CHEMBL3415621	ChEMBL	7.0	—	—	N#Cc1ccc(N2CCC(Nc3ccc(C(=O)NO)cc3)C2=O)cc1
E3 Binder	CHEMBL3357475	ChEMBL	6.34	—	—	N#Cc1ccc(NC2CCc3ccc(C(=O)NO)cc3C2)cc1Cl
E3 Binder	CHEMBL4856920	ChEMBL	8.34	—	—	N#Cc1ccc2c(c1)CCCCN2Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4874875	ChEMBL	8.89	—	—	N#Cc1ccc2c(c1)CCCN2Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4583466	ChEMBL	6.52	—	—	N#Cc1ccc2c(c1)SC(=S)N1CCN=C21
E3 Binder	CHEMBL5287395	ChEMBL	7.31	—	—	N#Cc1cccc(-c2cn(CCCCCCn3cccc(/C=C/C(=O)NO)c3=O)nn2)c1
E3 Binder	CHEMBL3110281	ChEMBL	6.45	—	—	N#Cc1cccc(-c2cn(CCCCCn3cccc(O)c3=S)nn2)c1
E3 Binder	CHEMBL4071528	ChEMBL	7.7	—	—	N#Cc1cccc(Nc2ncnc3cc(NC(=O)CCCCCCC(=O)NO)sc23)c1
E3 Binder	CHEMBL2047680	ChEMBL	6.0	—	—	N/N=C(\Cc1ccc(O)c(Br)c1)C(=O)NCCS
E3 Binder	CHEMBL568151	ChEMBL	7.41	—	—	N=C(N)NCCC[C@@H]1NC(=O)C[C@H](Cc2ccc(O)cc2)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCCCCC(=O)NO)NC1=O
E3 Binder	CHEMBL596216	ChEMBL	8.42	—	—	NC(/C=C/c1ccccc1)CN1CCN(c2ncc(C(=O)NO)cn2)CC1
E3 Binder	CHEMBL5208297	ChEMBL	6.29	—	—	NC(=O)/C=C/c1ccc(COc2ccc(-n3cc4cccc(C(N)=O)c4n3)cc2)cc1
E3 Binder	CHEMBL150236	ChEMBL	6.48	—	—	NC(=O)C(=O)NCCSSCCNC(=O)/C(Cc1ccc(O)c(Br)c1)=N/O
E3 Binder	CHEMBL3640699	ChEMBL	8.1	—	—	NC(=O)C1CCN(c2ncc(C(=O)NCCCCCCC(=O)NO)cn2)CC1
E3 Binder	CHEMBL2036473	ChEMBL	7.31	—	—	NC(=O)CCC(c1nc2ccccc2o1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL2018449	ChEMBL	8.39	—	—	NC(=O)CCCN1CCc2c(c3ccccc3n2Cc2ccc(C(=O)NO)cc2)C1
E3 Binder	CHEMBL2018447	ChEMBL	9.34	—	—	NC(=O)CCN1CCc2c(c3ccccc3n2Cc2ccc(C(=O)NO)cc2)C1
E3 Binder	CHEMBL2018448	ChEMBL	9.1	—	—	NC(=O)CN1CCc2c(c3ccccc3n2Cc2ccc(C(=O)NO)cc2)C1
E3 Binder	CHEMBL5177616	ChEMBL	6.27	—	—	NC(=O)c1ccc(COc2ccc(-n3cc4cccc(C(N)=O)c4n3)cc2)cc1
E3 Binder	CHEMBL4847663	ChEMBL	8.62	—	—	NC(=O)c1ccc2c(c1)CCCCN2Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4846435	ChEMBL	9.15	QRB	—	NC(=O)c1ccc2c(c1)CCCN2Cc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4859992	ChEMBL	7.7	—	—	NC(=O)c1ccc2c(c1)N(Cc1ccc(/C=C/C(=O)NO)cc1)c1ccccc1S2
E3 Binder	CHEMBL4862510	ChEMBL	8.34	—	—	NC(=O)c1ccc2c(c1)N(Cc1ccc(C(=O)NO)cc1)c1ccccc1S2
E3 Binder	CHEMBL4847771	ChEMBL	7.84	—	—	NC(=O)c1ccc2c(c1)N(Cc1ccc(C(=O)NO)cc1)c1ccccc1[S+]2[O-]
E3 Binder	CHEMBL184238	ChEMBL	6.06	—	—	NC(=O)c1cccc(-c2cccc(OC(=O)NC3CCCCC3)c2)c1
E3 Binder	CHEMBL428721	ChEMBL	6.57	—	—	NC1=NC(=O)C2N=C(CNc3ccc(C(=O)N[C@@H](CCC(=O)NCCSSCCCCCCC(=O)Nc4ncc(-c5ccccc5)s4)C(=O)O)cc3)C=NC2=N1
E3 Binder	CHEMBL3914588	ChEMBL	6.7	—	—	NCC(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3966183	ChEMBL	6.41	—	—	NCC(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCNC(=O)CS)cc1
E3 Binder	CHEMBL260653	ChEMBL	8.18	—	—	NCCCn1cc(CNc2ccc(C(=O)NCCCCCCC(=O)NO)cc2)nn1
E3 Binder	CHEMBL4589682	ChEMBL	8.4	—	—	NCc1ccc(-c2nnn(Cc3c(F)cc(C(=O)NO)cc3F)n2)cc1
E3 Binder	CHEMBL4471726	ChEMBL	8.7	—	—	NCc1ccc(-c2nnn(Cc3ccc(C(=O)NO)cc3)n2)cc1
E3 Binder	CHEMBL4591933	ChEMBL	6.16	P6V	—	NCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4777296	ChEMBL	9.4	N28	—	NCc1ccc(NC(=O)N(CCCCO)Cc2ccc(C(=O)NO)cc2)cc1
E3 Binder	CHEMBL454438	ChEMBL	6.31	—	—	NS(=O)(=O)NCCCCCC(=O)Nc1ccc2ncccc2c1
E3 Binder	CHEMBL507114	ChEMBL	6.41	—	—	NS(=O)(=O)NCCCCCC(=O)Nc1cccc2cccnc12
E3 Binder	CHEMBL475714	ChEMBL	6.15	—	—	NS(=O)(=O)NCCCCCC(=O)Nc1cnc2ccccc2c1
E3 Binder	CHEMBL493347	ChEMBL	6.05	—	—	NS(=O)(=O)NCCCCCC(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL514485	ChEMBL	6.82	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)Cc1ccccc1)C(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL515764	ChEMBL	6.43	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)NCc1ccc(F)cc1)C(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL474446	ChEMBL	6.25	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)Nc1ccccc1)C(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL516218	ChEMBL	6.28	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccc(Cl)cc1)C(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL475203	ChEMBL	6.55	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1cccc(Cl)c1)C(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL475391	ChEMBL	6.6	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1nc(-c2ccc(Cl)cc2)cs1
E3 Binder	CHEMBL475043	ChEMBL	6.35	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1nc(-c2ccccc2)c(-c2ccccc2)s1
E3 Binder	CHEMBL473836	ChEMBL	6.75	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL475861	ChEMBL	6.72	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1nc2ccccc2s1
E3 Binder	CHEMBL494138	ChEMBL	6.39	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1c[nH]c(-c2ccccc2)n1
E3 Binder	CHEMBL492312	ChEMBL	6.4	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1csc(-c2ccccc2)n1
E3 Binder	CHEMBL494139	ChEMBL	6.5	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1n[nH]c(-c2ccccc2)n1
E3 Binder	CHEMBL524193	ChEMBL	6.32	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1nc2cc(-c3cccs3)ccc2[nH]1
E3 Binder	CHEMBL494331	ChEMBL	7.0	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1ccccc1)c1nc2ccccc2[nH]1
E3 Binder	CHEMBL515452	ChEMBL	6.22	—	—	NS(=O)(=O)NCCCC[C@H](NC(=O)OCc1cccnc1)C(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL475618	ChEMBL	6.28	—	—	NS(=O)(=O)NCCCC[C@H](NS(=O)(=O)Cc1ccccc1)C(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL286738	ChEMBL	6.07	667	—	NS(=O)(=O)Oc1ccc2c3c(c(=O)oc2c1)CCCCC3
E3 Binder	CHEMBL389688	ChEMBL	8.27	—	—	N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3919705	ChEMBL	6.18	—	—	N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCNC(=O)CS)cc1
E3 Binder	CHEMBL227170	ChEMBL	8.05	—	—	N[C@@H](Cc1ccc(O)cc1)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL389687	ChEMBL	8.12	—	—	N[C@@H](Cc1ccccc1)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL3947997	ChEMBL	6.35	—	—	N[C@@H](Cc1ccccc1)C(=O)Nc1ccccc1-c1ccc(NC(=O)CCCCCNC(=O)CS)cc1
E3 Binder	CHEMBL4851389	ChEMBL	6.95	—	—	Nc1c(F)cc(C(=O)NO)cc1F
E3 Binder	CHEMBL3621988	ChEMBL	6.78	—	—	Nc1cc(F)ccc1NC(=O)c1ccc(CNC(=O)/C=C/c2cccnc2)cc1
E3 Binder	CHEMBL468841	ChEMBL	7.46	—	—	Nc1ccc(-c2cc(C(=O)NCCCCC(=O)NO)no2)cc1
E3 Binder	CHEMBL467793	ChEMBL	8.23	—	—	Nc1ccc(-c2cc(C(=O)NCCCCCCC(=O)NO)no2)cc1
E3 Binder	CHEMBL3286732	ChEMBL	7.8	—	—	Nc1ccc(-c2cccs2)cc1NC(=O)c1ccc(N2CCC3(CC2)CNC(=O)O3)nc1
E3 Binder	CHEMBL393242	ChEMBL	6.05	—	—	Nc1ccc(-c2cccs2)cc1NC(=O)c1ccc2nccnc2c1
E3 Binder	CHEMBL5174437	ChEMBL	7.89	—	—	Nc1ccc(-c2cn(Cc3ccc(C(=O)NO)cc3)c(=O)c(N3CCOCC3)n2)cc1
E3 Binder	CHEMBL5191006	ChEMBL	7.92	—	—	Nc1ccc(-c2cn(Cc3ccc(C(=O)NO)cc3)c(=O)c(N3CCOCC3)n2)cn1
E3 Binder	CHEMBL4552057	ChEMBL	8.61	—	—	Nc1ccc(-c2nc(N3CCOCC3)c3cnn(CCCCCCC(=O)NO)c3n2)cc1
E3 Binder	CHEMBL4785064	ChEMBL	8.34	—	—	Nc1ccc(-c2nc(N3CCOCC3)c3ncn(CCCCCCC(=O)NO)c3n2)cn1
E3 Binder	CHEMBL4568509	ChEMBL	8.52	—	—	Nc1ccc(-c2nnn(Cc3c(F)cc(C(=O)NO)cc3F)n2)cc1
E3 Binder	CHEMBL4574641	ChEMBL	9.0	—	—	Nc1ccc(-c2nnn(Cc3ccc(C(=O)NO)cc3)n2)cc1
E3 Binder	CHEMBL1094708	ChEMBL	8.6	—	—	Nc1ccc(-n2cc(-c3cccc(NC(=O)CCCCCCC(=O)NO)c3)nn2)cc1
E3 Binder	CHEMBL3980019	ChEMBL	7.0	—	—	Nc1ccc(C(=O)NCCNC(=O)CCCC(=O)NO)cc1
E3 Binder	CHEMBL3893547	ChEMBL	6.0	—	—	Nc1ccc(C(=O)NCCNC(=O)CCCCC(=O)NO)cc1
E3 Binder	CHEMBL155579	ChEMBL	6.41	—	—	Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4869421	ChEMBL	6.74	—	—	Nc1ccc(C(=O)NO)cc1F
E3 Binder	CHEMBL4864065	ChEMBL	6.62	—	—	Nc1ccc(C(=O)NO)cn1
E3 Binder	CHEMBL4520110	ChEMBL	7.07	—	—	Nc1ccc(CCc2nc(CCC(=O)NO)cs2)cc1
E3 Binder	CHEMBL4087968	ChEMBL	6.05	—	—	Nc1ccc(F)cc1NC(=O)c1ccc(CNC(=O)/C=C/c2cccnc2)cc1
E3 Binder	CHEMBL446512	ChEMBL	7.14	—	—	Nc1cccc(-c2cc(C(=O)NCCCCC(=O)NO)no2)c1
E3 Binder	CHEMBL468595	ChEMBL	8.6	—	—	Nc1cccc(-c2cc(C(=O)NCCCCCCC(=O)NO)no2)c1
E3 Binder	CHEMBL1630208	ChEMBL	8.48	—	—	Nc1cccc(-c2csc(NC(=O)CCCCCC(=O)NO)n2)c1
E3 Binder	CHEMBL468935	ChEMBL	8.52	—	—	Nc1cccc(-c2csc(NC(=O)CCCCCCC(=O)NO)n2)c1
E3 Binder	CHEMBL511432	ChEMBL	7.09	—	—	Nc1cccc(-c2csc(NC(=O)CCCCc3cc(C(=O)NO)no3)n2)c1
E3 Binder	CHEMBL3926370	ChEMBL	7.1	—	—	Nc1ccccc1-c1ccc(NC(=O)CCCCCCC(=O)NO)cc1
E3 Binder	CHEMBL5283204	ChEMBL	6.75	—	—	Nc1ccccc1NC(=O)/C=C/c1ccc(C(=O)NCC2CCN(Cc3ccccc3)CC2)cc1
E3 Binder	CHEMBL5072579	ChEMBL	6.2	—	—	Nc1ccccc1NC(=O)/C=C/c1cnc(-c2ccc3cc[nH]c3c2)s1
E3 Binder	CHEMBL4282111	ChEMBL	8.0	—	—	Nc1ccccc1NC(=O)CCCCCCC(=O)NO
E3 Binder	CHEMBL5275640	ChEMBL	6.34	—	—	Nc1ccccc1NC(=O)CCc1ccc(C(=O)NCC2CCN(Cc3ccccc3)CC2)cc1
E3 Binder	CHEMBL4291940	ChEMBL	7.17	—	—	Nc1ccccc1NC(=O)c1ccc(C(=O)NCCNc2nonc2/C(=N/O)Nc2ccc(F)c(Br)c2)cc1
E3 Binder	CHEMBL4460434	ChEMBL	6.0	—	—	Nc1ccccc1NC(=O)c1ccc(CN(CC(=O)NCc2ccccc2)C(=O)c2cccnc2)cc1
E3 Binder	CHEMBL27759	ChEMBL	7.47	—	—	Nc1ccccc1NC(=O)c1ccc(CNC(=O)OCc2cccnc2)cc1
E3 Binder	CHEMBL3670675	ChEMBL	8.7	—	—	Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2[nH]c(-c3ccc(O)cc3)cc2-c2ccoc2)cc1
E3 Binder	CHEMBL3670674	ChEMBL	8.8	—	—	Nc1ccccc1NC(=O)c1ccc(CNC(=O)c2[nH]c(-c3ccsc3)cc2-c2ccc(O)cc2)cc1
E3 Binder	CHEMBL3217993	ChEMBL	6.6	—	—	Nc1ccccc1NC(=O)c1ccc(COc2ccc3ncnc(Nc4cccc(Br)c4)c3c2)cc1
E3 Binder	CHEMBL4276962	ChEMBL	6.14	—	—	Nc1ccccc1NC(=O)c1ccc(CSC(=S)N2CCN(c3ccncc3)CC2)cc1
E3 Binder	CHEMBL4795285	ChEMBL	7.95	—	—	Nc1ccccc1NC(=O)c1ccc(Cn2cnc3c(Nc4ccc(C(=O)NO)cc4)nc(Cl)nc32)cc1
E3 Binder	CHEMBL5201523	ChEMBL	8.68	—	—	Nc1nc(-c2ccco2)c2cnn(Cc3cccc(OCCCCCCC(=O)NO)c3)c2n1
E3 Binder	CHEMBL5086791	ChEMBL	7.72	—	—	Nc1nc(N2CCN(CCc3ccc(C(=O)NO)cc3)CC2)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5090351	ChEMBL	7.97	—	—	Nc1nc(NCCCCCCC(=O)NO)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5094920	ChEMBL	8.31	—	—	Nc1nc(NCCCc2ccc(C(=O)NO)cc2)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5080901	ChEMBL	8.49	—	—	Nc1nc(NCCOc2ccc(C(=O)NO)cc2)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5077827	ChEMBL	7.16	—	—	Nc1nc(NCCc2ccc(/C=C/C(=O)NO)cc2)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5075704	ChEMBL	7.83	—	—	Nc1nc(NCCc2ccc(C(=O)NO)cc2)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5076540	ChEMBL	8.23	—	—	Nc1nc(NCCc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5087206	ChEMBL	6.88	—	—	Nc1nc(NCCc2ccc(OCCCC(=O)NO)cc2)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5082737	ChEMBL	7.43	—	—	Nc1nc(NCCc2ccc(OCCCCC(=O)NO)cc2)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5079065	ChEMBL	8.1	—	—	Nc1nc(NCCc2ccc(OCCCCCC(=O)NO)cc2)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5086912	ChEMBL	8.05	—	—	Nc1nc(NCc2ccc(/C=C/C(=O)NO)cc2)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5076402	ChEMBL	8.52	—	—	Nc1nc(NCc2ccc(C(=O)NO)cc2)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5081907	ChEMBL	7.46	—	—	Nc1nc(NCc2ccc(OCCCCC(=O)NO)cc2)nc2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5090390	ChEMBL	7.13	—	—	Nc1nc2c(cnn2CCCCC(=O)NO)c2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5087220	ChEMBL	7.82	—	—	Nc1nc2c(cnn2CCCCCC(=O)NO)c2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5092198	ChEMBL	8.18	—	—	Nc1nc2c(cnn2CCCCCCC(=O)NO)c2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5079449	ChEMBL	7.5	—	—	Nc1nc2c(cnn2CCN2CCC(c3ccc(C(=O)NO)cc3)CC2)c2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5090592	ChEMBL	7.1	—	—	Nc1nc2c(cnn2CCN2CCc3ccc(C(=O)NO)cc3C2)c2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5094087	ChEMBL	8.12	—	—	Nc1nc2c(cnn2CCc2ccc(C(=O)NO)cc2)c2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5093149	ChEMBL	8.23	—	—	Nc1nc2c(cnn2CCc2ccc(NC(=O)CCCCCCC(=O)NO)cc2)c2nc(-c3ccco3)nn12
E3 Binder	CHEMBL5086693	ChEMBL	7.8	—	—	Nc1nc2c(cnn2CCc2ccc(OCCCCCC(=O)NO)cc2)c2nc(-c3ccco3)nn12
E3 Binder	CHEMBL4862549	ChEMBL	7.07	—	—	Nc1nc2cc(-c3nn(CC4CCN(c5ncc(C(=O)NO)cn5)CC4)c4ncnc(N)c34)ccc2o1
E3 Binder	CHEMBL4846560	ChEMBL	8.82	—	—	Nc1nc2cc(-c3nn(CCCCCCC(=O)NO)c4ncnc(N)c34)ccc2o1
E3 Binder	CHEMBL3415961	ChEMBL	6.67	—	—	Nc1nc2ncc(CNc3ccc(C(=O)NCCCCC(=O)NO)cc3)nc2c(=O)[nH]1
E3 Binder	CHEMBL3415962	ChEMBL	7.36	—	—	Nc1nc2ncc(CNc3ccc(C(=O)NCCCCCC(=O)NO)cc3)nc2c(=O)[nH]1
E3 Binder	CHEMBL3415963	ChEMBL	7.91	—	—	Nc1nc2ncc(CNc3ccc(C(=O)NCCCCCCC(=O)NO)cc3)nc2c(=O)[nH]1
E3 Binder	CHEMBL3415964	ChEMBL	7.26	—	—	Nc1nc2ncc(CNc3ccc(C(=O)NCCCCCCCC(=O)NO)cc3)nc2c(=O)[nH]1
E3 Binder	CHEMBL3415965	ChEMBL	7.99	—	—	Nc1nc2ncc(CNc3ccc(C(=O)NCCCCCCCCC(=O)NO)cc3)nc2c(=O)[nH]1
E3 Binder	CHEMBL3415966	ChEMBL	6.32	—	—	Nc1nc2ncc(CNc3ccc(C(=O)NCCCCCCCCCC(=O)NO)cc3)nc2c(=O)[nH]1
E3 Binder	CHEMBL3415959	ChEMBL	7.75	—	—	Nc1nc2ncc(CNc3ccc(C(=O)NO)cc3)nc2c(=O)[nH]1
E3 Binder	CHEMBL3415968	ChEMBL	6.88	—	—	Nc1nc2ncc(CNc3ccc(C(=O)N[C@@H](CCC(=O)NCCCCCCC(=O)NO)C(=O)O)cc3)nc2c(=O)[nH]1
E3 Binder	CHEMBL3415969	ChEMBL	6.71	—	—	Nc1nc2ncc(CNc3ccc(C(=O)N[C@@H](CCC(=O)NCCCCCCCC(=O)NO)C(=O)O)cc3)nc2c(=O)[nH]1
E3 Binder	CHEMBL3415970	ChEMBL	6.75	—	—	Nc1nc2ncc(CNc3ccc(C(=O)N[C@@H](CCC(=O)NCCCCCCCCC(=O)NO)C(=O)O)cc3)nc2c(=O)[nH]1
E3 Binder	CHEMBL5172884	ChEMBL	7.7	—	—	Nc1ncc(-c2cc(N3CCOCC3)c(=O)n(Cc3ccc(C(=O)NO)cc3)c2)cn1
E3 Binder	CHEMBL5192044	ChEMBL	7.89	—	—	Nc1ncc(-c2cc(N3CCOCC3)c(=O)n(Cc3ccc(C(=O)NO)cc3)n2)cn1
E3 Binder	CHEMBL5183646	ChEMBL	6.96	—	—	Nc1ncc(-c2cn(CCCCCC(=O)NO)c(=O)c(N3CCOCC3)n2)cn1
E3 Binder	CHEMBL5187051	ChEMBL	7.27	—	—	Nc1ncc(-c2cn(CCCCCCC(=O)NO)c(=O)c(N3CCOCC3)n2)cn1
E3 Binder	CHEMBL5185319	ChEMBL	6.71	—	—	Nc1ncc(-c2cn(CCCCCCCC(=O)NO)c(=O)c(N3CCOCC3)n2)cn1
E3 Binder	CHEMBL5192159	ChEMBL	8.38	—	—	Nc1ncc(-c2cn(Cc3ccc(C(=O)NO)cc3)c(=O)c(N3CCCCC3)n2)cn1
E3 Binder	CHEMBL5179687	ChEMBL	7.82	—	—	Nc1ncc(-c2cn(Cc3ccc(C(=O)NO)cc3)c(=O)c(N3CCOCC3)n2)cn1
E3 Binder	CHEMBL5184950	ChEMBL	8.16	—	—	Nc1ncc(-c2cn(Cc3ccc(C(=O)NO)cc3)c(=O)c(Nc3ccccc3)n2)cn1
E3 Binder	CHEMBL5172866	ChEMBL	6.19	—	—	Nc1ncc(-c2cn(Cc3cccc(C(=O)NO)c3)c(=O)c(N3CCOCC3)n2)cn1
E3 Binder	CHEMBL4744689	ChEMBL	8.18	—	—	Nc1ncc(-c2nc(N3CCOCC3)c3ccn(CCCCCCC(=O)NO)c3n2)cn1
E3 Binder	CHEMBL4852256	ChEMBL	7.19	—	—	Nc1ncc(C(=O)NO)cn1
E3 Binder	CHEMBL1209431	ChEMBL	6.11	—	—	Nc1nccc(/C=C/c2ccccc2)n1
E3 Binder	CHEMBL2408778	ChEMBL	8.57	—	—	Nc1ncnc2c1c(-c1ccc(Cl)cc1)nn2-c1cccc(-c2cnnn2CCCCCC(=O)NO)c1
E3 Binder	CHEMBL4846776	ChEMBL	8.02	—	—	Nc1ncnc2c1c(-c1cnc3[nH]ccc3c1)nn2CCCCCCCCC(=O)NO
E3 Binder	CHEMBL3925604	ChEMBL	7.0	—	—	Nc1ncnc2c1nc(Sc1cc3c(cc1Br)OCO3)n2CCCCCC(=O)NO
E3 Binder	CHEMBL3975711	ChEMBL	6.0	—	—	Nc1ncnc2c1nc(Sc1cc3c(cc1Br)OCO3)n2CCOCCCCC(=O)NO
E3 Binder	CHEMBL3926697	ChEMBL	6.0	—	—	Nc1ncnc2c1nc(Sc1cc3c(cc1Br)OCO3)n2CCOCCCCCC(=O)NO
E3 Binder	CHEMBL3907592	ChEMBL	7.0	—	—	Nc1ncnc2c1nc(Sc1cc3c(cc1I)OCO3)n2CCNCCCCCC(=O)NO
E3 Binder	CHEMBL314389	ChEMBL	6.87	—	—	O=C(/C=C/C#Cc1ccc(NS(=O)(=O)c2ccccc2)cc1)NO
E3 Binder	CHEMBL5188463	ChEMBL	6.37	—	—	O=C(/C=C/C1CCN(Cc2ccc(Cl)cc2)CC1)NO
E3 Binder	CHEMBL1808673	ChEMBL	6.14	—	—	O=C(/C=C/C=C/CC/C=C/c1ccc2c(c1)OCO2)NO
E3 Binder	CHEMBL312098	ChEMBL	6.6	—	—	O=C(/C=C/C=C/c1ccc(Cl)cc1)NO
E3 Binder	CHEMBL448955	ChEMBL	7.54	—	—	O=C(/C=C/C=C/c1ccccc1)NCCCCCC(=O)NO
E3 Binder	CHEMBL84395	ChEMBL	6.55	—	—	O=C(/C=C/C=C/c1ccccc1)NO
E3 Binder	CHEMBL5206154	ChEMBL	6.8	—	—	O=C(/C=C/C=C/c1csc(Br)n1)NO
E3 Binder	CHEMBL571547	ChEMBL	6.49	—	—	O=C(/C=C/c1cc(/C=C/C(=O)c2ccccc2)ccn1)NO
E3 Binder	CHEMBL556332	ChEMBL	7.38	—	—	O=C(/C=C/c1ccc(-c2ccc(O)cc2)cc1)NO
E3 Binder	CHEMBL1630110	ChEMBL	6.64	—	—	O=C(/C=C/c1ccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)cc1)NO
E3 Binder	CHEMBL1630107	ChEMBL	6.64	—	—	O=C(/C=C/c1ccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)o1)NO
E3 Binder	CHEMBL3314860	ChEMBL	7.52	—	—	O=C(/C=C/c1ccc(-c2nnc(Cc3c[nH]c4ccccc34)o2)cc1)NO
E3 Binder	CHEMBL3314859	ChEMBL	7.22	—	—	O=C(/C=C/c1ccc(-c2nnc(Cc3cccc4ccccc34)o2)cc1)NO
E3 Binder	CHEMBL4285033	ChEMBL	6.17	—	—	O=C(/C=C/c1ccc(-n2[se]c3ccccc3c2=O)cc1)NO
E3 Binder	CHEMBL3758457	ChEMBL	7.57	—	—	O=C(/C=C/c1ccc(/C=C(/CNC2CC2)c2ccc(F)cc2)cc1)NO
E3 Binder	CHEMBL461763	ChEMBL	6.2	—	—	O=C(/C=C/c1ccc(/C=C/C(=O)c2ccc3ccccc3c2)o1)NO
E3 Binder	CHEMBL578393	ChEMBL	7.66	—	—	O=C(/C=C/c1ccc(/C=C/C(=O)c2ccccc2)cn1)NO
E3 Binder	CHEMBL472631	ChEMBL	6.52	—	—	O=C(/C=C/c1ccc(/C=N/OCCN2CCOCC2)cc1)NO
E3 Binder	CHEMBL471041	ChEMBL	6.18	—	—	O=C(/C=C/c1ccc(/C=N/OCc2c(F)c(F)c(F)c(F)c2F)cc1)NO
E3 Binder	CHEMBL471042	ChEMBL	6.91	—	—	O=C(/C=C/c1ccc(/C=N/OCc2ccc([N+](=O)[O-])cc2)cc1)NO
E3 Binder	CHEMBL1213457	ChEMBL	7.5	—	—	O=C(/C=C/c1ccc(C(=O)N/N=C/c2ccc(O)c(O)c2O)cc1)NO
E3 Binder	CHEMBL5192800	ChEMBL	6.77	—	—	O=C(/C=C/c1ccc(C(=O)N2CCC(N3C(=O)[C@H](c4ccccc4)[C@H]3c3ccccc3)CC2)cc1)NO
E3 Binder	CHEMBL4583327	ChEMBL	6.4	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)NC2CC2)cc1)NO
E3 Binder	CHEMBL4545703	ChEMBL	6.62	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)NC2CCCC2)cc1)NO
E3 Binder	CHEMBL4577653	ChEMBL	6.7	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)NCc2ccccc2)cc1)NO
E3 Binder	CHEMBL4542734	ChEMBL	7.72	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)Nc2ccc(Br)cc2)cc1)NO
E3 Binder	CHEMBL4592307	ChEMBL	6.25	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)Nc2ccc(C(F)(F)F)cc2)cc1)NO
E3 Binder	CHEMBL4574697	ChEMBL	7.46	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)Nc2ccc(Cl)cc2)cc1)NO
E3 Binder	CHEMBL4590924	ChEMBL	6.52	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)Nc2ccc(F)cc2)cc1)NO
E3 Binder	CHEMBL4563800	ChEMBL	7.28	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)Nc2ccc(I)cc2)cc1)NO
E3 Binder	CHEMBL4588104	ChEMBL	7.21	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)Nc2ccc3ccccc3c2)cc1)NO
E3 Binder	CHEMBL4592929	ChEMBL	7.11	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)Nc2cccc(Br)c2)cc1)NO
E3 Binder	CHEMBL4529623	ChEMBL	6.82	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)Nc2ccccc2)cc1)NO
E3 Binder	CHEMBL4563265	ChEMBL	6.89	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)Nc2ccccc2Br)cc1)NO
E3 Binder	CHEMBL4575399	ChEMBL	7.14	—	—	O=C(/C=C/c1ccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)Nc2ccncc2)cc1)NO
E3 Binder	CHEMBL5269960	ChEMBL	6.55	—	—	O=C(/C=C/c1ccc(C(=O)NCC2CCN(Cc3ccccc3)CC2)cc1)NO
E3 Binder	CHEMBL4568722	ChEMBL	6.64	—	—	O=C(/C=C/c1ccc(C(=O)NCCCOc2no[n+]([O-])c2S(=O)(=O)c2ccccc2)cc1)NO
E3 Binder	CHEMBL4519499	ChEMBL	6.82	—	—	O=C(/C=C/c1ccc(C(=O)NCCOc2no[n+]([O-])c2S(=O)(=O)c2ccccc2)cc1)NO
E3 Binder	CHEMBL4226835	ChEMBL	6.57	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CC1
E3 Binder	CHEMBL4227758	ChEMBL	6.6	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NC1CCCC1
E3 Binder	CHEMBL4226968	ChEMBL	7.66	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCCc1ccccc1
E3 Binder	CHEMBL4226914	ChEMBL	7.43	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCc1ccccc1
E3 Binder	CHEMBL4228565	ChEMBL	8.7	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccc(Br)cc1
E3 Binder	CHEMBL4229142	ChEMBL	8.24	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccc(Cl)cc1
E3 Binder	CHEMBL4228304	ChEMBL	8.7	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccc(F)cc1
E3 Binder	CHEMBL4224796	ChEMBL	7.53	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccc(I)cc1
E3 Binder	CHEMBL4225063	ChEMBL	8.09	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1cccc(Cl)c1
E3 Binder	CHEMBL4226126	ChEMBL	7.22	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1cccc2ccccc12
E3 Binder	CHEMBL4227898	ChEMBL	8.12	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccccc1
E3 Binder	CHEMBL4224735	ChEMBL	7.24	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccccc1Cl
E3 Binder	CHEMBL4227225	ChEMBL	7.43	—	—	O=C(/C=C/c1ccc(C(=O)NO)cc1)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccncc1
E3 Binder	CHEMBL492956	ChEMBL	7.26	—	—	O=C(/C=C/c1ccc(C(=O)Nc2cccc(Nc3ncc(-c4cccnc4)s3)c2)cc1)NO
E3 Binder	CHEMBL523684	ChEMBL	7.35	—	—	O=C(/C=C/c1ccc(C(=O)Nc2cccc(Nc3ncc(-c4cccnc4)s3)c2)s1)NO
E3 Binder	CHEMBL390908	ChEMBL	6.51	—	—	O=C(/C=C/c1ccc(C(=O)c2cc3ccccc3[nH]2)cc1)NO
E3 Binder	CHEMBL243181	ChEMBL	6.57	—	—	O=C(/C=C/c1ccc(C(=O)c2cc3ccccc3n2S(=O)(=O)c2ccccc2)cc1)NO
E3 Binder	CHEMBL243809	ChEMBL	6.35	—	—	O=C(/C=C/c1ccc(C(=O)c2cc3ccccc3o2)cc1)NO
E3 Binder	CHEMBL3394285	ChEMBL	6.74	—	—	O=C(/C=C/c1ccc(C(F)(F)F)cc1)NO
E3 Binder	CHEMBL5179574	ChEMBL	7.24	—	—	O=C(/C=C/c1ccc(CCCCCCc2n[nH]c(=O)c3cc(F)ccc23)cc1)NO
E3 Binder	CHEMBL4093350	ChEMBL	8.08	—	—	O=C(/C=C/c1ccc(CCNC(=O)c2c[nH]c3ncccc23)cc1)NO
E3 Binder	CHEMBL4067480	ChEMBL	7.76	—	—	O=C(/C=C/c1ccc(CCNC(=O)c2cc(C(F)(F)F)ccc2Cl)cc1)NO
E3 Binder	CHEMBL4096060	ChEMBL	8.09	—	—	O=C(/C=C/c1ccc(CCNC(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)cc1)NO
E3 Binder	CHEMBL4076931	ChEMBL	8.33	—	—	O=C(/C=C/c1ccc(CCNC(=O)c2ccc3[nH]cnc3c2)cc1)NO
E3 Binder	CHEMBL4075984	ChEMBL	7.93	—	—	O=C(/C=C/c1ccc(CCNC(=O)c2ccc3c(c2)OCCO3)cc1)NO
E3 Binder	CHEMBL4078380	ChEMBL	8.15	—	—	O=C(/C=C/c1ccc(CCNC(=O)c2ccc3c(c2)OCO3)cc1)NO
E3 Binder	CHEMBL4069152	ChEMBL	8.28	—	—	O=C(/C=C/c1ccc(CCNC(=O)c2ccc3ncccc3c2)cc1)NO
E3 Binder	CHEMBL4069669	ChEMBL	7.44	—	—	O=C(/C=C/c1ccc(CCNC(=O)c2cncc(F)c2)cc1)NO
E3 Binder	CHEMBL270118	ChEMBL	6.85	—	—	O=C(/C=C/c1ccc(CCc2nc3ccccc3[nH]2)cc1)NO
E3 Binder	CHEMBL4785378	ChEMBL	7.92	—	—	O=C(/C=C/c1ccc(CN(C(=O)c2c(F)c(F)c(F)c(F)c2F)C2CC2)cc1)NO
E3 Binder	CHEMBL2413295	ChEMBL	6.1	—	—	O=C(/C=C/c1ccc(CN(CCCOc2ccccc2)Cc2ccccc2)o1)NO
E3 Binder	CHEMBL143497	ChEMBL	6.56	—	—	O=C(/C=C/c1ccc(CN(CCCc2ccccc2)Cc2ccccn2)cc1)NO
E3 Binder	CHEMBL341826	ChEMBL	6.79	—	—	O=C(/C=C/c1ccc(CN(CCCc2ccccc2)Cc2cccnc2)cc1)NO
E3 Binder	CHEMBL356066	ChEMBL	8.23	—	—	O=C(/C=C/c1ccc(CN(CCO)CCc2c[nH]c3ccccc23)cc1)NO
E3 Binder	CHEMBL403323	ChEMBL	7.82	—	—	O=C(/C=C/c1ccc(CN(CCO)CCc2cc3ccccc3[nH]2)cc1)NO
E3 Binder	CHEMBL2413287	ChEMBL	6.4	—	—	O=C(/C=C/c1ccc(CN(CCO)CCc2ccc3c(c2)OCO3)o1)NO
E3 Binder	CHEMBL348256	ChEMBL	7.62	—	—	O=C(/C=C/c1ccc(CN(CCO)CCc2cnc3ccccc3c2)cc1)NO
E3 Binder	CHEMBL2413304	ChEMBL	7.05	—	—	O=C(/C=C/c1ccc(CN(CCO)Cc2ccc(-c3ccccc3)cc2)o1)NO
E3 Binder	CHEMBL2413292	ChEMBL	6.77	—	—	O=C(/C=C/c1ccc(CN(CCO)Cc2ccccc2)o1)NO
E3 Binder	CHEMBL143329	ChEMBL	6.43	—	—	O=C(/C=C/c1ccc(CN(CCOC(=O)NCc2ccoc2)CCc2c[nH]c3ccccc23)cc1)NO
E3 Binder	CHEMBL343091	ChEMBL	7.28	—	—	O=C(/C=C/c1ccc(CN(CCc2c[nH]c3ccccc23)C(CO)CO)cc1)NO
E3 Binder	CHEMBL143255	ChEMBL	7.7	—	—	O=C(/C=C/c1ccc(CN(CCc2c[nH]c3ccccc23)C2CCCCC2)cc1)NO
E3 Binder	CHEMBL357231	ChEMBL	8.0	—	—	O=C(/C=C/c1ccc(CN(CCc2c[nH]c3ccccc23)C2CCOCC2)cc1)NO
E3 Binder	CHEMBL421934	ChEMBL	7.07	—	—	O=C(/C=C/c1ccc(CN(CCc2c[nH]c3ccccc23)Cc2ccccc2)cc1)NO
E3 Binder	CHEMBL4758196	ChEMBL	6.74	—	—	O=C(/C=C/c1ccc(CN2C(=O)/C(=C3\Nc4ccccc4\C3=N/O)c3cc(Br)ccc32)cc1)NO
E3 Binder	CHEMBL4748486	ChEMBL	6.5	—	—	O=C(/C=C/c1ccc(CN2C(=O)/C(=C3\Nc4ccccc4\C3=N/O)c3cc(Cl)ccc32)cc1)NO
E3 Binder	CHEMBL4795999	ChEMBL	6.38	—	—	O=C(/C=C/c1ccc(CN2C(=O)/C(=C3\Nc4ccccc4\C3=N/O)c3cc(F)ccc32)cc1)NO
E3 Binder	CHEMBL4746171	ChEMBL	6.22	—	—	O=C(/C=C/c1ccc(CN2C(=O)/C(=C3\Nc4ccccc4\C3=N/O)c3cccc(Cl)c32)cc1)NO
E3 Binder	CHEMBL4781506	ChEMBL	7.02	—	—	O=C(/C=C/c1ccc(CN2C(=O)/C(=C3\Nc4ccccc4\C3=N/O)c3ccccc32)cc1)NO
E3 Binder	CHEMBL140811	ChEMBL	7.28	—	—	O=C(/C=C/c1ccc(CN2CCC(c3c[nH]c4ccccc34)CC2)cc1)NO
E3 Binder	CHEMBL4078014	ChEMBL	7.99	—	—	O=C(/C=C/c1ccc(CN2CCN(C(=O)c3cc(Cc4n[nH]c(=O)c5ccccc45)ccc3F)CC2)cc1)NO
E3 Binder	CHEMBL336674	ChEMBL	6.93	—	—	O=C(/C=C/c1ccc(CN2CCc3c([nH]c4ccccc34)C2)cc1)NO
E3 Binder	CHEMBL4867268	ChEMBL	6.33	—	—	O=C(/C=C/c1ccc(CN2c3ccccc3Sc3ccccc32)cc1)NO
E3 Binder	CHEMBL4765007	ChEMBL	7.85	—	—	O=C(/C=C/c1ccc(CNC(=O)c2c(F)c(F)c(F)c(F)c2F)cc1)NO
E3 Binder	CHEMBL152543	ChEMBL	6.69	—	—	O=C(/C=C/c1ccc(CNC(=O)c2ccc(N3CCCC3)cc2)cc1)NO
E3 Binder	CHEMBL152538	ChEMBL	6.24	—	—	O=C(/C=C/c1ccc(CNC(=O)c2ccc(N3CCN(Cc4cccnc4)CC3)cc2)cc1)NO
E3 Binder	CHEMBL347068	ChEMBL	6.03	—	—	O=C(/C=C/c1ccc(CNC(=O)c2ccccn2)cc1)NO
E3 Binder	CHEMBL346525	ChEMBL	6.43	—	—	O=C(/C=C/c1ccc(CNC(=O)c2cccnc2)cc1)NO
E3 Binder	CHEMBL143283	ChEMBL	7.43	—	—	O=C(/C=C/c1ccc(CNCCCCc2c[nH]c3ccccc23)cc1)NO
E3 Binder	CHEMBL139836	ChEMBL	7.28	—	—	O=C(/C=C/c1ccc(CNCCCc2c[nH]c3ccccc23)cc1)NO
E3 Binder	CHEMBL342474	ChEMBL	7.19	—	—	O=C(/C=C/c1ccc(CNCCCc2ccccc2)cc1)NO
E3 Binder	CHEMBL140900	ChEMBL	7.1	—	—	O=C(/C=C/c1ccc(CNCCCn2c3ccccc3c3ccccc32)cc1)NO
E3 Binder	CHEMBL140899	ChEMBL	7.16	—	—	O=C(/C=C/c1ccc(CNCCOc2ccccc2)cc1)NO
E3 Binder	CHEMBL140013	ChEMBL	7.85	—	—	O=C(/C=C/c1ccc(CNCCc2c[nH]c3ccc(F)cc23)cc1)NO
E3 Binder	CHEMBL141087	ChEMBL	7.52	—	—	O=C(/C=C/c1ccc(CNCCc2c[nH]c3ccc(OCc4ccccc4)cc23)cc1)NO
E3 Binder	CHEMBL344227	ChEMBL	7.2	—	—	O=C(/C=C/c1ccc(CNCCc2c[nH]c3ccccc23)cc1)NO
E3 Binder	CHEMBL142120	ChEMBL	7.34	—	—	O=C(/C=C/c1ccc(CNCCc2cc3ccccc3[nH]2)cc1)NO
E3 Binder	CHEMBL343068	ChEMBL	7.52	—	—	O=C(/C=C/c1ccc(CNCCc2ccc3c(c2)OCO3)cc1)NO
E3 Binder	CHEMBL141236	ChEMBL	7.08	—	—	O=C(/C=C/c1ccc(CNCCc2cn(CC3CC3)c3ccccc23)cc1)NO
E3 Binder	CHEMBL139663	ChEMBL	7.17	—	—	O=C(/C=C/c1ccc(CNCCc2cnc3ccccc3c2)cc1)NO
E3 Binder	CHEMBL140014	ChEMBL	7.8	—	—	O=C(/C=C/c1ccc(CNCCc2coc3ccccc23)cc1)NO
E3 Binder	CHEMBL341601	ChEMBL	7.18	—	—	O=C(/C=C/c1ccc(CNCCn2c3ccccc3c3ccccc32)cc1)NO
E3 Binder	CHEMBL140530	ChEMBL	7.23	—	—	O=C(/C=C/c1ccc(CNCc2c[nH]c3ccccc23)cc1)NO
E3 Binder	CHEMBL335812	ChEMBL	7.29	—	—	O=C(/C=C/c1ccc(CNCc2cc3ccccc3[nH]2)cc1)NO
E3 Binder	CHEMBL4094579	ChEMBL	7.44	—	—	O=C(/C=C/c1ccc(CNCc2ccc3cccc(Cl)c3n2)cc1)NO
E3 Binder	CHEMBL4079007	ChEMBL	7.3	—	—	O=C(/C=C/c1ccc(CNCc2ccc3ccccc3n2)cc1)NO
E3 Binder	CHEMBL358059	ChEMBL	7.4	—	—	O=C(/C=C/c1ccc(CN[C@@H](CO)Cc2c[nH]c3ccccc23)cc1)NO
E3 Binder	CHEMBL343823	ChEMBL	7.57	—	—	O=C(/C=C/c1ccc(CN[C@H](CO)Cc2c[nH]c3ccccc23)cc1)NO
E3 Binder	CHEMBL5205415	ChEMBL	7.89	—	—	O=C(/C=C/c1ccc(CNc2ccc3nc4n(c(=O)c3c2)CCCCC4)cc1)NO
E3 Binder	CHEMBL4096377	ChEMBL	7.38	—	—	O=C(/C=C/c1ccc(CNc2cccc3cccnc23)cc1)NO
E3 Binder	CHEMBL4069121	ChEMBL	7.6	—	—	O=C(/C=C/c1ccc(CNc2cccc3ncccc23)cc1)NO
E3 Binder	CHEMBL3752134	ChEMBL	7.16	—	—	O=C(/C=C/c1ccc(CNc2nccc(-c3cccnc3)n2)cc1)NO
E3 Binder	CHEMBL4459795	ChEMBL	7.0	—	—	O=C(/C=C/c1ccc(CONC(=O)c2ccc3ccccc3n2)cc1)NO
E3 Binder	CHEMBL4462881	ChEMBL	6.03	—	—	O=C(/C=C/c1ccc(CONC(=O)c2ccccc2)cc1)NO
E3 Binder	CHEMBL4776616	ChEMBL	6.61	—	—	O=C(/C=C/c1ccc(COc2ccc(-c3csc(N4N=C(c5ccccc5)/C(=N/Nc5nccs5)C4=O)n3)cc2)cc1)NO
E3 Binder	CHEMBL270327	ChEMBL	7.55	—	—	O=C(/C=C/c1ccc(Cc2nc3ccccc3[nH]2)cc1)NO
E3 Binder	CHEMBL3314861	ChEMBL	7.52	—	—	O=C(/C=C/c1ccc(Cc2nnc(Cc3cccc4ccccc34)o2)cc1)NO
E3 Binder	CHEMBL484489	ChEMBL	8.6	—	—	O=C(/C=C/c1ccc(Cl)cc1F)NCCCCCC(=O)NO
E3 Binder	CHEMBL4084164	ChEMBL	7.85	—	—	O=C(/C=C/c1ccc(Cn2c3c(c4ccccc42)CCN2C(=O)CCCC32)cc1)NO
E3 Binder	CHEMBL5208182	ChEMBL	7.13	—	—	O=C(/C=C/c1ccc(Cn2cc(C(=O)NC3C4CC5CC(C4)CC3C5)c3ccccc32)cc1)NO
E3 Binder	CHEMBL4540416	ChEMBL	7.2	—	—	O=C(/C=C/c1ccc(Cn2cc(Nc3ncc(Cl)c(Nc4ccc(F)cc4)n3)cn2)cc1)NO
E3 Binder	CHEMBL5285649	ChEMBL	6.82	—	—	O=C(/C=C/c1ccc(Cn2cnc3cc(F)ccc3c2=O)cc1)NO
E3 Binder	CHEMBL3426804	ChEMBL	8.0	—	—	O=C(/C=C/c1ccc(NC(=O)C(Cc2ccccc2)c2ccccc2)cn1)NO
E3 Binder	CHEMBL4550522	ChEMBL	7.82	—	—	O=C(/C=C/c1ccc(NC(=O)Cc2cccc3ccccc23)cn1)NO
E3 Binder	CHEMBL5087583	ChEMBL	6.78	—	—	O=C(/C=C/c1ccc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)cc1)NO
E3 Binder	CHEMBL552465	ChEMBL	8.09	—	—	O=C(/C=C/c1ccc(NC(=O)Nc2ccc(Cl)cc2)cc1)NO
E3 Binder	CHEMBL143179	ChEMBL	6.58	—	—	O=C(/C=C/c1ccc(NCCCc2c[nH]c3ccccc23)cc1)NO
E3 Binder	CHEMBL4059703	ChEMBL	6.83	—	—	O=C(/C=C/c1ccc(NCCCn2cc(-c3ncnc4[nH]ccc34)cn2)cc1)NO
E3 Binder	CHEMBL145891	ChEMBL	7.52	—	—	O=C(/C=C/c1ccc(NS(=O)(=O)c2ccc(-c3ccccc3)cc2)cc1)NO
E3 Binder	CHEMBL317814	ChEMBL	7.23	—	—	O=C(/C=C/c1ccc(NS(=O)(=O)c2ccccc2)cc1)NO
E3 Binder	CHEMBL284616	ChEMBL	6.87	—	—	O=C(/C=C/c1ccc(O)c(O)c1)O[C@@H]1C[C@](O)(C(=O)O)C[C@@H](O)[C@H]1O
E3 Binder	CHEMBL3975710	ChEMBL	7.0	—	—	O=C(/C=C/c1ccc(OCCOc2ccc3ncnc(Nc4ccc(F)c(Cl)c4)c3c2)cc1)NO
E3 Binder	CHEMBL3233697	ChEMBL	7.28	—	—	O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)CCc2ccccc2)cc1)NO
E3 Binder	CHEMBL3233696	ChEMBL	7.63	—	—	O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)Cc2ccccc2)cc1)NO
E3 Binder	CHEMBL3233704	ChEMBL	7.69	—	—	O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(Br)cc2)cc1)NO
E3 Binder	CHEMBL3233702	ChEMBL	6.68	—	—	O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(Cl)c(Cl)c2)cc1)NO
E3 Binder	CHEMBL3233698	ChEMBL	8.25	—	—	O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(Cl)cc2)cc1)NO
E3 Binder	CHEMBL3233701	ChEMBL	6.73	—	—	O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(Cl)cc2Cl)cc1)NO
E3 Binder	CHEMBL3233703	ChEMBL	8.17	—	—	O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(F)cc2)cc1)NO
E3 Binder	CHEMBL3233700	ChEMBL	6.83	—	—	O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2cccc(Cl)c2)cc1)NO
E3 Binder	CHEMBL3233687	ChEMBL	7.98	—	—	O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccccc2)cc1)NO
E3 Binder	CHEMBL3233699	ChEMBL	7.3	—	—	O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccccc2Cl)cc1)NO
E3 Binder	CHEMBL3233693	ChEMBL	7.68	—	—	O=C(/C=C/c1ccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccccc2O)cc1)NO
E3 Binder	CHEMBL3330000	ChEMBL	7.36	—	—	O=C(/C=C/c1ccc(S(=O)(=O)N2CCc3c([nH]c4ccccc34)C2)cc1)NO
E3 Binder	CHEMBL3262729	ChEMBL	6.07	—	—	O=C(/C=C/c1ccc(S(=O)(=O)N2CCc3cccnc32)cc1)NO
E3 Binder	CHEMBL4647028	ChEMBL	6.12	—	—	O=C(/C=C/c1ccc(S(=O)(=O)NCCCN2c3ccccc3CCc3ccc(Cl)cc32)cc1)NO
E3 Binder	CHEMBL3329998	ChEMBL	8.18	—	—	O=C(/C=C/c1ccc(S(=O)(=O)NCCc2c[nH]c3ccccc23)cc1)NO
E3 Binder	CHEMBL4069853	ChEMBL	8.08	—	—	O=C(/C=C/c1ccc(S(=O)(=O)NCCc2cccc3[nH]ccc23)cc1)NO
E3 Binder	CHEMBL5283395	ChEMBL	8.28	—	—	O=C(/C=C/c1ccc(S(=O)(=O)Nc2cc(F)cc(F)c2)cc1)NO
E3 Binder	CHEMBL434466	ChEMBL	7.18	—	—	O=C(/C=C/c1ccc(S(=O)(=O)Nc2ccc(-c3ccccc3)cc2)cc1)NO
E3 Binder	CHEMBL258824	ChEMBL	7.54	—	—	O=C(/C=C/c1ccc(S(=O)(=O)Nc2ccccc2)cc1)NO
E3 Binder	CHEMBL3262728	ChEMBL	6.62	—	—	O=C(/C=C/c1ccc(S(=O)(=O)n2ccc3cccnc32)cc1)NO
E3 Binder	CHEMBL3262726	ChEMBL	6.25	—	—	O=C(/C=C/c1ccc(S(=O)(=O)n2ccc3ccncc32)cc1)NO
E3 Binder	CHEMBL3262724	ChEMBL	6.3	—	—	O=C(/C=C/c1ccc(S(=O)(=O)n2ncc3ccccc32)cc1)NO
E3 Binder	CHEMBL244670	ChEMBL	6.47	—	—	O=C(/C=C/c1ccc2[nH]c(C(=O)c3ccccc3)cc2c1)NO
E3 Binder	CHEMBL2048759	ChEMBL	6.56	—	—	O=C(/C=C/c1ccc2[nH]cc(S(=O)(=O)c3ccccc3)c2c1)NO
E3 Binder	CHEMBL2425963	ChEMBL	7.39	—	—	O=C(/C=C/c1ccc2c(=O)n(CCc3ccccc3)c(C3CC3)nc2c1)NO
E3 Binder	CHEMBL2425960	ChEMBL	7.46	—	—	O=C(/C=C/c1ccc2c(=O)n(CCc3ccccc3)cnc2c1)NO
E3 Binder	CHEMBL1938445	ChEMBL	6.03	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)C1(CCN(Cc3ccccc3)CC1)O2)NO
E3 Binder	CHEMBL1938441	ChEMBL	6.66	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)C1(CCNCC1)O2)NO
E3 Binder	CHEMBL3758604	ChEMBL	6.78	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCCN(C(=O)c3ccccc3)C1)O2)NO
E3 Binder	CHEMBL3758233	ChEMBL	6.96	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCCN(C(=O)c3ccccc3)CC1)O2)NO
E3 Binder	CHEMBL3758184	ChEMBL	9.0	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCCN(CCc3ccccc3)C1)O2)NO
E3 Binder	CHEMBL3758515	ChEMBL	7.25	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCCN(CCc3ccccc3)CC1)O2)NO
E3 Binder	CHEMBL3758716	ChEMBL	7.47	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCCN(Cc3ccc(F)cc3)C1)O2)NO
E3 Binder	CHEMBL3759858	ChEMBL	6.83	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCCN(Cc3ccc(F)cc3)CC1)O2)NO
E3 Binder	CHEMBL3758450	ChEMBL	7.25	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCCN(Cc3ccccc3)C1)O2)NO
E3 Binder	CHEMBL3759808	ChEMBL	7.14	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCCN(Cc3ccccc3)CC1)O2)NO
E3 Binder	CHEMBL3759169	ChEMBL	6.87	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCCNC1)O2)NO
E3 Binder	CHEMBL3759976	ChEMBL	6.87	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCCNCC1)O2)NO
E3 Binder	CHEMBL3759066	ChEMBL	6.73	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCN(C(=O)c3ccccc3)C1)O2)NO
E3 Binder	CHEMBL1938434	ChEMBL	6.5	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCN(C(=O)c3ccccc3)CC1)O2)NO
E3 Binder	CHEMBL3759550	ChEMBL	7.57	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCN(CCc3ccccc3)C1)O2)NO
E3 Binder	CHEMBL2390996	ChEMBL	6.95	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCN(CCc3ccccc3)CC1)O2)NO
E3 Binder	CHEMBL3758891	ChEMBL	6.71	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCN(Cc3ccc(F)cc3)C1)O2)NO
E3 Binder	CHEMBL2390995	ChEMBL	6.97	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCN(Cc3ccc(F)cc3)CC1)O2)NO
E3 Binder	CHEMBL3758901	ChEMBL	7.58	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCN(Cc3ccccc3)C1)O2)NO
E3 Binder	CHEMBL1938433	ChEMBL	7.59	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCN(Cc3ccccc3)CC1)O2)NO
E3 Binder	CHEMBL3759091	ChEMBL	6.88	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCNC1)O2)NO
E3 Binder	CHEMBL1938429	ChEMBL	7.09	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CCNCC1)O2)NO
E3 Binder	CHEMBL3759521	ChEMBL	7.09	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CN(C(=O)c3ccccc3)C1)O2)NO
E3 Binder	CHEMBL3759583	ChEMBL	6.66	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CN(CCc3ccccc3)C1)O2)NO
E3 Binder	CHEMBL3758910	ChEMBL	6.89	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CN(Cc3ccc(F)cc3)C1)O2)NO
E3 Binder	CHEMBL3759197	ChEMBL	7.17	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CN(Cc3ccccc3)C1)O2)NO
E3 Binder	CHEMBL3760005	ChEMBL	6.64	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)CC1(CNC1)O2)NO
E3 Binder	CHEMBL198140	ChEMBL	6.75	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)N(CCc1ccccc1)C2=O)NO
E3 Binder	CHEMBL247653	ChEMBL	6.12	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)N(Cc1ccc(-c3ccccc3)cc1)C2)NO
E3 Binder	CHEMBL247654	ChEMBL	6.55	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)N(Cc1ccc(-c3cccnc3)cc1)C2)NO
E3 Binder	CHEMBL370695	ChEMBL	6.73	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)N(Cc1ccc(CO)cc1)C2=O)NO
E3 Binder	CHEMBL2390994	ChEMBL	6.19	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)N(Cc1ccccc1)C1(CCN(CCc3ccccc3)CC1)O2)NO
E3 Binder	CHEMBL2390993	ChEMBL	6.18	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)N(Cc1ccccc1)C1(CCN(Cc3ccc(F)cc3)CC1)O2)NO
E3 Binder	CHEMBL2390992	ChEMBL	6.27	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)N(Cc1ccccc1)C1(CCN(Cc3ccccc3)CC1)O2)NO
E3 Binder	CHEMBL2391007	ChEMBL	7.23	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)N(Cc1ccccc1)C1(CCNCC1)O2)NO
E3 Binder	CHEMBL247217	ChEMBL	6.64	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)N(Cc1ccccc1)C2)NO
E3 Binder	CHEMBL197774	ChEMBL	6.83	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)N(Cc1ccccc1)C2=O)NO
E3 Binder	CHEMBL197480	ChEMBL	6.12	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)N([C@H](COC(=O)c1ccccc1)c1ccccc1)C2=O)NO
E3 Binder	CHEMBL2391001	ChEMBL	7.04	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)NC1(CCN(CCc3ccccc3)CC1)O2)NO
E3 Binder	CHEMBL2391000	ChEMBL	6.99	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)NC1(CCN(Cc3ccc(F)cc3)CC1)O2)NO
E3 Binder	CHEMBL2390999	ChEMBL	7.08	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)NC1(CCN(Cc3ccccc3)CC1)O2)NO
E3 Binder	CHEMBL2390997	ChEMBL	7.11	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)NC1(CCNCC1)O2)NO
E3 Binder	CHEMBL4556817	ChEMBL	6.27	—	—	O=C(/C=C/c1ccc2c(c1)C(=O)c1ccccc1C2=O)NO
E3 Binder	CHEMBL2385394	ChEMBL	6.79	—	—	O=C(/C=C/c1ccc2c(c1)Cc1sc(NCCN3CCOCC3)nc1-2)NO
E3 Binder	CHEMBL2385389	ChEMBL	6.53	—	—	O=C(/C=C/c1ccc2c(c1)Cc1sc(Nc3cccnc3)nc1-2)NO
E3 Binder	CHEMBL1938440	ChEMBL	6.44	—	—	O=C(/C=C/c1ccc2c(c1)OC1(CCN(C(=O)c3ccccc3)CC1)CC2=O)NO
E3 Binder	CHEMBL1955942	ChEMBL	7.54	—	—	O=C(/C=C/c1ccc2c(c1)OCO2)NCCCCCC(=O)NO
E3 Binder	CHEMBL388429	ChEMBL	7.05	—	—	O=C(/C=C/c1ccc2c(c1)cc(C(=O)c1ccccc1)n2S(=O)(=O)c1ccccc1)NO
E3 Binder	CHEMBL491316	ChEMBL	7.7	—	—	O=C(/C=C/c1ccc2c(c1)nc(CCc1ccccc1)n2CCN1CCCC1)NO
E3 Binder	CHEMBL489332	ChEMBL	7.57	—	—	O=C(/C=C/c1ccc2c(c1)nc(CCc1ccccc1)n2CCN1CCCCC1)NO
E3 Binder	CHEMBL2048756	ChEMBL	6.73	—	—	O=C(/C=C/c1ccc2c(ccn2-c2ccccc2)c1)NO
E3 Binder	CHEMBL2048754	ChEMBL	6.12	—	—	O=C(/C=C/c1ccc2c(ccn2C(=O)c2ccccc2)c1)NO
E3 Binder	CHEMBL2048755	ChEMBL	7.49	—	—	O=C(/C=C/c1ccc2c(ccn2Cc2ccccc2)c1)NO
E3 Binder	CHEMBL2048751	ChEMBL	7.78	—	—	O=C(/C=C/c1ccc2c(ccn2S(=O)(=O)c2ccc(F)cc2)c1)NO
E3 Binder	CHEMBL2048752	ChEMBL	7.9	—	—	O=C(/C=C/c1ccc2c(ccn2S(=O)(=O)c2ccc([N+](=O)[O-])cc2)c1)NO
E3 Binder	CHEMBL2048746	ChEMBL	9.0	—	—	O=C(/C=C/c1ccc2c(ccn2S(=O)(=O)c2ccccc2)c1)NO
E3 Binder	CHEMBL4646266	ChEMBL	7.29	—	—	O=C(/C=C/c1ccc2cc(Oc3ccc([N+](=O)[O-])cc3)ccc2n1)NO
E3 Binder	CHEMBL490261	ChEMBL	8.15	—	—	O=C(/C=C/c1ccc2ccccc2c1)NCCCCCC(=O)NO
E3 Binder	CHEMBL1958437	ChEMBL	7.66	—	—	O=C(/C=C/c1ccc2ccccc2n1)NO
E3 Binder	CHEMBL484073	ChEMBL	8.47	—	—	O=C(/C=C/c1ccc2cccnc2c1)NCCCCCC(=O)NO
E3 Binder	CHEMBL2048747	ChEMBL	6.59	—	—	O=C(/C=C/c1ccc2ccn(S(=O)(=O)c3ccccc3)c2c1)NO
E3 Binder	CHEMBL501518	ChEMBL	7.44	—	—	O=C(/C=C/c1ccc2ncccc2c1)NCCCCCC(=O)NO
E3 Binder	CHEMBL397904	ChEMBL	6.08	—	—	O=C(/C=C/c1ccc2oc(C(=O)c3ccccc3)cc2c1)NO
E3 Binder	CHEMBL1630109	ChEMBL	7.33	—	—	O=C(/C=C/c1cccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)c1)NO
E3 Binder	CHEMBL1098042	ChEMBL	7.0	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3[nH]2)c1)NO
E3 Binder	CHEMBL1099094	ChEMBL	7.0	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2-c2ccc(Cl)cc2)c1)NO
E3 Binder	CHEMBL1094085	ChEMBL	7.3	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2-c2ccccc2)c1)NO
E3 Binder	CHEMBL1097369	ChEMBL	7.6	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2C2CCCCC2)c1)NO
E3 Binder	CHEMBL1094794	ChEMBL	7.4	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2C2CCCNC2)c1)NO
E3 Binder	CHEMBL1095076	ChEMBL	6.7	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2CC2CCNCC2)c1)NO
E3 Binder	CHEMBL1097761	ChEMBL	7.7	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2CCCc2ccccc2)c1)NO
E3 Binder	CHEMBL1099058	ChEMBL	7.2	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2CCN2CCCC2)c1)NO
E3 Binder	CHEMBL1099057	ChEMBL	7.4	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2CCN2CCCCC2)c1)NO
E3 Binder	CHEMBL1095075	ChEMBL	6.8	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2CCN2CCOCC2)c1)NO
E3 Binder	CHEMBL1099096	ChEMBL	7.51	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2CCc2ccccc2)c1)NO
E3 Binder	CHEMBL1097981	ChEMBL	7.2	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2Cc2ccccc2)c1)NO
E3 Binder	CHEMBL1095124	ChEMBL	7.1	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2[C@@H]2CCCNC2)c1)NO
E3 Binder	CHEMBL1094152	ChEMBL	7.6	—	—	O=C(/C=C/c1cccc(-c2nc3ccccc3n2[C@H]2CCCNC2)c1)NO
E3 Binder	CHEMBL569326	ChEMBL	7.07	—	—	O=C(/C=C/c1cccc(/C=C/C(=O)c2ccccc2)c1)NO
E3 Binder	CHEMBL569715	ChEMBL	7.7	—	—	O=C(/C=C/c1cccc(/C=C/C(=O)c2ccccc2)n1)NO
E3 Binder	CHEMBL4541704	ChEMBL	8.0	—	—	O=C(/C=C/c1cccc(C(=O)NC(Cc2c[nH]c3ccccc23)C(=O)Nc2ccc(Cl)cc2)c1)NO
E3 Binder	CHEMBL5268446	ChEMBL	7.17	—	—	O=C(/C=C/c1cccc(C(=O)NCC2CCN(Cc3ccccc3)CC2)c1)NO
E3 Binder	CHEMBL2381524	ChEMBL	7.68	—	—	O=C(/C=C/c1cccc(C(=O)NO)c1)Nc1ccccc1
E3 Binder	CHEMBL242533	ChEMBL	7.41	—	—	O=C(/C=C/c1cccc(C(=O)c2cc3ccccc3[nH]2)c1)NO
E3 Binder	CHEMBL390907	ChEMBL	7.47	—	—	O=C(/C=C/c1cccc(C(=O)c2cc3ccccc3n2S(=O)(=O)c2ccccc2)c1)NO
E3 Binder	CHEMBL390452	ChEMBL	7.24	—	—	O=C(/C=C/c1cccc(C(=O)c2cc3ccccc3o2)c1)NO
E3 Binder	CHEMBL270326	ChEMBL	6.82	—	—	O=C(/C=C/c1cccc(Cc2nc3ccccc3[nH]2)c1)NO
E3 Binder	CHEMBL270331	ChEMBL	6.97	—	—	O=C(/C=C/c1cccc(NS(=O)(=O)c2ccc(-c3ccccc3)cc2)c1)NO
E3 Binder	CHEMBL271785	ChEMBL	6.73	—	—	O=C(/C=C/c1cccc(NS(=O)(=O)c2ccccc2)c1)NO
E3 Binder	CHEMBL5271319	ChEMBL	6.25	—	—	O=C(/C=C/c1cccc(Nc2ncnc3cc4c(cc23)OCCO4)c1)NO
E3 Binder	CHEMBL3354911	ChEMBL	6.3	—	—	O=C(/C=C/c1cccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)CCCc2ccccc2)c1)NO
E3 Binder	CHEMBL3354910	ChEMBL	6.33	—	—	O=C(/C=C/c1cccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)CCc2ccccc2)c1)NO
E3 Binder	CHEMBL3354909	ChEMBL	6.35	—	—	O=C(/C=C/c1cccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)Cc2ccccc2)c1)NO
E3 Binder	CHEMBL3354918	ChEMBL	6.11	—	—	O=C(/C=C/c1cccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2cc(Cl)cc(Cl)c2)c1)NO
E3 Binder	CHEMBL3354912	ChEMBL	6.16	—	—	O=C(/C=C/c1cccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(Br)cc2)c1)NO
E3 Binder	CHEMBL3233711	ChEMBL	6.78	—	—	O=C(/C=C/c1cccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(Cl)cc2)c1)NO
E3 Binder	CHEMBL3354917	ChEMBL	6.59	—	—	O=C(/C=C/c1cccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(Cl)cc2Cl)c1)NO
E3 Binder	CHEMBL3233710	ChEMBL	6.35	—	—	O=C(/C=C/c1cccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccc(F)cc2)c1)NO
E3 Binder	CHEMBL3354916	ChEMBL	6.45	—	—	O=C(/C=C/c1cccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2cccc(Cl)c2)c1)NO
E3 Binder	CHEMBL3233709	ChEMBL	6.38	—	—	O=C(/C=C/c1cccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccccc2)c1)NO
E3 Binder	CHEMBL3354915	ChEMBL	7.09	—	—	O=C(/C=C/c1cccc(OC[C@H](Cc2c[nH]c3ccccc23)NC(=O)c2ccccc2Cl)c1)NO
E3 Binder	CHEMBL1958435	ChEMBL	6.57	—	—	O=C(/C=C/c1cccc(S(=O)(=O)N2CCN(Cc3ccc4c(c3)OCO4)CC2)c1)NO
E3 Binder	CHEMBL1958423	ChEMBL	6.83	—	—	O=C(/C=C/c1cccc(S(=O)(=O)N2CCN(c3ccc(Cl)cc3)CC2)c1)NO
E3 Binder	CHEMBL1958425	ChEMBL	6.73	—	—	O=C(/C=C/c1cccc(S(=O)(=O)N2CCN(c3cccc(Cl)c3)CC2)c1)NO
E3 Binder	CHEMBL1958432	ChEMBL	6.88	—	—	O=C(/C=C/c1cccc(S(=O)(=O)N2CCN(c3ccccc3)CC2)c1)NO
E3 Binder	CHEMBL1958428	ChEMBL	7.17	—	—	O=C(/C=C/c1cccc(S(=O)(=O)N2CCN(c3ccccc3Cl)CC2)c1)NO
E3 Binder	CHEMBL1958427	ChEMBL	6.72	—	—	O=C(/C=C/c1cccc(S(=O)(=O)N2CCN(c3ccccc3F)CC2)c1)NO
E3 Binder	CHEMBL1958424	ChEMBL	6.91	—	—	O=C(/C=C/c1cccc(S(=O)(=O)N2CCN(c3ccccn3)CC2)c1)NO
E3 Binder	CHEMBL1958422	ChEMBL	7.08	—	—	O=C(/C=C/c1cccc(S(=O)(=O)N2CCN(c3ncccn3)CC2)c1)NO
E3 Binder	CHEMBL3259849	ChEMBL	6.22	—	—	O=C(/C=C/c1cccc(S(=O)(=O)N2CCc3cccnc32)c1)NO
E3 Binder	CHEMBL4649439	ChEMBL	6.09	—	—	O=C(/C=C/c1cccc(S(=O)(=O)NCCCN2c3ccccc3CCc3ccc(Cl)cc32)c1)NO
E3 Binder	CHEMBL270733	ChEMBL	7.47	—	—	O=C(/C=C/c1cccc(S(=O)(=O)NCc2ccccc2)c1)NO
E3 Binder	CHEMBL270734	ChEMBL	7.27	—	—	O=C(/C=C/c1cccc(S(=O)(=O)Nc2ccc(-c3ccccc3)cc2)c1)NO
E3 Binder	CHEMBL1958438	ChEMBL	7.38	—	—	O=C(/C=C/c1cccc(S(=O)(=O)Nc2ccc(Cl)cc2)c1)NO
E3 Binder	CHEMBL1958429	ChEMBL	8.0	—	—	O=C(/C=C/c1cccc(S(=O)(=O)Nc2ccc(OC(F)F)cc2)c1)NO
E3 Binder	CHEMBL1958436	ChEMBL	7.7	—	—	O=C(/C=C/c1cccc(S(=O)(=O)Nc2cccc(F)c2)c1)NO
E3 Binder	CHEMBL408513	ChEMBL	8.8	5OG	—	O=C(/C=C/c1cccc(S(=O)(=O)Nc2ccccc2)c1)NO
E3 Binder	CHEMBL3925939	ChEMBL	8.23	—	—	O=C(/C=C/c1cccc(S(=O)(=O)c2ccc3cccc(F)c3n2)c1)NO
E3 Binder	CHEMBL3973951	ChEMBL	9.54	—	—	O=C(/C=C/c1cccc(S(=O)(=O)c2ccc3ccccc3n2)c1)NO
E3 Binder	CHEMBL3262722	ChEMBL	6.29	—	—	O=C(/C=C/c1cccc(S(=O)(=O)n2ccc3ccccc32)c1)NO
E3 Binder	CHEMBL3262727	ChEMBL	8.28	—	—	O=C(/C=C/c1cccc(S(=O)(=O)n2ccc3cccnc32)c1)NO
E3 Binder	CHEMBL3262725	ChEMBL	6.55	—	—	O=C(/C=C/c1cccc(S(=O)(=O)n2ccc3ccncc32)c1)NO
E3 Binder	CHEMBL3262723	ChEMBL	6.64	—	—	O=C(/C=C/c1cccc(S(=O)(=O)n2ncc3ccccc32)c1)NO
E3 Binder	CHEMBL2048745	ChEMBL	6.77	—	—	O=C(/C=C/c1cccc2c1ccn2S(=O)(=O)c1ccccc1)NO
E3 Binder	CHEMBL483260	ChEMBL	7.6	—	—	O=C(/C=C/c1cccc2cccnc12)NCCCCCC(=O)NO
E3 Binder	CHEMBL453755	ChEMBL	7.7	—	—	O=C(/C=C/c1ccccc1)NCCCCCC(=O)NO
E3 Binder	CHEMBL154574	ChEMBL	7.66	—	—	O=C(/C=C/c1ccccc1)NO
E3 Binder	CHEMBL2032251	ChEMBL	7.0	TB8	—	O=C(/C=C/c1ccccc1Cl)NO
E3 Binder	CHEMBL451583	ChEMBL	7.34	—	—	O=C(/C=C/c1ccccn1)NCCCCCC(=O)NO.O=C(O)C(=O)O
E3 Binder	CHEMBL3427661	ChEMBL	6.68	—	—	O=C(/C=C/c1cccn(CCCc2ccc(Br)cc2)c1=O)NO
E3 Binder	CHEMBL4082995	ChEMBL	8.61	—	—	O=C(/C=C/c1cccn(CCCc2ccc3ccccc3c2)c1=O)NO
E3 Binder	CHEMBL3427660	ChEMBL	7.0	—	—	O=C(/C=C/c1cccn(CCCc2cccc(Br)c2)c1=O)NO
E3 Binder	CHEMBL3427659	ChEMBL	6.32	—	—	O=C(/C=C/c1cccn(CCCc2ccccc2Br)c1=O)NO
E3 Binder	CHEMBL3427667	ChEMBL	6.24	—	—	O=C(/C=C/c1cccn(CCCc2cccnc2)c1=O)NO
E3 Binder	CHEMBL3427650	ChEMBL	6.44	—	—	O=C(/C=C/c1cccn(CCc2ccc(Br)cc2)c1=O)NO
E3 Binder	CHEMBL4577107	ChEMBL	7.29	—	—	O=C(/C=C/c1cccn(CCc2ccc3ccccc3c2)c1=O)NO
E3 Binder	CHEMBL3427649	ChEMBL	6.8	—	—	O=C(/C=C/c1cccn(CCc2cccc(Br)c2)c1=O)NO
E3 Binder	CHEMBL3427639	ChEMBL	7.0	—	—	O=C(/C=C/c1cccn(Cc2ccc(Br)cc2)c1=O)NO
E3 Binder	CHEMBL3427648	ChEMBL	7.52	—	—	O=C(/C=C/c1cccn(Cc2ccc3ccccc3n2)c1=O)NO
E3 Binder	CHEMBL3427638	ChEMBL	6.42	—	—	O=C(/C=C/c1cccn(Cc2cccc(Br)c2)c1=O)NO
E3 Binder	CHEMBL3427637	ChEMBL	6.72	—	—	O=C(/C=C/c1cccn(Cc2ccccc2Br)c1=O)NO
E3 Binder	CHEMBL3427645	ChEMBL	6.34	—	—	O=C(/C=C/c1cccn(Cc2ccccn2)c1=O)NO
E3 Binder	CHEMBL3427646	ChEMBL	6.52	—	—	O=C(/C=C/c1cccn(Cc2cccnc2)c1=O)NO
E3 Binder	CHEMBL3427647	ChEMBL	6.38	—	—	O=C(/C=C/c1cccn(Cc2ccncc2)c1=O)NO
E3 Binder	CHEMBL490260	ChEMBL	6.85	—	—	O=C(/C=C/c1cccnc1)NCCCCCC(=O)NO.O=C(O)C(=O)O
E3 Binder	CHEMBL521766	ChEMBL	7.0	—	—	O=C(/C=C/c1ccncc1)NCCCCCC(=O)NO.O=C(O)C(=O)O
E3 Binder	CHEMBL1808165	ChEMBL	7.27	—	—	O=C(/C=C/c1cn(C(/C=C/c2ccccc2)C2CCC2)nn1)NO
E3 Binder	CHEMBL1808166	ChEMBL	6.94	—	—	O=C(/C=C/c1cn(C(/C=C/c2ccccc2)C2CCCC2)nn1)NO
E3 Binder	CHEMBL1808173	ChEMBL	7.03	—	—	O=C(/C=C/c1cn(C(/C=C/c2ccccc2)Cc2ccc3ccccc3c2)nn1)NO
E3 Binder	CHEMBL1808170	ChEMBL	6.39	—	—	O=C(/C=C/c1cn(C(/C=C/c2ccccc2)Cc2cccc(-c3ccccc3)c2)nn1)NO
E3 Binder	CHEMBL1808171	ChEMBL	6.29	—	—	O=C(/C=C/c1cn(C(/C=C/c2ccccc2)Cc2cccc(Oc3ccccc3)c2)nn1)NO
E3 Binder	CHEMBL1808172	ChEMBL	6.96	—	—	O=C(/C=C/c1cn(C(/C=C/c2ccccc2)Cc2cccc3ccccc23)nn1)NO
E3 Binder	CHEMBL1808168	ChEMBL	7.11	—	—	O=C(/C=C/c1cn(C(/C=C/c2ccccc2)Cc2ccccc2)nn1)NO
E3 Binder	CHEMBL1808169	ChEMBL	6.77	—	—	O=C(/C=C/c1cn(C(/C=C/c2ccccc2)Cc2nccs2)nn1)NO
E3 Binder	CHEMBL2036477	ChEMBL	6.66	—	—	O=C(/C=C/c1cn(C(Cc2ccccc2)c2nc3ccccc3o2)nn1)NO
E3 Binder	CHEMBL487962	ChEMBL	6.98	—	—	O=C(/C=C/c1cn(C/C=C/c2ccccc2)nn1)NO
E3 Binder	CHEMBL2036472	ChEMBL	6.75	—	—	O=C(/C=C/c1cn(Cc2nc3ccccc3[nH]2)nn1)NO
E3 Binder	CHEMBL2036471	ChEMBL	6.98	—	—	O=C(/C=C/c1cn(Cc2nc3ccccc3o2)nn1)NO
E3 Binder	CHEMBL2036470	ChEMBL	7.39	—	—	O=C(/C=C/c1cn(Cc2nc3ccccc3s2)nn1)NO
E3 Binder	CHEMBL5084994	ChEMBL	6.03	—	—	O=C(/C=C/c1cnc(-c2ccc(F)cc2F)s1)NO
E3 Binder	CHEMBL5077333	ChEMBL	6.26	—	—	O=C(/C=C/c1cnc(-c2ccc(N3CCOCC3)cc2)s1)NO
E3 Binder	CHEMBL5085234	ChEMBL	6.17	—	—	O=C(/C=C/c1cnc(-c2ccc3c(c2)OCCO3)s1)NO
E3 Binder	CHEMBL5078499	ChEMBL	6.05	—	—	O=C(/C=C/c1cnc(-c2ccc3c(c2)OCO3)s1)NO
E3 Binder	CHEMBL399738	ChEMBL	7.3	—	—	O=C(/C=C/c1cnc(N2CCN(S(=O)(=O)c3ccc4ccccc4c3)CC2)s1)NO
E3 Binder	CHEMBL250995	ChEMBL	6.36	—	—	O=C(/C=C/c1cnc(N2CCN(S(=O)(=O)c3ccccc3)CC2)s1)NO
E3 Binder	CHEMBL5204550	ChEMBL	6.77	—	—	O=C(/C=C/c1csc(Br)n1)NO
E3 Binder	CHEMBL1958440	ChEMBL	7.32	—	—	O=C(/C=C/c1nc2ccccc2o1)NO
E3 Binder	CHEMBL485513	ChEMBL	6.7	—	—	O=C(C=C(c1ccccc1)c1ccccc1)NCCCCCC(=O)NO
E3 Binder	CHEMBL485514	ChEMBL	8.7	—	—	O=C(C=C1c2ccccc2-c2ccccc21)NCCCCCC(=O)NO
E3 Binder	CHEMBL519210	ChEMBL	6.47	—	—	O=C(C=C1c2ccccc2CCc2ccccc21)NCCCCCC(=O)NO
E3 Binder	CHEMBL3960127	ChEMBL	7.0	—	—	O=C(CCC(=O)NCc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL5288573	ChEMBL	6.7	—	—	O=C(CCC(=O)Nc1nnc(-c2ccc(Cl)cc2)s1)NO
E3 Binder	CHEMBL5269957	ChEMBL	6.7	—	—	O=C(CCC(=O)Nc1nnc(-c2ccc(O)cc2)s1)NO
E3 Binder	CHEMBL4284448	ChEMBL	6.85	—	—	O=C(CCC(CCCC(=O)Nc1ccccc1)Cc1ccccc1)NO
E3 Binder	CHEMBL4295105	ChEMBL	6.96	—	—	O=C(CCC(CCCC(=O)Nc1ccccc1)c1ccccc1)NO
E3 Binder	CHEMBL250195	ChEMBL	6.7	—	—	O=C(CCC1=CCCN(CCCCc2ccc(-c3ccccc3)cc2)C1=O)NO
E3 Binder	CHEMBL250396	ChEMBL	6.96	—	—	O=C(CCC1=CCCN(CCCCc2cccc3ccccc23)C1=O)NO
E3 Binder	CHEMBL226224	ChEMBL	6.89	—	—	O=C(CCC1=CCCN(CCCCc2ccccc2)C1=O)NO
E3 Binder	CHEMBL250193	ChEMBL	6.57	—	—	O=C(CCC1=CCCN(CCCc2ccc(-c3ccccc3)cc2)C1=O)NO
E3 Binder	CHEMBL428054	ChEMBL	7.52	—	—	O=C(CCC1=CCCN(CCCc2ccc3ccccc3c2)C1=O)NO
E3 Binder	CHEMBL388174	ChEMBL	6.57	—	—	O=C(CCC1=CCCN(CCCc2ccccc2)C1=O)NO
E3 Binder	CHEMBL249580	ChEMBL	6.64	—	—	O=C(CCC1=CCCN(CCc2ccc(-c3ccccc3)cc2)C1=O)NO
E3 Binder	CHEMBL249993	ChEMBL	7.43	—	—	O=C(CCC1=CCCN(CCc2ccc3ccccc3c2)C1=O)NO
E3 Binder	CHEMBL400139	ChEMBL	6.5	—	—	O=C(CCC1=CCCN(CCc2cccc3ccccc23)C1=O)NO
E3 Binder	CHEMBL214049	ChEMBL	6.46	—	—	O=C(CCC1=CCCN(CCc2ccccc2)C1=O)NO
E3 Binder	CHEMBL250676	ChEMBL	6.35	—	—	O=C(CCC1=CCCN(Cc2ccc(Br)cc2)C1=O)NO
E3 Binder	CHEMBL251033	ChEMBL	6.25	—	—	O=C(CCC1=CCCN(Cc2ccc(F)cc2)C1=O)NO
E3 Binder	CHEMBL399347	ChEMBL	6.29	—	—	O=C(CCC1=CCCN(Cc2ccc(NC(=O)c3ccccc3)cc2)C1=O)NO
E3 Binder	CHEMBL249382	ChEMBL	6.64	—	—	O=C(CCC1=CCCN(Cc2ccc([N+](=O)[O-])cc2)C1=O)NO
E3 Binder	CHEMBL213997	ChEMBL	6.17	—	—	O=C(CCC1=CCCN(Cc2ccccc2)C1=O)NO
E3 Binder	CHEMBL1668018	ChEMBL	6.1	—	—	O=C(CCC1=CCN(CCCc2ccc3ccccc3c2)C1=O)NO
E3 Binder	CHEMBL4537466	ChEMBL	8.01	—	—	O=C(CCC1C(=O)N(Cc2ccccc2)C(=O)N1Cc1ccc(Br)cc1)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4459226	ChEMBL	7.78	—	—	O=C(CCC1C(=O)N(c2ccc(Cl)cc2)C(=O)N1Cc1ccc(Br)cc1)NCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4444176	ChEMBL	8.01	—	—	O=C(CCC1C(=O)N(c2ccc(Cl)cc2)C(=O)N1Cc1ccc(Br)cc1)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4439468	ChEMBL	7.9	—	—	O=C(CCC1C(=O)N(c2ccc(Cl)cc2)C(=O)N1Cc1ccccc1)NCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4450285	ChEMBL	8.12	—	—	O=C(CCC1C(=O)N(c2ccc(Cl)cc2)C(=O)N1Cc1ccccc1)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4587714	ChEMBL	7.87	—	—	O=C(CCC1C(=O)N(c2ccccc2)C(=O)N1Cc1ccc(Br)cc1)NCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3086768	ChEMBL	6.41	—	—	O=C(CCCC(=O)NCCc1ccccc1)NO
E3 Binder	CHEMBL3905089	ChEMBL	7.0	—	—	O=C(CCCC(=O)NCc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL3971412	ChEMBL	7.0	—	—	O=C(CCCC(=O)Nc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL4102833	ChEMBL	6.57	—	—	O=C(CCCC(CCC(=O)Nc1ccccc1)Cc1ccccc1)NO
E3 Binder	CHEMBL599968	ChEMBL	6.29	—	—	O=C(CCCC/C=C(\F)CS)Nc1ccccc1
E3 Binder	CHEMBL1760913	ChEMBL	6.58	—	—	O=C(CCCC1CCN(C(=O)Cc2ccccc2)CC1)NO
E3 Binder	CHEMBL1760915	ChEMBL	7.05	—	—	O=C(CCCC1CCN(C(=O)NCc2ccccc2)CC1)NO
E3 Binder	CHEMBL1760914	ChEMBL	7.0	—	—	O=C(CCCC1CCN(C(=O)Nc2ccccc2)CC1)NO
E3 Binder	CHEMBL1760910	ChEMBL	6.08	—	—	O=C(CCCC1CCN(S(=O)(=O)Cc2ccccc2)CC1)NO
E3 Binder	CHEMBL1910049	ChEMBL	6.89	—	—	O=C(CCCC1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1)NO
E3 Binder	CHEMBL1910042	ChEMBL	6.67	—	—	O=C(CCCC1CCN(S(=O)(=O)c2cccc(-c3cnco3)c2)CC1)NO
E3 Binder	CHEMBL1910050	ChEMBL	6.74	—	—	O=C(CCCC1CCN(S(=O)(=O)c2cccc3ccccc23)CC1)NO
E3 Binder	CHEMBL1760911	ChEMBL	6.27	—	—	O=C(CCCC1CCN(S(=O)(=O)c2ccccc2)CC1)NO
E3 Binder	CHEMBL1909951	ChEMBL	6.76	—	—	O=C(CCCC1CCN(S(=O)(=O)c2ccccc2Cl)CC1)NO
E3 Binder	CHEMBL3417188	ChEMBL	6.07	—	—	O=C(CCCCC(=O)N1C/C=C/CCOc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO
E3 Binder	CHEMBL3417193	ChEMBL	6.4	—	—	O=C(CCCCC(=O)N1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO
E3 Binder	CHEMBL3984522	ChEMBL	7.0	—	—	O=C(CCCCC(=O)NCc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL3948777	ChEMBL	6.0	—	—	O=C(CCCCC(=O)Nc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL3339009	ChEMBL	6.25	—	—	O=C(CCCCC(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2s1)NO
E3 Binder	CHEMBL3621296	ChEMBL	8.79	—	—	O=C(CCCCC(=O)Nc1ccc2c(c1)/C(=C/c1ccc[nH]1)C(=O)N2)NO
E3 Binder	CHEMBL2204666	ChEMBL	6.46	—	—	O=C(CCCCC(CC(=O)Nc1ccccc1)c1ccccc1)NO
E3 Binder	CHEMBL597443	ChEMBL	6.44	—	—	O=C(CCCCC/C=C(\F)CS)Nc1ccccc1
E3 Binder	CHEMBL126465	ChEMBL	6.0	—	—	O=C(CCCCC/C=C/c1ccc(-c2ccccc2)cc1)c1ncco1
E3 Binder	CHEMBL5174162	ChEMBL	7.62	—	—	O=C(CCCCC/C=C/c1csc(Br)n1)NO
E3 Binder	CHEMBL5193020	ChEMBL	8.4	—	—	O=C(CCCCC/C=C\c1csc(Br)n1)NO
E3 Binder	CHEMBL1243289	ChEMBL	6.12	—	—	O=C(CCCCC1CC(C(=O)NO)=NO1)Nc1ccccc1
E3 Binder	CHEMBL3675756	ChEMBL	7.17	—	—	O=C(CCCCC=C(c1ccccn1)c1ccccn1)NO
E3 Binder	CHEMBL5274330	ChEMBL	8.94	—	—	O=C(CCCCCC(=O)N(Cc1ccc(Br)s1)c1ccc(OCCN2CCOCC2)cc1)NO
E3 Binder	CHEMBL3759982	ChEMBL	9.22	—	—	O=C(CCCCCC(=O)N/N=C/c1ccc(-c2ccccc2)cc1)NO
E3 Binder	CHEMBL3759794	ChEMBL	9.3	—	—	O=C(CCCCCC(=O)N/N=C/c1ccc(-c2cccnc2)cc1)NO
E3 Binder	CHEMBL4636051	ChEMBL	7.21	—	—	O=C(CCCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc21)NO
E3 Binder	CHEMBL3946124	ChEMBL	7.0	—	—	O=C(CCCCCC(=O)Nc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL3339013	ChEMBL	7.52	—	—	O=C(CCCCCC(=O)Nc1cc2c(Nc3ccc(Cl)c(C(F)(F)F)c3)ncnc2s1)NO
E3 Binder	CHEMBL3339010	ChEMBL	7.62	—	—	O=C(CCCCCC(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2s1)NO
E3 Binder	CHEMBL3339021	ChEMBL	7.57	—	—	O=C(CCCCCC(=O)Nc1cc2c(Nc3ccccc3)ncnc2s1)NO
E3 Binder	CHEMBL3933593	ChEMBL	8.6	—	—	O=C(CCCCCC(=O)Nc1ccc(NCCOc2ccc3cc2COC/C=C/COCc2cccc(c2)-c2ccnc(n2)N3)cc1)NO
E3 Binder	CHEMBL1630846	ChEMBL	7.36	—	—	O=C(CCCCCC(=O)Nc1cccc2cccnc12)NS
E3 Binder	CHEMBL126289	ChEMBL	6.51	—	—	O=C(CCCCCC(=O)c1ncco1)Nc1cccc(-c2ccccc2)c1
E3 Binder	CHEMBL561604	ChEMBL	7.7	—	—	O=C(CCCCCC(c1c[nH]c2ccc([N+](=O)[O-])cc12)c1c[nH]c2ccc([N+](=O)[O-])cc12)NO
E3 Binder	CHEMBL564876	ChEMBL	8.22	—	—	O=C(CCCCCC(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12)NO
E3 Binder	CHEMBL1631912	ChEMBL	8.03	—	—	O=C(CCCCCC1OCCCCCCCOc2ccccc2NC1=O)NO
E3 Binder	CHEMBL1631911	ChEMBL	8.0	—	—	O=C(CCCCCC1OCCCCCCOc2ccccc2NC1=O)NO
E3 Binder	CHEMBL1631910	ChEMBL	7.81	—	—	O=C(CCCCCC1OCCCCCOc2ccccc2NC1=O)NO
E3 Binder	CHEMBL3675759	ChEMBL	7.66	—	—	O=C(CCCCCC=C(c1ccccn1)c1ccccn1)NO
E3 Binder	CHEMBL331158	ChEMBL	6.52	—	—	O=C(CCCCCCC(=O)C(F)(F)F)Nc1ccc(Oc2ccccc2)cc1
E3 Binder	CHEMBL115011	ChEMBL	6.42	—	—	O=C(CCCCCCC(=O)C(F)(F)F)Nc1cccc(-c2ccccc2)c1
E3 Binder	CHEMBL116702	ChEMBL	6.51	—	—	O=C(CCCCCCC(=O)C(F)(F)F)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL5075729	ChEMBL	6.4	—	—	O=C(CCCCCCC(=O)N/N=C/c1ccc(N(c2ccccc2)c2ccccc2)cc1)NO
E3 Binder	CHEMBL5188297	ChEMBL	9.4	—	—	O=C(CCCCCCC(=O)N/N=C/c1cnc(N(c2ccccc2)c2ccccc2)nc1)NO
E3 Binder	CHEMBL3417189	ChEMBL	6.51	—	—	O=C(CCCCCCC(=O)N1C/C=C/CCOc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO
E3 Binder	CHEMBL3417194	ChEMBL	6.53	—	—	O=C(CCCCCCC(=O)N1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO
E3 Binder	CHEMBL2408694	ChEMBL	6.75	—	—	O=C(CCCCCCC(=O)N1CCN=C(c2ccccc2)c2ccccc21)NO
E3 Binder	CHEMBL4570814	ChEMBL	6.82	—	—	O=C(CCCCCCC(=O)NC(Cc1c[nH]c2ccccc12)C(=O)Nc1ccc(Cl)cc1)NO
E3 Binder	CHEMBL1630845	ChEMBL	6.38	—	—	O=C(CCCCCCC(=O)NC12CC3CC(CC(C3)C1)C2)NO
E3 Binder	CHEMBL3098696	ChEMBL	7.12	—	—	O=C(CCCCCCC(=O)NC1CCCC1)NO
E3 Binder	CHEMBL5280795	ChEMBL	6.23	—	—	O=C(CCCCCCC(=O)NCC1CCN(Cc2ccccc2)CC1)NO
E3 Binder	CHEMBL4636526	ChEMBL	6.18	—	—	O=C(CCCCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc21)NO
E3 Binder	CHEMBL483477	ChEMBL	7.6	—	—	O=C(CCCCCCC(=O)NCCc1ccccc1)NO
E3 Binder	CHEMBL2387320	ChEMBL	6.92	—	—	O=C(CCCCCCC(=O)NC[C@H]1O[C@@H]2O[C@H]3[C@H](O)[C@@H](O)[C@@H](O[C@H]4[C@H](O)[C@@H](O)[C@@H](O[C@H]5[C@H](O)[C@@H](O)[C@@H](O[C@H]6[C@H](O)[C@@H](O)[C@@H](O[C@H]7[C@H](O)[C@@H](O)[C@@H](O[C@H]8[C@H](O)[C@@H](O)[C@@H](O[C@H]1[C@H](O)[C@H]2O)O[C@@H]8CO)O[C@@H]7CO)O[C@@H]6CO)O[C@@H]5CO)O[C@@H]4CO)O[C@@H]3CO)NO
E3 Binder	CHEMBL3949983	ChEMBL	7.0	—	—	O=C(CCCCCCC(=O)NCc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL320497	ChEMBL	7.84	—	—	O=C(CCCCCCC(=O)NO)NO
E3 Binder	CHEMBL3339034	ChEMBL	7.82	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Cl)ncnc2s1)NO
E3 Binder	CHEMBL3339017	ChEMBL	8.05	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3ccc(Br)cc3F)ncnc2s1)NO
E3 Binder	CHEMBL3339014	ChEMBL	7.94	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3ccc(Cl)c(C(F)(F)F)c3)ncnc2s1)NO
E3 Binder	CHEMBL3339016	ChEMBL	8.25	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3ccc(Cl)cc3F)ncnc2s1)NO
E3 Binder	CHEMBL3339011	ChEMBL	7.66	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2s1)NO
E3 Binder	CHEMBL3339015	ChEMBL	8.1	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3ccc(F)cc3F)ncnc2s1)NO
E3 Binder	CHEMBL3339018	ChEMBL	8.18	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3ccc(I)cc3F)ncnc2s1)NO
E3 Binder	CHEMBL3339032	ChEMBL	8.03	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3ccc(N4CCCC4)c(F)c3)ncnc2s1)NO
E3 Binder	CHEMBL3339033	ChEMBL	8.14	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3ccc(N4CCCC4)cc3)ncnc2s1)NO
E3 Binder	CHEMBL3339031	ChEMBL	8.47	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3ccc(N4CCCCC4)c(F)c3)ncnc2s1)NO
E3 Binder	CHEMBL3339030	ChEMBL	8.72	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3ccc(O[C@H]4CCOC4)c(Cl)c3)ncnc2s1)NO
E3 Binder	CHEMBL3339020	ChEMBL	8.07	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3cccc(Cl)c3)ncnc2s1)NO
E3 Binder	CHEMBL3339019	ChEMBL	8.07	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3cccc(Cl)c3F)ncnc2s1)NO
E3 Binder	CHEMBL3339022	ChEMBL	7.92	—	—	O=C(CCCCCCC(=O)Nc1cc2c(Nc3ccccc3)ncnc2s1)NO
E3 Binder	CHEMBL4091531	ChEMBL	7.43	—	—	O=C(CCCCCCC(=O)Nc1cc2ncnc(Nc3ccc(Cl)cc3F)c2s1)NO
E3 Binder	CHEMBL4101744	ChEMBL	7.72	—	—	O=C(CCCCCCC(=O)Nc1cc2ncnc(Nc3ccc(F)cc3F)c2s1)NO
E3 Binder	CHEMBL4079625	ChEMBL	7.77	—	—	O=C(CCCCCCC(=O)Nc1cc2ncnc(Nc3cccc(Br)c3)c2s1)NO
E3 Binder	CHEMBL4097655	ChEMBL	7.47	—	—	O=C(CCCCCCC(=O)Nc1cc2ncnc(Nc3cccc(Cl)c3)c2s1)NO
E3 Binder	CHEMBL4086244	ChEMBL	7.37	—	—	O=C(CCCCCCC(=O)Nc1cc2ncnc(Nc3cccc(F)c3)c2s1)NO
E3 Binder	CHEMBL512644	ChEMBL	8.3	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2ccccc2)cc1)NO
E3 Binder	CHEMBL2417781	ChEMBL	7.8	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2ccccc2NC(=O)[C@@H]2CCCN2)cc1)NO
E3 Binder	CHEMBL4285223	ChEMBL	7.64	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2ccnc(Nc3ccc(N4CCCCC4)cc3)n2)cc1)NO
E3 Binder	CHEMBL4286867	ChEMBL	8.92	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2ccnc(Nc3ccc(N4CCOCC4)cc3)n2)cc1)NO
E3 Binder	CHEMBL4277267	ChEMBL	8.05	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2ccnc(Nc3cccc(N4CCCCC4)c3)n2)cc1)NO
E3 Binder	CHEMBL4278951	ChEMBL	8.84	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2ccnc(Nc3ccccc3)n2)cc1)NO
E3 Binder	CHEMBL519491	ChEMBL	8.89	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2cn(-c3ccccc3)nn2)cc1)NO
E3 Binder	CHEMBL483495	ChEMBL	8.36	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2cn(CC(O)c3cccc(Br)c3)nn2)cc1)NO
E3 Binder	CHEMBL483494	ChEMBL	8.72	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2cn(Cc3ccc(F)cc3)nn2)cc1)NO
E3 Binder	CHEMBL487533	ChEMBL	8.32	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2cn(Cc3ccccc3)nn2)cc1)NO
E3 Binder	CHEMBL487742	ChEMBL	8.46	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2cnnn2-c2ccccc2)cc1)NO
E3 Binder	CHEMBL487943	ChEMBL	8.38	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2cnnn2CC(O)c2cccc(Br)c2)cc1)NO
E3 Binder	CHEMBL487741	ChEMBL	8.14	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2cnnn2Cc2ccc(F)cc2)cc1)NO
E3 Binder	CHEMBL519746	ChEMBL	8.51	—	—	O=C(CCCCCCC(=O)Nc1ccc(-c2cnnn2Cc2ccccc2)cc1)NO
E3 Binder	CHEMBL5076638	ChEMBL	7.72	—	—	O=C(CCCCCCC(=O)Nc1ccc(C(=O)NC2CCNCC2)cc1)NO
E3 Binder	CHEMBL5078990	ChEMBL	6.64	—	—	O=C(CCCCCCC(=O)Nc1ccc(C(=O)NCCN2CCOCC2)cc1)NO
E3 Binder	CHEMBL3589699	ChEMBL	6.64	—	—	O=C(CCCCCCC(=O)Nc1ccc(C2=C(c3ccc(O)cc3)C3CC(S(=O)(=O)Oc4ccc(Br)cc4)C2O3)cc1)NO
E3 Binder	CHEMBL3589701	ChEMBL	6.49	—	—	O=C(CCCCCCC(=O)Nc1ccc(C2=C(c3ccc(O)cc3)C3CC(S(=O)(=O)Oc4ccc5ccccc5c4)C2O3)cc1)NO
E3 Binder	CHEMBL3589700	ChEMBL	7.52	—	—	O=C(CCCCCCC(=O)Nc1ccc(C2=C(c3ccc(O)cc3)C3CC(S(=O)(=O)Oc4cccc5ccccc45)C2O3)cc1)NO
E3 Binder	CHEMBL4091233	ChEMBL	9.05	—	—	O=C(CCCCCCC(=O)Nc1ccc(CCCn2cc(-c3ncnc4[nH]ccc34)cn2)cc1)NO
E3 Binder	CHEMBL4205840	ChEMBL	6.21	—	—	O=C(CCCCCCC(=O)Nc1ccc(N(CCCl)CCCl)cc1)NO
E3 Binder	CHEMBL4084049	ChEMBL	6.26	—	—	O=C(CCCCCCC(=O)Nc1ccc(NC(=O)CCCn2cc(-c3ncnc4[nH]ccc34)cn2)cc1)NO
E3 Binder	CHEMBL4098975	ChEMBL	9.85	—	—	O=C(CCCCCCC(=O)Nc1ccc(NCCCn2cc(-c3ncnc4[nH]ccc34)cn2)cc1)NO
E3 Binder	CHEMBL3972157	ChEMBL	8.64	—	—	O=C(CCCCCCC(=O)Nc1ccc(NCCOc2ccc3cc2COC/C=C/COCc2cccc(c2)-c2ccnc(n2)N3)cc1)NO
E3 Binder	CHEMBL4243347	ChEMBL	9.7	—	—	O=C(CCCCCCC(=O)Nc1ccc(Nc2nc(-c3cn[nH]c3)c3cc[nH]c3n2)cc1)NO
E3 Binder	CHEMBL4250122	ChEMBL	8.02	—	—	O=C(CCCCCCC(=O)Nc1ccc(Nc2nc(-c3cnn(CC4CCCC4)c3)c3cc[nH]c3n2)cc1)NO
E3 Binder	CHEMBL4243822	ChEMBL	7.8	—	—	O=C(CCCCCCC(=O)Nc1ccc(Nc2nc(-c3cnn(CCCCCCOc4ccccc4)c3)c3cc[nH]c3n2)cc1)NO
E3 Binder	CHEMBL4248054	ChEMBL	8.28	—	—	O=C(CCCCCCC(=O)Nc1ccc(Nc2nc(-c3cnn(CCCCCOc4ccccc4)c3)c3cc[nH]c3n2)cc1)NO
E3 Binder	CHEMBL4240012	ChEMBL	8.15	—	—	O=C(CCCCCCC(=O)Nc1ccc(Nc2nc(-c3cnn(CCCCOc4ccccc4)c3)c3cc[nH]c3n2)cc1)NO
E3 Binder	CHEMBL4438378	ChEMBL	8.23	—	—	O=C(CCCCCCC(=O)Nc1ccc(Nc2nc(NC3CCN(Cc4ccccc4)CC3)c3sccc3n2)cc1)NO
E3 Binder	CHEMBL3589351	ChEMBL	6.72	—	—	O=C(CCCCCCC(=O)Nc1ccc(OS(=O)(=O)C2CC3OC2C(c2ccc(O)cc2)=C3c2ccc(O)cc2)cc1)NO
E3 Binder	CHEMBL1923808	ChEMBL	7.3	—	—	O=C(CCCCCCC(=O)Nc1ccc([19F])cc1)NO
E3 Binder	CHEMBL469187	ChEMBL	7.55	—	—	O=C(CCCCCCC(=O)Nc1ccc([C@H]2O[C@@H](CSc3ccncc3)C[C@@H](c3ccccc3)O2)cc1)NO
E3 Binder	CHEMBL356769	ChEMBL	9.05	—	—	O=C(CCCCCCC(=O)Nc1ccc([C@H]2O[C@@H](CSc3nc(-c4ccccc4)c(-c4ccccc4)o3)C[C@@H](c3ccc(CO)cc3)O2)cc1)NO
E3 Binder	CHEMBL3311464	ChEMBL	7.18	—	—	O=C(CCCCCCC(=O)Nc1ccc2[nH]c(=O)ccc2c1)NO
E3 Binder	CHEMBL3621294	ChEMBL	9.49	—	—	O=C(CCCCCCC(=O)Nc1ccc2c(c1)/C(=C/c1ccc[nH]1)C(=O)N2)NO
E3 Binder	CHEMBL3311465	ChEMBL	6.2	—	—	O=C(CCCCCCC(=O)Nc1ccc2c(c1)CCC(=O)N2)NO
E3 Binder	CHEMBL3601340	ChEMBL	7.53	—	—	O=C(CCCCCCC(=O)Nc1ccc2ccnc(N3CCOCC3)c2c1)NO
E3 Binder	CHEMBL3601331	ChEMBL	8.17	—	—	O=C(CCCCCCC(=O)Nc1ccc2ccnc(Nc3ccc(Br)cc3F)c2c1)NO
E3 Binder	CHEMBL3601334	ChEMBL	8.29	—	—	O=C(CCCCCCC(=O)Nc1ccc2ccnc(Nc3ccc4ccccc4c3)c2c1)NO
E3 Binder	CHEMBL3601332	ChEMBL	8.1	—	—	O=C(CCCCCCC(=O)Nc1ccc2ccnc(Nc3cccc(Cl)c3F)c2c1)NO
E3 Binder	CHEMBL3601338	ChEMBL	7.96	—	—	O=C(CCCCCCC(=O)Nc1ccc2ccnc(Nc3ccccc3F)c2c1)NO
E3 Binder	CHEMBL473270	ChEMBL	8.05	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2ccccc2)c1)NO
E3 Binder	CHEMBL1088736	ChEMBL	8.72	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cn(-c3cc(CO)cc(CO)c3)nn2)c1)NO
E3 Binder	CHEMBL1091815	ChEMBL	8.77	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cn(-c3cc(F)cc(F)c3)nn2)c1)NO
E3 Binder	CHEMBL1088734	ChEMBL	8.54	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cn(-c3ccc(C(F)(F)F)cc3)nn2)c1)NO
E3 Binder	CHEMBL1091474	ChEMBL	8.08	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cn(-c3ccc(F)cc3)nn2)c1)NO
E3 Binder	CHEMBL1091475	ChEMBL	8.66	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cn(-c3ccc(I)cc3)nn2)c1)NO
E3 Binder	CHEMBL519668	ChEMBL	8.02	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cn(-c3ccccc3)nn2)c1)NO
E3 Binder	CHEMBL1094707	ChEMBL	8.48	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cn(C3CCCCC3)nn2)c1)NO
E3 Binder	CHEMBL483893	ChEMBL	8.72	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cn(CC(O)c3cccc(Br)c3)nn2)c1)NO
E3 Binder	CHEMBL483892	ChEMBL	8.59	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cn(Cc3ccc(F)cc3)nn2)c1)NO
E3 Binder	CHEMBL1088735	ChEMBL	8.12	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cn(Cc3ccc(O)cc3)nn2)c1)NO
E3 Binder	CHEMBL483693	ChEMBL	8.51	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cn(Cc3ccccc3)nn2)c1)NO
E3 Binder	CHEMBL520056	ChEMBL	8.12	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cnnn2-c2ccccc2)c1)NO
E3 Binder	CHEMBL487107	ChEMBL	8.55	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cnnn2CC(O)c2cccc(Br)c2)c1)NO
E3 Binder	CHEMBL487106	ChEMBL	8.42	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cnnn2Cc2ccc(F)cc2)c1)NO
E3 Binder	CHEMBL488747	ChEMBL	8.48	—	—	O=C(CCCCCCC(=O)Nc1cccc(-c2cnnn2Cc2ccccc2)c1)NO
E3 Binder	CHEMBL1094709	ChEMBL	8.51	—	—	O=C(CCCCCCC(=O)Nc1cccc(-n2cc(-c3ccccc3)nn2)c1)NO
E3 Binder	CHEMBL1094710	ChEMBL	8.37	—	—	O=C(CCCCCCC(=O)Nc1cccc(-n2cc(C3CCCCC3)nn2)c1)NO
E3 Binder	CHEMBL1089495	ChEMBL	8.22	—	—	O=C(CCCCCCC(=O)Nc1cccc(C(F)(F)F)c1)NO
E3 Binder	CHEMBL98	ChEMBL	9.0	SHH	—	O=C(CCCCCCC(=O)Nc1ccccc1)NO
E3 Binder	CHEMBL1164069	ChEMBL	6.6	—	—	O=C(CCCCCCC(=O)Nc1ccccc1)NOC(=O)c1csc(=S)s1
E3 Binder	CHEMBL181459	ChEMBL	7.38	—	—	O=C(CCCCCCC(=O)Nc1ccccc1C(=O)NO)Nc1ccccc1
E3 Binder	CHEMBL164872	ChEMBL	6.61	—	—	O=C(CCCCCCC(=O)Nc1ccccn1)NO
E3 Binder	CHEMBL353581	ChEMBL	8.32	—	—	O=C(CCCCCCC(=O)Nc1cccnc1)NO
E3 Binder	CHEMBL165162	ChEMBL	6.51	—	—	O=C(CCCCCCC(=O)Nc1ccncc1)NO
E3 Binder	CHEMBL4778689	ChEMBL	8.36	—	—	O=C(CCCCCCC(=O)Nc1cnc(N(c2ccccc2)c2ccccc2)nc1)NO
E3 Binder	CHEMBL387924	ChEMBL	8.43	—	—	O=C(CCCCCCC(=O)Nc1nc(-c2cccc([N+](=O)[O-])c2)cs1)NO
E3 Binder	CHEMBL511212	ChEMBL	8.52	—	—	O=C(CCCCCCC(=O)Nc1nc(-c2ccccc2)cs1)NO
E3 Binder	CHEMBL3954624	ChEMBL	7.4	—	—	O=C(CCCCCCC(=O)Nc1nc(-c2ccccc2[N+](=O)[O-])cs1)NO
E3 Binder	CHEMBL5199007	ChEMBL	8.34	—	—	O=C(CCCCCCC(=O)Nc1nc2c(s1)C[C@@H](NC(=O)c1cccc3ccccc13)CC2)NO
E3 Binder	CHEMBL5189571	ChEMBL	6.92	—	—	O=C(CCCCCCC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1)NO
E3 Binder	CHEMBL423515	ChEMBL	6.5	—	—	O=C(CCCCCCC(=O)c1ncco1)Nc1ccc(Cl)cc1
E3 Binder	CHEMBL126777	ChEMBL	6.24	—	—	O=C(CCCCCCC(=O)c1ncco1)Nc1ccc(Oc2ccccc2)cc1
E3 Binder	CHEMBL125416	ChEMBL	7.22	—	—	O=C(CCCCCCC(=O)c1ncco1)Nc1cccc(-c2ccccc2)c1
E3 Binder	CHEMBL3417190	ChEMBL	6.45	—	—	O=C(CCCCCCCC(=O)N1C/C=C/CCOc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO
E3 Binder	CHEMBL3417195	ChEMBL	6.48	—	—	O=C(CCCCCCCC(=O)N1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO
E3 Binder	CHEMBL4537089	ChEMBL	6.77	—	—	O=C(CCCCCCCC(=O)NC(Cc1c[nH]c2ccccc12)C(=O)Nc1ccc(Cl)cc1)NO
E3 Binder	CHEMBL5289255	ChEMBL	6.37	—	—	O=C(CCCCCCCC(=O)NCC1CCN(Cc2ccccc2)CC1)NO
E3 Binder	CHEMBL4642616	ChEMBL	6.84	—	—	O=C(CCCCCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc21)NO
E3 Binder	CHEMBL4633944	ChEMBL	6.85	—	—	O=C(CCCCCCCCC(=O)NCCCN1c2ccccc2CCc2ccc(Cl)cc21)NO
E3 Binder	CHEMBL4070306	ChEMBL	7.06	—	—	O=C(CCCCCCCCCCn1cc(-c2ncnc3[nH]ccc23)cn1)NO
E3 Binder	CHEMBL591525	ChEMBL	6.83	—	—	O=C(CCCCCCCCn1cc(-c2cccc(-c3ccccc3)c2)nn1)NO
E3 Binder	CHEMBL591746	ChEMBL	7.26	—	—	O=C(CCCCCCCCn1cc(-c2ccccc2)nn1)NO
E3 Binder	CHEMBL3973966	ChEMBL	6.0	—	—	O=C(CCCCCCCNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL3693705	ChEMBL	8.22	—	—	O=C(CCCCCCCNC(=O)c1ccc(N(c2ncccn2)c2ncccn2)cc1)NO
E3 Binder	CHEMBL490254	ChEMBL	7.55	—	—	O=C(CCCCCCCNC(=O)c1ccc2ccccc2c1)NO
E3 Binder	CHEMBL3939518	ChEMBL	6.87	—	—	O=C(CCCCCCCNC(=O)c1nc(-c2nccs2)sc1C1CC1)NO
E3 Binder	CHEMBL3963327	ChEMBL	7.0	—	—	O=C(CCCCCCCNCc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL3980430	ChEMBL	7.0	—	—	O=C(CCCCCCCNCc1ccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)o1)NO
E3 Binder	CHEMBL4649511	ChEMBL	7.89	—	—	O=C(CCCCCCCNc1nc2cc(C(=O)O)ccc2c2cnccc12)NO.O=C(O)C(F)(F)F
E3 Binder	CHEMBL5078723	ChEMBL	6.95	—	—	O=C(CCCCCCCNc1nn2c(=O)c3cc(Br)ccc3nc2c2ccccc12)NO
E3 Binder	CHEMBL5093545	ChEMBL	6.94	—	—	O=C(CCCCCCCNc1nn2c(=O)c3cc(Cl)ccc3nc2c2ccccc12)NO
E3 Binder	CHEMBL5072785	ChEMBL	6.93	—	—	O=C(CCCCCCCNc1nn2c(=O)c3cc(F)ccc3nc2c2ccccc12)NO
E3 Binder	CHEMBL5084865	ChEMBL	7.36	—	—	O=C(CCCCCCCNc1nn2c(=O)c3ccccc3nc2c2ccccc12)NO
E3 Binder	CHEMBL4784916	ChEMBL	6.87	—	—	O=C(CCCCCCCOc1ccc(-c2csc(N3N=C(c4ccccc4)/C(=N/Nc4nccs4)C3=O)n2)cc1)NO
E3 Binder	CHEMBL3099244	ChEMBL	6.31	—	—	O=C(CCCCCCCOc1ccc(-c2nc(N3CCOCC3)c3sccc3n2)cc1)NO
E3 Binder	CHEMBL5085582	ChEMBL	7.7	—	—	O=C(CCCCCCCOc1ccc(-c2nc3ccc(-c4nc5ccccc5[nH]4)cc3[nH]2)cc1)NO
E3 Binder	CHEMBL5081018	ChEMBL	7.31	—	—	O=C(CCCCCCCOc1ccc(-c2nc3ccccc3[nH]2)cc1)NO
E3 Binder	CHEMBL3945293	ChEMBL	7.8	—	—	O=C(CCCCCCCOc1ccc2cc1COC/C=C/COCc1cccc(c1)-c1ccnc(n1)N2)NO
E3 Binder	CHEMBL3099245	ChEMBL	6.21	—	—	O=C(CCCCCCCOc1cccc(-c2nc(N3CCOCC3)c3sccc3n2)c1)NO
E3 Binder	CHEMBL5094029	ChEMBL	8.14	—	—	O=C(CCCCCCCOc1cccc(-c2nc3ccc(-c4nc5ccccc5[nH]4)cc3[nH]2)c1)NO
E3 Binder	CHEMBL5077171	ChEMBL	8.1	—	—	O=C(CCCCCCCOc1cccc(-c2nc3ccccc3[nH]2)c1)NO
E3 Binder	CHEMBL326433	ChEMBL	7.16	—	—	O=C(CCCCCCCS)Nc1ccccc1
E3 Binder	CHEMBL589664	ChEMBL	6.67	—	—	O=C(CCCCCCCn1cc(-c2ccc(-c3ccncc3)cc2)nn1)NO
E3 Binder	CHEMBL592469	ChEMBL	6.96	—	—	O=C(CCCCCCCn1cc(-c2cccc(-c3ccccc3)c2)nn1)NO
E3 Binder	CHEMBL591747	ChEMBL	6.44	—	—	O=C(CCCCCCCn1cc(-c2ccccc2)nn1)NO
E3 Binder	CHEMBL591821	ChEMBL	6.37	—	—	O=C(CCCCCCCn1cc(-c2cccnc2)nn1)NO
E3 Binder	CHEMBL4069283	ChEMBL	8.74	—	—	O=C(CCCCCCCn1cc(-c2ncnc3[nH]ccc23)cn1)NO
E3 Binder	CHEMBL4584008	ChEMBL	7.42	—	—	O=C(CCCCCCCn1cc(Nc2ncc(Cl)c(Nc3ccc(F)cc3)n2)cn1)NO
E3 Binder	CHEMBL4163681	ChEMBL	8.21	—	—	O=C(CCCCCCN(Cc1ccc(F)cc1)c1ncc(C(=O)NCCCn2ccnc2)s1)NO
E3 Binder	CHEMBL3675760	ChEMBL	7.72	—	—	O=C(CCCCCCN(c1ccccn1)c1cc(-c2ccccc2)ccn1)NO
E3 Binder	CHEMBL3675765	ChEMBL	8.52	—	—	O=C(CCCCCCN(c1ccccn1)c1cc(OCc2ccccc2)ccn1)NO
E3 Binder	CHEMBL3675764	ChEMBL	8.7	—	—	O=C(CCCCCCN(c1ccccn1)c1cc2ccccc2cn1)NO
E3 Binder	CHEMBL3675762	ChEMBL	7.24	—	—	O=C(CCCCCCN(c1ccccn1)c1ccc(OCc2ccccc2)cn1)NO
E3 Binder	CHEMBL3675758	ChEMBL	7.8	—	—	O=C(CCCCCCN(c1ccccn1)c1ccc2ccccc2n1)NO
E3 Binder	CHEMBL3675757	ChEMBL	8.05	—	—	O=C(CCCCCCN(c1ccccn1)c1ccccn1)NO
E3 Binder	CHEMBL4746933	ChEMBL	8.4	—	—	O=C(CCCCCCN1C(=O)/C(=C2\Nc3ccccc3\C2=N/O)c2cc(Br)ccc21)NO
E3 Binder	CHEMBL4788217	ChEMBL	8.52	—	—	O=C(CCCCCCN1C(=O)/C(=C2\Nc3ccccc3\C2=N/O)c2cc(Cl)ccc21)NO
E3 Binder	CHEMBL4781515	ChEMBL	7.85	—	—	O=C(CCCCCCN1C(=O)/C(=C2\Nc3ccccc3\C2=N/O)c2cc(F)ccc21)NO
E3 Binder	CHEMBL4756818	ChEMBL	8.15	—	—	O=C(CCCCCCN1C(=O)/C(=C2\Nc3ccccc3\C2=N/O)c2cccc(Cl)c21)NO
E3 Binder	CHEMBL4761187	ChEMBL	7.66	—	—	O=C(CCCCCCN1C(=O)/C(=C2\Nc3ccccc3\C2=N/O)c2ccccc21)NO
E3 Binder	CHEMBL4172557	ChEMBL	6.58	—	—	O=C(CCCCCCN1C(=O)NC2(CCCc3ccccc32)C1=O)NO
E3 Binder	CHEMBL149606	ChEMBL	6.45	—	—	O=C(CCCCCCN1C(=O)c2ccccc2C1=O)NO
E3 Binder	CHEMBL3417187	ChEMBL	7.06	—	—	O=C(CCCCCCN1C/C=C/CCOc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO
E3 Binder	CHEMBL3414599	ChEMBL	6.8	—	—	O=C(CCCCCCN1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO
E3 Binder	CHEMBL5219000	ChEMBL	7.85	—	—	O=C(CCCCCCN1CC(=O)N2[C@H](CC3c4ccccc4NC3[C@H]2c2ccc(Br)cc2)C1=O)NO
E3 Binder	CHEMBL5275513	ChEMBL	8.04	—	—	O=C(CCCCCCN1CC(=O)N2[C@H](c3ccc(Cl)cc3)c3[nH]c4ccccc4c3C[C@@H]2C1=O)NO
E3 Binder	CHEMBL5178922	ChEMBL	8.37	—	—	O=C(CCCCCCN1CC(c2ccc3ncnc(Nc4ccc(Br)cc4F)c3c2)N=N1)NO
E3 Binder	CHEMBL147655	ChEMBL	8.0	—	—	O=C(CCCCCCN1c2cccc3cccc(c23)S1(=O)=O)NO
E3 Binder	CHEMBL146446	ChEMBL	7.53	—	—	O=C(CCCCCCNC(=O)C1Cc2ccccc2O1)NO
E3 Binder	CHEMBL3621293	ChEMBL	8.74	—	—	O=C(CCCCCCNC(=O)Cn1cnc2c(Nc3ccccc3)nc(Nc3ccccc3)nc21)NO
E3 Binder	CHEMBL294464	ChEMBL	7.43	—	—	O=C(CCCCCCNC(=O)c1c[nH]c2ccccc12)NO
E3 Binder	CHEMBL4225451	ChEMBL	7.66	—	—	O=C(CCCCCCNC(=O)c1cc(-c2ccc(F)cc2)[nH]n1)NO
E3 Binder	CHEMBL3897288	ChEMBL	7.0	—	—	O=C(CCCCCCNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL301223	ChEMBL	8.46	—	—	O=C(CCCCCCNC(=O)c1cc2cc(Br)ccc2[nH]1)NO
E3 Binder	CHEMBL59316	ChEMBL	7.82	—	—	O=C(CCCCCCNC(=O)c1cc2cc(Cl)ccc2o1)NO
E3 Binder	CHEMBL58487	ChEMBL	8.27	—	—	O=C(CCCCCCNC(=O)c1cc2cc(F)ccc2[nH]1)NO
E3 Binder	CHEMBL56157	ChEMBL	7.84	—	—	O=C(CCCCCCNC(=O)c1cc2ccccc2[nH]1)NO
E3 Binder	CHEMBL4753330	ChEMBL	7.0	—	—	O=C(CCCCCCNC(=O)c1ccc(-c2csc(N3N=C(c4ccccc4)/C(=N/Nc4nccs4)C3=O)n2)cc1)NO
E3 Binder	CHEMBL3693774	ChEMBL	8.15	—	—	O=C(CCCCCCNC(=O)c1ccc(C(CO)(c2ccccc2)c2ccccc2)cc1)NO
E3 Binder	CHEMBL3640654	ChEMBL	8.4	—	—	O=C(CCCCCCNC(=O)c1ccc(C(O)(c2cc(F)cc(F)c2)c2cc(F)cc(F)c2)cc1)NO
E3 Binder	CHEMBL3640667	ChEMBL	8.3	—	—	O=C(CCCCCCNC(=O)c1ccc(C(O)(c2ccc(F)cc2)C(F)(F)F)cc1)NO
E3 Binder	CHEMBL3693778	ChEMBL	8.52	—	—	O=C(CCCCCCNC(=O)c1ccc(C(O)(c2ccc(F)cc2)c2ccc(F)cc2)cc1)NO
E3 Binder	CHEMBL3640660	ChEMBL	8.52	—	—	O=C(CCCCCCNC(=O)c1ccc(C(O)(c2ccc(F)cc2)c2ccccn2)cc1)NO
E3 Binder	CHEMBL3640650	ChEMBL	8.3	—	—	O=C(CCCCCCNC(=O)c1ccc(C(O)(c2ccc(F)cc2F)c2ccc(F)cc2F)cc1)NO
E3 Binder	CHEMBL3693795	ChEMBL	8.3	—	—	O=C(CCCCCCNC(=O)c1ccc(C(O)(c2cccc(F)c2)c2cccc(F)c2)cc1)NO
E3 Binder	CHEMBL3693773	ChEMBL	8.0	—	—	O=C(CCCCCCNC(=O)c1ccc(C(O)(c2ccccc2)c2ccccc2)cc1)NO
E3 Binder	CHEMBL3693775	ChEMBL	8.4	—	—	O=C(CCCCCCNC(=O)c1ccc(C(O)(c2ccccc2)c2ccncc2)cc1)NO
E3 Binder	CHEMBL3693812	ChEMBL	8.52	—	—	O=C(CCCCCCNC(=O)c1ccc(C(O)(c2ccccc2F)c2ccccc2F)cc1)NO
E3 Binder	CHEMBL3693783	ChEMBL	8.4	—	—	O=C(CCCCCCNC(=O)c1ccc(C(O)(c2ccccn2)c2ccccn2)cc1)NO
E3 Binder	CHEMBL3640664	ChEMBL	8.3	—	—	O=C(CCCCCCNC(=O)c1ccc(C(O)(c2nccs2)c2nccs2)cc1)NO
E3 Binder	CHEMBL3693791	ChEMBL	7.66	—	—	O=C(CCCCCCNC(=O)c1ccc(C(c2ccccc2)c2ccccc2)cc1)NO
E3 Binder	CHEMBL3640669	ChEMBL	8.52	—	—	O=C(CCCCCCNC(=O)c1ccc(C2(c3ccc(F)cc3)CCCO2)cc1)NO
E3 Binder	CHEMBL3640680	ChEMBL	7.96	—	—	O=C(CCCCCCNC(=O)c1ccc(C2(c3ccccc3)OC(=O)c3ccccc32)cc1)NO
E3 Binder	CHEMBL3693777	ChEMBL	8.7	—	—	O=C(CCCCCCNC(=O)c1ccc(N(C(=O)c2ccccc2)c2ccccc2)cc1)NO
E3 Binder	CHEMBL3693793	ChEMBL	8.3	—	—	O=C(CCCCCCNC(=O)c1ccc(N(C(=O)c2ccccn2)c2ccccc2)cc1)NO
E3 Binder	CHEMBL3693723	ChEMBL	6.07	—	—	O=C(CCCCCCNC(=O)c1ccc(N(c2cccc(Cl)c2)c2cccc(Cl)c2)cc1)NO
E3 Binder	CHEMBL3693735	ChEMBL	7.82	—	—	O=C(CCCCCCNC(=O)c1ccc(N(c2ccccc2)S(=O)(=O)c2ccccc2)cc1)NO
E3 Binder	CHEMBL3693701	ChEMBL	7.75	—	—	O=C(CCCCCCNC(=O)c1ccc(N(c2ccccc2)c2ccccc2)cc1)NO
E3 Binder	CHEMBL3693734	ChEMBL	7.85	—	—	O=C(CCCCCCNC(=O)c1ccc(N(c2ccccc2)c2ccccn2)cc1)NO
E3 Binder	CHEMBL3693736	ChEMBL	7.68	—	—	O=C(CCCCCCNC(=O)c1ccc(N(c2ccccc2)c2cccnc2)cc1)NO
E3 Binder	CHEMBL3693732	ChEMBL	7.85	—	—	O=C(CCCCCCNC(=O)c1ccc(N(c2ccccc2)c2cnccn2)cc1)NO
E3 Binder	CHEMBL3693729	ChEMBL	7.92	—	—	O=C(CCCCCCNC(=O)c1ccc(N(c2ccccc2)c2cncnc2)cc1)NO
E3 Binder	CHEMBL3693717	ChEMBL	8.52	—	—	O=C(CCCCCCNC(=O)c1ccc(N(c2ccccc2)c2ncccn2)cc1)NO
E3 Binder	CHEMBL3693702	ChEMBL	6.76	—	—	O=C(CCCCCCNC(=O)c1ccc(N(c2ncccn2)c2ncccn2)cc1)NO
E3 Binder	CHEMBL255686	ChEMBL	8.34	—	—	O=C(CCCCCCNC(=O)c1ccc(NCc2cn(CCCNC(=S)Nc3ccc(-c4c5ccc(=O)cc-5oc5ccccc45)c(C(=O)O)c3)nn2)cc1)NO
E3 Binder	CHEMBL3693716	ChEMBL	8.52	—	—	O=C(CCCCCCNC(=O)c1ccc(Nc2c(Cl)cccc2Cl)cc1)NO
E3 Binder	CHEMBL3693722	ChEMBL	8.52	—	—	O=C(CCCCCCNC(=O)c1ccc(Nc2c(F)cccc2F)cc1)NO
E3 Binder	CHEMBL3693745	ChEMBL	8.15	—	—	O=C(CCCCCCNC(=O)c1ccc(Nc2ccccc2)cc1)NO
E3 Binder	CHEMBL3693731	ChEMBL	8.52	—	—	O=C(CCCCCCNC(=O)c1ccc(Nc2nc3ccccc3o2)cc1)NO
E3 Binder	CHEMBL3693741	ChEMBL	7.92	—	—	O=C(CCCCCCNC(=O)c1ccc(Nc2nc3ccccc3s2)cc1)NO
E3 Binder	CHEMBL3311471	ChEMBL	6.55	—	—	O=C(CCCCCCNC(=O)c1ccc2[nH]c(=O)ccc2c1)NO
E3 Binder	CHEMBL55499	ChEMBL	7.5	—	—	O=C(CCCCCCNC(=O)c1ccc2[nH]ccc2c1)NO
E3 Binder	CHEMBL3311472	ChEMBL	6.37	—	—	O=C(CCCCCCNC(=O)c1ccc2c(c1)CCC(=O)N2)NO
E3 Binder	CHEMBL54867	ChEMBL	7.25	—	—	O=C(CCCCCCNC(=O)c1ccc2cc[nH]c2c1)NO
E3 Binder	CHEMBL490255	ChEMBL	7.7	—	—	O=C(CCCCCCNC(=O)c1ccc2ccccc2c1)NO
E3 Binder	CHEMBL55234	ChEMBL	6.28	—	—	O=C(CCCCCCNC(=O)c1ccc[nH]1)NO
E3 Binder	CHEMBL3640665	ChEMBL	7.75	—	—	O=C(CCCCCCNC(=O)c1cccc(C(O)(c2ccc(F)cc2)c2ccc(F)cc2)c1)NO
E3 Binder	CHEMBL3640671	ChEMBL	7.39	—	—	O=C(CCCCCCNC(=O)c1cccc(C(O)(c2ccccn2)c2ccccn2)c1)NO
E3 Binder	CHEMBL54543	ChEMBL	7.09	—	—	O=C(CCCCCCNC(=O)c1cccc2[nH]ccc12)NO
E3 Binder	CHEMBL55728	ChEMBL	7.39	—	—	O=C(CCCCCCNC(=O)c1cccc2cc[nH]c12)NO
E3 Binder	CHEMBL57107	ChEMBL	6.25	—	—	O=C(CCCCCCNC(=O)c1ccccc1)NO
E3 Binder	CHEMBL5091193	ChEMBL	6.02	—	—	O=C(CCCCCCNC(=O)c1cnc(-c2ccc(Cl)cc2)s1)NO
E3 Binder	CHEMBL5086629	ChEMBL	6.16	—	—	O=C(CCCCCCNC(=O)c1cnc(-c2ccc(OC(F)(F)F)cc2)s1)NO
E3 Binder	CHEMBL5079545	ChEMBL	6.1	—	—	O=C(CCCCCCNC(=O)c1cnc(-c2ccc(Oc3ccccc3)cc2)s1)NO
E3 Binder	CHEMBL3640684	ChEMBL	8.1	—	—	O=C(CCCCCCNC(=O)c1cnc(N(CCO)CC(c2ccc(F)cc2)c2ccc(F)cc2)nc1)NO
E3 Binder	CHEMBL3640685	ChEMBL	8.52	—	—	O=C(CCCCCCNC(=O)c1cnc(N(CCO)CCc2c[nH]c3ccccc23)nc1)NO
E3 Binder	CHEMBL3640670	ChEMBL	8.1	—	—	O=C(CCCCCCNC(=O)c1cnc(N(CCO)c2ccccc2)nc1)NO
E3 Binder	CHEMBL3640675	ChEMBL	7.92	—	—	O=C(CCCCCCNC(=O)c1cnc(N(c2ccc(F)cc2)c2ccc(F)cc2)nc1)NO
E3 Binder	CHEMBL2364628	ChEMBL	9.0	AH4	—	O=C(CCCCCCNC(=O)c1cnc(N(c2ccccc2)c2ccccc2)nc1)NO
E3 Binder	CHEMBL3693786	ChEMBL	8.66	X4U	—	O=C(CCCCCCNC(=O)c1cnc(N(c2ccccc2)c2ccccc2Cl)nc1)NO
E3 Binder	CHEMBL3640700	ChEMBL	8.4	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCC(O)(c3ccc(Cl)cc3)CC2)nc1)NO
E3 Binder	CHEMBL3639395	ChEMBL	8.4	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCC(O)(c3ccccc3)CC2)nc1)NO
E3 Binder	CHEMBL3640706	ChEMBL	8.3	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCCCC2)nc1)NO
E3 Binder	CHEMBL3640705	ChEMBL	7.72	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCCNCC2)nc1)NO
E3 Binder	CHEMBL3640698	ChEMBL	8.15	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCC[C@@H](O)C2)nc1)NO
E3 Binder	CHEMBL3640702	ChEMBL	8.15	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCC[C@H]2CO)nc1)NO
E3 Binder	CHEMBL3640682	ChEMBL	8.22	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCCc3ccccc32)nc1)NO
E3 Binder	CHEMBL3640690	ChEMBL	7.89	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCN(CCO)CC2)nc1)NO
E3 Binder	CHEMBL3640689	ChEMBL	8.22	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCN(Cc3ccccc3)CC2)nc1)NO
E3 Binder	CHEMBL3640704	ChEMBL	8.3	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCN(c3ccc(F)cc3)CC2)nc1)NO
E3 Binder	CHEMBL3640693	ChEMBL	8.4	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCN(c3ccccc3)CC2)nc1)NO
E3 Binder	CHEMBL3640696	ChEMBL	8.15	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCN(c3nccc(C(F)(F)F)n3)CC2)nc1)NO
E3 Binder	CHEMBL3640688	ChEMBL	7.68	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCNCC2)nc1)NO
E3 Binder	CHEMBL3640697	ChEMBL	8.15	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCOC(CO)C2)nc1)NO
E3 Binder	CHEMBL3640686	ChEMBL	8.1	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCOCC2)nc1)NO
E3 Binder	CHEMBL3640683	ChEMBL	8.52	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCc3ccccc3C2)nc1)NO
E3 Binder	CHEMBL3640692	ChEMBL	7.85	—	—	O=C(CCCCCCNC(=O)c1cnc(N2CCn3c(nnc3C(F)(F)F)C2)nc1)NO
E3 Binder	CHEMBL3640681	ChEMBL	8.3	—	—	O=C(CCCCCCNC(=O)c1cnc(NC(c2ccc(F)cc2)c2ccc(F)cc2)nc1)NO
E3 Binder	CHEMBL5172507	ChEMBL	8.22	—	—	O=C(CCCCCCNC(=O)c1csc(Br)n1)NO
E3 Binder	CHEMBL3961271	ChEMBL	7.31	—	—	O=C(CCCCCCNC(=O)c1nc(-c2nc3c(s2)CCCC3)sc1C1CC1)NO
E3 Binder	CHEMBL3911545	ChEMBL	8.0	—	—	O=C(CCCCCCNC(=O)c1nc(-c2nccs2)sc1C1CC1)NO
E3 Binder	CHEMBL3984477	ChEMBL	7.0	—	—	O=C(CCCCCCNCc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL3967081	ChEMBL	7.0	—	—	O=C(CCCCCCNCc1ccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)o1)NO
E3 Binder	CHEMBL127179	ChEMBL	6.37	—	—	O=C(CCCCCCNc1ccc2ccccc2c1)c1ncco1
E3 Binder	CHEMBL5289915	ChEMBL	6.11	—	—	O=C(CCCCCCNc1ccc2ncnc(Nc3ccc(F)cc3)c2n1)NO
E3 Binder	CHEMBL5269112	ChEMBL	7.35	—	—	O=C(CCCCCCNc1nc2ccccc2nc1-c1nc2ccccc2o1)NO
E3 Binder	CHEMBL4102051	ChEMBL	8.15	—	—	O=C(CCCCCCNc1ncnc2ccc(Cl)cc12)NO
E3 Binder	CHEMBL4094315	ChEMBL	8.1	—	—	O=C(CCCCCCNc1ncnc2ccc(F)cc12)NO
E3 Binder	CHEMBL5090447	ChEMBL	7.21	—	—	O=C(CCCCCCNc1nn2c(=O)c3cc(Br)ccc3nc2c2ccccc12)NO
E3 Binder	CHEMBL5076796	ChEMBL	7.18	—	—	O=C(CCCCCCNc1nn2c(=O)c3cc(Cl)ccc3nc2c2ccccc12)NO
E3 Binder	CHEMBL5093737	ChEMBL	7.15	—	—	O=C(CCCCCCNc1nn2c(=O)c3cc(F)ccc3nc2c2ccccc12)NO
E3 Binder	CHEMBL5087773	ChEMBL	7.37	—	—	O=C(CCCCCCNc1nn2c(=O)c3ccccc3nc2c2ccccc12)NO
E3 Binder	CHEMBL3894186	ChEMBL	7.0	—	—	O=C(CCCCCCOc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL1163161	ChEMBL	8.0	—	—	O=C(CCCCCCOc1ccc(-c2cc(=S)ss2)cc1)NO
E3 Binder	CHEMBL114184	ChEMBL	7.7	—	—	O=C(CCCCCCOc1ccc(-c2ccccc2)cc1)NO
E3 Binder	CHEMBL4756429	ChEMBL	7.39	—	—	O=C(CCCCCCOc1ccc(-c2csc(N3N=C(c4ccccc4)/C(=N/Nc4nccs4)C3=O)n2)cc1)NO
E3 Binder	CHEMBL5087772	ChEMBL	8.12	—	—	O=C(CCCCCCOc1ccc(-c2nc3ccc(-c4nc5ccccc5[nH]4)cc3[nH]2)cc1)NO
E3 Binder	CHEMBL5078111	ChEMBL	7.39	—	—	O=C(CCCCCCOc1ccc(-c2nc3ccccc3[nH]2)cc1)NO
E3 Binder	CHEMBL5179735	ChEMBL	7.19	—	—	O=C(CCCCCCOc1ccc(-c2nnc(-c3ccccc3)s2)cc1)NO
E3 Binder	CHEMBL4278151	ChEMBL	6.74	—	—	O=C(CCCCCCOc1ccc(-n2[se]c3ccccc3c2=O)cc1)NO
E3 Binder	CHEMBL3917405	ChEMBL	8.68	—	—	O=C(CCCCCCOc1ccc2cc1COC/C=C/COCc1cccc(c1)-c1ccnc(n1)N2)NO
E3 Binder	CHEMBL127328	ChEMBL	6.28	—	—	O=C(CCCCCCOc1ccc2ccccc2c1)c1ncco1
E3 Binder	CHEMBL604094	ChEMBL	8.36	—	—	O=C(CCCCCCOc1ccc2ncnc(Nc3ccc(F)c(Cl)c3)c2c1)NO
E3 Binder	CHEMBL127351	ChEMBL	6.21	—	—	O=C(CCCCCCOc1cccc(-c2ccccc2)c1)c1ncco1
E3 Binder	CHEMBL3099243	ChEMBL	6.42	—	—	O=C(CCCCCCOc1cccc(-c2nc(N3CCOCC3)c3sccc3n2)c1)NO
E3 Binder	CHEMBL5079630	ChEMBL	7.75	—	—	O=C(CCCCCCOc1cccc(-c2nc3ccc(-c4nc5ccccc5[nH]4)cc3[nH]2)c1)NO
E3 Binder	CHEMBL5086208	ChEMBL	7.88	—	—	O=C(CCCCCCOc1cccc(-c2nc3ccccc3[nH]2)c1)NO
E3 Binder	CHEMBL5193360	ChEMBL	6.73	—	—	O=C(CCCCCCOc1cccc(-c2nnc(-c3ccccc3)s2)c1)NO
E3 Binder	CHEMBL5204591	ChEMBL	7.52	—	—	O=C(CCCCCCOc1cccc(-c2nnc(-c3ccccc3Cl)s2)c1)NO
E3 Binder	CHEMBL340721	ChEMBL	6.21	—	—	O=C(CCCCCCS(=O)(=O)c1ccc2ccccc2c1)c1ncco1
E3 Binder	CHEMBL3356930	ChEMBL	7.06	—	—	O=C(CCCCCCS)NC1CCCC1
E3 Binder	CHEMBL112129	ChEMBL	6.21	—	—	O=C(CCCCCCS)Nc1ccc(Oc2ccccc2)cc1
E3 Binder	CHEMBL320323	ChEMBL	7.12	—	—	O=C(CCCCCCS)Nc1cccc(-c2ccccc2)c1
E3 Binder	CHEMBL322504	ChEMBL	6.68	—	—	O=C(CCCCCCS)Nc1cccc(Oc2ccccc2)c1
E3 Binder	CHEMBL325676	ChEMBL	7.72	—	—	O=C(CCCCCCS)Nc1ccccc1
E3 Binder	CHEMBL332246	ChEMBL	6.96	—	—	O=C(CCCCCCS)Nc1cccnc1
E3 Binder	CHEMBL112234	ChEMBL	7.14	—	—	O=C(CCCCCCS)Nc1cnc2ccccc2c1
E3 Binder	CHEMBL3288489	ChEMBL	6.26	—	—	O=C(CCCCCCS)Nc1nc(-c2ccc(F)cc2)cs1
E3 Binder	CHEMBL3288484	ChEMBL	6.82	—	—	O=C(CCCCCCS)Nc1nc(-c2cccc(F)c2)cs1
E3 Binder	CHEMBL419758	ChEMBL	6.77	—	—	O=C(CCCCCCS)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL178779	ChEMBL	6.47	—	—	O=C(CCCCCCS)Nc1nc2ccccc2s1
E3 Binder	CHEMBL127606	ChEMBL	6.27	—	—	O=C(CCCCCCSc1ccc2ccccc2c1)c1ncco1
E3 Binder	CHEMBL201131	ChEMBL	6.42	—	—	O=C(CCCCCC[S+]([O-])c1ccc(Cl)cc1)NO
E3 Binder	CHEMBL339796	ChEMBL	7.92	—	—	O=C(CCCCCCc1cnc(-c2ccc(-c3ccccc3)cc2)o1)NO
E3 Binder	CHEMBL123905	ChEMBL	8.36	—	—	O=C(CCCCCCc1cnc(-c2ccc(Br)cc2)o1)NO
E3 Binder	CHEMBL338776	ChEMBL	7.64	—	—	O=C(CCCCCCc1cnc(-c2ccc(F)cc2)o1)NO
E3 Binder	CHEMBL124593	ChEMBL	7.05	—	—	O=C(CCCCCCc1cnc(-c2ccc(OC(F)(F)F)cc2)o1)NO
E3 Binder	CHEMBL127184	ChEMBL	7.89	—	—	O=C(CCCCCCc1cnc(-c2ccccc2)o1)NO
E3 Binder	CHEMBL126274	ChEMBL	7.96	—	—	O=C(CCCCCCc1nc(-c2ccc(-c3ccccc3)cc2)cs1)NO
E3 Binder	CHEMBL340835	ChEMBL	8.07	—	—	O=C(CCCCCCc1nc(-c2ccc(Br)cc2)cs1)NO
E3 Binder	CHEMBL126273	ChEMBL	7.38	—	—	O=C(CCCCCCc1nc(-c2ccc(C(F)(F)F)cc2)cs1)NO
E3 Binder	CHEMBL123506	ChEMBL	7.13	—	—	O=C(CCCCCCc1nc(-c2ccc(OC(F)(F)F)cc2)cs1)NO
E3 Binder	CHEMBL340885	ChEMBL	8.37	—	—	O=C(CCCCCCc1nc(-c2ccc3ccccc3c2)cs1)NO
E3 Binder	CHEMBL125042	ChEMBL	8.24	—	—	O=C(CCCCCCc1nc(-c2cccc(Br)c2)cs1)NO
E3 Binder	CHEMBL124909	ChEMBL	7.72	—	—	O=C(CCCCCCc1nc(-c2ccccc2)cs1)NO
E3 Binder	CHEMBL2414098	ChEMBL	8.72	—	—	O=C(CCCCCCc1nc2ccc(Br)cc2[nH]1)NO
E3 Binder	CHEMBL124650	ChEMBL	8.17	—	—	O=C(CCCCCCc1ncc(-c2ccc(-c3ccc(Cl)cc3)cc2)o1)NO
E3 Binder	CHEMBL339720	ChEMBL	8.57	—	—	O=C(CCCCCCc1ncc(-c2ccc(Br)cc2)o1)NO
E3 Binder	CHEMBL127846	ChEMBL	8.01	—	—	O=C(CCCCCCc1ncc(-c2ccccc2)o1)NO
E3 Binder	CHEMBL127627	ChEMBL	6.6	—	—	O=C(CCCCCCc1nnc(-c2ccc(-c3ccccc3)cc2)o1)c1ncco1
E3 Binder	CHEMBL4282673	ChEMBL	7.72	—	—	O=C(CCCCCCn1[se]c2ccccc2c1=O)NO
E3 Binder	CHEMBL5180181	ChEMBL	8.16	—	—	O=C(CCCCCCn1c(C(=O)NC2C3CC4CC(C3)CC2C4)cc2cc(Cl)ccc21)NO
E3 Binder	CHEMBL5171482	ChEMBL	8.33	—	—	O=C(CCCCCCn1c(C(=O)NC2C3CC4CC(C3)CC2C4)cc2ccc(Br)cc21)NO
E3 Binder	CHEMBL5169341	ChEMBL	8.61	—	—	O=C(CCCCCCn1c(C(=O)NC2C3CC4CC(C3)CC2C4)cc2ccccc21)NO
E3 Binder	CHEMBL5191345	ChEMBL	8.28	—	—	O=C(CCCCCCn1c(C(=O)NC2C3CC4CC(C3)CC2C4)nc2ccccc21)NO
E3 Binder	CHEMBL3675752	ChEMBL	8.22	—	—	O=C(CCCCCCn1c2ccccc2c2ccccc21)NO
E3 Binder	CHEMBL477283	ChEMBL	7.78	—	—	O=C(CCCCCCn1cc(-c2ccc(-c3ccncc3)cc2)nn1)NO
E3 Binder	CHEMBL4241141	ChEMBL	8.54	—	—	O=C(CCCCCCn1cc(-c2ccc(Nc3c4ccccc4nc4ccccc34)cc2)nn1)NO
E3 Binder	CHEMBL4863294	ChEMBL	8.37	—	—	O=C(CCCCCCn1cc(-c2ccc3ncnc(Nc4ccc(Br)cc4F)c3c2)nn1)NO
E3 Binder	CHEMBL3957055	ChEMBL	8.08	—	—	O=C(CCCCCCn1cc(-c2ccc3ncnc(Nc4ccc(F)c(Cl)c4)c3c2)nn1)NO
E3 Binder	CHEMBL3911796	ChEMBL	7.71	—	—	O=C(CCCCCCn1cc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)nn1)NO
E3 Binder	CHEMBL3902778	ChEMBL	7.87	—	—	O=C(CCCCCCn1cc(-c2ccc3ncnc(Nc4ccc(OCc5nccs5)c(Cl)c4)c3c2)nn1)NO
E3 Binder	CHEMBL3930620	ChEMBL	8.49	—	—	O=C(CCCCCCn1cc(-c2ccc3ncnc(Nc4cccc(Cl)c4F)c3c2)nn1)NO
E3 Binder	CHEMBL477101	ChEMBL	8.27	—	—	O=C(CCCCCCn1cc(-c2cccc(-c3ccccc3)c2)nn1)NO
E3 Binder	CHEMBL4240694	ChEMBL	8.3	—	—	O=C(CCCCCCn1cc(-c2cccc(Nc3c4ccccc4nc4ccccc34)c2)nn1)NO
E3 Binder	CHEMBL478109	ChEMBL	8.02	—	—	O=C(CCCCCCn1cc(-c2ccccc2)nn1)NO
E3 Binder	CHEMBL478309	ChEMBL	7.62	—	—	O=C(CCCCCCn1cc(-c2ccccn2)nn1)NO
E3 Binder	CHEMBL589605	ChEMBL	6.44	—	—	O=C(CCCCCCn1cc(-c2cccnc2)nn1)NO
E3 Binder	CHEMBL4060201	ChEMBL	8.85	—	—	O=C(CCCCCCn1cc(-c2ncnc3[nH]ccc23)cn1)NO
E3 Binder	CHEMBL5173771	ChEMBL	8.12	—	—	O=C(CCCCCCn1cc(C(=O)N2CCOCC2)c2ccccc21)NO
E3 Binder	CHEMBL5208269	ChEMBL	8.72	—	—	O=C(CCCCCCn1cc(C(=O)NC23CC4CC(CC(C4)C2)C3)c2ccccc21)NO
E3 Binder	CHEMBL5206239	ChEMBL	8.77	—	—	O=C(CCCCCCn1cc(C(=O)NC2C3CC4CC(C3)CC2C4)c2ccccc21)NO
E3 Binder	CHEMBL5197455	ChEMBL	8.63	—	—	O=C(CCCCCCn1cc(C(=O)NC2CCCCC2)c2ccccc21)NO
E3 Binder	CHEMBL5174843	ChEMBL	8.68	—	—	O=C(CCCCCCn1cc(C(=O)NC2CCCCCC2)c2ccccc21)NO
E3 Binder	CHEMBL5185898	ChEMBL	8.74	—	—	O=C(CCCCCCn1cc(C(=O)NC2CCCCCCC2)c2ccccc21)NO
E3 Binder	CHEMBL5189457	ChEMBL	8.81	—	—	O=C(CCCCCCn1cc(C(=O)NCc2ccc(Cl)cc2)c2ccccc21)NO
E3 Binder	CHEMBL5171183	ChEMBL	8.43	—	—	O=C(CCCCCCn1cc(C(=O)Nc2ccc(Cl)cc2Cl)c2ccccc21)NO
E3 Binder	CHEMBL4581017	ChEMBL	7.39	—	—	O=C(CCCCCCn1cc(Nc2ncc(C(F)(F)F)c(Nc3ccc(F)cc3)n2)cn1)NO
E3 Binder	CHEMBL4562491	ChEMBL	7.4	—	—	O=C(CCCCCCn1cc(Nc2ncc(Cl)c(N3CCCCC3)n2)cn1)NO
E3 Binder	CHEMBL4556463	ChEMBL	7.43	—	—	O=C(CCCCCCn1cc(Nc2ncc(Cl)c(N3CCOCC3)n2)cn1)NO
E3 Binder	CHEMBL4466059	ChEMBL	7.89	—	—	O=C(CCCCCCn1cc(Nc2ncc(Cl)c(NC3CC3)n2)cn1)NO
E3 Binder	CHEMBL4575813	ChEMBL	8.7	—	—	O=C(CCCCCCn1cc(Nc2ncc(Cl)c(Nc3ccc(Cl)cc3)n2)cn1)NO
E3 Binder	CHEMBL4520721	ChEMBL	8.52	—	—	O=C(CCCCCCn1cc(Nc2ncc(Cl)c(Nc3ccc(F)cc3)n2)cn1)NO
E3 Binder	CHEMBL4471710	ChEMBL	7.7	—	—	O=C(CCCCCCn1cc(Nc2ncc(Cl)c(Nc3cccc(Cl)c3)n2)cn1)NO
E3 Binder	CHEMBL4443462	ChEMBL	7.72	—	—	O=C(CCCCCCn1cc(Nc2ncc(Cl)c(Nc3ccccc3)n2)cn1)NO
E3 Binder	CHEMBL4533614	ChEMBL	8.0	—	—	O=C(CCCCCCn1cc(Nc2ncc(Cl)c(Nc3ccccc3Cl)n2)cn1)NO
E3 Binder	CHEMBL4538220	ChEMBL	8.52	—	—	O=C(CCCCCCn1cc(Nc2ncc(F)c(Nc3ccc(F)cc3)n2)cn1)NO
E3 Binder	CHEMBL5083776	ChEMBL	7.7	—	—	O=C(CCCCCCn1cc(Nc2ncc3ccn(-c4ccc(Br)cc4)c3n2)cn1)NO
E3 Binder	CHEMBL5076046	ChEMBL	7.48	—	—	O=C(CCCCCCn1cc(Nc2ncc3ccn(-c4ccc(Cl)cc4)c3n2)cn1)NO
E3 Binder	CHEMBL5091553	ChEMBL	7.67	—	—	O=C(CCCCCCn1cc(Nc2ncc3ccn(-c4ccc(F)cc4)c3n2)cn1)NO
E3 Binder	CHEMBL5081471	ChEMBL	7.88	—	—	O=C(CCCCCCn1cc(Nc2ncc3ccn(-c4ccccc4)c3n2)cn1)NO
E3 Binder	CHEMBL5089674	ChEMBL	7.66	—	—	O=C(CCCCCCn1cc(Nc2ncc3ccn(C4CCCC4)c3n2)cn1)NO
E3 Binder	CHEMBL5075022	ChEMBL	7.8	—	—	O=C(CCCCCCn1cc(Nc2ncc3ccn(CC4CC4)c3n2)cn1)NO
E3 Binder	CHEMBL5079677	ChEMBL	7.06	—	—	O=C(CCCCCCn1cc(Nc2ncc3ccn(CC4CCCCC4)c3n2)cn1)NO
E3 Binder	CHEMBL5073935	ChEMBL	7.43	—	—	O=C(CCCCCCn1cc(Nc2ncc3ccn(Cc4cccc(Cl)c4)c3n2)cn1)NO
E3 Binder	CHEMBL5087239	ChEMBL	7.83	—	—	O=C(CCCCCCn1cc(Nc2ncc3ccn(Cc4cccc(F)c4)c3n2)cn1)NO
E3 Binder	CHEMBL5078586	ChEMBL	7.9	—	—	O=C(CCCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4)c3n2)cn1)NO
E3 Binder	CHEMBL5092838	ChEMBL	7.38	—	—	O=C(CCCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4Cl)c3n2)cn1)NO
E3 Binder	CHEMBL5076728	ChEMBL	8.08	—	—	O=C(CCCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4F)c3n2)cn1)NO
E3 Binder	CHEMBL4441124	ChEMBL	7.75	—	—	O=C(CCCCCCn1cc(Nc2nccc(Nc3ccc(F)cc3)n2)cn1)NO
E3 Binder	CHEMBL3936496	ChEMBL	7.0	—	—	O=C(CCCCCCn1ccc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)cc1=O)NO
E3 Binder	CHEMBL4749655	ChEMBL	8.38	—	—	O=C(CCCCCCn1cnc2c(N3CCOCC3)nc(-c3cccc(CO)c3)nc21)NO
E3 Binder	CHEMBL5180263	ChEMBL	8.56	—	—	O=C(CCCCCCn1nc(C(=O)NC2C3CC4CC(C3)CC2C4)c2ccccc21)NO
E3 Binder	CHEMBL4095157	ChEMBL	6.22	—	—	O=C(CCCCCN(CC(=O)NC1CCCCC1)C(=O)c1cccc2ccccc12)NO
E3 Binder	CHEMBL4160632	ChEMBL	9.19	—	—	O=C(CCCCCN1C(=O)c2cccc3c(N4CCOCC4)ccc(c23)C1=O)NO
E3 Binder	CHEMBL4532304	ChEMBL	8.46	—	—	O=C(CCCCCN1C(=O)c2cccc3c(NCc4ccccc4)ccc(c23)C1=O)NO
E3 Binder	CHEMBL4461622	ChEMBL	7.85	—	—	O=C(CCCCCN1C(=O)c2cccc3c(Nc4cccc(F)c4)ccc(c23)C1=O)NO
E3 Binder	CHEMBL4526647	ChEMBL	7.89	—	—	O=C(CCCCCN1C(=O)c2cccc3c(Nc4ccccc4)ccc(c23)C1=O)NO
E3 Binder	CHEMBL4864538	ChEMBL	7.92	—	—	O=C(CCCCCN1C(=O)c2cccc3c(OCc4ccc(C(F)(F)F)cc4)ccc(c23)C1=O)NO
E3 Binder	CHEMBL4465218	ChEMBL	8.24	—	—	O=C(CCCCCN1C(=O)c2cccc3c([N+](=O)[O-])ccc(c23)C1=O)NO
E3 Binder	CHEMBL96051	ChEMBL	9.6	—	—	O=C(CCCCCN1C(=O)c2cccc3cccc(c23)C1=O)NO
E3 Binder	CHEMBL2063489	ChEMBL	6.96	—	—	O=C(CCCCCN1C(=O)c2ccccc2C(F)(F)c2ccccc21)NO
E3 Binder	CHEMBL2063487	ChEMBL	7.28	—	—	O=C(CCCCCN1C(=O)c2ccccc2C(F)c2ccccc21)NO
E3 Binder	CHEMBL2063486	ChEMBL	7.22	—	—	O=C(CCCCCN1C(=O)c2ccccc2C(O)c2ccccc21)NO
E3 Binder	CHEMBL146202	ChEMBL	6.29	—	—	O=C(CCCCCN1C(=O)c2ccccc2C1=O)NO
E3 Binder	CHEMBL2063484	ChEMBL	7.38	—	—	O=C(CCCCCN1C(=O)c2ccccc2Cc2ccccc21)NO
E3 Binder	CHEMBL1688188	ChEMBL	6.08	—	—	O=C(CCCCCN1C(=O)c2ccccc2Nc2ccc(Cl)cc21)NO
E3 Binder	CHEMBL1688193	ChEMBL	6.42	—	—	O=C(CCCCCN1C(=O)c2ccccc2Oc2ccc(Cl)cc21)NO
E3 Binder	CHEMBL1688184	ChEMBL	7.52	—	—	O=C(CCCCCN1C(=O)c2ccccc2S(=O)(=O)c2ccc(Cl)cc21)NO
E3 Binder	CHEMBL1688189	ChEMBL	6.3	—	—	O=C(CCCCCN1C(=O)c2ccccc2S(=O)(=O)c2ccccc21)NO
E3 Binder	CHEMBL1688191	ChEMBL	6.47	—	—	O=C(CCCCCN1C(=O)c2ccccc2Sc2ccc(Cl)cc21)NO
E3 Binder	CHEMBL1688187	ChEMBL	6.37	—	—	O=C(CCCCCN1C(=O)c2ccccc2Sc2ccccc21)NO
E3 Binder	CHEMBL3417186	ChEMBL	6.82	—	—	O=C(CCCCCN1C/C=C/CCOc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO
E3 Binder	CHEMBL3417192	ChEMBL	6.91	—	—	O=C(CCCCCN1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO
E3 Binder	CHEMBL5219389	ChEMBL	7.21	—	—	O=C(CCCCCN1CC(=O)N2[C@@H](CC3c4ccccc4NC3[C@@H]2c2ccc(Br)cc2)C1=O)NO
E3 Binder	CHEMBL5289022	ChEMBL	7.21	—	—	O=C(CCCCCN1CC(=O)N2[C@H](c3ccc(Br)cc3)c3[nH]c4ccccc4c3C[C@@H]2C1=O)NO
E3 Binder	CHEMBL3917105	ChEMBL	7.0	—	—	O=C(CCCCCN1CCN(Cc2ccc(-c3cc4c(NCc5ccccc5)ncnc4[nH]3)cc2)CC1)NO
E3 Binder	CHEMBL5276050	ChEMBL	7.84	—	—	O=C(CCCCCN1CCN2[C@H](Cc3c([nH]c4ccccc34)[C@H]2c2ccc(Br)cc2)C1)NO
E3 Binder	CHEMBL504898	ChEMBL	7.21	—	—	O=C(CCCCCNC(=O)CC#Cc1ccccc1)NO
E3 Binder	CHEMBL484487	ChEMBL	6.2	—	—	O=C(CCCCCNC(=O)CC/C=C/c1ccccc1)NO
E3 Binder	CHEMBL3621287	ChEMBL	8.59	—	—	O=C(CCCCCNC(=O)Cn1cnc2c(N3CCOCC3)nc(Nc3ccccc3)nc21)NO
E3 Binder	CHEMBL3621292	ChEMBL	8.42	—	—	O=C(CCCCCNC(=O)Cn1cnc2c(Nc3ccccc3)nc(Nc3ccccc3)nc21)NO
E3 Binder	CHEMBL1083086	ChEMBL	8.1	—	—	O=C(CCCCCNC(=O)NC(=O)c1ccc(Br)cc1)NO
E3 Binder	CHEMBL1083439	ChEMBL	8.15	—	—	O=C(CCCCCNC(=O)NC(=O)c1ccccc1)NO
E3 Binder	CHEMBL227118	ChEMBL	7.14	—	—	O=C(CCCCCNC(=O)NC12CC3CC(CC(C3)C1)C2)NO
E3 Binder	CHEMBL270120	ChEMBL	7.72	—	—	O=C(CCCCCNC(=O)Nc1cccc(-c2nc3cc(C(F)(F)F)ccc3o2)c1)NO
E3 Binder	CHEMBL272638	ChEMBL	8.1	—	—	O=C(CCCCCNC(=O)Nc1cccc(-c2nc3cc(F)ccc3o2)c1)NO
E3 Binder	CHEMBL411264	ChEMBL	8.05	—	—	O=C(CCCCCNC(=O)Nc1cccc(-c2nc3ccc(F)cc3o2)c1)NO
E3 Binder	CHEMBL271114	ChEMBL	8.1	—	—	O=C(CCCCCNC(=O)Nc1cccc(-c2nc3ccccc3o2)c1)NO
E3 Binder	CHEMBL98428	ChEMBL	6.18	—	—	O=C(CCCCCNC(=O)[C@H](Cc1ccccc1)N1C(=O)CCC1=O)NO
E3 Binder	CHEMBL4226433	ChEMBL	7.54	—	—	O=C(CCCCCNC(=O)c1cc(-c2ccc(F)cc2)[nH]n1)NO
E3 Binder	CHEMBL3934468	ChEMBL	7.0	—	—	O=C(CCCCCNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL143327	ChEMBL	7.42	—	—	O=C(CCCCCNC(=O)c1ccc(-c2ccccc2)cc1)NO
E3 Binder	CHEMBL4780328	ChEMBL	7.06	—	—	O=C(CCCCCNC(=O)c1ccc(-c2csc(N3N=C(c4ccccc4)/C(=N/Nc4nccs4)C3=O)n2)cc1)NO
E3 Binder	CHEMBL143734	ChEMBL	6.43	—	—	O=C(CCCCCNC(=O)c1ccc(Cl)cc1)NO
E3 Binder	CHEMBL167455	ChEMBL	6.83	—	—	O=C(CCCCCNC(=O)c1ccc(O)cc1)NO
E3 Binder	CHEMBL162344	ChEMBL	6.66	—	—	O=C(CCCCCNC(=O)c1ccc(OCc2ccccc2)cc1)NO
E3 Binder	CHEMBL5287236	ChEMBL	6.78	—	—	O=C(CCCCCNC(=O)c1ccc2cccc(OCc3ccc(Br)cc3)c2n1)NO
E3 Binder	CHEMBL5279091	ChEMBL	6.78	—	—	O=C(CCCCCNC(=O)c1ccc2cccc(OCc3ccccc3)c2n1)NO
E3 Binder	CHEMBL454719	ChEMBL	7.68	—	—	O=C(CCCCCNC(=O)c1ccc2ccccc2c1)NO
E3 Binder	CHEMBL5206589	ChEMBL	8.66	—	—	O=C(CCCCCNC(=O)c1cccc2cc3ccccc3nc12)NO
E3 Binder	CHEMBL143849	ChEMBL	6.62	—	—	O=C(CCCCCNC(=O)c1ccccc1)NO
E3 Binder	CHEMBL3903212	ChEMBL	6.98	—	—	O=C(CCCCCNC(=O)c1nc(-c2nccs2)sc1C1CC1)NO
E3 Binder	CHEMBL4776969	ChEMBL	7.33	—	—	O=C(CCCCCNC(=S)N/N=C(\c1ccccc1)c1cccc([N+](=O)[O-])c1)NO
E3 Binder	CHEMBL3987181	ChEMBL	7.0	—	—	O=C(CCCCCNCc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL3936512	ChEMBL	7.0	—	—	O=C(CCCCCNCc1ccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)o1)NO
E3 Binder	CHEMBL2311792	ChEMBL	6.05	—	—	O=C(CCCCCONC(=O)Nc1cccc2ccccc12)NO
E3 Binder	CHEMBL2311793	ChEMBL	7.29	—	—	O=C(CCCCCONC(=O)Nc1cnc2ccccc2c1)NO
E3 Binder	CHEMBL4863947	ChEMBL	6.37	—	—	O=C(CCCCCONC(=O)c1[nH]nc2ccccc12)NO
E3 Binder	CHEMBL4635256	ChEMBL	6.46	—	—	O=C(CCCCCONC(=O)c1c(Cl)cncc1Cl)NO
E3 Binder	CHEMBL4846633	ChEMBL	6.09	—	—	O=C(CCCCCONC(=O)c1c[nH]c2ccccc12)NO
E3 Binder	CHEMBL4639388	ChEMBL	6.92	—	—	O=C(CCCCCONC(=O)c1cc(Br)cc(Br)c1)NO
E3 Binder	CHEMBL4638018	ChEMBL	6.25	—	—	O=C(CCCCCONC(=O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1)NO
E3 Binder	CHEMBL4638555	ChEMBL	7.0	—	—	O=C(CCCCCONC(=O)c1cc(F)cc(F)c1)NO
E3 Binder	CHEMBL4636427	ChEMBL	6.48	—	—	O=C(CCCCCONC(=O)c1cc(I)cc(I)c1I)NO
E3 Binder	CHEMBL4850081	ChEMBL	7.89	—	—	O=C(CCCCCONC(=O)c1cc2ccccc2[nH]1)NO
E3 Binder	CHEMBL4848096	ChEMBL	6.35	—	—	O=C(CCCCCONC(=O)c1ccc2[nH]ccc2c1)NO
E3 Binder	CHEMBL4876613	ChEMBL	6.4	—	—	O=C(CCCCCONC(=O)c1ccc2cc[nH]c2c1)NO
E3 Binder	CHEMBL4876405	ChEMBL	7.96	—	—	O=C(CCCCCONC(=O)c1ccc2ccccc2c1)NO
E3 Binder	CHEMBL4866536	ChEMBL	7.6	—	—	O=C(CCCCCONC(=O)c1ccc2ccccc2n1)NO
E3 Binder	CHEMBL4863503	ChEMBL	6.32	—	—	O=C(CCCCCONC(=O)c1cccc2[nH]ccc12)NO
E3 Binder	CHEMBL4849008	ChEMBL	6.34	—	—	O=C(CCCCCONC(=O)c1cccc2cc[nH]c12)NO
E3 Binder	CHEMBL4875953	ChEMBL	7.75	—	—	O=C(CCCCCONC(=O)c1cnc2ccccc2n1)NO
E3 Binder	CHEMBL4870868	ChEMBL	6.76	—	—	O=C(CCCCCONC(=O)c1nccc2ccccc12)NO
E3 Binder	CHEMBL3977601	ChEMBL	6.0	—	—	O=C(CCCCCOc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL4758680	ChEMBL	7.12	—	—	O=C(CCCCCOc1ccc(-c2csc(N3N=C(c4ccccc4)/C(=N/Nc4nccs4)C3=O)n2)cc1)NO
E3 Binder	CHEMBL5080255	ChEMBL	7.36	—	—	O=C(CCCCCOc1ccc(-c2nc3ccc(-c4nc5ccccc5[nH]4)cc3[nH]2)cc1)NO
E3 Binder	CHEMBL5088764	ChEMBL	7.12	—	—	O=C(CCCCCOc1ccc(-c2nc3ccccc3[nH]2)cc1)NO
E3 Binder	CHEMBL4280514	ChEMBL	6.29	—	—	O=C(CCCCCOc1ccc(-n2[se]c3ccccc3c2=O)cc1)NO
E3 Binder	CHEMBL5218611	ChEMBL	7.3	—	—	O=C(CCCCCOc1ccc2c(c1)N=C(NC(=O)c1ccccc1)N1CCN=C21)NO
E3 Binder	CHEMBL3951291	ChEMBL	7.55	—	—	O=C(CCCCCOc1ccc2cc1COC/C=C/COCc1cccc(c1)-c1ccnc(n1)N2)NO
E3 Binder	CHEMBL5080983	ChEMBL	7.56	—	—	O=C(CCCCCOc1cccc(-c2nc3ccc(-c4nc5ccccc5[nH]4)cc3[nH]2)c1)NO
E3 Binder	CHEMBL5069427	ChEMBL	6.93	—	—	O=C(CCCCCOc1cccc(-c2nc3ccccc3[nH]2)c1)NO
E3 Binder	CHEMBL5182740	ChEMBL	7.7	—	—	O=C(CCCCCOc1cccc(-c2nnc(-c3ccccc3)s2)c1)NO
E3 Binder	CHEMBL3426906	ChEMBL	8.13	—	—	O=C(CCCCCOc1no[n+]([O-])c1S(=O)(=O)c1ccccc1)NO
E3 Binder	CHEMBL203207	ChEMBL	7.4	—	—	O=C(CCCCCS(=O)(=O)c1ccccc1)NO
E3 Binder	CHEMBL109654	ChEMBL	7.17	—	—	O=C(CCCCCS)Nc1ccccc1
E3 Binder	CHEMBL200980	ChEMBL	6.58	—	—	O=C(CCCCCSc1ccc(Cl)cc1)NO
E3 Binder	CHEMBL371212	ChEMBL	6.96	—	—	O=C(CCCCCSc1ccc(NS(=O)(=O)c2ccc(Cl)cc2)cc1)NO
E3 Binder	CHEMBL203028	ChEMBL	6.92	—	—	O=C(CCCCCSc1ccccc1)NO
E3 Binder	CHEMBL4593437	ChEMBL	8.05	—	—	O=C(CCCCCSc1nc(-c2ccc(-c3ccccc3)cc2)cc(=O)[nH]1)NO
E3 Binder	CHEMBL4469596	ChEMBL	7.77	—	—	O=C(CCCCCSc1nc(-c2ccc3ccccc3c2)cc(=O)[nH]1)NO
E3 Binder	CHEMBL589918	ChEMBL	6.62	—	—	O=C(CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@@H]2CCCCCCCCCCCC[C@@H](NC1=O)C(=O)N2)NO
E3 Binder	CHEMBL589311	ChEMBL	6.55	—	—	O=C(CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@@H]2CCCCCCCCCCC[C@@H](NC1=O)C(=O)N2)NO
E3 Binder	CHEMBL592719	ChEMBL	6.39	—	—	O=C(CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@@H]2CCCCCCCCCC[C@@H](NC1=O)C(=O)N2)NO
E3 Binder	CHEMBL598363	ChEMBL	6.48	—	—	O=C(CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@@H]2CCCCCCCCC[C@@H](NC1=O)C(=O)N2)NO
E3 Binder	CHEMBL99392	ChEMBL	8.7	—	—	O=C(CCCCC[C@@H]1NC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccccc2)NC1=O)NO
E3 Binder	CHEMBL3098694	ChEMBL	8.4	—	—	O=C(CCCCC[C@H](NC(=O)C1C(=O)NCC1c1ccccc1)C(=O)Nc1ccccc1)NO
E3 Binder	CHEMBL3098692	ChEMBL	7.72	—	—	O=C(CCCCC[C@H](NC(=O)C1CCCNC1=O)C(=O)Nc1ccccc1)NO
E3 Binder	CHEMBL3098693	ChEMBL	8.4	—	—	O=C(CCCCC[C@H](NC(=O)C1CCNC1=O)C(=O)Nc1ccccc1)NO
E3 Binder	CHEMBL3098695	ChEMBL	8.52	—	—	O=C(CCCCC[C@H](NC(=O)[C@@H]1CC(=O)N1)C(=O)Nc1ccccc1)NO
E3 Binder	CHEMBL3098691	ChEMBL	8.52	—	—	O=C(CCCCC[C@H](NC(=O)[C@@H]1CCC(=O)N1)C(=O)Nc1ccccc1)NO
E3 Binder	CHEMBL3098697	ChEMBL	7.51	—	—	O=C(CCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)NC1CCCC1)NO
E3 Binder	CHEMBL3098687	ChEMBL	8.1	—	—	O=C(CCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)NCCc1ccccc1)NO
E3 Binder	CHEMBL3098689	ChEMBL	8.3	—	—	O=C(CCCCC[C@H](NC(=O)[C@@H]1CCCC(=O)N1)C(=O)Nc1ccccc1)NO
E3 Binder	CHEMBL3098688	ChEMBL	8.22	—	—	O=C(CCCCC[C@H](NC(=O)[C@H]1CCC(=O)N1)C(=O)NCCc1ccccc1)NO
E3 Binder	CHEMBL3098602	ChEMBL	8.7	—	—	O=C(CCCCC[C@H](NC(=O)[C@H]1CCC(=O)N1)C(=O)Nc1cccc(C(F)(F)F)c1)NO
E3 Binder	CHEMBL3098690	ChEMBL	8.1	—	—	O=C(CCCCC[C@H](NC(=O)[C@H]1CCC(=O)N1)C(=O)Nc1ccccc1)NO
E3 Binder	CHEMBL221655	ChEMBL	6.97	—	—	O=C(CCCCC[C@H](NC(=O)c1cc2ccccc2[nH]1)C(=O)Nc1cccc2cccnc12)NO
E3 Binder	CHEMBL198350	ChEMBL	6.82	—	—	O=C(CCCCC[S+]([O-])c1ccc(Cl)cc1)NO
E3 Binder	CHEMBL201473	ChEMBL	7.22	—	—	O=C(CCCCC[S+]([O-])c1ccccc1)NO
E3 Binder	CHEMBL3890846	ChEMBL	7.43	—	—	O=C(CCCCCc1ccc2c(c1)OCO2)NO
E3 Binder	CHEMBL550625	ChEMBL	6.22	—	—	O=C(CCCCCc1nc2cc3ccccc3cc2[nH]1)C(F)(F)F
E3 Binder	CHEMBL4293957	ChEMBL	6.74	—	—	O=C(CCCCCn1[se]c2ccccc2c1=O)NO
E3 Binder	CHEMBL2063485	ChEMBL	6.82	—	—	O=C(CCCCCn1c(=O)c2ccccc2c(=O)c2ccccc21)NO
E3 Binder	CHEMBL3675747	ChEMBL	7.05	—	—	O=C(CCCCCn1c2c(c3ccccc31)CCCC2)NO
E3 Binder	CHEMBL1290142	ChEMBL	7.39	—	—	O=C(CCCCCn1c2ccccc2c2ccccc21)NO
E3 Binder	CHEMBL479183	ChEMBL	7.28	—	—	O=C(CCCCCn1cc(-c2ccc(-c3ccccc3)cc2)nn1)NO
E3 Binder	CHEMBL477268	ChEMBL	8.64	—	—	O=C(CCCCCn1cc(-c2ccc(-c3ccncc3)cc2)nn1)NO
E3 Binder	CHEMBL4237410	ChEMBL	8.59	—	—	O=C(CCCCCn1cc(-c2ccc(Nc3c4ccccc4nc4ccccc34)cc2)nn1)NO
E3 Binder	CHEMBL518585	ChEMBL	8.68	—	—	O=C(CCCCCn1cc(-c2ccc3ccccc3n2)nn1)NO
E3 Binder	CHEMBL478163	ChEMBL	6.82	—	—	O=C(CCCCCn1cc(-c2ccc3cccnc3c2)nn1)NO
E3 Binder	CHEMBL5280359	ChEMBL	8.37	—	—	O=C(CCCCCn1cc(-c2ccc3ncnc(Nc4ccc(Br)cc4F)c3c2)nn1)NO
E3 Binder	CHEMBL3920583	ChEMBL	8.02	—	—	O=C(CCCCCn1cc(-c2ccc3ncnc(Nc4ccc(F)c(Cl)c4)c3c2)nn1)NO
E3 Binder	CHEMBL3964033	ChEMBL	7.03	—	—	O=C(CCCCCn1cc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)nn1)NO
E3 Binder	CHEMBL3939771	ChEMBL	7.84	—	—	O=C(CCCCCn1cc(-c2ccc3ncnc(Nc4ccc(OCc5nccs5)c(Cl)c4)c3c2)nn1)NO
E3 Binder	CHEMBL3929484	ChEMBL	8.39	—	—	O=C(CCCCCn1cc(-c2ccc3ncnc(Nc4cccc(Cl)c4F)c3c2)nn1)NO
E3 Binder	CHEMBL477093	ChEMBL	8.72	—	—	O=C(CCCCCn1cc(-c2cccc(-c3ccccc3)c2)nn1)NO
E3 Binder	CHEMBL4251261	ChEMBL	8.47	—	—	O=C(CCCCCn1cc(-c2cccc(Nc3c4ccccc4nc4ccccc34)c2)nn1)NO
E3 Binder	CHEMBL478108	ChEMBL	7.85	—	—	O=C(CCCCCn1cc(-c2ccccc2)nn1)NO
E3 Binder	CHEMBL477102	ChEMBL	6.79	—	—	O=C(CCCCCn1cc(-c2ccccc2-c2ccccc2)nn1)NO
E3 Binder	CHEMBL478308	ChEMBL	7.17	—	—	O=C(CCCCCn1cc(-c2ccccn2)nn1)NO
E3 Binder	CHEMBL478117	ChEMBL	6.54	—	—	O=C(CCCCCn1cc(-c2cccnc2)nn1)NO
E3 Binder	CHEMBL499754	ChEMBL	7.5	—	—	O=C(CCCCCn1cc(-c2cccs2)nn1)NO
E3 Binder	CHEMBL478307	ChEMBL	6.95	—	—	O=C(CCCCCn1cc(-c2ccncc2)nn1)NO
E3 Binder	CHEMBL4060602	ChEMBL	8.54	—	—	O=C(CCCCCn1cc(-c2ncnc3[nH]ccc23)cn1)NO
E3 Binder	CHEMBL5192298	ChEMBL	7.98	—	—	O=C(CCCCCn1cc(C(=O)NC2C3CC4CC(C3)CC2C4)c2ccccc21)NO
E3 Binder	CHEMBL4526274	ChEMBL	8.7	—	—	O=C(CCCCCn1cc(Nc2ncc(Cl)c(Nc3ccc(Cl)cc3)n2)cn1)NO
E3 Binder	CHEMBL4564021	ChEMBL	7.58	—	—	O=C(CCCCCn1cc(Nc2ncc(Cl)c(Nc3ccc(F)cc3)n2)cn1)NO
E3 Binder	CHEMBL4462229	ChEMBL	8.4	—	—	O=C(CCCCCn1cc(Nc2ncc(Cl)c(Nc3cccc(Cl)c3)n2)cn1)NO
E3 Binder	CHEMBL4559926	ChEMBL	7.75	—	—	O=C(CCCCCn1cc(Nc2ncc(Cl)c(Nc3ccccc3Cl)n2)cn1)NO
E3 Binder	CHEMBL5093859	ChEMBL	7.95	—	—	O=C(CCCCCn1cc(Nc2ncc3ccn(-c4ccc(Br)cc4)c3n2)cn1)NO
E3 Binder	CHEMBL5093906	ChEMBL	7.46	—	—	O=C(CCCCCn1cc(Nc2ncc3ccn(Cc4cccc(Cl)c4)c3n2)cn1)NO
E3 Binder	CHEMBL5092781	ChEMBL	7.86	—	—	O=C(CCCCCn1cc(Nc2ncc3ccn(Cc4cccc(F)c4)c3n2)cn1)NO
E3 Binder	CHEMBL5078697	ChEMBL	7.86	—	—	O=C(CCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4)c3n2)cn1)NO
E3 Binder	CHEMBL5070551	ChEMBL	7.35	—	—	O=C(CCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4Cl)c3n2)cn1)NO
E3 Binder	CHEMBL5083330	ChEMBL	7.82	—	—	O=C(CCCCCn1cc(Nc2ncc3ccn(Cc4ccccc4F)c3n2)cn1)NO
E3 Binder	CHEMBL3901188	ChEMBL	7.0	—	—	O=C(CCCCCn1ccc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)cc1=O)NO
E3 Binder	CHEMBL4084736	ChEMBL	6.24	—	—	O=C(CCCCN1C(=O)[C@@H](CS)N=C(c2ccccc2)c2ccccc21)NO
E3 Binder	CHEMBL4086281	ChEMBL	6.0	—	—	O=C(CCCCN1C(=O)[C@H](CCC(=O)NC(c2ccccc2)(c2ccccc2)c2ccccc2)N=C(c2ccccc2)c2ccccc21)NO
E3 Binder	CHEMBL3417185	ChEMBL	6.6	—	—	O=C(CCCCN1C/C=C/CCOc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO
E3 Binder	CHEMBL3417191	ChEMBL	6.8	—	—	O=C(CCCCN1C/C=C/COCc2cccc(c2)-c2ccnc(n2)Nc2cccc(c2)C1)NO
E3 Binder	CHEMBL5278646	ChEMBL	7.21	—	—	O=C(CCCCN1CC(=O)N2[C@H](c3ccc(Br)cc3)c3[nH]c4ccccc4c3C[C@@H]2C1=O)NO
E3 Binder	CHEMBL4227275	ChEMBL	6.56	—	—	O=C(CCCCNC(=O)c1cc(-c2ccc(F)cc2)[nH]n1)NO
E3 Binder	CHEMBL467998	ChEMBL	7.21	—	—	O=C(CCCCNC(=O)c1cc(-c2ccccc2)on1)NO
E3 Binder	CHEMBL4778142	ChEMBL	6.68	—	—	O=C(CCCCNC(=O)c1ccc(-c2csc(N3N=C(c4ccccc4)/C(=N/Nc4nccs4)C3=O)n2)cc1)NO
E3 Binder	CHEMBL3963714	ChEMBL	6.22	—	—	O=C(CCCCNC(=O)c1csc(-c2cccs2)n1)NO
E3 Binder	CHEMBL3968861	ChEMBL	6.73	—	—	O=C(CCCCNC(=O)c1nc(-c2nc(-c3ccccc3)cs2)sc1C1CC1)NO
E3 Binder	CHEMBL3906734	ChEMBL	6.48	—	—	O=C(CCCCNC(=O)c1nc(-c2nc(C3CC3)cs2)sc1C1CC1)NO
E3 Binder	CHEMBL3930328	ChEMBL	6.31	—	—	O=C(CCCCNC(=O)c1nc(-c2ncc(-c3ccccc3)s2)sc1C1CC1)NO
E3 Binder	CHEMBL3287258	ChEMBL	6.3	—	—	O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccc(F)cc1)NO
E3 Binder	CHEMBL3915628	ChEMBL	6.33	—	—	O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1cccc([N+](=O)[O-])c1)NO
E3 Binder	CHEMBL3287257	ChEMBL	6.33	—	—	O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccccc1)NO
E3 Binder	CHEMBL3891112	ChEMBL	6.11	—	—	O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1/C=C/c1ccccc1)NO
E3 Binder	CHEMBL3287255	ChEMBL	7.21	—	—	O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1C1CC1)NO
E3 Binder	CHEMBL3287256	ChEMBL	6.13	—	—	O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1C1CCCCC1)NO
E3 Binder	CHEMBL3287263	ChEMBL	6.02	—	—	O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1CCOCc1ccccc1)NO
E3 Binder	CHEMBL513160	ChEMBL	7.3	—	—	O=C(CCCCOCc1cc(-c2ccccc2)on1)NO
E3 Binder	CHEMBL3925515	ChEMBL	7.0	—	—	O=C(CCCCONC(=O)c1ccc(F)c(F)c1Nc1ccc(I)cc1F)NO
E3 Binder	CHEMBL3968341	ChEMBL	7.0	—	—	O=C(CCCCOc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL1165020	ChEMBL	7.1	—	—	O=C(CCCCOc1ccc(-c2cc(=S)ss2)cc1)NO
E3 Binder	CHEMBL4797324	ChEMBL	6.93	—	—	O=C(CCCCOc1ccc(-c2csc(N3N=C(c4ccccc4)/C(=N/Nc4nccs4)C3=O)n2)cc1)NO
E3 Binder	CHEMBL5087595	ChEMBL	6.66	—	—	O=C(CCCCOc1ccc(-c2nc3ccc(-c4nc5ccccc5[nH]4)cc3[nH]2)cc1)NO
E3 Binder	CHEMBL5086631	ChEMBL	6.72	—	—	O=C(CCCCOc1ccc(-c2nc3ccccc3[nH]2)cc1)NO
E3 Binder	CHEMBL3980203	ChEMBL	6.97	—	—	O=C(CCCCOc1ccc2cc1COC/C=C/COCc1cccc(c1)-c1ccnc(n1)N2)NO
E3 Binder	CHEMBL3905086	ChEMBL	7.0	—	—	O=C(CCCCOc1ccc2ncnc(Nc3ccc(F)c(Cl)c3)c2c1)NO
E3 Binder	CHEMBL5074277	ChEMBL	6.52	—	—	O=C(CCCCOc1cccc(-c2nc3ccc(-c4nc5ccccc5[nH]4)cc3[nH]2)c1)NO
E3 Binder	CHEMBL5077786	ChEMBL	6.71	—	—	O=C(CCCCOc1cccc(-c2nc3ccccc3[nH]2)c1)NO
E3 Binder	CHEMBL5205120	ChEMBL	7.5	—	—	O=C(CCCCOc1cccc(-c2nnc(-c3ccccc3)s2)c1)NO
E3 Binder	CHEMBL3426803	ChEMBL	8.15	—	—	O=C(CCCCSc1nc(-c2ccc(-c3ccccc3)cc2)cc(=O)[nH]1)NO
E3 Binder	CHEMBL4476057	ChEMBL	7.92	—	—	O=C(CCCCSc1nc(-c2ccc3ccccc3c2)cc(=O)[nH]1)NO
E3 Binder	CHEMBL468527	ChEMBL	6.05	—	—	O=C(CCCCc1cc(C(=O)NO)no1)Nc1ccc(-c2ccccc2)cc1
E3 Binder	CHEMBL1243261	ChEMBL	6.37	—	—	O=C(CCCCc1cc(C(=O)NO)no1)Nc1ccccc1
E3 Binder	CHEMBL511715	ChEMBL	7.29	—	—	O=C(CCCCc1cc(C(=O)NO)no1)Nc1cnc2ccccc2c1
E3 Binder	CHEMBL469134	ChEMBL	7.17	—	—	O=C(CCCCc1cc(C(=O)NO)no1)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL190014	ChEMBL	6.6	—	—	O=C(CCCCc1ccccc1)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3335288	ChEMBL	7.19	—	—	O=C(CCCCc1ccn(-c2ccccc2)n1)NO
E3 Binder	CHEMBL3335300	ChEMBL	7.47	—	—	O=C(CCCCc1ccn(Cc2ccc(-c3ccccc3)cc2)n1)NO
E3 Binder	CHEMBL3335298	ChEMBL	6.8	—	—	O=C(CCCCc1ccn(Cc2ccc(-n3ccc4ccccc43)cc2)n1)NO
E3 Binder	CHEMBL3335299	ChEMBL	7.19	—	—	O=C(CCCCc1ccn(Cc2ccc(Nc3ccccc3)cc2)n1)NO
E3 Binder	CHEMBL5187023	ChEMBL	8.22	—	—	O=C(CCCCc1nnc(-c2cc3c([nH]c4ccccc43)c(-c3ccc(C(F)(F)F)cc3)n2)o1)NO
E3 Binder	CHEMBL4286053	ChEMBL	6.45	—	—	O=C(CCCCn1[se]c2ccccc2c1=O)NO
E3 Binder	CHEMBL5201054	ChEMBL	8.37	—	—	O=C(CCCCn1cc(-c2ccc3ncnc(Nc4ccccc4F)c3c2)nn1)NO
E3 Binder	CHEMBL477943	ChEMBL	6.96	—	—	O=C(CCCCn1cc(-c2ccccc2)nn1)NO
E3 Binder	CHEMBL4088824	ChEMBL	8.22	—	—	O=C(CCCCn1cc(-c2ncnc3[nH]ccc23)cn1)NO
E3 Binder	CHEMBL5176749	ChEMBL	7.4	—	—	O=C(CCCCn1cc(C(=O)NC2C3CC4CC(C3)CC2C4)c2ccccc21)NO
E3 Binder	CHEMBL4568644	ChEMBL	6.51	—	—	O=C(CCCCn1cc(Nc2ncc(Cl)c(Nc3ccc(F)cc3)n2)cn1)NO
E3 Binder	CHEMBL3898427	ChEMBL	6.0	—	—	O=C(CCCCn1ccc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)cc1=O)NO
E3 Binder	CHEMBL3912163	ChEMBL	6.0	—	—	O=C(CCCNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL4867598	ChEMBL	6.89	—	—	O=C(CCCO/N=C1C(=C2/C(=O)Nc3ccccc32)/Nc2ccccc2/1)NO
E3 Binder	CHEMBL3967834	ChEMBL	6.0	—	—	O=C(CCCONC(=O)c1ccc(F)c(F)c1Nc1ccc(I)cc1F)NO
E3 Binder	CHEMBL3939256	ChEMBL	6.0	—	—	O=C(CCCOc1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL4761391	ChEMBL	6.17	—	—	O=C(CCCOc1ccc(-c2csc(N3N=C(c4ccccc4)/C(=N/Nc4nccs4)C3=O)n2)cc1)NO
E3 Binder	CHEMBL5079152	ChEMBL	6.01	—	—	O=C(CCCOc1ccc(-c2nc3ccccc3[nH]2)cc1)NO
E3 Binder	CHEMBL4288401	ChEMBL	6.04	—	—	O=C(CCCOc1ccc(-n2[se]c3ccccc3c2=O)cc1)NO
E3 Binder	CHEMBL3942555	ChEMBL	6.29	—	—	O=C(CCCOc1ccc2cc1COC/C=C/COCc1cccc(c1)-c1ccnc(n1)N2)NO
E3 Binder	CHEMBL5093425	ChEMBL	7.3	—	—	O=C(CCCOc1cccc(-c2nc3ccc(-c4nc5ccccc5[nH]4)cc3[nH]2)c1)NO
E3 Binder	CHEMBL5093054	ChEMBL	6.31	—	—	O=C(CCCOc1cccc(-c2nc3ccccc3[nH]2)c1)NO
E3 Binder	CHEMBL5088034	ChEMBL	7.71	—	—	O=C(CCCSC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1cccc2ccccc12)NO
E3 Binder	CHEMBL5093258	ChEMBL	7.69	—	—	O=C(CCCSC[C@H](NC(=O)OCc1ccccc1)C(=O)Nc1ccccc1)NO
E3 Binder	CHEMBL5089854	ChEMBL	7.86	—	—	O=C(CCCSC[C@H](NC(=O)c1ccccc1)C(=O)Nc1ccccc1)NO
E3 Binder	CHEMBL347734	ChEMBL	6.28	—	—	O=C(CCCc1ccccc1)NCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL55895	ChEMBL	6.82	4R9	—	O=C(CCCc1ccccc1)NO
E3 Binder	CHEMBL143336	ChEMBL	7.36	—	—	O=C(CCCc1ccccc1)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL3792392	ChEMBL	6.7	—	—	O=C(CCCc1csc(/C=C/c2ccccc2)n1)NO
E3 Binder	CHEMBL4458196	ChEMBL	7.02	—	—	O=C(CCCc1csc(CCc2ccccc2)n1)NO
E3 Binder	CHEMBL4446737	ChEMBL	6.08	—	—	O=C(CCCc1csc(Cc2ccccc2)n1)NO
E3 Binder	CHEMBL4089113	ChEMBL	6.22	—	—	O=C(CCCn1cc(-c2ncnc3[nH]ccc23)cn1)NO
E3 Binder	CHEMBL3952662	ChEMBL	6.0	—	—	O=C(CCCn1ccc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)cc1=O)NO
E3 Binder	CHEMBL4577419	ChEMBL	7.9	—	—	O=C(CCN(Cc1ccc(C(=O)NO)cc1)C(=O)c1ccccc1)NCc1ccccc1
E3 Binder	CHEMBL3593627	ChEMBL	6.9	—	—	O=C(CCN1C(=O)C2(OCCCO2)c2cc(Br)ccc21)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL2047684	ChEMBL	7.02	—	—	O=C(CCNC(=O)/C(Cc1ccc(O)c(Br)c1)=N/O)NO
E3 Binder	CHEMBL3909453	ChEMBL	6.0	—	—	O=C(CCNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)cc2)ccn1)NO
E3 Binder	CHEMBL3930226	ChEMBL	6.0	—	—	O=C(CCOc1ccc2ncnc(Nc3ccc(F)c(Cl)c3)c2c1)NO
E3 Binder	CHEMBL4287851	ChEMBL	7.32	—	—	O=C(CC[C@@H](CCCC(=O)Nc1ccccc1)Cc1ccccc1)NO
E3 Binder	CHEMBL4283418	ChEMBL	7.02	—	—	O=C(CC[C@H](CCCC(=O)Nc1ccccc1)Cc1ccccc1)NO
E3 Binder	CHEMBL4520424	ChEMBL	7.51	—	—	O=C(CCc1cc(C(=O)NO)no1)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL5288873	ChEMBL	6.0	—	—	O=C(CCc1ccc(C(=O)NCC2CCN(Cc3ccccc3)CC2)cc1)NO
E3 Binder	CHEMBL4860339	ChEMBL	6.46	—	—	O=C(CCc1ccc(CN2c3ccccc3Sc3ccccc32)cc1)NO
E3 Binder	CHEMBL142048	ChEMBL	6.28	—	—	O=C(CCc1ccc(NC(=O)CCCc2ccccc2)cc1)NO
E3 Binder	CHEMBL356579	ChEMBL	6.17	—	—	O=C(CCc1ccc(NC(=O)Cc2ccccc2)cc1)NO
E3 Binder	CHEMBL4740829	ChEMBL	6.98	—	—	O=C(CCc1ccc(NC(=O)Nc2ccc(Cl)cc2)cc1)NO
E3 Binder	CHEMBL4248676	ChEMBL	7.0	—	—	O=C(CCc1ccc(Nc2c3ccccc3nc3ccccc23)cc1)NO
E3 Binder	CHEMBL194851	ChEMBL	6.39	—	—	O=C(CCc1ccc2c(c1)C(=O)N(Cc1ccccc1)C2=O)NO
E3 Binder	CHEMBL2048758	ChEMBL	6.39	—	—	O=C(CCc1ccc2c(ccn2S(=O)(=O)c2ccccc2)c1)NO
E3 Binder	CHEMBL5270654	ChEMBL	6.33	—	—	O=C(CCc1cccc(C(=O)NCC2CCN(Cc3ccccc3)CC2)c1)NO
E3 Binder	CHEMBL152162	ChEMBL	6.35	—	—	O=C(CCc1ccccc1)NO
E3 Binder	CHEMBL189912	ChEMBL	6.96	—	—	O=C(CCc1ccccc1)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4542710	ChEMBL	6.93	—	—	O=C(CCc1csc(/C=C/c2c[nH]c3ccccc23)n1)NO
E3 Binder	CHEMBL4445910	ChEMBL	6.51	—	—	O=C(CCc1csc(/C=C/c2ccc(Br)cc2)n1)NO
E3 Binder	CHEMBL4450477	ChEMBL	6.23	—	—	O=C(CCc1csc(/C=C/c2ccc(Cl)cc2)n1)NO
E3 Binder	CHEMBL4436629	ChEMBL	7.37	—	—	O=C(CCc1csc(/C=C/c2ccc(F)cc2)n1)NO
E3 Binder	CHEMBL4439017	ChEMBL	7.27	—	—	O=C(CCc1csc(CCc2c[nH]c3ccccc23)n1)NO
E3 Binder	CHEMBL4565948	ChEMBL	7.8	—	—	O=C(CCc1csc(CCc2ccc(Br)cc2)n1)NO
E3 Binder	CHEMBL4582980	ChEMBL	7.41	—	—	O=C(CCc1csc(CCc2ccc(C(F)(F)F)cc2)n1)NO
E3 Binder	CHEMBL4538156	ChEMBL	7.81	—	—	O=C(CCc1csc(CCc2ccc(Cl)cc2)n1)NO
E3 Binder	CHEMBL4591740	ChEMBL	7.69	—	—	O=C(CCc1csc(CCc2ccc(F)c(F)c2)n1)NO
E3 Binder	CHEMBL4516093	ChEMBL	7.67	—	—	O=C(CCc1csc(CCc2ccc(F)cc2)n1)NO
E3 Binder	CHEMBL4474608	ChEMBL	6.25	—	—	O=C(CCc1csc(CCc2ccc(O)c(O)c2)n1)NO
E3 Binder	CHEMBL4446389	ChEMBL	7.25	—	—	O=C(CCc1csc(CCc2ccc(O)cc2)n1)NO
E3 Binder	CHEMBL4435558	ChEMBL	7.36	—	—	O=C(CCc1csc(CCc2ccc([N+](=O)[O-])cc2)n1)NO
E3 Binder	CHEMBL4435211	ChEMBL	7.42	—	—	O=C(CCc1csc(CCc2cccc(F)c2)n1)NO
E3 Binder	CHEMBL4570194	ChEMBL	7.51	—	—	O=C(CCc1csc(CCc2ccccc2)n1)NO
E3 Binder	CHEMBL4467027	ChEMBL	7.0	—	—	O=C(CCc1csc(CCc2ccco2)n1)NO
E3 Binder	CHEMBL4514922	ChEMBL	7.47	—	—	O=C(CCc1csc(CCc2cccs2)n1)NO
E3 Binder	CHEMBL4849235	ChEMBL	7.3	—	—	O=C(CN(Cc1ccc(C(=O)NO)cc1)C(=O)Cc1ccccc1)NC1CCCCC1
E3 Binder	CHEMBL4851776	ChEMBL	7.52	—	—	O=C(CN(Cc1ccc(C(=O)NO)cc1)C(=O)Cc1ccccc1)NCc1ccccc1
E3 Binder	CHEMBL4854577	ChEMBL	8.0	—	—	O=C(CN(Cc1ccc(C(=O)NO)cc1)C(=O)c1cccc2ccccc12)NCc1ccccc1
E3 Binder	CHEMBL5187865	ChEMBL	7.57	—	—	O=C(CN(Cc1ccc(C(=O)NO)cc1F)C(=O)c1ccccc1C(F)(F)F)NC1CCCCC1
E3 Binder	CHEMBL5184839	ChEMBL	7.75	—	—	O=C(CN(Cc1ccc(C(=O)NO)cc1F)C(=O)c1ccccc1F)NC1CCCCC1
E3 Binder	CHEMBL4532891	ChEMBL	6.47	—	—	O=C(CNC(=O)CNC(=O)OCc1ccccc1)NCc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4515619	ChEMBL	6.01	—	—	O=C(CNC(=S)N/N=C1\C(=O)Nc2ccc(Cl)cc21)NO
E3 Binder	CHEMBL5093666	ChEMBL	6.8	—	—	O=C(COc1ccc(-c2nc3ccccc3[nH]2)cc1)NO
E3 Binder	CHEMBL3601776	ChEMBL	6.26	—	—	O=C(COc1ccc(C(=O)NO)cc1)Nc1ccc2ccnc(Nc3ccc4ccccc4c3)c2c1
E3 Binder	CHEMBL5185297	ChEMBL	7.85	—	—	O=C(COc1ccc(CNCCc2c[nH]c3ccccc23)c(F)c1)NO
E3 Binder	CHEMBL402451	ChEMBL	6.82	—	—	O=C(CS)CCCCCCC(=O)Nc1ccccc1
E3 Binder	CHEMBL4096524	ChEMBL	6.27	—	—	O=C(CS)NCC(S)CCCn1ccc2cc(Cl)c(Cl)cc21
E3 Binder	CHEMBL194777	ChEMBL	6.18	—	—	O=C(CS)NCCCC(=O)Nc1cnc2ccccc2c1
E3 Binder	CHEMBL3938429	ChEMBL	6.68	—	—	O=C(CS)NCCCCCC(=O)Nc1ccc(-c2ccccc2NC(=O)[C@@H]2CCCN2)cc1
E3 Binder	CHEMBL178858	ChEMBL	6.05	—	—	O=C(CS)NCCCCCC(=O)Nc1ccc2ncccc2c1
E3 Binder	CHEMBL178456	ChEMBL	7.7	—	—	O=C(CS)NCCCCCC(=O)Nc1cccc2cccnc12
E3 Binder	CHEMBL178727	ChEMBL	6.41	9Z8	—	O=C(CS)NCCCCCC(=O)Nc1ccccc1
E3 Binder	CHEMBL4079113	ChEMBL	6.62	—	—	O=C(CS)NCCCCCCn1cc(Cl)c2cc(Cl)c(Cl)cc21
E3 Binder	CHEMBL4102024	ChEMBL	7.19	—	—	O=C(CS)NCCCCCCn1ccc2cc(Cl)c(Cl)cc21
E3 Binder	CHEMBL4094909	ChEMBL	7.19	—	—	O=C(CS)NCCCCCCn1ccc2cc(F)c(Cl)cc21
E3 Binder	CHEMBL4094664	ChEMBL	7.83	—	—	O=C(CS)NCCCCCNc1c(Cl)cc(Cl)c2cccnc12
E3 Binder	CHEMBL4066042	ChEMBL	7.48	—	—	O=C(CS)NCCCCCOc1c(Cl)cc(Cl)c2cccnc12
E3 Binder	CHEMBL4065147	ChEMBL	7.96	W45	—	O=C(CS)NCCCCCn1ccc2cc(Cl)c(Cl)cc21
E3 Binder	CHEMBL4076426	ChEMBL	8.55	—	—	O=C(CS)NCCCCNc1c(Cl)cc(Cl)c2cccnc12
E3 Binder	CHEMBL3758407	ChEMBL	6.06	—	—	O=C(CS)NCCCNC(=O)c1cc(-c2ccc(F)cc2)[nH]n1
E3 Binder	CHEMBL242894	ChEMBL	7.0	—	—	O=C(CSC(=S)Sc1ccccc1)c1ccc(Cl)c(Cl)c1
E3 Binder	CHEMBL3905394	ChEMBL	7.0	—	—	O=C(CSSCC(=O)NCCCCCC(=O)Nc1nc(-c2ccccc2)cs1)NCCCCCC(=O)Nc1nc(-c2ccccc2)cs1
E3 Binder	CHEMBL3347686	ChEMBL	6.87	—	—	O=C(CSSCC(=O)c1ccc(Br)cc1)c1ccc(Br)cc1
E3 Binder	CHEMBL4077645	ChEMBL	8.22	—	—	O=C(Cc1ccc(C(=O)NO)cc1)NC1=CC(=O)c2ccccc2C1=O
E3 Binder	CHEMBL4075511	ChEMBL	6.89	—	—	O=C(Cc1ccc(CN2CCN(C(=O)c3cc(Cc4n[nH]c(=O)c5ccccc45)ccc3F)CC2)cc1)NO
E3 Binder	CHEMBL3675753	ChEMBL	6.52	—	—	O=C(Cc1ccc(Cn2c3ccccc3c3ccccc32)cc1)NO
E3 Binder	CHEMBL4757768	ChEMBL	7.13	—	—	O=C(Cc1ccc(Nc2c3ccccc3nc3ccccc23)cc1)NO
E3 Binder	CHEMBL2047675	ChEMBL	6.0	—	—	O=C(Cc1ccc(O)c(Br)c1)C(=O)NCCS
E3 Binder	CHEMBL4745420	ChEMBL	6.34	—	—	O=C(Cc1ccc(OCCCn2c3c(c4cccc(Cl)c42)CCNC3)cc1)NO
E3 Binder	CHEMBL4521590	ChEMBL	7.58	—	—	O=C(Cc1cccc2ccccc12)Nc1ccc(C(=O)NO)nc1
E3 Binder	CHEMBL356824	ChEMBL	6.96	—	—	O=C(Cc1ccccc1)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL4435005	ChEMBL	7.43	—	—	O=C(Cc1ccccc1)Nc1ccc(C(=O)NO)nc1
E3 Binder	CHEMBL5269889	ChEMBL	6.62	—	—	O=C(Cc1cnc(N2CCC(CN3CC(=O)N4[C@H](c5ccc6c(c5)OCO6)c5[nH]c6ccccc6c5C[C@@H]4C3=O)CC2)nc1)NO
E3 Binder	CHEMBL462202	ChEMBL	6.15	—	—	O=C(Cc1noc(-c2ccc(C(=O)C(F)(F)F)s2)n1)N1CCCC1
E3 Binder	CHEMBL386473	ChEMBL	8.15	—	—	O=C(Cn1ccc(-c2ccc(C(=O)NO)s2)n1)Nc1cccc2cccnc12
E3 Binder	CHEMBL385406	ChEMBL	7.68	—	—	O=C(Cn1ccc(-c2ccc(C(=O)NO)s2)n1)Nc1ccccc1
E3 Binder	CHEMBL4543038	ChEMBL	8.12	—	—	O=C(NC(CCCCCSSCCCCCC(NC(=O)OCc1ccccc1)C(=O)Nc1cccc2cccnc12)C(=O)Nc1cccc2cccnc12)OCc1ccccc1
E3 Binder	CHEMBL4438404	ChEMBL	8.49	—	—	O=C(NC(CCCCCSSCCO)C(=O)Nc1cccc2cccnc12)OCc1ccccc1
E3 Binder	CHEMBL5187827	ChEMBL	6.63	—	—	O=C(NC1C2CC3CC(C2)CC1C3)c1cn(CCCCCCCS)c2ccccc12
E3 Binder	CHEMBL5173462	ChEMBL	7.72	—	—	O=C(NC1C2CC3CC(C2)CC1C3)c1cn(CCCCCCS)c2ccccc12
E3 Binder	CHEMBL3110004	ChEMBL	6.05	NU9	—	O=C(NCC1(c2nc(-c3ccccc3)cs2)CCOCC1)c1cccc(-c2noc(C(F)(F)F)n2)c1
E3 Binder	CHEMBL275380	ChEMBL	6.51	—	—	O=C(NCC1CCC(C(=O)NO)CC1)c1ccc(-c2ccccc2)cc1
E3 Binder	CHEMBL497331	ChEMBL	6.34	—	—	O=C(NCC1CCCCC1)c1ccc(C(=O)C(F)(F)F)s1
E3 Binder	CHEMBL3770504	ChEMBL	7.75	—	—	O=C(NCCCCC(=O)C(F)(F)F)c1nc(-c2nc3c(s2)CCCC3)sc1C1CC1
E3 Binder	CHEMBL3770287	ChEMBL	7.68	—	—	O=C(NCCCCC(=O)C(F)(F)F)c1nc(-c2nccs2)sc1C1CC1
E3 Binder	CHEMBL3771288	ChEMBL	7.23	—	—	O=C(NCCCCC(=O)C(F)(F)F)c1nc(-c2nccs2)sc1Cc1ccccc1
E3 Binder	CHEMBL609609	ChEMBL	6.54	—	—	O=C(NCCCCC/C=C(\F)CS)c1ccccc1
E3 Binder	CHEMBL3770531	ChEMBL	6.84	—	—	O=C(NCCCCCC(=O)C(F)(F)F)c1nc(-c2nccs2)sc1C1CC1
E3 Binder	CHEMBL338816	ChEMBL	6.47	—	—	O=C(NCCCCCC(=O)c1ncco1)c1cc2ccccc2[nH]1
E3 Binder	CHEMBL340725	ChEMBL	7.05	—	—	O=C(NCCCCCCC(=O)c1ncco1)c1cc2ccccc2[nH]1
E3 Binder	CHEMBL3759322	ChEMBL	7.48	—	—	O=C(NCCCCCCS)c1cc(-c2c[nH]c3ccccc23)n[nH]1
E3 Binder	CHEMBL3758334	ChEMBL	7.37	—	—	O=C(NCCCCCCS)c1cc(-c2ccc(-c3ccccc3)cc2)n[nH]1
E3 Binder	CHEMBL3758445	ChEMBL	6.66	—	—	O=C(NCCCCCCS)c1cc(-c2ccc(F)cc2)n(CCCCO)n1
E3 Binder	CHEMBL3760074	ChEMBL	6.07	—	—	O=C(NCCCCCCS)c1cc(-c2ccc(F)cc2)n(CCCO)n1
E3 Binder	CHEMBL3758444	ChEMBL	6.61	—	—	O=C(NCCCCCCS)c1cc(-c2ccc(F)cc2)n[nH]1
E3 Binder	CHEMBL3758692	ChEMBL	6.85	—	—	O=C(NCCCCCCS)c1cc(-c2ccc(F)cc2)nn1CCCCO
E3 Binder	CHEMBL3758842	ChEMBL	6.33	—	—	O=C(NCCCCCCS)c1cc(-c2ccc(F)cc2)nn1CCCO
E3 Binder	CHEMBL3758642	ChEMBL	6.16	—	—	O=C(NCCCCCCS)c1cc(-c2ccc(F)cc2)nn1CCO
E3 Binder	CHEMBL3759880	ChEMBL	6.06	—	—	O=C(NCCCCCCS)c1cc(-c2ccc(F)cc2)on1
E3 Binder	CHEMBL3759836	ChEMBL	6.99	—	—	O=C(NCCCCCCS)c1cc(-c2ccc3ccccc3c2)n[nH]1
E3 Binder	CHEMBL3758595	ChEMBL	6.61	—	—	O=C(NCCCCCCS)c1cc(-c2cccc3ccccc23)n[nH]1
E3 Binder	CHEMBL3759791	ChEMBL	7.64	—	—	O=C(NCCCCCCS)c1cc(-c2ccccc2)n[nH]1
E3 Binder	CHEMBL3758261	ChEMBL	7.57	—	—	O=C(NCCCCCCS)c1cc(-c2ccccn2)n[nH]1
E3 Binder	CHEMBL3758882	ChEMBL	7.82	—	—	O=C(NCCCCCCS)c1cc(-c2cccnc2)n[nH]1
E3 Binder	CHEMBL3759562	ChEMBL	8.1	—	—	O=C(NCCCCCCS)c1cc(-c2ccncc2)n[nH]1
E3 Binder	CHEMBL3760013	ChEMBL	7.75	—	—	O=C(NCCCCCCS)c1cc(-c2cnccn2)n[nH]1
E3 Binder	CHEMBL3758451	ChEMBL	6.62	—	—	O=C(NCCCCCCS)c1cc(C2CCCCC2)n[nH]1
E3 Binder	CHEMBL113159	ChEMBL	7.0	—	—	O=C(NCCCCCCS)c1cc2ccccc2[nH]1
E3 Binder	CHEMBL112105	ChEMBL	7.1	—	—	O=C(NCCCCCCS)c1cc2ccccc2o1
E3 Binder	CHEMBL113421	ChEMBL	7.07	—	—	O=C(NCCCCCCS)c1ccc2ccccc2c1
E3 Binder	CHEMBL112364	ChEMBL	6.44	—	—	O=C(NCCCCCCS)c1ccccc1
E3 Binder	CHEMBL3759941	ChEMBL	7.09	—	—	O=C(NCCCCCCS)c1ccn[nH]1
E3 Binder	CHEMBL2047701	ChEMBL	6.1	—	—	O=C(NCCS)/C(Cc1cc(Br)c(O)c(Br)c1)=N/O
E3 Binder	CHEMBL2047700	ChEMBL	6.13	—	—	O=C(NCCS)/C(Cc1cc(Br)cc([N+](=O)[O-])c1)=N/O
E3 Binder	CHEMBL2047692	ChEMBL	6.19	—	—	O=C(NCCS)/C(Cc1ccc(F)c(Br)c1)=N/O
E3 Binder	CHEMBL2047540	ChEMBL	6.44	—	—	O=C(NCCS)/C(Cc1ccc(O)c(Br)c1)=N/O
E3 Binder	CHEMBL4460345	ChEMBL	6.55	—	—	O=C(NCCSSCCNC(=O)/C(Cc1ccc(Cl)cc1Cl)=N/O)/C(Cc1ccc(Cl)cc1Cl)=N/O
E3 Binder	CHEMBL83747	ChEMBL	8.4	—	—	O=C(NCCSSCCNC(=O)/C(Cc1ccc(O)c(Br)c1)=N/O)/C(Cc1ccc(O)c(Br)c1)=N/O
E3 Binder	CHEMBL1818029	ChEMBL	6.92	—	—	O=C(NCCSSCCNC(=O)/C(Cc1ccc(O)cc1)=N/O)/C(Cc1ccc(O)cc1)=N/O
E3 Binder	CHEMBL4450983	ChEMBL	6.89	—	—	O=C(NCCSSCCNC(=O)/C(Cc1ccc2c(c1)OCO2)=N/O)/C(Cc1ccc2c(c1)OCO2)=N/O
E3 Binder	CHEMBL4475727	ChEMBL	6.57	—	—	O=C(NCCSSCCNC(=O)/C(Cc1cccc(C(F)(F)F)c1)=N/O)/C(Cc1cccc(C(F)(F)F)c1)=N/O
E3 Binder	CHEMBL4443774	ChEMBL	6.68	—	—	O=C(NCCSSCCNC(=O)/C(Cc1cccc(Cl)c1)=N/O)/C(Cc1cccc(Cl)c1)=N/O
E3 Binder	CHEMBL4557651	ChEMBL	6.17	—	—	O=C(NCCSSCCNC(=O)c1cc(-c2ccc(O)c(Br)c2)[nH]n1)c1cc(-c2ccc(O)c(Br)c2)[nH]n1
E3 Binder	CHEMBL4469488	ChEMBL	7.92	JNN	—	O=C(NCCc1cc(C(=O)NO)no1)c1ccc(Cl)c(Cl)c1
E3 Binder	CHEMBL4556111	ChEMBL	8.0	—	—	O=C(NCCc1cc(C(=O)NO)no1)c1ccc2ccccc2c1
E3 Binder	CHEMBL4483795	ChEMBL	7.62	—	—	O=C(NCCc1cc(C(=O)NO)no1)c1cccc(-c2ccccc2)c1
E3 Binder	CHEMBL4584312	ChEMBL	6.72	—	—	O=C(NCCc1cc(C(=O)NO)no1)c1ccccc1
E3 Binder	CHEMBL523588	ChEMBL	6.68	—	—	O=C(NCCc1ccccc1)c1ccc(C(=O)C(F)(F)F)s1
E3 Binder	CHEMBL455455	ChEMBL	6.43	—	—	O=C(NCc1ccccc1)c1ccc(C(=O)C(F)(F)F)s1
E3 Binder	CHEMBL519738	ChEMBL	6.72	—	—	O=C(NCc1ccccc1Cl)c1ccc(C(=O)C(F)(F)F)s1
E3 Binder	CHEMBL583967	ChEMBL	6.05	—	—	O=C(NO)C(c1ccc2c(c1)CCO2)c1ccc2c(c1)CCO2
E3 Binder	CHEMBL2333346	ChEMBL	7.52	FBJ	—	O=C(NO)C1=CCCC1
E3 Binder	CHEMBL2333344	ChEMBL	7.92	FBM	—	O=C(NO)C1=CCCCC1
E3 Binder	CHEMBL2333345	ChEMBL	6.42	F9P	—	O=C(NO)C1CCCCC1
E3 Binder	CHEMBL3961053	ChEMBL	6.05	—	—	O=C(NO)C1CCN(CCOc2ccc3cc2COC/C=C/COCc2cccc(c2)-c2ccnc(n2)N3)CC1
E3 Binder	CHEMBL4551620	ChEMBL	6.16	—	—	O=C(NO)c1cc(CCCCN2CCCc3cc(Cl)ccc32)on1
E3 Binder	CHEMBL4470946	ChEMBL	6.7	—	—	O=C(NO)c1cc(CCCOc2ccc(Cl)c(Cl)c2)on1
E3 Binder	CHEMBL4515782	ChEMBL	8.4	—	—	O=C(NO)c1cc(F)c(Cc2nnc(-c3ccncc3)s2)c(F)c1
E3 Binder	CHEMBL4548513	ChEMBL	8.0	—	—	O=C(NO)c1cc(F)c(Cn2nnc(-c3ccc4ccccc4n3)n2)c(F)c1
E3 Binder	CHEMBL4440341	ChEMBL	8.15	—	—	O=C(NO)c1cc(F)c(Cn2nnc(-c3ccccn3)n2)c(F)c1
E3 Binder	CHEMBL4458053	ChEMBL	8.52	—	—	O=C(NO)c1cc(F)c(Cn2nnc(-c3ccco3)n2)c(F)c1
E3 Binder	CHEMBL4439065	ChEMBL	7.66	—	—	O=C(NO)c1cc(F)c(Cn2nnc(-c3nccc4ccccc34)n2)c(F)c1
E3 Binder	CHEMBL4470373	ChEMBL	8.3	V05	—	O=C(NO)c1cc(F)c(Cn2nnc(-c3ncccn3)n2)c(F)c1
E3 Binder	CHEMBL4862563	ChEMBL	7.72	—	—	O=C(NO)c1cc(F)c(Cn2nnnc2-c2cccs2)c(F)c1
E3 Binder	CHEMBL4852905	ChEMBL	9.0	—	—	O=C(NO)c1cc(F)c2c(c1)CCN(C1CCC1)C2
E3 Binder	CHEMBL4847638	ChEMBL	9.0	—	—	O=C(NO)c1cc(F)c2c(c1)CCn1cccc1-2
E3 Binder	CHEMBL2431921	ChEMBL	7.44	—	—	O=C(NO)c1cc2c(s1)CCN(C(=O)C1CCCCC1)C2
E3 Binder	CHEMBL2431918	ChEMBL	7.7	—	—	O=C(NO)c1cc2c(s1)CN(C(=O)C1CCCCC1)CC2
E3 Binder	CHEMBL3353058	ChEMBL	7.0	—	—	O=C(NO)c1cc2n(c1)CCN(C(=O)C1CCCCC1)C2
E3 Binder	CHEMBL3353059	ChEMBL	6.55	—	—	O=C(NO)c1cc2n(c1)CCN(C(=O)c1cc3ccccc3[nH]1)C2
E3 Binder	CHEMBL3353056	ChEMBL	7.41	—	—	O=C(NO)c1cc2n(c1)CCN(C(=O)c1cc3ccccc3s1)C2
E3 Binder	CHEMBL3353062	ChEMBL	7.5	—	—	O=C(NO)c1cc2n(c1)CCN(C(=O)c1ccc(-c3ccccc3)cc1)C2
E3 Binder	CHEMBL3353055	ChEMBL	6.96	—	—	O=C(NO)c1cc2n(c1)CCN(C(=O)c1cccs1)C2
E3 Binder	CHEMBL2403453	ChEMBL	6.25	—	—	O=C(NO)c1cc2sccc2s1
E3 Binder	CHEMBL4113837	ChEMBL	8.46	—	—	O=C(NO)c1ccc(-c2c[nH]c3cncnc23)cc1
E3 Binder	CHEMBL4110772	ChEMBL	7.85	—	—	O=C(NO)c1ccc(-c2c[nH]c3ncncc23)cc1
E3 Binder	CHEMBL3981584	ChEMBL	7.0	—	—	O=C(NO)c1ccc(-c2cc3c(NCc4ccccc4)ncnc3[nH]2)cc1
E3 Binder	CHEMBL1630118	ChEMBL	7.3	—	—	O=C(NO)c1ccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)s1
E3 Binder	CHEMBL3960054	ChEMBL	7.96	—	—	O=C(NO)c1ccc(-c2ccc[nH]2)cc1
E3 Binder	CHEMBL216509	ChEMBL	6.61	—	—	O=C(NO)c1ccc(-c2ccccn2)s1
E3 Binder	CHEMBL218080	ChEMBL	7.47	—	—	O=C(NO)c1ccc(-c2ccn(CCCc3ccccc3)n2)s1
E3 Binder	CHEMBL217004	ChEMBL	8.3	—	—	O=C(NO)c1ccc(-c2ccn(CCNCc3ccc(-c4ccccn4)cc3)n2)s1
E3 Binder	CHEMBL217098	ChEMBL	8.05	—	—	O=C(NO)c1ccc(-c2ccn(CCNCc3ccc(-n4ccnc4)cc3)n2)s1
E3 Binder	CHEMBL218511	ChEMBL	8.3	—	—	O=C(NO)c1ccc(-c2ccn(CCNCc3ccc4[nH]ccc4c3)n2)s1
E3 Binder	CHEMBL217716	ChEMBL	7.54	—	—	O=C(NO)c1ccc(-c2ccn(CCNCc3ccc4c(c3)OCO4)n2)s1
E3 Binder	CHEMBL386135	ChEMBL	7.48	—	—	O=C(NO)c1ccc(-c2ccn(CCNCc3ccccc3)n2)s1
E3 Binder	CHEMBL217468	ChEMBL	7.7	—	—	O=C(NO)c1ccc(-c2ccn(CCOCc3ccccc3)n2)s1
E3 Binder	CHEMBL218514	ChEMBL	7.66	—	—	O=C(NO)c1ccc(-c2ccn(CCOc3ccccc3)n2)s1
E3 Binder	CHEMBL216359	ChEMBL	7.0	—	—	O=C(NO)c1ccc(-c2ccn(CCc3ccccc3)n2)s1
E3 Binder	CHEMBL218236	ChEMBL	6.82	—	—	O=C(NO)c1ccc(-c2ccn(Cc3ccccc3)n2)s1
E3 Binder	CHEMBL4160840	ChEMBL	6.38	—	—	O=C(NO)c1ccc(-c2ccnc(Nc3ccc(N4CCOCC4)cc3)n2)cc1
E3 Binder	CHEMBL3907669	ChEMBL	7.45	—	—	O=C(NO)c1ccc(-c2ccncc2)cc1
E3 Binder	CHEMBL4754714	ChEMBL	6.24	—	—	O=C(NO)c1ccc(-c2csc(N3N=C(c4ccccc4)/C(=N/Nc4nccs4)C3=O)n2)cc1
E3 Binder	CHEMBL4529659	ChEMBL	6.18	—	—	O=C(NO)c1ccc(-c2nnc(-c3ccccc3)o2)cc1
E3 Binder	CHEMBL4548553	ChEMBL	7.85	—	—	O=C(NO)c1ccc(-n2cnc3ncncc32)cc1
E3 Binder	CHEMBL5177483	ChEMBL	6.89	—	—	O=C(NO)c1ccc(/C=C/C(=O)N2CCC(N3C(=O)[C@H](c4ccccc4)[C@H]3c3ccccc3)CC2)cc1
E3 Binder	CHEMBL5087823	ChEMBL	6.62	—	—	O=C(NO)c1ccc(/C=C/c2cccc(-c3cc(F)ccc3O)c2)cc1
E3 Binder	CHEMBL5092482	ChEMBL	6.7	—	—	O=C(NO)c1ccc(/C=C/c2cccc(-c3cccc(O)c3)c2)cc1
E3 Binder	CHEMBL5087779	ChEMBL	6.75	—	—	O=C(NO)c1ccc(/C=C/c2cccc(-c3ccccc3O)c2)cc1
E3 Binder	CHEMBL5094326	ChEMBL	6.89	—	—	O=C(NO)c1ccc(/C=C/c2ccnc(-c3cc(F)ccc3O)c2)cc1
E3 Binder	CHEMBL5087466	ChEMBL	7.47	—	—	O=C(NO)c1ccc(/C=C/c2ccnc(-c3cccc(CO)c3)c2)cc1
E3 Binder	CHEMBL5081674	ChEMBL	7.72	—	—	O=C(NO)c1ccc(/C=C/c2ccnc(-c3cccc(O)c3)c2)cc1
E3 Binder	CHEMBL5075646	ChEMBL	7.33	—	—	O=C(NO)c1ccc(/C=C/c2ccnc(-c3ccccc3O)c2)cc1
E3 Binder	CHEMBL5083395	ChEMBL	7.85	—	—	O=C(NO)c1ccc(/C=C/c2ccnc(-c3cccnc3)c2)cc1
E3 Binder	CHEMBL5085680	ChEMBL	7.27	—	—	O=C(NO)c1ccc(/C=C/c2ccnc(-c3ccsc3)c2)cc1
E3 Binder	CHEMBL5081459	ChEMBL	6.5	—	—	O=C(NO)c1ccc(/C=C/c2ccnc(Br)c2)cc1
E3 Binder	CHEMBL5076948	ChEMBL	6.89	—	—	O=C(NO)c1ccc(/C=C/c2ccncc2)cc1
E3 Binder	CHEMBL5087997	ChEMBL	7.89	—	—	O=C(NO)c1ccc(/C=C/c2cncc(-c3ccccc3O)c2)cc1
E3 Binder	CHEMBL5192518	ChEMBL	7.82	—	—	O=C(NO)c1ccc(/C=N/NC(=O)c2cc(N3CCOCC3)nc(-c3cccc(O)c3)n2)cc1
E3 Binder	CHEMBL5182686	ChEMBL	7.46	—	—	O=C(NO)c1ccc(/C=N/NC(=O)c2cc(N3CCOCC3)nc(-c3cccc4[nH]ncc34)n2)cc1
E3 Binder	CHEMBL5174964	ChEMBL	7.73	—	—	O=C(NO)c1ccc(/C=N/NC(=O)c2ccnc(-c3ccccc3)n2)cc1
E3 Binder	CHEMBL3800411	ChEMBL	6.82	—	—	O=C(NO)c1ccc(Br)c(NC(=O)c2ccccc2)c1
E3 Binder	CHEMBL5284034	ChEMBL	6.85	—	—	O=C(NO)c1ccc(C(=O)NCC2CCN(Cc3ccccc3)CC2)cc1
E3 Binder	CHEMBL4640986	ChEMBL	6.35	—	—	O=C(NO)c1ccc(C(=O)NCCCN2c3ccccc3CCc3ccc(Cl)cc32)cc1
E3 Binder	CHEMBL2333340	ChEMBL	8.4	—	—	O=C(NO)c1ccc(C(=O)NCCc2ccccc2)cc1
E3 Binder	CHEMBL2333339	ChEMBL	8.1	—	—	O=C(NO)c1ccc(C(=O)NCCc2ccncc2)cc1
E3 Binder	CHEMBL2333341	ChEMBL	8.15	—	—	O=C(NO)c1ccc(C(=O)NCc2ccccc2)cc1
E3 Binder	CHEMBL475051	ChEMBL	7.04	—	—	O=C(NO)c1ccc(C(=O)Nc2cccc(Nc3ncc(-c4cccnc4)s3)c2)cc1
E3 Binder	CHEMBL4088663	ChEMBL	6.58	—	—	O=C(NO)c1ccc(C(=O)Nc2cccc3cccnc23)cc1
E3 Binder	CHEMBL4060433	ChEMBL	6.28	—	—	O=C(NO)c1ccc(C(=O)Nc2cccc3ncccc23)cc1
E3 Binder	CHEMBL2333342	ChEMBL	7.43	—	—	O=C(NO)c1ccc(C(=O)Nc2ccccc2)cc1
E3 Binder	CHEMBL4215505	ChEMBL	6.42	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4c(Cl)cccc4Cl)ccc23)cc1
E3 Binder	CHEMBL4203935	ChEMBL	6.53	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4cc(Cl)cc(Cl)c4)ccc23)cc1
E3 Binder	CHEMBL4207699	ChEMBL	6.75	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4cc(Cl)ccc4Cl)ccc23)cc1
E3 Binder	CHEMBL4205375	ChEMBL	6.99	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4ccc(C(F)(F)F)cc4)ccc23)cc1
E3 Binder	CHEMBL4213207	ChEMBL	6.83	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4ccc(Cl)c(Cl)c4)ccc23)cc1
E3 Binder	CHEMBL4203741	ChEMBL	7.01	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4ccc(Cl)c(F)c4)ccc23)cc1
E3 Binder	CHEMBL4217088	ChEMBL	6.55	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4ccc(Cl)cc4)ccc23)cc1
E3 Binder	CHEMBL4212219	ChEMBL	7.16	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4cccc(Cl)c4)ccc23)cc1
E3 Binder	CHEMBL4208276	ChEMBL	6.8	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4cccc(Cl)c4Cl)ccc23)cc1
E3 Binder	CHEMBL4210396	ChEMBL	6.66	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4cccc(OC(F)(F)F)c4)ccc23)cc1
E3 Binder	CHEMBL4211477	ChEMBL	7.42	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4ccccc4)ccc23)cc1
E3 Binder	CHEMBL4217618	ChEMBL	7.23	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4ccccc4Cl)ccc23)cc1
E3 Binder	CHEMBL4214775	ChEMBL	7.19	—	—	O=C(NO)c1ccc(C(=O)Nc2n[nH]c3cc(-c4ccccc4F)ccc23)cc1
E3 Binder	CHEMBL3799728	ChEMBL	6.85	—	—	O=C(NO)c1ccc(C(F)(F)F)c(NC(=O)c2ccccc2)c1
E3 Binder	CHEMBL4515845	ChEMBL	7.78	—	—	O=C(NO)c1ccc(C2(NC(=O)c3nc(-c4nccs4)sc3C3CC3)CC2)cc1
E3 Binder	CHEMBL3921742	ChEMBL	6.27	—	—	O=C(NO)c1ccc(C2CCCC2)cc1
E3 Binder	CHEMBL5194437	ChEMBL	7.6	—	—	O=C(NO)c1ccc(CC(=O)N(CCO)C(=O)Cc2ccccc2)cc1
E3 Binder	CHEMBL4066043	ChEMBL	7.6	5OJ	—	O=C(NO)c1ccc(CC(=O)N(CCO)c2ccccc2)cc1
E3 Binder	CHEMBL5181949	ChEMBL	6.92	—	—	O=C(NO)c1ccc(CC(=O)N2CCC(N3C(=O)[C@H](c4ccccc4)[C@H]3c3ccccc3)CC2)cc1
E3 Binder	CHEMBL5189806	ChEMBL	7.04	—	—	O=C(NO)c1ccc(CC(=O)N2CCC(N3CC(c4ccccc4)(c4ccccc4)C3=O)CC2)cc1
E3 Binder	CHEMBL4782147	ChEMBL	6.64	—	—	O=C(NO)c1ccc(CC(=O)N2CCC3(CC2)CN(Cc2ccccc2)c2ccccc23)cc1
E3 Binder	CHEMBL4750725	ChEMBL	6.74	—	—	O=C(NO)c1ccc(CCCN2CC(CN[C@H]3C[C@@H]3c3ccccc3)C2)cc1
E3 Binder	CHEMBL4762346	ChEMBL	7.51	—	—	O=C(NO)c1ccc(CCCN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1
E3 Binder	CHEMBL4796905	ChEMBL	7.0	—	—	O=C(NO)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(-c4ccc(C(F)(F)F)nc4)cc3)CC2)cc1
E3 Binder	CHEMBL4789904	ChEMBL	7.72	—	—	O=C(NO)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(-c4ccc(Cl)cc4)cc3)CC2)cc1
E3 Binder	CHEMBL4790127	ChEMBL	7.23	—	—	O=C(NO)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(-c4ccc(F)cc4)cc3)CC2)cc1
E3 Binder	CHEMBL4791396	ChEMBL	6.67	—	—	O=C(NO)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(C(=O)N4CCCCC4)cc3)CC2)cc1
E3 Binder	CHEMBL4777594	ChEMBL	6.54	—	—	O=C(NO)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(C(=O)N4CCOCC4)cc3)CC2)cc1
E3 Binder	CHEMBL4785144	ChEMBL	7.29	—	—	O=C(NO)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(F)cc3)CC2)cc1
E3 Binder	CHEMBL4741826	ChEMBL	7.92	—	—	O=C(NO)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccc(OCc4ccc(F)cc4)cc3)CC2)cc1
E3 Binder	CHEMBL4749146	ChEMBL	7.32	—	—	O=C(NO)c1ccc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1
E3 Binder	CHEMBL4744667	ChEMBL	6.74	—	—	O=C(NO)c1ccc(CCCN2CCc3cc(CN[C@H]4C[C@@H]4c4ccc(F)cc4)ccc3C2)cc1
E3 Binder	CHEMBL4165684	ChEMBL	6.86	—	—	O=C(NO)c1ccc(CCN2C(=O)c3cccc4c(N5CCOCC5)ccc(c34)C2=O)cc1
E3 Binder	CHEMBL4750898	ChEMBL	6.31	—	—	O=C(NO)c1ccc(CCN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1
E3 Binder	CHEMBL4534310	ChEMBL	6.87	—	—	O=C(NO)c1ccc(CCN2c3ccccc3Sc3ccccc32)cc1
E3 Binder	CHEMBL4065354	ChEMBL	7.38	—	—	O=C(NO)c1ccc(CCc2cccc3cccnc23)cc1
E3 Binder	CHEMBL3675754	ChEMBL	6.75	—	—	O=C(NO)c1ccc(CCn2c3ccccc3c3ccccc32)cc1
E3 Binder	CHEMBL4761127	ChEMBL	7.74	—	—	O=C(NO)c1ccc(CN(C(=O)c2c(F)c(F)c(F)c(F)c2F)C2CC2)cc1
E3 Binder	CHEMBL5192119	ChEMBL	7.82	—	—	O=C(NO)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)c(Cl)c(F)c(Cl)c2F)cc1
E3 Binder	CHEMBL5189543	ChEMBL	7.16	—	—	O=C(NO)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)c(F)c(Cl)c(F)c2F)cc1
E3 Binder	CHEMBL5193507	ChEMBL	9.05	—	—	O=C(NO)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL5176422	ChEMBL	8.0	—	—	O=C(NO)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)c(F)cc(F)c2F)cc1
E3 Binder	CHEMBL5181605	ChEMBL	8.05	—	—	O=C(NO)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)cc(F)c(Cl)c2F)cc1
E3 Binder	CHEMBL5176705	ChEMBL	8.1	—	—	O=C(NO)c1ccc(CN(C2CC2)S(=O)(=O)c2c(F)cc(F)cc2F)cc1
E3 Binder	CHEMBL5201529	ChEMBL	7.85	—	—	O=C(NO)c1ccc(CN(C2CC2)S(=O)(=O)c2cc(F)c(F)c(F)c2)cc1
E3 Binder	CHEMBL5192865	ChEMBL	8.19	—	—	O=C(NO)c1ccc(CN(C2CC2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL5193014	ChEMBL	7.96	—	—	O=C(NO)c1ccc(CN(C2CC2)S(=O)(=O)c2ccc(F)cc2)cc1
E3 Binder	CHEMBL5199669	ChEMBL	7.3	—	—	O=C(NO)c1ccc(CN(C2CCCC2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL4177129	ChEMBL	9.3	—	—	O=C(NO)c1ccc(CN(CCCCO)C(=O)Nc2ccccc2)cc1
E3 Binder	CHEMBL4783802	ChEMBL	7.51	—	—	O=C(NO)c1ccc(CN(CCCO)C(=O)Cc2ccccc2)cc1
E3 Binder	CHEMBL4079541	ChEMBL	7.6	AGJ	—	O=C(NO)c1ccc(CN(CCO)C(=O)Cc2ccccc2)cc1
E3 Binder	CHEMBL2179619	ChEMBL	7.85	—	—	O=C(NO)c1ccc(CN(CCc2ccccc2)C(=O)Nc2ccccc2)cc1
E3 Binder	CHEMBL5085571	ChEMBL	7.35	—	—	O=C(NO)c1ccc(CN(Cc2ccc(C(F)(F)F)cc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL5080599	ChEMBL	7.89	—	—	O=C(NO)c1ccc(CN(Cc2ccc(F)cc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL5087501	ChEMBL	7.68	—	—	O=C(NO)c1ccc(CN(Cc2ccc(F)cc2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL5070393	ChEMBL	7.85	—	—	O=C(NO)c1ccc(CN(Cc2cccc(F)c2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL5080426	ChEMBL	8.05	—	—	O=C(NO)c1ccc(CN(Cc2ccccc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL5092466	ChEMBL	8.3	—	—	O=C(NO)c1ccc(CN(Cc2ccccc2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL5094501	ChEMBL	8.0	—	—	O=C(NO)c1ccc(CN(Cc2ccccc2F)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL5093071	ChEMBL	8.22	—	—	O=C(NO)c1ccc(CN(Cc2ccccn2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL5075135	ChEMBL	9.15	TO3	—	O=C(NO)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL5086440	ChEMBL	7.85	—	—	O=C(NO)c1ccc(CN(Cc2ccncc2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL5089527	ChEMBL	7.96	—	—	O=C(NO)c1ccc(CN(Cc2ccncc2)S(=O)(=O)c2cc(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL4748093	ChEMBL	7.16	—	—	O=C(NO)c1ccc(CN(Cc2nnnn2C2CCCCC2)C(=O)c2ccccc2)cc1
E3 Binder	CHEMBL4786332	ChEMBL	7.52	—	—	O=C(NO)c1ccc(CN(Cc2nnnn2Cc2ccccc2)C(=O)c2ccccc2)cc1
E3 Binder	CHEMBL4800426	ChEMBL	7.52	P5Y	—	O=C(NO)c1ccc(CN(Cc2nnnn2Cc2ccccc2)C(=O)c2ccccc2C(F)(F)F)cc1
E3 Binder	CHEMBL4764495	ChEMBL	7.62	—	—	O=C(NO)c1ccc(CN2C(=O)/C(=C3\Nc4ccccc4\C3=N/O)c3cc(Br)ccc32)cc1
E3 Binder	CHEMBL4777783	ChEMBL	7.8	—	—	O=C(NO)c1ccc(CN2C(=O)/C(=C3\Nc4ccccc4\C3=N/O)c3cc(Cl)ccc32)cc1
E3 Binder	CHEMBL4743446	ChEMBL	7.37	—	—	O=C(NO)c1ccc(CN2C(=O)/C(=C3\Nc4ccccc4\C3=N/O)c3cc(F)ccc32)cc1
E3 Binder	CHEMBL4762257	ChEMBL	7.31	—	—	O=C(NO)c1ccc(CN2C(=O)/C(=C3\Nc4ccccc4\C3=N/O)c3cccc(Cl)c32)cc1
E3 Binder	CHEMBL4797488	ChEMBL	8.15	—	—	O=C(NO)c1ccc(CN2C(=O)/C(=C3\Nc4ccccc4\C3=N/O)c3ccccc32)cc1
E3 Binder	CHEMBL4871920	ChEMBL	7.7	—	—	O=C(NO)c1ccc(CN2C(=O)C(Cc3ccccc3)N(CCc3ccccc3)C2=O)cc1
E3 Binder	CHEMBL4851023	ChEMBL	8.22	—	—	O=C(NO)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3ccc(Cl)cc3)C2=O)cc1
E3 Binder	CHEMBL4854096	ChEMBL	7.6	—	—	O=C(NO)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3ccc4ccccc4c3)C2=O)cc1
E3 Binder	CHEMBL4846062	ChEMBL	7.54	—	—	O=C(NO)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3cccc4ccccc34)C2=O)cc1
E3 Binder	CHEMBL4854541	ChEMBL	7.67	—	—	O=C(NO)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3ccccc3)C2=O)cc1
E3 Binder	CHEMBL4858289	ChEMBL	8.32	—	—	O=C(NO)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3ccccn3)C2=O)cc1
E3 Binder	CHEMBL4866683	ChEMBL	8.68	—	—	O=C(NO)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3cccnc3)C2=O)cc1
E3 Binder	CHEMBL4878288	ChEMBL	7.86	—	—	O=C(NO)c1ccc(CN2C(=O)C(Cc3ccccc3)N(Cc3ccncc3)C2=O)cc1
E3 Binder	CHEMBL4846714	ChEMBL	9.1	—	—	O=C(NO)c1ccc(CN2C(=O)CCCc3cc(Cl)ccc32)cc1
E3 Binder	CHEMBL4857825	ChEMBL	9.05	—	—	O=C(NO)c1ccc(CN2C(=O)CCc3cc(Br)ccc32)cc1
E3 Binder	CHEMBL4847122	ChEMBL	8.57	—	—	O=C(NO)c1ccc(CN2C(=O)CCc3cc(C4CC4)ccc32)cc1
E3 Binder	CHEMBL4859648	ChEMBL	8.54	—	—	O=C(NO)c1ccc(CN2C(=O)CCc3cc(Cl)ccc32)cc1
E3 Binder	CHEMBL4858911	ChEMBL	7.66	—	—	O=C(NO)c1ccc(CN2C(=O)CN(CCc3ccccc3)C2=O)cc1
E3 Binder	CHEMBL4854752	ChEMBL	8.08	—	—	O=C(NO)c1ccc(CN2C(=O)CN(Cc3ccc(Cl)cc3)C2=O)cc1
E3 Binder	CHEMBL4863833	ChEMBL	7.9	—	—	O=C(NO)c1ccc(CN2C(=O)CN(Cc3ccccc3)C2=O)cc1
E3 Binder	CHEMBL481719	ChEMBL	6.96	—	—	O=C(NO)c1ccc(CN2C(=O)CNC(=O)[C@H]2Cc2c[nH]c3ccccc23)cc1
E3 Binder	CHEMBL481718	ChEMBL	6.77	—	—	O=C(NO)c1ccc(CN2C(=O)CNC(=O)[C@H]2Cc2ccccc2)cc1
E3 Binder	CHEMBL481726	ChEMBL	6.8	—	—	O=C(NO)c1ccc(CN2C(=O)CNC(=O)[C@H]2Cc2cccs2)cc1
E3 Binder	CHEMBL5172211	ChEMBL	7.68	—	—	O=C(NO)c1ccc(CN2C(=O)CSC2=O)cc1
E3 Binder	CHEMBL4845845	ChEMBL	7.61	—	—	O=C(NO)c1ccc(CN2C(=O)NC(CCc3ccccc3)(c3ccccc3)C2=O)cc1
E3 Binder	CHEMBL4849507	ChEMBL	7.27	—	—	O=C(NO)c1ccc(CN2C(=O)NC(Cc3ccc(Cl)cc3)(c3ccccc3)C2=O)cc1
E3 Binder	CHEMBL4871002	ChEMBL	7.13	—	—	O=C(NO)c1ccc(CN2C(=O)NC(Cc3ccc4ccccc4c3)(c3ccccc3)C2=O)cc1
E3 Binder	CHEMBL4865529	ChEMBL	7.04	—	—	O=C(NO)c1ccc(CN2C(=O)NC(Cc3cccc4ccccc34)(c3ccccc3)C2=O)cc1
E3 Binder	CHEMBL4860720	ChEMBL	7.14	—	—	O=C(NO)c1ccc(CN2C(=O)NC(Cc3ccccc3)(c3ccccc3)C2=O)cc1
E3 Binder	CHEMBL3971359	ChEMBL	7.59	—	—	O=C(NO)c1ccc(CN2C(=O)N[C@@H](Cc3ccccc3)C2=O)cc1
E3 Binder	CHEMBL4176291	ChEMBL	8.57	—	—	O=C(NO)c1ccc(CN2C(=O)c3cccc4c(N5CCOCC5)ccc(c34)C2=O)cc1
E3 Binder	CHEMBL5285323	ChEMBL	7.93	—	—	O=C(NO)c1ccc(CN2CC(=O)N(Cc3ccc(Cl)cc3)[C@H](Cc3ccccc3)C2=O)cc1
E3 Binder	CHEMBL5266137	ChEMBL	7.98	—	—	O=C(NO)c1ccc(CN2CC(=O)N(Cc3cccc(Cl)c3)[C@H](Cc3ccccc3)C2=O)cc1
E3 Binder	CHEMBL5289315	ChEMBL	8.01	—	—	O=C(NO)c1ccc(CN2CC(=O)N(Cc3ccccc3)[C@H](Cc3ccccc3)C2=O)cc1
E3 Binder	CHEMBL5286689	ChEMBL	8.0	—	—	O=C(NO)c1ccc(CN2CC(=O)N(Cc3ccccc3Cl)[C@H](Cc3ccccc3)C2=O)cc1
E3 Binder	CHEMBL5284275	ChEMBL	7.79	—	—	O=C(NO)c1ccc(CN2CC(=O)N(c3ccccc3)C(CCc3ccccc3)C2=O)cc1
E3 Binder	CHEMBL4283913	ChEMBL	7.39	—	—	O=C(NO)c1ccc(CN2CC3(CCCCC3)c3ccccc32)cc1
E3 Binder	CHEMBL4862465	ChEMBL	9.0	—	—	O=C(NO)c1ccc(CN2CC3(CCOC3)C2)c(F)c1
E3 Binder	CHEMBL4795265	ChEMBL	6.63	—	—	O=C(NO)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1
E3 Binder	CHEMBL4782002	ChEMBL	6.33	—	—	O=C(NO)c1ccc(CN2CCC3(CC2)CN(C(=O)c2ccccc2)c2c(-c4ccccc4)cccc23)cc1
E3 Binder	CHEMBL4785718	ChEMBL	6.81	—	—	O=C(NO)c1ccc(CN2CCC3(CC2)CN(C(=O)c2ccccc2)c2ccccc23)cc1
E3 Binder	CHEMBL4787293	ChEMBL	6.25	—	—	O=C(NO)c1ccc(CN2CCC3(CC2)CN(Cc2ccccc2)c2ccccc23)cc1
E3 Binder	CHEMBL3918458	ChEMBL	6.27	—	—	O=C(NO)c1ccc(CN2CCCC2)cc1
E3 Binder	CHEMBL4866436	ChEMBL	7.77	—	—	O=C(NO)c1ccc(CN2CCCCc3cc(-c4cc[nH]n4)ccc32)cc1
E3 Binder	CHEMBL4856207	ChEMBL	8.05	—	—	O=C(NO)c1ccc(CN2CCCCc3cc(Br)ccc32)cc1
E3 Binder	CHEMBL4856735	ChEMBL	9.0	—	—	O=C(NO)c1ccc(CN2CCCCc3cc(Cl)ccc32)cc1
E3 Binder	CHEMBL4878252	ChEMBL	6.89	—	—	O=C(NO)c1ccc(CN2CCCCc3ccc(-c4ccccc4)cc32)cc1
E3 Binder	CHEMBL4857891	ChEMBL	7.37	—	—	O=C(NO)c1ccc(CN2CCCCc3ccc(Br)cc32)cc1
E3 Binder	CHEMBL4862419	ChEMBL	7.35	—	—	O=C(NO)c1ccc(CN2CCCCc3ccc(C4CC4)cc32)cc1
E3 Binder	CHEMBL4875969	ChEMBL	7.85	—	—	O=C(NO)c1ccc(CN2CCCCc3ccc(Cl)cc32)cc1
E3 Binder	CHEMBL4862139	ChEMBL	7.72	—	—	O=C(NO)c1ccc(CN2CCCCc3ccc(F)cc32)cc1
E3 Binder	CHEMBL4847454	ChEMBL	8.3	—	—	O=C(NO)c1ccc(CN2CCCCc3ccccc32)cc1
E3 Binder	CHEMBL4873296	ChEMBL	8.21	—	—	O=C(NO)c1ccc(CN2CCCOc3ccccc32)cc1
E3 Binder	CHEMBL4858994	ChEMBL	8.74	—	—	O=C(NO)c1ccc(CN2CCCSc3ccccc32)cc1
E3 Binder	CHEMBL4876815	ChEMBL	7.89	—	—	O=C(NO)c1ccc(CN2CCC[S+]([O-])c3ccccc32)cc1
E3 Binder	CHEMBL4863515	ChEMBL	9.52	—	—	O=C(NO)c1ccc(CN2CCCc3cc(-c4cc[nH]n4)ccc32)cc1
E3 Binder	CHEMBL4536605	ChEMBL	9.3	—	—	O=C(NO)c1ccc(CN2CCCc3cc(Cl)ccc32)cc1
E3 Binder	CHEMBL4860333	ChEMBL	8.64	—	—	O=C(NO)c1ccc(CN2CCCc3ccccc32)cc1
E3 Binder	CHEMBL4853358	ChEMBL	7.0	—	—	O=C(NO)c1ccc(CN2CCCc3ccccc3C2)cc1
E3 Binder	CHEMBL5281081	ChEMBL	7.85	—	—	O=C(NO)c1ccc(CN2CCN(C(=O)c3c[nH]c4cc(F)ccc34)CC2)cc1
E3 Binder	CHEMBL5272622	ChEMBL	7.63	—	—	O=C(NO)c1ccc(CN2CCN(C(=O)c3c[nH]c4cc(OCc5ccccc5)ccc34)CC2)cc1
E3 Binder	CHEMBL5286805	ChEMBL	7.58	—	—	O=C(NO)c1ccc(CN2CCN(C(=O)c3c[nH]c4ccc(Cl)cc34)CC2)cc1
E3 Binder	CHEMBL5278328	ChEMBL	7.11	—	—	O=C(NO)c1ccc(CN2CCN(C(=O)c3c[nH]c4cccc(Cc5ccccc5)c34)CC2)cc1
E3 Binder	CHEMBL5276052	ChEMBL	7.84	—	—	O=C(NO)c1ccc(CN2CCN(C(=O)c3c[nH]c4ccccc34)CC2)cc1
E3 Binder	CHEMBL4097093	ChEMBL	7.78	—	—	O=C(NO)c1ccc(CN2CCN(C(=O)c3cc(Cc4n[nH]c(=O)c5ccccc45)ccc3F)CC2)cc1
E3 Binder	CHEMBL5285262	ChEMBL	7.05	—	—	O=C(NO)c1ccc(CN2CCN(C(=O)c3cc4ccccc4[nH]3)CC2)cc1
E3 Binder	CHEMBL4848981	ChEMBL	6.59	—	—	O=C(NO)c1ccc(CN2CCc3ccccc3CC2)cc1
E3 Binder	CHEMBL4447453	ChEMBL	6.94	—	—	O=C(NO)c1ccc(CN2N=C(Cl)C=C3Sc4ccccc4N=C32)cc1
E3 Binder	CHEMBL4436946	ChEMBL	7.72	—	—	O=C(NO)c1ccc(CN2N=CC=C3Sc4ccccc4N=C32)cc1
E3 Binder	CHEMBL4450128	ChEMBL	7.96	—	—	O=C(NO)c1ccc(CN2c3cc(C(F)(F)F)ccc3CCC[C@@H]3CCCC[C@H]32)cc1
E3 Binder	CHEMBL4445312	ChEMBL	8.09	—	—	O=C(NO)c1ccc(CN2c3ccccc3C3C2CCS3(=O)=O)cc1
E3 Binder	CHEMBL4557665	ChEMBL	8.1	—	—	O=C(NO)c1ccc(CN2c3ccccc3CCC[C@@H]3CCCC[C@H]32)cc1
E3 Binder	CHEMBL4469098	ChEMBL	8.22	—	—	O=C(NO)c1ccc(CN2c3ccccc3CC[C@@H]3CCCC[C@H]32)cc1
E3 Binder	CHEMBL4579366	ChEMBL	7.48	—	—	O=C(NO)c1ccc(CN2c3ccccc3C[C@@H]3CCCCC[C@H]32)cc1
E3 Binder	CHEMBL4471619	ChEMBL	7.44	—	—	O=C(NO)c1ccc(CN2c3ccccc3C[C@@H]3CCCC[C@H]32)cc1
E3 Binder	CHEMBL516600	ChEMBL	6.66	—	—	O=C(NO)c1ccc(CN2c3ccccc3NC(=O)[C@@H]2Cc2ccccc2)cc1
E3 Binder	CHEMBL519943	ChEMBL	6.51	—	—	O=C(NO)c1ccc(CN2c3ccccc3NC(=O)[C@@H]2Cc2cccs2)cc1
E3 Binder	CHEMBL482358	ChEMBL	8.0	—	—	O=C(NO)c1ccc(CN2c3ccccc3NC(=O)[C@H]2CCc2ccccc2)cc1
E3 Binder	CHEMBL481018	ChEMBL	7.4	—	—	O=C(NO)c1ccc(CN2c3ccccc3NC(=O)[C@H]2Cc2ccc(F)c(F)c2)cc1
E3 Binder	CHEMBL481538	ChEMBL	8.0	—	—	O=C(NO)c1ccc(CN2c3ccccc3NC(=O)[C@H]2Cc2ccc(O)cc2)cc1
E3 Binder	CHEMBL479842	ChEMBL	8.0	—	—	O=C(NO)c1ccc(CN2c3ccccc3NC(=O)[C@H]2Cc2ccccc2)cc1
E3 Binder	CHEMBL518957	ChEMBL	7.4	—	—	O=C(NO)c1ccc(CN2c3ccccc3NC(=O)[C@H]2Cc2cccs2)cc1
E3 Binder	CHEMBL4744479	ChEMBL	8.1	—	—	O=C(NO)c1ccc(CN2c3ccccc3S(=O)(=O)C[C@@H]3CCCC[C@@H]32)cc1
E3 Binder	CHEMBL4104247	ChEMBL	8.1	—	—	O=C(NO)c1ccc(CN2c3ccccc3S(=O)(=O)C[C@H]3CCCC[C@H]32)cc1
E3 Binder	CHEMBL4444811	ChEMBL	7.89	—	—	O=C(NO)c1ccc(CN2c3ccccc3S(=O)(=O)c3ccccc32)cc1
E3 Binder	CHEMBL4581606	ChEMBL	7.75	—	—	O=C(NO)c1ccc(CN2c3ccccc3Sc3cc(Cl)nnc32)cc1
E3 Binder	CHEMBL4874716	ChEMBL	7.52	—	—	O=C(NO)c1ccc(CN2c3ccccc3Sc3ccc(C(=O)Nc4ccc(Br)cn4)cc32)cc1
E3 Binder	CHEMBL4852441	ChEMBL	7.4	—	—	O=C(NO)c1ccc(CN2c3ccccc3Sc3ccc(C(=O)Nc4ccccn4)cc32)cc1
E3 Binder	CHEMBL4472834	ChEMBL	7.85	—	—	O=C(NO)c1ccc(CN2c3ccccc3Sc3ccc(C(F)(F)F)cc32)cc1
E3 Binder	CHEMBL4530950	ChEMBL	8.02	—	—	O=C(NO)c1ccc(CN2c3ccccc3Sc3ccc(Cl)cc32)cc1
E3 Binder	CHEMBL4450965	ChEMBL	7.8	—	—	O=C(NO)c1ccc(CN2c3ccccc3Sc3cccc(Cl)c32)cc1
E3 Binder	CHEMBL4438566	ChEMBL	8.12	—	—	O=C(NO)c1ccc(CN2c3ccccc3Sc3ccccc32)cc1
E3 Binder	CHEMBL4858133	ChEMBL	7.96	—	—	O=C(NO)c1ccc(CN2c3ccccc3Sc3ccccc32)nc1
E3 Binder	CHEMBL4457162	ChEMBL	8.3	—	—	O=C(NO)c1ccc(CN2c3ccccc3Sc3cccnc32)cc1
E3 Binder	CHEMBL4468273	ChEMBL	8.15	—	—	O=C(NO)c1ccc(CN2c3ccccc3Sc3ccncc32)cc1
E3 Binder	CHEMBL4443794	ChEMBL	7.96	—	—	O=C(NO)c1ccc(CN2c3ccccc3Sc3ccnnc32)cc1
E3 Binder	CHEMBL4442266	ChEMBL	7.77	—	—	O=C(NO)c1ccc(CN2c3ccccc3Sc3nccnc32)cc1
E3 Binder	CHEMBL4877023	ChEMBL	7.71	—	—	O=C(NO)c1ccc(CN2c3ccccc3[S+]([O-])c3ccc(C(F)(F)F)cc32)cc1
E3 Binder	CHEMBL4874671	ChEMBL	8.01	—	—	O=C(NO)c1ccc(CN2c3ccccc3[S+]([O-])c3ccc(Cl)cc32)cc1
E3 Binder	CHEMBL4473451	ChEMBL	7.69	—	—	O=C(NO)c1ccc(CN2c3ccccc3[S+]([O-])c3ccccc32)cc1
E3 Binder	CHEMBL4546254	ChEMBL	7.85	—	—	O=C(NO)c1ccc(CN2c3cccnc3Sc3cccnc32)cc1
E3 Binder	CHEMBL4556275	ChEMBL	8.05	—	—	O=C(NO)c1ccc(CN2c3ccncc3Sc3ccncc32)cc1
E3 Binder	CHEMBL4439108	ChEMBL	7.92	—	—	O=C(NO)c1ccc(CN2c3ccncc3Sc3ncccc32)cc1
E3 Binder	CHEMBL2431864	ChEMBL	7.12	—	—	O=C(NO)c1ccc(CNC(=O)C2CCCCC2)cc1
E3 Binder	CHEMBL5206603	ChEMBL	6.57	—	—	O=C(NO)c1ccc(CNC(=O)N2CCC(N3C(=O)CC3c3cccc(Cl)c3)CC2)cc1
E3 Binder	CHEMBL5184498	ChEMBL	7.68	—	—	O=C(NO)c1ccc(CNC(=O)N2CCC(N3C(=O)[C@H](c4ccccc4)[C@H]3c3ccccc3)CC2)cc1
E3 Binder	CHEMBL5188540	ChEMBL	8.47	—	—	O=C(NO)c1ccc(CNC(=O)N2CCC(N3CC(c4ccccc4)(c4ccccc4)C3=O)CC2)cc1
E3 Binder	CHEMBL4790624	ChEMBL	6.96	—	—	O=C(NO)c1ccc(CNC(=O)N2CCC3(CC2)CN(Cc2ccccc2)c2ccccc23)cc1
E3 Binder	CHEMBL3670661	ChEMBL	7.28	—	—	O=C(NO)c1ccc(CNC(=O)c2[nH]c(-c3ccc(O)cc3)cc2-c2ccoc2)cc1
E3 Binder	CHEMBL3670665	ChEMBL	7.97	—	—	O=C(NO)c1ccc(CNC(=O)c2[nH]c(-c3ccc(O)cc3)cc2-c2ccsc2)cc1
E3 Binder	CHEMBL4784006	ChEMBL	8.23	—	—	O=C(NO)c1ccc(CNC(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL4225914	ChEMBL	9.0	—	—	O=C(NO)c1ccc(CNC(=O)c2cc(-c3ccc(F)cc3)[nH]n2)cc1
E3 Binder	CHEMBL4531853	ChEMBL	9.21	—	—	O=C(NO)c1ccc(CNC(=O)c2cc(Cn3c4ccccc4c4ccccc43)on2)cc1
E3 Binder	CHEMBL26844	ChEMBL	6.62	—	—	O=C(NO)c1ccc(CNC(=O)c2ccc(-c3ccccc3)cc2)cc1
E3 Binder	CHEMBL4794290	ChEMBL	7.2	—	—	O=C(NO)c1ccc(CNC(=O)c2ccc(-c3csc(N4N=C(c5ccccc5)/C(=N/Nc5nccs5)C4=O)n3)cc2)cc1
E3 Binder	CHEMBL4447715	ChEMBL	8.7	—	—	O=C(NO)c1ccc(CNC(=O)c2ccc(Cl)c(Cl)c2)cc1
E3 Binder	CHEMBL5288929	ChEMBL	7.27	—	—	O=C(NO)c1ccc(CNC(=O)c2ccc3cccc(OCc4ccc(Br)cc4)c3n2)cc1
E3 Binder	CHEMBL5280863	ChEMBL	7.48	—	—	O=C(NO)c1ccc(CNC(=O)c2ccc3cccc(OCc4ccc(F)cc4)c3n2)cc1
E3 Binder	CHEMBL5268755	ChEMBL	7.21	—	—	O=C(NO)c1ccc(CNC(=O)c2ccc3cccc(OCc4ccccc4)c3n2)cc1
E3 Binder	CHEMBL27556	ChEMBL	7.36	—	—	O=C(NO)c1ccc(CNC(=O)c2ccc3ccccc3c2)cc1
E3 Binder	CHEMBL28280	ChEMBL	6.08	—	—	O=C(NO)c1ccc(CNC(=O)c2cccc3ccccc23)cc1
E3 Binder	CHEMBL4475378	ChEMBL	7.77	P6Y	—	O=C(NO)c1ccc(CNC(=O)c2cccnc2C(F)(F)F)cc1
E3 Binder	CHEMBL3919448	ChEMBL	7.12	—	—	O=C(NO)c1ccc(CNC(=O)c2nc(-c3nc4c(s3)CCCC4)sc2C2CC2)cc1
E3 Binder	CHEMBL3977346	ChEMBL	7.7	—	—	O=C(NO)c1ccc(CNC(=O)c2nc(-c3nccs3)sc2C2CC2)cc1
E3 Binder	CHEMBL4760090	ChEMBL	6.92	—	—	O=C(NO)c1ccc(CNC(c2ccccc2)c2nnnn2C2CCCCC2)cc1
E3 Binder	CHEMBL4780849	ChEMBL	7.0	—	—	O=C(NO)c1ccc(CNC(c2ccccc2)c2nnnn2Cc2ccccc2)cc1
E3 Binder	CHEMBL5181507	ChEMBL	6.68	—	—	O=C(NO)c1ccc(CNCc2ccccc2)cc1
E3 Binder	CHEMBL5208700	ChEMBL	6.8	—	—	O=C(NO)c1ccc(CNCc2cccs2)cc1
E3 Binder	CHEMBL5208990	ChEMBL	6.75	LSL	—	O=C(NO)c1ccc(CNCc2ccsc2)cc1
E3 Binder	CHEMBL4462652	ChEMBL	7.85	—	—	O=C(NO)c1ccc(CNCc2csc3ccccc23)cc1
E3 Binder	CHEMBL4754868	ChEMBL	6.92	—	—	O=C(NO)c1ccc(CNCc2nnnn2C2CCCCC2)cc1
E3 Binder	CHEMBL4752076	ChEMBL	7.0	—	—	O=C(NO)c1ccc(CNCc2nnnn2Cc2ccccc2)cc1
E3 Binder	CHEMBL5082396	ChEMBL	6.41	—	—	O=C(NO)c1ccc(CNS(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL4073165	ChEMBL	8.37	—	—	O=C(NO)c1ccc(CNc2ccc3ccccc3n2)cc1
E3 Binder	CHEMBL4079874	ChEMBL	8.49	—	—	O=C(NO)c1ccc(CNc2ccc3cccnc3c2)cc1
E3 Binder	CHEMBL4068310	ChEMBL	8.32	—	—	O=C(NO)c1ccc(CNc2ccc3ncccc3c2)cc1
E3 Binder	CHEMBL4082487	ChEMBL	7.71	—	—	O=C(NO)c1ccc(CNc2cccc3c2CCC3)cc1
E3 Binder	CHEMBL4060607	ChEMBL	7.6	—	—	O=C(NO)c1ccc(CNc2cccc3c2CCCC3)cc1
E3 Binder	CHEMBL4104117	ChEMBL	9.54	—	—	O=C(NO)c1ccc(CNc2cccc3cccnc23)cc1
E3 Binder	CHEMBL4085971	ChEMBL	8.47	—	—	O=C(NO)c1ccc(CNc2cccc3ccncc23)cc1
E3 Binder	CHEMBL4101436	ChEMBL	8.45	—	—	O=C(NO)c1ccc(CNc2cccc3cn[nH]c23)cc1
E3 Binder	CHEMBL4091237	ChEMBL	8.63	—	—	O=C(NO)c1ccc(CNc2cccc3cnccc23)cc1
E3 Binder	CHEMBL4095667	ChEMBL	9.1	—	—	O=C(NO)c1ccc(CNc2cccc3ncccc23)cc1
E3 Binder	CHEMBL4083449	ChEMBL	8.23	—	—	O=C(NO)c1ccc(CNc2cccc3nccnc23)cc1
E3 Binder	CHEMBL4083577	ChEMBL	7.67	—	—	O=C(NO)c1ccc(CNc2ccnc3ccccc23)cc1
E3 Binder	CHEMBL4061807	ChEMBL	6.39	—	—	O=C(NO)c1ccc(CNc2cnc3ccccc3c2)cc1
E3 Binder	CHEMBL4063376	ChEMBL	8.64	—	—	O=C(NO)c1ccc(CNc2cncc3ccccc23)cc1
E3 Binder	CHEMBL2407730	ChEMBL	7.38	—	—	O=C(NO)c1ccc(CNc2nccc(-c3cccnc3)n2)cc1
E3 Binder	CHEMBL5176595	ChEMBL	7.73	—	—	O=C(NO)c1ccc(COC(=O)N2CCC(N3CC(c4ccccc4)(c4ccccc4)C3=O)CC2)cc1
E3 Binder	CHEMBL4794313	ChEMBL	7.31	—	—	O=C(NO)c1ccc(COC(=O)N2CCC3(CC2)CN(Cc2ccccc2)c2ccccc23)cc1
E3 Binder	CHEMBL4796822	ChEMBL	6.83	—	—	O=C(NO)c1ccc(COc2c(-c3ccccc3)c3ccccc3[nH]c2=O)cc1
E3 Binder	CHEMBL4785403	ChEMBL	6.06	—	—	O=C(NO)c1ccc(COc2c(-c3ccccc3)c3ccccc3n(C3CCN(Cc4ccccc4)CC3)c2=O)cc1
E3 Binder	CHEMBL4790834	ChEMBL	6.75	—	—	O=C(NO)c1ccc(COc2c(-c3ccccc3)c3ccccc3n(Cc3ccccc3)c2=O)cc1
E3 Binder	CHEMBL4743692	ChEMBL	7.08	—	—	O=C(NO)c1ccc(COc2c(-c3ccccc3)c3ccccc3n(Cc3ccncc3)c2=O)cc1
E3 Binder	CHEMBL4750401	ChEMBL	7.59	—	—	O=C(NO)c1ccc(COc2c(-c3cccnc3)c3ccccc3n(Cc3ccccc3)c2=O)cc1
E3 Binder	CHEMBL4793901	ChEMBL	7.34	—	—	O=C(NO)c1ccc(COc2c(-c3cccnc3)c3ccccc3n(Cc3ccncc3)c2=O)cc1
E3 Binder	CHEMBL4779693	ChEMBL	7.07	—	—	O=C(NO)c1ccc(COc2ccc(-c3csc(N4N=C(c5ccccc5)/C(=N/Nc5nccs5)C4=O)n3)cc2)cc1
E3 Binder	CHEMBL4098833	ChEMBL	8.55	—	—	O=C(NO)c1ccc(COc2cccc3cccnc23)cc1
E3 Binder	CHEMBL4080790	ChEMBL	8.02	—	—	O=C(NO)c1ccc(CSc2cccc3cccnc23)cc1
E3 Binder	CHEMBL3898702	ChEMBL	7.45	—	—	O=C(NO)c1ccc(Cc2ccncc2)cc1
E3 Binder	CHEMBL4581909	ChEMBL	6.43	—	—	O=C(NO)c1ccc(Cc2nc(-c3ccc(Cl)cc3)nn2Cc2ccccc2)cc1
E3 Binder	CHEMBL4574536	ChEMBL	8.3	—	—	O=C(NO)c1ccc(Cc2nnc(-c3ccccc3)[nH]2)cc1
E3 Binder	CHEMBL4440425	ChEMBL	8.4	—	—	O=C(NO)c1ccc(Cc2nnc(-c3ccccc3)o2)cc1
E3 Binder	CHEMBL4460868	ChEMBL	7.8	—	—	O=C(NO)c1ccc(Cc2nnc(-c3ccccc3)s2)cc1
E3 Binder	CHEMBL4439302	ChEMBL	6.7	—	—	O=C(NO)c1ccc(Cc2nnc[nH]2)cc1
E3 Binder	CHEMBL4524728	ChEMBL	8.22	—	—	O=C(NO)c1ccc(Cc2noc(-c3ccccc3)n2)cc1
E3 Binder	CHEMBL3800615	ChEMBL	7.05	—	—	O=C(NO)c1ccc(Cl)c(NC(=O)c2ccc(Cl)cc2)c1
E3 Binder	CHEMBL3797232	ChEMBL	6.1	GT2	—	O=C(NO)c1ccc(Cl)c(NC(=O)c2ccc(Cl)cc2Cl)c1
E3 Binder	CHEMBL3799183	ChEMBL	6.82	—	—	O=C(NO)c1ccc(Cl)c(NC(=O)c2ccc(Oc3ccccc3)cc2)c1
E3 Binder	CHEMBL3798027	ChEMBL	6.52	—	—	O=C(NO)c1ccc(Cl)c(NC(=O)c2cccc(Oc3ccccc3)c2)c1
E3 Binder	CHEMBL4160522	ChEMBL	7.28	GQW	—	O=C(NO)c1ccc(Cl)c(NC(=O)c2cccc3ccsc23)c1
E3 Binder	CHEMBL3797843	ChEMBL	6.92	T61	—	O=C(NO)c1ccc(Cl)c(NC(=O)c2ccccc2)c1
E3 Binder	CHEMBL4288702	ChEMBL	6.23	—	—	O=C(NO)c1ccc(Cn2[se]c3ccc(C(F)(F)F)cc3c2=O)cc1
E3 Binder	CHEMBL4282039	ChEMBL	6.75	—	—	O=C(NO)c1ccc(Cn2[se]c3ccc(F)cc3c2=O)cc1
E3 Binder	CHEMBL4280808	ChEMBL	6.73	—	—	O=C(NO)c1ccc(Cn2[se]c3ccc(O)cc3c2=O)cc1
E3 Binder	CHEMBL4277089	ChEMBL	7.43	—	—	O=C(NO)c1ccc(Cn2[se]c3ccccc3c2=O)cc1
E3 Binder	CHEMBL4759780	ChEMBL	7.91	—	—	O=C(NO)c1ccc(Cn2c(=O)c(F)cn(C3CCCO3)c2=O)cc1
E3 Binder	CHEMBL4746040	ChEMBL	6.51	—	—	O=C(NO)c1ccc(Cn2c(=O)c(O)c(-c3ccccc3)c3ccccc32)cc1
E3 Binder	CHEMBL4741473	ChEMBL	6.53	—	—	O=C(NO)c1ccc(Cn2c(=O)c(O)c(-c3cccnc3)c3ccccc32)cc1
E3 Binder	CHEMBL4782170	ChEMBL	7.07	—	—	O=C(NO)c1ccc(Cn2c(=O)c(OCc3ccccc3)c(-c3ccccc3)c3ccccc32)cc1
E3 Binder	CHEMBL4453971	ChEMBL	7.64	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccc(F)cc3)c(=O)c3ccccc32)cc1
E3 Binder	CHEMBL4462263	ChEMBL	8.3	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccc(O)cc3)c(=O)c3ccccc32)cc1
E3 Binder	CHEMBL4564622	ChEMBL	7.62	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3cccc(C(F)(F)F)c3)c(=O)c3ccccc32)cc1
E3 Binder	CHEMBL4442777	ChEMBL	8.0	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3cccc(F)c3)c(=O)c3ccccc32)cc1
E3 Binder	CHEMBL4464975	ChEMBL	7.46	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3cc(Cl)ccc32)cc1
E3 Binder	CHEMBL4470654	ChEMBL	7.24	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3cc(F)ccc32)cc1
E3 Binder	CHEMBL4513424	ChEMBL	6.2	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3ccc(C(F)(F)F)cc32)cc1
E3 Binder	CHEMBL4474286	ChEMBL	6.78	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3ccc(C4CC4)cc32)cc1
E3 Binder	CHEMBL4565933	ChEMBL	7.66	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3ccc(Cl)cc32)cc1
E3 Binder	CHEMBL4579683	ChEMBL	8.1	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3ccc(F)cc32)cc1
E3 Binder	CHEMBL4441436	ChEMBL	7.5	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3ccc(O)cc32)cc1
E3 Binder	CHEMBL4550214	ChEMBL	8.8	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3ccccc32)cc1
E3 Binder	CHEMBL4552452	ChEMBL	7.7	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3ccccc32)s1
E3 Binder	CHEMBL4438057	ChEMBL	8.41	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3cccnc32)cc1
E3 Binder	CHEMBL4457790	ChEMBL	7.82	—	—	O=C(NO)c1ccc(Cn2c(=O)n(CCc3ccccc3)c(=O)c3ccsc32)cc1
E3 Binder	CHEMBL5220934	ChEMBL	7.55	—	—	O=C(NO)c1ccc(Cn2c([C@@H]3CC4(CC4)CN3c3ncnc4[nH]cnc34)nc3cccc(F)c3c2=O)cc1
E3 Binder	CHEMBL4531108	ChEMBL	8.43	—	—	O=C(NO)c1ccc(Cn2c3c(c4cc(F)ccc42)CS(=O)(=O)CC3)cc1
E3 Binder	CHEMBL4537561	ChEMBL	7.66	—	—	O=C(NO)c1ccc(Cn2c3c(c4cc(F)ccc42)CSCC3)cc1
E3 Binder	CHEMBL4283105	ChEMBL	8.03	—	—	O=C(NO)c1ccc(Cn2c3c(c4cc(F)ccc42)C[S+]([O-])CC3)cc1
E3 Binder	CHEMBL4081647	ChEMBL	8.19	—	—	O=C(NO)c1ccc(Cn2c3c(c4ccccc42)C2CCN(C3)C2)cc1.O=C(O)C(F)(F)F
E3 Binder	CHEMBL4475240	ChEMBL	7.2	—	—	O=C(NO)c1ccc(Cn2c3c(c4ccccc42)CCCC3)cc1
E3 Binder	CHEMBL2018452	ChEMBL	9.06	—	—	O=C(NO)c1ccc(Cn2c3c(c4ccccc42)CCN(Cc2ccccc2)C3)cc1
E3 Binder	CHEMBL4062461	ChEMBL	7.52	—	—	O=C(NO)c1ccc(Cn2c3c(c4ccccc42)CCN2C(=O)CCCC32)cc1
E3 Binder	CHEMBL2018450	ChEMBL	8.6	—	—	O=C(NO)c1ccc(Cn2c3c(c4ccccc42)CCNC3)cc1
E3 Binder	CHEMBL2018443	ChEMBL	8.84	—	—	O=C(NO)c1ccc(Cn2c3c(c4ccccc42)CN(Cc2ccccc2)CC3)cc1
E3 Binder	CHEMBL2018446	ChEMBL	9.23	—	—	O=C(NO)c1ccc(Cn2c3c(c4ccccc42)CN(Cc2ccncc2)CC3)cc1
E3 Binder	CHEMBL2018304	ChEMBL	8.18	—	—	O=C(NO)c1ccc(Cn2c3c(c4ccccc42)CNCC3)cc1
E3 Binder	CHEMBL4531802	ChEMBL	7.7	—	—	O=C(NO)c1ccc(Cn2c3c(c4ccccc42)COCC3)cc1
E3 Binder	CHEMBL4577299	ChEMBL	8.72	—	—	O=C(NO)c1ccc(Cn2c3c(c4ccccc42)CS(=O)(=O)CC3)cc1
E3 Binder	CHEMBL4438279	ChEMBL	6.9	—	—	O=C(NO)c1ccc(Cn2c3c(c4ccccc42)CSCC3)cc1
E3 Binder	CHEMBL4069287	ChEMBL	8.1	—	—	O=C(NO)c1ccc(Cn2c3c(c4ccccc42)S(=O)(=O)CC3)cc1
E3 Binder	CHEMBL2170166	ChEMBL	7.72	—	—	O=C(NO)c1ccc(Cn2c3ccccc3c3ccccc32)cc1
E3 Binder	CHEMBL4090165	ChEMBL	7.96	—	—	O=C(NO)c1ccc(Cn2cc(-c3ccc(CN4CCCC4)cc3)nn2)cc1
E3 Binder	CHEMBL5204426	ChEMBL	7.82	—	—	O=C(NO)c1ccc(Cn2cc(-c3ccc(CO)cc3)nc(N3CCOCC3)c2=O)cc1
E3 Binder	CHEMBL5175778	ChEMBL	7.85	—	—	O=C(NO)c1ccc(Cn2cc(-c3ccc(O)cc3)nc(N3CCOCC3)c2=O)cc1
E3 Binder	CHEMBL5206969	ChEMBL	7.85	—	—	O=C(NO)c1ccc(Cn2cc(-c3cccc(CO)c3)nc(N3CCOCC3)c2=O)cc1
E3 Binder	CHEMBL5170590	ChEMBL	7.64	—	—	O=C(NO)c1ccc(Cn2cc(-c3cccc(O)c3)nc(N3CCOCC3)c2=O)cc1
E3 Binder	CHEMBL5180796	ChEMBL	8.35	—	—	O=C(NO)c1ccc(Cn2cc(-c3cccc4[nH]ncc34)nc(N3CCOCC3)c2=O)cc1
E3 Binder	CHEMBL5194733	ChEMBL	7.82	—	—	O=C(NO)c1ccc(Cn2cc(-c3cccnc3)nc(N3CCOCC3)c2=O)cc1
E3 Binder	CHEMBL5180870	ChEMBL	8.1	—	—	O=C(NO)c1ccc(Cn2cc(-c3ccoc3)nc(N3CCOCC3)c2=O)cc1
E3 Binder	CHEMBL5186022	ChEMBL	7.52	—	—	O=C(NO)c1ccc(Cn2cc(-c3cn[nH]c3)nc(N3CCOCC3)c2=O)cc1
E3 Binder	CHEMBL5202781	ChEMBL	7.46	—	—	O=C(NO)c1ccc(Cn2cc(-c3cncnc3)nc(N3CCOCC3)c2=O)cc1
E3 Binder	CHEMBL5188338	ChEMBL	8.28	—	—	O=C(NO)c1ccc(Cn2cc(C(=O)NC3C4CC5CC(C4)CC3C5)c3ccccc32)cc1
E3 Binder	CHEMBL4466930	ChEMBL	7.5	TWS	—	O=C(NO)c1ccc(Cn2cc(CCO)c3ccccc32)cc1
E3 Binder	CHEMBL4578278	ChEMBL	6.8	—	—	O=C(NO)c1ccc(Cn2cc(CN3CCCC3)c3ccccc32)cc1
E3 Binder	CHEMBL3948680	ChEMBL	7.53	—	—	O=C(NO)c1ccc(Cn2cc(Cc3ccccc3)c3ccccc32)cc1
E3 Binder	CHEMBL4563723	ChEMBL	7.89	—	—	O=C(NO)c1ccc(Cn2cc(Nc3ncc(Cl)c(Nc4ccc(F)cc4)n3)cn2)cc1
E3 Binder	CHEMBL4206537	ChEMBL	8.17	—	—	O=C(NO)c1ccc(Cn2ccc3cc(C(=O)c4ccc(Cl)cc4)ccc32)cc1
E3 Binder	CHEMBL4215954	ChEMBL	8.03	—	—	O=C(NO)c1ccc(Cn2ccc3cc(C(=O)c4ccc(F)cc4)ccc32)cc1
E3 Binder	CHEMBL3958794	ChEMBL	8.01	TWP	—	O=C(NO)c1ccc(Cn2ccc3ccccc32)cc1
E3 Binder	CHEMBL3976023	ChEMBL	7.5	—	—	O=C(NO)c1ccc(Cn2cccc2)cc1
E3 Binder	CHEMBL3970950	ChEMBL	7.96	—	—	O=C(NO)c1ccc(Cn2cccn2)cc1
E3 Binder	CHEMBL5280669	ChEMBL	7.84	—	—	O=C(NO)c1ccc(Cn2cnc(-c3c(F)cccc3F)n2)cc1
E3 Binder	CHEMBL5271970	ChEMBL	7.71	—	—	O=C(NO)c1ccc(Cn2cnc(-c3cc(F)cc(F)c3)n2)cc1
E3 Binder	CHEMBL5273396	ChEMBL	7.9	—	—	O=C(NO)c1ccc(Cn2cnc(-c3ccc(F)cc3)n2)cc1
E3 Binder	CHEMBL5279952	ChEMBL	7.96	—	—	O=C(NO)c1ccc(Cn2cnc(-c3cccc(-c4ccccc4)c3)n2)cc1
E3 Binder	CHEMBL5274088	ChEMBL	8.34	—	—	O=C(NO)c1ccc(Cn2cnc(-c3cccc(C(F)(F)F)c3)n2)cc1
E3 Binder	CHEMBL5271520	ChEMBL	8.19	—	—	O=C(NO)c1ccc(Cn2cnc(-c3cccc(Cl)c3)n2)cc1
E3 Binder	CHEMBL5271793	ChEMBL	8.06	—	—	O=C(NO)c1ccc(Cn2cnc(-c3cccc(F)c3)n2)cc1
E3 Binder	CHEMBL5267739	ChEMBL	7.91	—	—	O=C(NO)c1ccc(Cn2cnc(-c3cccc(O)c3)n2)cc1
E3 Binder	CHEMBL5285879	ChEMBL	7.88	—	—	O=C(NO)c1ccc(Cn2cnc(-c3cccc(OC(F)(F)F)c3)n2)cc1
E3 Binder	CHEMBL5281142	ChEMBL	7.91	—	—	O=C(NO)c1ccc(Cn2cnc(-c3ccccc3)n2)c(F)c1
E3 Binder	CHEMBL5266236	ChEMBL	8.04	—	—	O=C(NO)c1ccc(Cn2cnc(-c3ccccc3)n2)cc1
E3 Binder	CHEMBL5290601	ChEMBL	7.69	—	—	O=C(NO)c1ccc(Cn2cnc(-c3ccccc3)n2)nc1
E3 Binder	CHEMBL5274634	ChEMBL	8.15	—	—	O=C(NO)c1ccc(Cn2cnc(-c3ccccc3F)n2)c(F)c1
E3 Binder	CHEMBL5268616	ChEMBL	8.0	—	—	O=C(NO)c1ccc(Cn2cnc(-c3ccccc3F)n2)cc1
E3 Binder	CHEMBL5285996	ChEMBL	7.55	—	—	O=C(NO)c1ccc(Cn2cnc(-c3cccnc3)n2)cc1
E3 Binder	CHEMBL5291256	ChEMBL	7.98	—	—	O=C(NO)c1ccc(Cn2cnc(-c3cccs3)n2)cc1
E3 Binder	CHEMBL5287254	ChEMBL	7.36	—	—	O=C(NO)c1ccc(Cn2cnc(Br)n2)cc1
E3 Binder	CHEMBL3927508	ChEMBL	7.53	—	—	O=C(NO)c1ccc(Cn2cnc3ccccc32)cc1
E3 Binder	CHEMBL3909186	ChEMBL	8.46	—	—	O=C(NO)c1ccc(Cn2cnc3cncnc32)cc1
E3 Binder	CHEMBL3909854	ChEMBL	7.85	—	—	O=C(NO)c1ccc(Cn2cnc3ncncc32)cc1
E3 Binder	CHEMBL5267379	ChEMBL	7.04	—	—	O=C(NO)c1ccc(Cn2cncn2)cc1
E3 Binder	CHEMBL4226489	ChEMBL	6.49	—	—	O=C(NO)c1ccc(Cn2nc(-c3ccc(F)cc3)cc2Cc2ccccc2)cc1
E3 Binder	CHEMBL4229043	ChEMBL	6.38	—	—	O=C(NO)c1ccc(Cn2nc(Cc3ccccc3)cc2-c2ccc(F)cc2)cc1
E3 Binder	CHEMBL5284689	ChEMBL	7.77	—	—	O=C(NO)c1ccc(Cn2ncnc2-c2ccccc2)cc1
E3 Binder	CHEMBL5271343	ChEMBL	7.93	—	—	O=C(NO)c1ccc(Cn2ncnc2-c2ccccc2F)cc1
E3 Binder	CHEMBL5287109	ChEMBL	7.74	—	—	O=C(NO)c1ccc(Cn2ncnc2-c2cccs2)cc1
E3 Binder	CHEMBL4580311	ChEMBL	7.96	—	—	O=C(NO)c1ccc(Cn2nnc(-c3ccc(C(F)(F)F)cc3)n2)cc1
E3 Binder	CHEMBL4454925	ChEMBL	7.6	—	—	O=C(NO)c1ccc(Cn2nnc(-c3ccc(S(F)(F)(F)(F)F)cc3)n2)cc1
E3 Binder	CHEMBL4529251	ChEMBL	7.7	—	—	O=C(NO)c1ccc(Cn2nnc(-c3ccc4ccccc4n3)n2)cc1
E3 Binder	CHEMBL4515650	ChEMBL	7.58	—	—	O=C(NO)c1ccc(Cn2nnc(-c3cccc(S(F)(F)(F)(F)F)c3)n2)cc1
E3 Binder	CHEMBL4456695	ChEMBL	8.52	—	—	O=C(NO)c1ccc(Cn2nnc(-c3ccccc3)n2)cc1
E3 Binder	CHEMBL4514075	ChEMBL	8.05	—	—	O=C(NO)c1ccc(Cn2nnc(-c3ccccn3)n2)cc1
E3 Binder	CHEMBL4535144	ChEMBL	7.7	—	—	O=C(NO)c1ccc(Cn2nnc(-c3nccc4ccccc34)n2)cc1
E3 Binder	CHEMBL4453121	ChEMBL	8.15	—	—	O=C(NO)c1ccc(Cn2nnc(-c3ncccn3)n2)cc1
E3 Binder	CHEMBL4464235	ChEMBL	7.28	—	—	O=C(NO)c1ccc(Cn2nnc(Cc3ccccc3)n2)cc1
E3 Binder	CHEMBL4551484	ChEMBL	7.6	—	—	O=C(NO)c1ccc(Cn2nnc(Cc3ccccn3)n2)cc1
E3 Binder	CHEMBL4551987	ChEMBL	8.05	—	—	O=C(NO)c1ccc(Cn2nnnc2-c2ccccc2)cc1
E3 Binder	CHEMBL4448410	ChEMBL	7.77	UZW	—	O=C(NO)c1ccc(Cn2nnnc2-c2cccs2)cc1
E3 Binder	CHEMBL5185889	ChEMBL	8.52	—	—	O=C(NO)c1ccc(Cn2sc3ccccc3c2=O)cc1
E3 Binder	CHEMBL3798925	ChEMBL	6.3	—	—	O=C(NO)c1ccc(F)c(NC(=O)c2ccccc2)c1
E3 Binder	CHEMBL4563091	ChEMBL	7.07	—	—	O=C(NO)c1ccc(N(Cc2ccc(C(F)(F)F)cc2)C(=O)CN(Cc2c(F)c(F)c(F)c(F)c2F)S(=O)(=O)c2ccc(F)cc2)cc1
E3 Binder	CHEMBL4578694	ChEMBL	6.73	—	—	O=C(NO)c1ccc(N(Cc2ccc(C(F)(F)F)cc2)C(=O)CN(Cc2ccccc2C(F)(F)F)S(=O)(=O)c2ccc(F)c(F)c2)cc1
E3 Binder	CHEMBL4561439	ChEMBL	7.03	—	—	O=C(NO)c1ccc(N(Cc2ccc(C(F)(F)F)cc2)C(=O)CN(Cc2ccccc2C(F)(F)F)S(=O)(=O)c2ccc(F)cc2)cc1
E3 Binder	CHEMBL4447317	ChEMBL	6.82	—	—	O=C(NO)c1ccc(N(Cc2ccc(C(F)(F)F)cc2)C(=O)CN(Cc2ccccc2C(F)(F)F)S(=O)(=O)c2ccc(F)cc2F)cc1
E3 Binder	CHEMBL4641390	ChEMBL	6.65	—	—	O=C(NO)c1ccc(N(Cc2cccc(C(F)(F)F)c2)C(=O)c2cccc(C(F)(F)F)c2)cc1
E3 Binder	CHEMBL4563224	ChEMBL	8.83	—	—	O=C(NO)c1ccc(N(Cc2ccccc2)C(=O)CN(Cc2c(F)c(F)c(F)c(F)c2F)S(=O)(=O)c2ccc(F)cc2)cc1
E3 Binder	CHEMBL4640205	ChEMBL	6.76	—	—	O=C(NO)c1ccc(N(Cc2ccccc2)C(=O)c2cccc(C(F)(F)F)c2)cc1
E3 Binder	CHEMBL4460979	ChEMBL	6.27	—	—	O=C(NO)c1ccc(N2CCCC2)cc1
E3 Binder	CHEMBL1270140	ChEMBL	7.35	—	—	O=C(NO)c1ccc(N2C[C@H]3CN(Cc4ccc5ccccc5c4)C[C@H]3C2)nc1
E3 Binder	CHEMBL5192082	ChEMBL	6.69	—	—	O=C(NO)c1ccc(NC(=O)N2CCC(N3C(=O)[C@H](c4ccccc4)[C@H]3c3ccccc3)CC2)cc1
E3 Binder	CHEMBL5272475	ChEMBL	6.46	—	—	O=C(NO)c1ccc(NC(=O)[C@@H](NC(=O)c2ccc(Cl)cc2)c2ccccc2)cc1
E3 Binder	CHEMBL5274036	ChEMBL	7.84	—	—	O=C(NO)c1ccc(NC(=O)[C@@H](NC(=O)c2ccc3ccccc3c2)c2ccccc2)cc1
E3 Binder	CHEMBL5273740	ChEMBL	7.86	—	—	O=C(NO)c1ccc(NC(=O)[C@@H](NC(=O)c2cccc(Br)c2)c2ccccc2)cc1
E3 Binder	CHEMBL5268468	ChEMBL	7.81	—	—	O=C(NO)c1ccc(NC(=O)[C@@H](NS(=O)(=O)c2cccc3ccccc23)c2ccccc2)cc1
E3 Binder	CHEMBL4750701	ChEMBL	8.84	—	—	O=C(NO)c1ccc(NC(=O)c2c(F)c(F)c(F)c(F)c2F)cc1
E3 Binder	CHEMBL4636672	ChEMBL	6.95	—	—	O=C(NO)c1ccc(NC(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1
E3 Binder	CHEMBL4780745	ChEMBL	7.65	—	—	O=C(NO)c1ccc(NC(=O)c2ccc(C(F)(F)F)cc2)cc1
E3 Binder	CHEMBL4747455	ChEMBL	8.55	—	—	O=C(NO)c1ccc(NC(=O)c2ccc(C3CC3)cc2)cc1
E3 Binder	CHEMBL4790223	ChEMBL	7.58	—	—	O=C(NO)c1ccc(NC(=O)c2ccc(C3CCCCC3)cc2)cc1
E3 Binder	CHEMBL4760306	ChEMBL	8.17	—	—	O=C(NO)c1ccc(NC(=O)c2ccc(F)cc2)cc1
E3 Binder	CHEMBL4788731	ChEMBL	7.01	—	—	O=C(NO)c1ccc(NC(=O)c2ccc(N3CCOCC3)cc2)cc1
E3 Binder	CHEMBL4641253	ChEMBL	7.22	—	—	O=C(NO)c1ccc(NC(=O)c2cccc(C(F)(F)F)c2)cc1
E3 Binder	CHEMBL191227	ChEMBL	6.68	—	—	O=C(NO)c1ccc(NC(=O)c2ccccc2)cc1
E3 Binder	CHEMBL3415452	ChEMBL	6.62	—	—	O=C(NO)c1ccc(NC2CCN(CCc3ccccc3)C2=O)cc1
E3 Binder	CHEMBL3415451	ChEMBL	6.29	—	—	O=C(NO)c1ccc(NC2CCN(Cc3ccccc3)C2=O)cc1
E3 Binder	CHEMBL3415618	ChEMBL	6.6	—	—	O=C(NO)c1ccc(NC2CCN(c3ccc(C(F)(F)F)cc3)C2=O)cc1
E3 Binder	CHEMBL3415619	ChEMBL	7.2	—	—	O=C(NO)c1ccc(NC2CCN(c3ccc(Cl)c(Cl)c3)C2=O)cc1
E3 Binder	CHEMBL3415625	ChEMBL	6.07	—	—	O=C(NO)c1ccc(NC2CCN(c3ccc(Cl)cc3)C2)cc1
E3 Binder	CHEMBL3415453	ChEMBL	6.8	—	—	O=C(NO)c1ccc(NC2CCN(c3ccc(Cl)cc3)C2=O)cc1
E3 Binder	CHEMBL3415454	ChEMBL	7.05	—	—	O=C(NO)c1ccc(NC2CCN(c3cccc(Cl)c3)C2=O)cc1
E3 Binder	CHEMBL3415446	ChEMBL	6.42	—	—	O=C(NO)c1ccc(NC2CCN(c3ccccc3)C2=O)cc1
E3 Binder	CHEMBL3415456	ChEMBL	6.44	—	—	O=C(NO)c1ccc(NC2CCN(c3ccccc3Cl)C2=O)cc1
E3 Binder	CHEMBL3915689	ChEMBL	6.4	—	—	O=C(NO)c1ccc(NCCOc2ccc3cc2COC/C=C/COCc2cccc(c2)-c2ccnc(n2)N3)cc1
E3 Binder	CHEMBL4093020	ChEMBL	8.13	—	—	O=C(NO)c1ccc(NCc2cccc3cccnc23)cc1
E3 Binder	CHEMBL4103801	ChEMBL	7.43	—	—	O=C(NO)c1ccc(NCc2csc3ccc(Br)cc23)cc1
E3 Binder	CHEMBL4649617	ChEMBL	7.85	—	—	O=C(NO)c1ccc(NCc2csc3ccccc23)cc1
E3 Binder	CHEMBL4866346	ChEMBL	6.49	—	—	O=C(NO)c1ccc(NCc2nc(-c3cc4ccccc4s3)nn2-c2ccccc2)cc1
E3 Binder	CHEMBL4865551	ChEMBL	6.74	—	—	O=C(NO)c1ccc(NCc2nc(-c3ccc(Cl)cc3)nn2-c2ccccc2)cc1
E3 Binder	CHEMBL4870410	ChEMBL	6.94	—	—	O=C(NO)c1ccc(NCc2nc(-c3ccc(F)cc3)nn2-c2ccccc2)cc1
E3 Binder	CHEMBL4871535	ChEMBL	6.94	—	—	O=C(NO)c1ccc(NCc2nc(-c3cccc(Cl)c3)nn2-c2ccccc2)cc1
E3 Binder	CHEMBL4862609	ChEMBL	6.56	—	—	O=C(NO)c1ccc(NCc2nc(-c3ccccc3)nn2-c2ccc(F)cc2)cc1
E3 Binder	CHEMBL4855023	ChEMBL	6.17	—	—	O=C(NO)c1ccc(NCc2nc(-c3ccccc3)nn2-c2cccc(Cl)c2)cc1
E3 Binder	CHEMBL4849763	ChEMBL	6.95	—	—	O=C(NO)c1ccc(NCc2nc(-c3ccccc3)nn2-c2ccccc2)cc1
E3 Binder	CHEMBL4849003	ChEMBL	6.17	—	—	O=C(NO)c1ccc(NCc2nc(-c3ccccc3)nn2-c2ccccc2Cl)cc1
E3 Binder	CHEMBL4860861	ChEMBL	6.73	—	—	O=C(NO)c1ccc(NCc2nc(-c3ccccc3Cl)nn2-c2ccccc2)cc1
E3 Binder	CHEMBL4854288	ChEMBL	7.47	—	—	O=C(NO)c1ccc(NCc2nc(-c3cccs3)nn2-c2ccc(O)cc2)cc1
E3 Binder	CHEMBL4863879	ChEMBL	7.26	—	—	O=C(NO)c1ccc(NCc2nc(-c3sccc3Br)nn2-c2ccccc2)cc1
E3 Binder	CHEMBL4796066	ChEMBL	7.58	—	—	O=C(NO)c1ccc(Nc2c3ccccc3nc3ccc(Br)cc23)cc1
E3 Binder	CHEMBL4757035	ChEMBL	7.54	—	—	O=C(NO)c1ccc(Nc2c3ccccc3nc3ccc(F)cc23)cc1
E3 Binder	CHEMBL4751082	ChEMBL	7.54	—	—	O=C(NO)c1ccc(Nc2c3ccccc3nc3ccc(OC(F)(F)F)cc23)cc1
E3 Binder	CHEMBL4761847	ChEMBL	6.66	—	—	O=C(NO)c1ccc(Nc2c3ccccc3nc3ccc(OCc4ccccc4)cc23)cc1
E3 Binder	CHEMBL4762873	ChEMBL	7.6	—	—	O=C(NO)c1ccc(Nc2c3ccccc3nc3ccccc23)cc1
E3 Binder	CHEMBL4073021	ChEMBL	6.89	—	—	O=C(NO)c1ccc(Nc2cccc3cccnc23)cc1
E3 Binder	CHEMBL4752558	ChEMBL	7.41	—	—	O=C(NO)c1ccc(Nc2ccnc3ccccc23)cc1
E3 Binder	CHEMBL4530238	ChEMBL	6.87	—	—	O=C(NO)c1ccc(Nc2nnc(-c3ccccc3)o2)cc1
E3 Binder	CHEMBL4436726	ChEMBL	7.18	—	—	O=C(NO)c1ccc(Nc2nnc(-c3ccccc3)s2)cc1
E3 Binder	CHEMBL3924682	ChEMBL	7.18	—	—	O=C(NO)c1ccc(OCCOc2ccc3cc2COC/C=C/COCc2cccc(c2)-c2ccnc(n2)N3)cc1
E3 Binder	CHEMBL5282067	ChEMBL	6.35	—	—	O=C(NO)c1ccc(S(=O)(=O)NCC2CCN(Cc3ccccc3)CC2)cc1
E3 Binder	CHEMBL4455244	ChEMBL	6.79	—	—	O=C(NO)c1ccc(Sc2nc(C3CC3)n(-c3ccccc3)n2)cc1
E3 Binder	CHEMBL4550551	ChEMBL	7.21	—	—	O=C(NO)c1ccc(Sc2ncc(-c3ccccc3)s2)cc1
E3 Binder	CHEMBL4545033	ChEMBL	7.25	—	—	O=C(NO)c1ccc(Sc2nnc(-c3ccccc3)n2-c2ccccc2)cc1
E3 Binder	CHEMBL4559109	ChEMBL	8.22	—	—	O=C(NO)c1ccc(Sc2nnc(-c3ccccc3)o2)cc1
E3 Binder	CHEMBL4466468	ChEMBL	8.22	—	—	O=C(NO)c1ccc(Sc2nnc(-c3ccccc3)s2)cc1
E3 Binder	CHEMBL566099	ChEMBL	8.81	—	—	O=C(NO)c1ccc2[nH]c(=O)c(CCCc3ccccc3)nc2c1
E3 Binder	CHEMBL4437432	ChEMBL	7.25	—	—	O=C(NO)c1ccc2c(c1)C(=O)c1ccccc1C2=O
E3 Binder	CHEMBL3357484	ChEMBL	6.0	—	—	O=C(NO)c1ccc2c(c1)CC(NS(=O)(=O)c1cccc(F)c1)CC2
E3 Binder	CHEMBL3357481	ChEMBL	6.03	—	—	O=C(NO)c1ccc2c(c1)CC(Nc1nccc(-c3ccccc3Cl)n1)CC2
E3 Binder	CHEMBL3415445	ChEMBL	7.92	—	—	O=C(NO)c1ccc2c(c1)CC(Nc1nccc(-c3cccnc3)n1)CN2
E3 Binder	CHEMBL3357477	ChEMBL	6.14	—	—	O=C(NO)c1ccc2c(c1)CC(Nc1ncccn1)CC2
E3 Binder	CHEMBL4447120	ChEMBL	7.0	—	—	O=C(NO)c1ccc2c(c1)CC1(CC2)CCN(Cc2cc(Cl)ccc2Cl)C1=O
E3 Binder	CHEMBL4469656	ChEMBL	7.0	—	—	O=C(NO)c1ccc2c(c1)CC1(CC2)CCN(Cc2ccccc2OC(F)(F)F)C1=O
E3 Binder	CHEMBL2431914	ChEMBL	6.47	—	—	O=C(NO)c1ccc2c(c1)CCCN(C(=O)C1CCCCCC1)C2
E3 Binder	CHEMBL2431915	ChEMBL	6.92	—	—	O=C(NO)c1ccc2c(c1)CCCN(C(=O)c1ccc(-c3ccccc3)cc1)C2
E3 Binder	CHEMBL2431903	ChEMBL	7.3	—	—	O=C(NO)c1ccc2c(c1)CCN(C(=O)C1CCCCC1)C2
E3 Binder	CHEMBL2431905	ChEMBL	7.27	—	—	O=C(NO)c1ccc2c(c1)CCN(C(=O)C1CCCCCC1)C2
E3 Binder	CHEMBL2431910	ChEMBL	6.92	—	—	O=C(NO)c1ccc2c(c1)CCN(C(=O)C1CCCCCC1)CC2
E3 Binder	CHEMBL2431911	ChEMBL	7.23	—	—	O=C(NO)c1ccc2c(c1)CCN(C(=O)c1ccc(-c3ccccc3)cc1)CC2
E3 Binder	CHEMBL5202970	ChEMBL	7.3	—	—	O=C(NO)c1ccc2c(c1)CCN(S(=O)(=O)c1cc(F)c(F)c(F)c1F)C2
E3 Binder	CHEMBL2431904	ChEMBL	7.22	—	—	O=C(NO)c1ccc2c(c1)CCN(S(=O)(=O)c1ccc(C(F)(F)F)cc1)C2
E3 Binder	CHEMBL3338404	ChEMBL	7.3	—	—	O=C(NO)c1ccc2c(c1)CN(Cc1ccc(-c3cccc([N+](=O)[O-])c3)o1)CC2
E3 Binder	CHEMBL3338417	ChEMBL	7.4	—	—	O=C(NO)c1ccc2c(c1)C[C@@H](Nc1nccc(-c3cccnc3)n1)CC2
E3 Binder	CHEMBL3338418	ChEMBL	7.32	—	—	O=C(NO)c1ccc2c(c1)C[C@H](Nc1nccc(-c3cccnc3)n1)CC2
E3 Binder	CHEMBL5084881	ChEMBL	6.4	—	—	O=C(NO)c1cccc(/C=C/c2ccnc(-c3cc(F)ccc3O)c2)c1
E3 Binder	CHEMBL5070176	ChEMBL	6.41	—	—	O=C(NO)c1cccc(/C=C/c2ccnc(-c3ccccc3O)c2)c1
E3 Binder	CHEMBL5274269	ChEMBL	6.1	—	—	O=C(NO)c1cccc(C(=O)NCC2CCN(Cc3ccccc3)CC2)c1
E3 Binder	CHEMBL2381517	ChEMBL	7.44	—	—	O=C(NO)c1cccc(C(=O)NCCc2ccccc2)c1
E3 Binder	CHEMBL2381518	ChEMBL	7.23	—	—	O=C(NO)c1cccc(C(=O)NCCc2cccnc2)c1
E3 Binder	CHEMBL2381519	ChEMBL	7.47	—	—	O=C(NO)c1cccc(C(=O)NCc2ccccc2)c1
E3 Binder	CHEMBL2381520	ChEMBL	7.24	GQZ	—	O=C(NO)c1cccc(C(=O)Nc2ccccc2)c1
E3 Binder	CHEMBL5192945	ChEMBL	6.31	—	—	O=C(NO)c1cccc(CN(C2CC2)S(=O)(=O)c2c(F)c(F)c(F)c(F)c2F)c1
E3 Binder	CHEMBL5281671	ChEMBL	6.82	—	—	O=C(NO)c1cccc(Cn2ncnc2-c2ccccc2)c1
E3 Binder	CHEMBL4850382	ChEMBL	6.34	—	—	O=C(NO)c1cccc(F)c1
E3 Binder	CHEMBL16300	ChEMBL	6.94	BHO	—	O=C(NO)c1ccccc1
E3 Binder	CHEMBL504369	ChEMBL	6.17	—	—	O=C(NO)c1cccnc1
E3 Binder	CHEMBL5281688	ChEMBL	6.0	—	—	O=C(NO)c1cn(C2CCN(C(=O)Cc3ccc4ccccc4c3)CC2)nn1
E3 Binder	CHEMBL3353067	ChEMBL	7.19	—	—	O=C(NO)c1cn2c(n1)CN(C(=O)c1cc3ccccc3s1)CC2
E3 Binder	CHEMBL3353068	ChEMBL	7.06	—	—	O=C(NO)c1cn2c(n1)CN(C(=O)c1ccc(-c3ccccc3)cc1)CC2
E3 Binder	CHEMBL4797268	ChEMBL	8.52	—	—	O=C(NO)c1cnc(C2(c3ccccc3)CCC(F)(F)CC2)nc1
E3 Binder	CHEMBL4798455	ChEMBL	6.29	—	—	O=C(NO)c1cnc(CCCN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)s1
E3 Binder	CHEMBL1801253	ChEMBL	7.5	—	—	O=C(NO)c1cnc(N2CC3C(CNCc4ccc5ccccc5c4)C3C2)nc1
E3 Binder	CHEMBL5277907	ChEMBL	7.1	—	—	O=C(NO)c1cnc(N2CCC(CN3CC(=O)N4C(Cc5c([nH]c6ccccc56)C4c4ccc5c(c4)OCO5)C3=O)CC2)nc1
E3 Binder	CHEMBL594542	ChEMBL	8.82	—	—	O=C(NO)c1cnc(N2CCC(CNC(/C=C/c3ccccc3)CO)CC2)nc1
E3 Binder	CHEMBL4289912	ChEMBL	6.35	—	—	O=C(NO)c1cnc(N2CCC(Cn3[se]c4ccccc4c3=O)CC2)nc1
E3 Binder	CHEMBL592902	ChEMBL	8.15	—	—	O=C(NO)c1cnc(N2CCC(NC(/C=C/c3ccccc3)CO)CC2)nc1
E3 Binder	CHEMBL5172182	ChEMBL	7.8	—	—	O=C(NO)c1cnc(N2CCC(NC(=O)c3cnc(-n4cccn4)nc3O)CC2)nc1
E3 Binder	CHEMBL4292239	ChEMBL	6.01	—	—	O=C(NO)c1cnc(N2CCC(n3[se]c4ccccc4c3=O)CC2)nc1
E3 Binder	CHEMBL605110	ChEMBL	9.05	—	—	O=C(NO)c1cnc(N2CCN(C(/C=C/c3ccc(-c4ccccc4)cc3)CO)CC2)nc1
E3 Binder	CHEMBL594317	ChEMBL	8.68	—	—	O=C(NO)c1cnc(N2CCN(C(/C=C/c3ccc(C(F)(F)F)cc3)CO)CC2)nc1
E3 Binder	CHEMBL604796	ChEMBL	8.92	—	—	O=C(NO)c1cnc(N2CCN(C(/C=C/c3ccc(Cl)cc3)CO)CC2)nc1
E3 Binder	CHEMBL594544	ChEMBL	8.98	—	—	O=C(NO)c1cnc(N2CCN(C(/C=C/c3ccc(F)cc3)CO)CC2)nc1
E3 Binder	CHEMBL608416	ChEMBL	8.92	—	—	O=C(NO)c1cnc(N2CCN(C(/C=C/c3cccc(F)c3)CO)CC2)nc1
E3 Binder	CHEMBL593859	ChEMBL	8.15	—	—	O=C(NO)c1cnc(N2CCN(C(/C=C/c3ccccc3)C(=O)N3CCOCC3)CC2)nc1
E3 Binder	CHEMBL595480	ChEMBL	7.96	—	—	O=C(NO)c1cnc(N2CCN(C(/C=C/c3ccccc3)CN3CCOCC3)CC2)nc1
E3 Binder	CHEMBL595910	ChEMBL	9.0	—	—	O=C(NO)c1cnc(N2CCN(C(/C=C/c3ccccc3)CO)CC2)nc1
E3 Binder	CHEMBL594543	ChEMBL	8.7	—	—	O=C(NO)c1cnc(N2CCN(C(/C=C/c3ccccc3F)CO)CC2)nc1
E3 Binder	CHEMBL594743	ChEMBL	8.82	—	—	O=C(NO)c1cnc(N2CCN(Cc3ccc4ccccc4c3)CC2)nc1
E3 Binder	CHEMBL250987	ChEMBL	6.7	—	—	O=C(NO)c1cnc(N2CCN(S(=O)(=O)c3ccc(-c4ccccc4)cc3)CC2)s1
E3 Binder	CHEMBL401078	ChEMBL	6.82	—	—	O=C(NO)c1cnc(N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)s1
E3 Binder	CHEMBL251381	ChEMBL	6.4	—	—	O=C(NO)c1cnc(N2CCN(S(=O)(=O)c3ccc([N+](=O)[O-])cc3)CC2)s1
E3 Binder	CHEMBL609583	ChEMBL	8.22	—	—	O=C(NO)c1cnc(N2CCN(S(=O)(=O)c3ccc4ccccc4c3)CC2)nc1
E3 Binder	CHEMBL250587	ChEMBL	6.66	—	—	O=C(NO)c1cnc(N2CCN(S(=O)(=O)c3ccc4ccccc4c3)CC2)s1
E3 Binder	CHEMBL400873	ChEMBL	6.24	—	—	O=C(NO)c1cnc(N2CCN(S(=O)(=O)c3ccccc3)CC2)s1
E3 Binder	CHEMBL596456	ChEMBL	8.1	—	—	O=C(NO)c1cnc(N2CCOC(CNC(/C=C/c3ccccc3)CO)C2)nc1
E3 Binder	CHEMBL4751524	ChEMBL	9.22	—	—	O=C(NO)c1cnc(N2CCc3ncccc3C2)c(F)c1
E3 Binder	CHEMBL1271349	ChEMBL	6.36	—	—	O=C(NO)c1cnc(N2C[C@@H]3CN(S(=O)(=O)c4cc(C(F)(F)F)cc(C(F)(F)F)c4)C[C@@H]3C2)nc1
E3 Binder	CHEMBL1271350	ChEMBL	6.91	—	—	O=C(NO)c1cnc(N2C[C@@H]3CN(S(=O)(=O)c4ccc(OC(F)(F)F)cc4)C[C@@H]3C2)nc1
E3 Binder	CHEMBL1269033	ChEMBL	7.19	—	—	O=C(NO)c1cnc(N2C[C@@H]3CN(S(=O)(=O)c4ccc5ccccc5c4)C[C@@H]3C2)nc1
E3 Binder	CHEMBL1801174	ChEMBL	7.89	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NC(=O)c2ccc3ccccc3c2)nc1
E3 Binder	CHEMBL1801232	ChEMBL	7.24	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NC(=O)c2ccccc2)nc1
E3 Binder	CHEMBL1801175	ChEMBL	7.4	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NC(=O)c2cccs2)nc1
E3 Binder	CHEMBL1801236	ChEMBL	7.36	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCC2CCCCC2)nc1
E3 Binder	CHEMBL1801235	ChEMBL	7.47	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCCc2ccccc2)nc1
E3 Binder	CHEMBL1801246	ChEMBL	7.8	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2cc(C(F)(F)F)cc(C(F)(F)F)c2)nc1
E3 Binder	CHEMBL1801241	ChEMBL	7.8	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2cc(F)cc(F)c2)nc1
E3 Binder	CHEMBL1801248	ChEMBL	7.85	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2ccc(-c3ccccc3)cc2)nc1
E3 Binder	CHEMBL1801239	ChEMBL	7.85	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2ccc(Br)cc2)nc1
E3 Binder	CHEMBL1801240	ChEMBL	7.47	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2ccc(C(F)(F)F)cc2)nc1
E3 Binder	CHEMBL1801238	ChEMBL	7.89	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2ccc(Cl)cc2)nc1
E3 Binder	CHEMBL1801237	ChEMBL	7.57	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2ccc(F)cc2)nc1
E3 Binder	CHEMBL1801243	ChEMBL	7.82	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2ccc(OC(F)(F)F)cc2)nc1
E3 Binder	CHEMBL1801247	ChEMBL	7.8	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2ccc(Oc3ccccc3)cc2)nc1
E3 Binder	CHEMBL1801250	ChEMBL	8.32	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2ccc3cc(F)ccc3n2)nc1
E3 Binder	CHEMBL1801233	ChEMBL	7.91	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2ccc3ccccc3c2)nc1
E3 Binder	CHEMBL1801249	ChEMBL	8.05	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2ccc3ccccc3n2)nc1
E3 Binder	CHEMBL1801234	ChEMBL	8.0	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NCc2ccccc2)nc1
E3 Binder	CHEMBL1801172	ChEMBL	8.19	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NS(=O)(=O)c2ccc3ccccc3c2)nc1
E3 Binder	CHEMBL1801173	ChEMBL	7.57	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3NS(=O)(=O)c2cccs2)nc1
E3 Binder	CHEMBL1801252	ChEMBL	7.75	—	—	O=C(NO)c1cnc(N2C[C@@H]3[C@H](C2)[C@H]3Nc2ccc3ccccc3n2)nc1
E3 Binder	CHEMBL1271458	ChEMBL	6.91	—	—	O=C(NO)c1cnc(N2C[C@H]3CN(C(=O)CCCOc4ccccc4)C[C@H]3C2)nc1
E3 Binder	CHEMBL1271457	ChEMBL	7.92	—	—	O=C(NO)c1cnc(N2C[C@H]3CN(C(=O)c4ccc5ccccc5c4)C[C@H]3C2)nc1
E3 Binder	CHEMBL1269926	ChEMBL	7.3	—	—	O=C(NO)c1cnc(N2C[C@H]3CN(Cc4cc(Cl)cc(Cl)c4)C[C@H]3C2)nc1
E3 Binder	CHEMBL1270033	ChEMBL	7.38	—	—	O=C(NO)c1cnc(N2C[C@H]3CN(Cc4ccc(Cl)cc4)C[C@H]3C2)nc1
E3 Binder	CHEMBL1270139	ChEMBL	7.89	—	—	O=C(NO)c1cnc(N2C[C@H]3CN(Cc4ccc5ccccc5c4)C[C@H]3C2)nc1
E3 Binder	CHEMBL3655966	ChEMBL	8.52	—	—	O=C(NO)c1cnc(NC(c2ccc(F)cc2)c2ccc(F)cc2)nc1
E3 Binder	CHEMBL3655942	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NC(c2ccccc2)c2ccccc2)nc1
E3 Binder	CHEMBL3655986	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NC2(Cc3ccccc3)CC2)nc1
E3 Binder	CHEMBL4749714	ChEMBL	9.37	—	—	O=C(NO)c1cnc(NC2(c3c(F)cccc3F)CC2)c(F)c1
E3 Binder	CHEMBL3655993	ChEMBL	9.0	—	—	O=C(NO)c1cnc(NC2(c3c(F)cccc3F)CC2)nc1
E3 Binder	CHEMBL3656014	ChEMBL	8.22	—	—	O=C(NO)c1cnc(NC2(c3cc(C(F)(F)F)cc(C(F)(F)F)c3)CC2)nc1
E3 Binder	CHEMBL3655995	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NC2(c3cc(C(F)(F)F)ccc3F)CC2)nc1
E3 Binder	CHEMBL3656015	ChEMBL	8.52	—	—	O=C(NO)c1cnc(NC2(c3cc(Cl)cc(Cl)c3)CC2)nc1
E3 Binder	CHEMBL3656001	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NC2(c3cc(F)cc(F)c3)CC2)nc1
E3 Binder	CHEMBL3944941	ChEMBL	8.54	—	—	O=C(NO)c1cnc(NC2(c3cc(F)cc(F)c3)CCCCC2)nc1
E3 Binder	CHEMBL3656024	ChEMBL	8.15	—	—	O=C(NO)c1cnc(NC2(c3cc(F)cc(F)c3)CCOCC2)nc1
E3 Binder	CHEMBL3920532	ChEMBL	8.62	—	—	O=C(NO)c1cnc(NC2(c3cc(F)ccc3F)CCOCC2)nc1
E3 Binder	CHEMBL3655979	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NC2(c3cc4ccccc4s3)CC2)nc1
E3 Binder	CHEMBL3656006	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NC2(c3ccc(C(F)(F)F)c(F)c3)CC2)nc1
E3 Binder	CHEMBL3656004	ChEMBL	8.15	—	—	O=C(NO)c1cnc(NC2(c3ccc(C(F)(F)F)cc3)CC2)nc1
E3 Binder	CHEMBL3655974	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NC2(c3ccc(CO)cc3)CC2)nc1
E3 Binder	CHEMBL3656010	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NC2(c3ccc(Cl)c(Cl)c3)CC2)nc1
E3 Binder	CHEMBL3656005	ChEMBL	8.52	—	—	O=C(NO)c1cnc(NC2(c3ccc(Cl)cc3)CC2)nc1
E3 Binder	CHEMBL3656000	ChEMBL	8.52	—	—	O=C(NO)c1cnc(NC2(c3ccc(F)c(Cl)c3)CC2)nc1
E3 Binder	CHEMBL3656009	ChEMBL	8.15	—	—	O=C(NO)c1cnc(NC2(c3ccc(F)c(F)c3)CC2)nc1
E3 Binder	CHEMBL3655958	ChEMBL	8.52	—	—	O=C(NO)c1cnc(NC2(c3ccc(F)cc3)CC2)nc1
E3 Binder	CHEMBL3656017	ChEMBL	8.52	—	—	O=C(NO)c1cnc(NC2(c3ccc(F)cc3)CCCC2)nc1
E3 Binder	CHEMBL3655977	ChEMBL	8.05	—	—	O=C(NO)c1cnc(NC2(c3ccc(F)cc3)CCCCC2)nc1
E3 Binder	CHEMBL3656019	ChEMBL	8.3	—	—	O=C(NO)c1cnc(NC2(c3ccc(F)cc3)CCOCC2)nc1
E3 Binder	CHEMBL3656013	ChEMBL	8.52	—	—	O=C(NO)c1cnc(NC2(c3ccc(F)cc3Cl)CC2)nc1
E3 Binder	CHEMBL3655992	ChEMBL	8.52	—	—	O=C(NO)c1cnc(NC2(c3ccc(F)cc3F)CC2)nc1
E3 Binder	CHEMBL3655997	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NC2(c3ccc4c(c3)OCO4)CC2)nc1
E3 Binder	CHEMBL3655990	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NC2(c3cccc(C(F)(F)F)c3)CC2)nc1
E3 Binder	CHEMBL3655971	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NC2(c3cccc(Cl)c3)CC2)nc1
E3 Binder	CHEMBL3656022	ChEMBL	8.1	—	—	O=C(NO)c1cnc(NC2(c3cccc(Cl)c3)CCCC2)nc1
E3 Binder	CHEMBL3655964	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NC2(c3cccc(F)c3)CC2)nc1
E3 Binder	CHEMBL3903253	ChEMBL	8.41	—	—	O=C(NO)c1cnc(NC2(c3cccc(F)c3)CCC3(CC2)OCCO3)nc1
E3 Binder	CHEMBL3656020	ChEMBL	8.52	—	—	O=C(NO)c1cnc(NC2(c3cccc(F)c3)CCCC2)nc1
E3 Binder	CHEMBL3655978	ChEMBL	8.15	—	—	O=C(NO)c1cnc(NC2(c3cccc(F)c3)CCCCC2)nc1
E3 Binder	CHEMBL3656018	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NC2(c3cccc(F)c3)CCOCC2)nc1
E3 Binder	CHEMBL3656012	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NC2(c3cccc(F)c3F)CC2)nc1
E3 Binder	CHEMBL3655994	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NC2(c3cccc(OC(F)(F)F)c3)CC2)nc1
E3 Binder	CHEMBL3655950	ChEMBL	8.77	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CC2)nc1
E3 Binder	CHEMBL3935992	ChEMBL	8.52	AH7	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCC(F)(F)CC2)nc1
E3 Binder	CHEMBL3655999	ChEMBL	8.52	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCC2)nc1
E3 Binder	CHEMBL3655965	ChEMBL	8.52	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCCC2)nc1
E3 Binder	CHEMBL3655961	ChEMBL	8.15	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCCCC2)nc1
E3 Binder	CHEMBL3891420	ChEMBL	8.55	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(C(=O)Cc3c[nH]c4ccccc34)CC2)nc1
E3 Binder	CHEMBL3935353	ChEMBL	8.3	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(C(=O)Cc3cc4ccccc4[nH]3)CC2)nc1
E3 Binder	CHEMBL3916028	ChEMBL	8.43	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(C(=O)Nc3c(F)cccc3F)CC2)nc1
E3 Binder	CHEMBL3939779	ChEMBL	7.85	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(C(=O)Nc3ccc(Cl)c(Cl)c3)CC2)nc1
E3 Binder	CHEMBL3961733	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(C(=O)Nc3ccc(F)cc3)CC2)nc1
E3 Binder	CHEMBL3934237	ChEMBL	8.6	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(C(=O)Nc3cccc(F)c3)CC2)nc1
E3 Binder	CHEMBL3963102	ChEMBL	8.72	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(C(=O)Nc3ccccc3)CC2)nc1
E3 Binder	CHEMBL3977741	ChEMBL	8.77	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(C(=O)Nc3ccccc3F)CC2)nc1
E3 Binder	CHEMBL3906837	ChEMBL	8.59	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(C(=O)OCc3ccccc3)CC2)nc1
E3 Binder	CHEMBL3952742	ChEMBL	8.62	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(C(=S)Nc3ccccc3)CC2)nc1
E3 Binder	CHEMBL3910638	ChEMBL	8.14	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(S(=O)(=O)c3ccc(C(F)(F)F)cc3)CC2)nc1
E3 Binder	CHEMBL3892568	ChEMBL	8.3	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)nc1
E3 Binder	CHEMBL3925038	ChEMBL	8.29	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(S(=O)(=O)c3cccc(F)c3)CC2)nc1
E3 Binder	CHEMBL3947383	ChEMBL	8.34	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(S(=O)(=O)c3ccccc3)CC2)nc1
E3 Binder	CHEMBL3948528	ChEMBL	8.68	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCN(c3ccccc3)CC2)nc1
E3 Binder	CHEMBL3655972	ChEMBL	8.52	—	—	O=C(NO)c1cnc(NC2(c3ccccc3)CCOCC2)nc1
E3 Binder	CHEMBL3655968	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NC2(c3ccccc3C(F)(F)F)CC2)nc1
E3 Binder	CHEMBL3655967	ChEMBL	9.0	—	—	O=C(NO)c1cnc(NC2(c3ccccc3Cl)CC2)nc1
E3 Binder	CHEMBL3655959	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NC2(c3ccccc3F)CC2)nc1
E3 Binder	CHEMBL3655976	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NC2(c3ccco3)CC2)nc1
E3 Binder	CHEMBL3655975	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NC2(c3cccs3)CC2)nc1
E3 Binder	CHEMBL3656023	ChEMBL	8.3	—	—	O=C(NO)c1cnc(NC2(c3cccs3)CCCCC2)nc1
E3 Binder	CHEMBL3655940	ChEMBL	8.05	—	—	O=C(NO)c1cnc(NC23CC4CC(CC(C4)C2)C3)nc1
E3 Binder	CHEMBL3655980	ChEMBL	7.34	—	—	O=C(NO)c1cnc(NC2CCCCC2)nc1
E3 Binder	CHEMBL3655981	ChEMBL	7.31	—	—	O=C(NO)c1cnc(NC2CCOCC2)nc1
E3 Binder	CHEMBL3655988	ChEMBL	7.72	—	—	O=C(NO)c1cnc(NC2c3ccccc3-c3ccccc32)nc1
E3 Binder	CHEMBL3655945	ChEMBL	7.72	—	—	O=C(NO)c1cnc(NCCc2c(Cl)cccc2Cl)nc1
E3 Binder	CHEMBL3655926	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NCCc2c[nH]c3ccccc23)nc1
E3 Binder	CHEMBL3655927	ChEMBL	7.96	—	—	O=C(NO)c1cnc(NCCc2ccc(Cl)cc2)nc1
E3 Binder	CHEMBL3655925	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NCCc2cccc(Cl)c2)nc1
E3 Binder	CHEMBL3655924	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NCCc2ccccc2)nc1
E3 Binder	CHEMBL3655941	ChEMBL	7.4	—	—	O=C(NO)c1cnc(NCCc2ccccc2-c2ccccc2)nc1
E3 Binder	CHEMBL3655922	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NCCc2ccccc2Cl)nc1
E3 Binder	CHEMBL3655934	ChEMBL	7.96	—	—	O=C(NO)c1cnc(NCc2c(CO)cccc2CO)nc1
E3 Binder	CHEMBL3655931	ChEMBL	8.15	—	—	O=C(NO)c1cnc(NCc2c(Cl)cccc2Cl)nc1
E3 Binder	CHEMBL3655984	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NCc2ccc(-c3ccccc3)cc2)nc1
E3 Binder	CHEMBL3655920	ChEMBL	8.3	—	—	O=C(NO)c1cnc(NCc2ccc(C(F)(F)F)cc2)nc1
E3 Binder	CHEMBL3655919	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NCc2ccc(Cl)cc2)nc1
E3 Binder	CHEMBL3655936	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NCc2ccc(F)c(Cl)c2)nc1
E3 Binder	CHEMBL3655939	ChEMBL	8.22	—	—	O=C(NO)c1cnc(NCc2ccc(F)cc2C(F)(F)F)nc1
E3 Binder	CHEMBL3655929	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NCc2ccc3c(c2)OCO3)nc1
E3 Binder	CHEMBL3655923	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NCc2cccc(C(F)(F)F)c2)nc1
E3 Binder	CHEMBL3655917	ChEMBL	9.0	—	—	O=C(NO)c1cnc(NCc2cccc(Cl)c2)nc1
E3 Binder	CHEMBL3655918	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NCc2ccccc2)nc1
E3 Binder	CHEMBL3655938	ChEMBL	8.1	—	—	O=C(NO)c1cnc(NCc2ccccc2-c2ccccc2)nc1
E3 Binder	CHEMBL3655921	ChEMBL	8.15	—	—	O=C(NO)c1cnc(NCc2ccccc2C(F)(F)F)nc1
E3 Binder	CHEMBL3655916	ChEMBL	8.7	—	—	O=C(NO)c1cnc(NCc2ccccc2Cl)nc1
E3 Binder	CHEMBL3655930	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NCc2ccccc2OC(F)(F)F)nc1
E3 Binder	CHEMBL3655985	ChEMBL	8.3	—	—	O=C(NO)c1cnc(NCc2ccccn2)nc1
E3 Binder	CHEMBL3655983	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NCc2cccnc2)nc1
E3 Binder	CHEMBL3655982	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NCc2cccs2)nc1
E3 Binder	CHEMBL3655946	ChEMBL	8.3	—	—	O=C(NO)c1cnc(NCc2ccncc2)nc1
E3 Binder	CHEMBL3655954	ChEMBL	8.4	—	—	O=C(NO)c1cnc(NCc2cnccn2)nc1
E3 Binder	CHEMBL4756236	ChEMBL	9.46	—	—	O=C(NO)c1cnc(N[C@@H](c2ccccn2)C2CC2)c(F)c1
E3 Binder	CHEMBL4748025	ChEMBL	9.56	—	—	O=C(NO)c1cnc(N[C@H](c2ccccc2)C2CC2)c(F)c1
E3 Binder	CHEMBL3652240	ChEMBL	6.06	—	—	O=C(NO)c1cnc(Nc2c(Cl)cccc2Cl)nc1
E3 Binder	CHEMBL3652236	ChEMBL	7.68	—	—	O=C(NO)c1cnc(Nc2c(F)c(F)cc(F)c2F)nc1
E3 Binder	CHEMBL3652235	ChEMBL	7.85	—	—	O=C(NO)c1cnc(Nc2cc(C(F)(F)F)cc(C(F)(F)F)c2)nc1
E3 Binder	CHEMBL3655908	ChEMBL	8.0	—	—	O=C(NO)c1cnc(Nc2cc(Cl)cc(C(F)(F)F)c2)nc1
E3 Binder	CHEMBL3655910	ChEMBL	8.15	—	—	O=C(NO)c1cnc(Nc2cc(Cl)cc(OC(F)(F)F)c2)nc1
E3 Binder	CHEMBL3652234	ChEMBL	7.82	—	—	O=C(NO)c1cnc(Nc2cc(Cl)ccc2Cl)nc1
E3 Binder	CHEMBL3655909	ChEMBL	8.3	—	—	O=C(NO)c1cnc(Nc2cc(F)cc(C(F)(F)F)c2)nc1
E3 Binder	CHEMBL3652238	ChEMBL	7.89	—	—	O=C(NO)c1cnc(Nc2cc(F)cc(F)c2)nc1
E3 Binder	CHEMBL3652226	ChEMBL	8.3	—	—	O=C(NO)c1cnc(Nc2ccc(Cl)c(Cl)c2)nc1
E3 Binder	CHEMBL3652230	ChEMBL	7.7	—	—	O=C(NO)c1cnc(Nc2ccc(Cl)cc2)nc1
E3 Binder	CHEMBL3652227	ChEMBL	8.1	—	—	O=C(NO)c1cnc(Nc2ccc(F)cc2)nc1
E3 Binder	CHEMBL3652233	ChEMBL	8.0	—	—	O=C(NO)c1cnc(Nc2ccc([N+](=O)[O-])c(C(F)(F)F)c2)nc1
E3 Binder	CHEMBL3655911	ChEMBL	8.4	—	—	O=C(NO)c1cnc(Nc2cccc(-c3ccccc3)c2)nc1
E3 Binder	CHEMBL3655913	ChEMBL	8.52	—	—	O=C(NO)c1cnc(Nc2cccc(-c3ccncc3)c2)nc1
E3 Binder	CHEMBL3652242	ChEMBL	8.52	—	—	O=C(NO)c1cnc(Nc2cccc(C(F)(F)F)c2)nc1
E3 Binder	CHEMBL3652237	ChEMBL	8.3	—	—	O=C(NO)c1cnc(Nc2cccc(Cl)c2)nc1
E3 Binder	CHEMBL3655912	ChEMBL	8.1	—	—	O=C(NO)c1cnc(Nc2cccc(N3CCOCC3)c2)nc1
E3 Binder	CHEMBL3652225	ChEMBL	8.15	—	—	O=C(NO)c1cnc(Nc2ccccc2)nc1
E3 Binder	CHEMBL3652231	ChEMBL	7.38	—	—	O=C(NO)c1cnc(Nc2ccccc2Cl)nc1
E3 Binder	CHEMBL3771326	ChEMBL	7.05	—	—	O=C(NO)c1coc(-c2ccc(-c3ccccc3)cc2)n1
E3 Binder	CHEMBL3770095	ChEMBL	7.23	P7V	—	O=C(NO)c1coc(-c2ccc(Br)cc2)n1
E3 Binder	CHEMBL3771189	ChEMBL	7.09	—	—	O=C(NO)c1coc(-c2ccc(Cl)cc2)n1
E3 Binder	CHEMBL3770763	ChEMBL	6.96	—	—	O=C(NO)c1coc(-c2ccc(F)cc2)n1
E3 Binder	CHEMBL3769820	ChEMBL	7.05	—	—	O=C(NO)c1coc(-c2ccc3ccccc3c2)n1
E3 Binder	CHEMBL3771355	ChEMBL	6.3	—	—	O=C(NO)c1coc(-c2cccc(-c3ccccc3)c2)n1
E3 Binder	CHEMBL3769783	ChEMBL	6.57	—	—	O=C(NO)c1coc(-c2ccccc2)n1
E3 Binder	CHEMBL3770566	ChEMBL	6.51	—	—	O=C(NO)c1coc(-c2cccs2)n1
E3 Binder	CHEMBL4874713	ChEMBL	6.05	—	—	O=C(NO)c1coc(CN2c3ccccc3Sc3ccccc32)n1
E3 Binder	CHEMBL3771312	ChEMBL	6.52	—	—	O=C(NO)c1csc(-c2cccnc2)n1
E3 Binder	CHEMBL3770180	ChEMBL	6.95	—	—	O=C(NO)c1noc(-c2ccccc2)n1
E3 Binder	CHEMBL449493	ChEMBL	6.5	—	—	O=C(N[C@@H](CCCCCB(O)O)C(=O)Nc1cccc(-c2ccccc2)c1)c1cccnc1
E3 Binder	CHEMBL492097	ChEMBL	6.96	—	—	O=C(N[C@@H](CCCCCB(O)O)C(=O)Nc1cccc(-c2ccccc2)c1)c1cncs1
E3 Binder	CHEMBL3187798	ChEMBL	6.73	—	—	O=C(Nc1cc2cc[nH]c2cn1)c1ccccc1
E3 Binder	CHEMBL2046610	ChEMBL	6.92	—	—	O=C(Nc1ccc(C(=O)N2CCc3nc(C(=O)NO)sc3C2)cc1)c1ccc(-c2ccccc2)s1
E3 Binder	CHEMBL4793248	ChEMBL	7.68	—	—	O=C(Nc1ccc(Cl)cc1)Nc1ccc(C(=O)NO)cc1
E3 Binder	CHEMBL239767	ChEMBL	6.21	—	—	O=C(Nc1ccc([N+](=O)[O-])cc1O)Nc1ccccc1Br
E3 Binder	CHEMBL5078716	ChEMBL	6.08	—	—	O=C(Nc1ccc2c(c1)CCN2c1ccc(C(=O)NO)cc1)Nc1ccc(Cl)c(C(F)(F)F)c1
E3 Binder	CHEMBL5086690	ChEMBL	6.6	—	—	O=C(Nc1ccc2c(c1)N(Cc1ccc(C(=O)NO)cc1)CC2)Nc1ccc(Cl)c(C(F)(F)F)c1
E3 Binder	CHEMBL556667	ChEMBL	6.48	BK0	—	O=C(Nc1cccc(Cl)c1)c1ccccn1
E3 Binder	CHEMBL27246	ChEMBL	8.09	TCA	—	O=C(O)/C=C/c1ccccc1
E3 Binder	CHEMBL150237	ChEMBL	8.7	—	—	O=C(O)C(=O)NCCSSCCNC(=O)/C(Cc1ccc(O)c(Br)c1)=N/O
E3 Binder	CHEMBL2036480	ChEMBL	6.85	—	—	O=C(O)CC(c1nc2ccccc2o1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL2036481	ChEMBL	6.48	—	—	O=C(O)CCC(c1nc2ccccc2o1)n1cc(/C=C/C(=O)NO)nn1
E3 Binder	CHEMBL3589364	ChEMBL	6.19	—	—	O=C(O)CCCCCCC(=O)Nc1ccc(C2=C(c3ccc(O)cc3)C3CC(S(=O)(=O)Oc4ccc(C(F)(F)F)cc4)C2O3)cc1
E3 Binder	CHEMBL3589357	ChEMBL	7.15	—	—	O=C(O)CCCCCCC(=O)Nc1ccc(C2=C(c3ccc(O)cc3)C3CC(S(=O)(=O)Oc4cccc(O)c4)C2O3)cc1
E3 Binder	CHEMBL162423	ChEMBL	6.57	—	—	O=C(O)CCCCCCC(=O)c1ccccc1
E3 Binder	CHEMBL565289	ChEMBL	6.0	—	—	O=C(O)CCCCC[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)C[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2cccc3ccccc23)NC1=O
E3 Binder	CHEMBL565304	ChEMBL	6.1	—	—	O=C(O)CCCCC[C@@H]1NC(=O)[C@H]2CCCCN2C(=O)C[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC1=O
E3 Binder	CHEMBL3758354	ChEMBL	7.1	—	—	O=C(O)CCCn1nc(-c2ccc(F)cc2)cc1C(=O)NCCCCCCS
E3 Binder	CHEMBL3758311	ChEMBL	6.35	—	—	O=C(O)CCCn1nc(C(=O)NCCCCCCS)cc1-c1ccc(F)cc1
E3 Binder	CHEMBL3759543	ChEMBL	6.68	—	—	O=C(O)CCn1nc(-c2ccc(F)cc2)cc1C(=O)NCCCCCCS
E3 Binder	CHEMBL3758912	ChEMBL	6.48	—	—	O=C(O)CCn1nc(C(=O)NCCCCCCS)cc1-c1ccc(F)cc1
E3 Binder	CHEMBL3759067	ChEMBL	7.4	—	—	O=C(O)Cn1nc(-c2ccc(F)cc2)cc1C(=O)NCCCCCCS
E3 Binder	CHEMBL3758778	ChEMBL	6.6	—	—	O=C(O)Cn1nc(C(=O)NCCCCCCS)cc1-c1ccc(F)cc1
E3 Binder	CHEMBL88712	ChEMBL	6.18	QY1	—	O=C(O)[C@@H](c1ccc(OCc2ccc3ccccc3n2)cc1)C1CCCC1
E3 Binder	CHEMBL569192	ChEMBL	7.57	—	—	O=C(O)c1ccc(-c2ccc(C(=O)C(F)(F)F)s2)cc1
E3 Binder	CHEMBL569193	ChEMBL	7.16	—	—	O=C(O)c1cccc(-c2ccc(C(=O)C(F)(F)F)s2)c1
E3 Binder	CHEMBL4559028	ChEMBL	7.92	—	—	O=C(O)c1cccc(-c2nnn(Cc3ccc(C(=O)NO)cc3)n2)c1
E3 Binder	CHEMBL256997	ChEMBL	6.52	JBF	—	O=C(O)c1cccc(-c2noc(-c3ccccc3F)n2)c1
E3 Binder	CHEMBL3617543	ChEMBL	6.82	WAF	—	O=C(O)c1cccc(=S)n1O
E3 Binder	CHEMBL1170610	ChEMBL	6.03	—	—	O=C(Oc1cccc2cccnc12)c1ccccc1
E3 Binder	CHEMBL566092	ChEMBL	7.43	—	—	O=C(c1ccc(-c2ccc3c(c2)OCCO3)s1)C(F)(F)F
E3 Binder	CHEMBL571505	ChEMBL	7.82	—	—	O=C(c1ccc(-c2ccc3nccnc3c2)s1)C(F)(F)F
E3 Binder	CHEMBL585554	ChEMBL	6.77	—	—	O=C(c1ccc(-c2ccccc2)s1)C(F)(F)F
E3 Binder	CHEMBL450362	ChEMBL	6.57	—	—	O=C(c1ccc(-c2nc(-c3ccc(F)cc3)no2)s1)C(F)(F)F
E3 Binder	CHEMBL460088	ChEMBL	6.24	—	—	O=C(c1ccc(-c2nc(-c3ccc(F)cc3F)no2)s1)C(F)(F)F
E3 Binder	CHEMBL462210	ChEMBL	6.24	—	—	O=C(c1ccc(-c2nc(-c3ccccc3)no2)s1)C(F)(F)F
E3 Binder	CHEMBL512043	ChEMBL	6.3	—	—	O=C(c1ccc(-c2nc(-c3ccccn3)no2)s1)C(F)(F)F
E3 Binder	CHEMBL462370	ChEMBL	6.08	—	—	O=C(c1ccc(-c2nc(-c3cccnc3)no2)s1)C(F)(F)F
E3 Binder	CHEMBL454671	ChEMBL	6.17	—	—	O=C(c1ccc(-c2nc(-c3cccs3)no2)s1)C(F)(F)F
E3 Binder	CHEMBL461333	ChEMBL	6.24	—	—	O=C(c1ccc(-c2nc(-c3ccncc3)no2)s1)C(F)(F)F
E3 Binder	CHEMBL518821	ChEMBL	6.55	—	—	O=C(c1ccc(-c2nc(COc3ccc(-c4nnco4)cc3)no2)s1)C(F)(F)F
E3 Binder	CHEMBL512517	ChEMBL	6.16	—	—	O=C(c1ccc(-c2nc(CS(=O)(=O)Cc3ccc(F)cc3)no2)s1)C(F)(F)F
E3 Binder	CHEMBL471174	ChEMBL	6.28	—	—	O=C(c1ccc(-c2nc(CS(=O)(=O)c3cccs3)no2)s1)C(F)(F)F
E3 Binder	CHEMBL504161	ChEMBL	6.77	—	—	O=C(c1ccc(-c2nc(Cc3cccs3)no2)s1)C(F)(F)F
E3 Binder	CHEMBL462223	ChEMBL	6.48	—	—	O=C(c1ccc(-c2nnc(-c3ccccc3)o2)s1)C(F)(F)F
E3 Binder	CHEMBL454672	ChEMBL	6.8	—	—	O=C(c1ccc(-c2nnc(-c3cccs3)o2)s1)C(F)(F)F
E3 Binder	CHEMBL493784	ChEMBL	6.24	—	—	O=C(c1ccc(C(=O)C(F)(F)F)[nH]1)N1CCc2ccccc21
E3 Binder	CHEMBL485771	ChEMBL	6.8	—	—	O=C(c1ccc(C(=O)C(F)(F)F)s1)N1CCC(c2nnc(-c3ccccc3)o2)CC1
E3 Binder	CHEMBL525529	ChEMBL	6.89	—	—	O=C(c1ccc(C(=O)C(F)(F)F)s1)N1CCc2ccccc21
E3 Binder	CHEMBL496094	ChEMBL	6.51	—	—	O=C(c1ccc(C(=O)C(F)(F)F)s1)N1CCn2c(-c3ccccc3)cnc2C1
E3 Binder	CHEMBL497760	ChEMBL	7.82	—	—	O=C(c1ccc(C(=O)N2CCc3ccccc32)s1)C(F)F
E3 Binder	CHEMBL574365	ChEMBL	6.68	—	—	O=C(c1cnc(-c2ccccc2)s1)C(F)(F)F
E3 Binder	CHEMBL487347	ChEMBL	6.39	—	—	O=C(c1ncc(C(=O)C(F)(F)F)s1)N1CCc2ccccc21
E3 Binder	CHEMBL3356939	ChEMBL	6.24	—	—	O=C1CCC[C@@H](C(=O)N[C@@H](CCCCCS)C(=O)N2CCc3ccccc3C2)N1
E3 Binder	CHEMBL3356931	ChEMBL	8.22	—	—	O=C1CCC[C@@H](C(=O)N[C@@H](CCCCCS)C(=O)NC2CCCC2)N1
E3 Binder	CHEMBL3356933	ChEMBL	6.86	—	—	O=C1CCC[C@@H](C(=O)N[C@@H](CCCCCS)C(=O)NCc2ccc(C(F)(F)F)cc2)N1
E3 Binder	CHEMBL3356935	ChEMBL	7.08	—	—	O=C1CCC[C@@H](C(=O)N[C@@H](CCCCCS)C(=O)NCc2cccc(OCc3ccccc3)c2)N1
E3 Binder	CHEMBL3356523	ChEMBL	8.22	—	—	O=C1CCC[C@@H](C(=O)N[C@@H](CCCCCS)C(=O)Nc2ccccc2)N1
E3 Binder	CHEMBL3356524	ChEMBL	8.3	—	—	O=C1CCC[C@H](C(=O)N[C@@H](CCCCCS)C(=O)Nc2ccccc2)N1
E3 Binder	CHEMBL3356918	ChEMBL	9.0	—	—	O=C1CC[C@@H](C(=O)N[C@@H](CCCCCS)C(=O)Nc2ccccc2)N1
E3 Binder	CHEMBL3356919	ChEMBL	8.52	—	—	O=C1CC[C@@H](C(=O)N[C@H](CCCCCS)C(=O)Nc2ccccc2)N1
E3 Binder	CHEMBL3353927	ChEMBL	8.3	—	—	O=C1CC[C@H](C(=O)N[C@@H](CCCCCS)C(=O)Nc2cccc(C(F)(F)F)c2)N1
E3 Binder	CHEMBL3353925	ChEMBL	8.52	—	—	O=C1CC[C@H](C(=O)N[C@@H](CCCCCS)C(=O)Nc2ccccc2)N1
E3 Binder	CHEMBL3356920	ChEMBL	7.68	—	—	O=C1CC[C@H](C(=O)N[C@H](CCCCCS)C(=O)Nc2ccccc2)N1
E3 Binder	CHEMBL5268638	ChEMBL	9.14	—	—	O=C1CN(Cc2ccc(C(=O)NO)cc2)C(=O)[C@@H](Cc2c[nH]c3ccccc23)N1
E3 Binder	CHEMBL5273674	ChEMBL	8.06	—	—	O=C1CN(Cc2ccc(C(=O)NO)cc2)C(=O)[C@@H](Cc2ccccc2)N1
E3 Binder	CHEMBL5270958	ChEMBL	8.18	—	—	O=C1CN(Cc2ccc(C(=O)NO)cc2)C(=O)[C@H](Cc2c[nH]c3ccccc23)N1
E3 Binder	CHEMBL5273465	ChEMBL	7.76	—	—	O=C1CN(Cc2ccc(C(=O)NO)cc2)C(=O)[C@H](Cc2ccccc2)N1
E3 Binder	CHEMBL481802	ChEMBL	6.82	—	—	O=C1CN(Cc2ccc(C(=O)NO)cc2)c2ccccc2N1
E3 Binder	CHEMBL462203	ChEMBL	6.39	—	—	O=C1COc2ccccc2N1Cc1noc(-c2ccc(C(=O)C(F)(F)F)s2)n1
E3 Binder	CHEMBL3356929	ChEMBL	8.7	—	—	O=C1C[C@@H](C(=O)N[C@@H](CCCCCS)C(=O)Nc2ccccc2)N1
E3 Binder	CHEMBL3356915	ChEMBL	9.0	—	—	O=C1NCCC[C@@H]1C(=O)N[C@@H](CCCCCS)C(=O)Nc1ccccc1
E3 Binder	CHEMBL3356527	ChEMBL	9.0	—	—	O=C1NCCC[C@H]1C(=O)N[C@@H](CCCCCS)C(=O)Nc1ccccc1
E3 Binder	CHEMBL3356925	ChEMBL	8.4	—	—	O=C1NC[C@@H](c2ccccc2)[C@@H]1C(=O)N[C@@H](CCCCCS)C(=O)Nc1ccccc1
E3 Binder	CHEMBL3356928	ChEMBL	7.46	—	—	O=C1NC[C@@H](c2ccccc2)[C@H]1C(=O)N[C@@H](CCCCCS)C(=O)Nc1ccccc1
E3 Binder	CHEMBL3356927	ChEMBL	8.4	—	—	O=C1NC[C@H](c2ccccc2)[C@@H]1C(=O)N[C@@H](CCCCCS)C(=O)Nc1ccccc1
E3 Binder	CHEMBL3356926	ChEMBL	6.8	—	—	O=C1NC[C@H](c2ccccc2)[C@H]1C(=O)N[C@@H](CCCCCS)C(=O)Nc1ccccc1
E3 Binder	CHEMBL2158742	ChEMBL	6.48	—	—	O=C1N[C@@H]2CCOCCSSCCCCC[C@@H]1NC(=O)[C@H]1CCCN1C(=O)[C@H](Cc1ccccc1)NC2=O
E3 Binder	CHEMBL409450	ChEMBL	6.16	BRW	—	O=C1Nc2cc(Br)ccc2/C1=C1/Nc2ccccc2/C1=N\O
E3 Binder	CHEMBL216543	ChEMBL	6.42	—	—	O=C1Nc2ccccc2/C1=C1/Nc2ccccc2/C1=N\O
E3 Binder	CHEMBL336935	ChEMBL	6.21	—	—	O=CN(O)CCCCCC(C(=O)Nc1ccc2ncccc2c1)C(=O)Nc1ccc2ncccc2c1
E3 Binder	CHEMBL140525	ChEMBL	6.11	—	—	O=CN(O)CCCCCC(C(=O)Nc1cnc2ccccc2c1)C(=O)Nc1cnc2ccccc2c1
E3 Binder	CHEMBL141909	ChEMBL	6.04	—	—	O=CN(O)CCCCCCCC(=O)Nc1ccc2ccccc2c1
E3 Binder	CHEMBL343717	ChEMBL	6.22	—	—	O=CN(O)CCCCCNC(=O)c1ccc2ccccc2c1
E3 Binder	CHEMBL5202641	ChEMBL	7.85	—	—	O=S(=O)(N1CCN(C2COC2)CC1)N(Cc1ccc(-c2nnc(C(F)(F)F)o2)cn1)c1ccc(F)c(Cl)c1
E3 Binder	CHEMBL5198435	ChEMBL	7.36	—	—	O=S(=O)(N1CCNCC1)N(Cc1ccc(-c2nnc(C(F)(F)F)o2)cc1F)c1cccnc1
E3 Binder	CHEMBL3692643	ChEMBL	6.36	—	—	O=S(=O)(Nc1ccc(F)cc1)c1ccc(-c2noc(C(F)(F)F)n2)cc1
E3 Binder	CHEMBL3692641	ChEMBL	6.34	—	—	O=S(=O)(Nc1cccc(Cl)c1)c1ccc(-c2noc(C(F)(F)F)n2)cc1
E3 Binder	CHEMBL3692630	ChEMBL	6.4	—	—	O=S(=O)(Nc1ccccc1)c1ccc(-c2noc(C(F)(F)F)n2)cc1
E3 Binder	CHEMBL3692638	ChEMBL	6.11	—	—	O=S(=O)(Nc1ccccc1Cl)c1ccc(-c2noc(C(F)(F)F)n2)cc1
E3 Binder	CHEMBL3692645	ChEMBL	6.24	—	—	O=S(=O)(Nc1ccccc1F)c1ccc(-c2noc(C(F)(F)F)n2)cc1
E3 Binder	CHEMBL8145	ChEMBL	6.04	ZF1	—	O=c1c(-c2ccc(O)cc2)coc2cc(O)ccc12
E3 Binder	CHEMBL50	ChEMBL	6.09	QUE	—	O=c1c(O)c(-c2ccc(O)c(O)c2)oc2cc(O)cc(O)c12
E3 Binder	CHEMBL2408237	ChEMBL	6.28	—	—	O=c1c(O)ccccc1-c1ccccc1
E3 Binder	CHEMBL85139	ChEMBL	6.14	—	—	O=c1c2ccccc2nc2n1CCc1c-2[nH]c2ccccc12
E3 Binder	CHEMBL117	ChEMBL	6.27	57D	—	O=c1cc(-c2ccccc2)oc2cc(O)cc(O)c12
E3 Binder	CHEMBL3545157	ChEMBL	6.0	—	—	O=c1sn(-c2cccc3ccccc23)c(=O)n1Cc1ccccc1
E3 Binder	CHEMBL1555354	ChEMBL	6.25	—	—	OCc1ccc(-c2ccc(-c3ccc(CO)s3)o2)s1
E3 Binder	CHEMBL69863	ChEMBL	6.05	PIT	—	Oc1cc(O)cc(/C=C/c2ccc(O)c(O)c2)c1
E3 Binder	CHEMBL402341	ChEMBL	6.35	—	—	Oc1ccc(-c2cc(=S)ss2)cc1
E3 Binder	CHEMBL188528	ChEMBL	6.07	—	—	Oc1ccc(-c2nc3cc(O)cc(Br)c3o2)cc1
E3 Binder	CHEMBL1388	ChEMBL	6.0	—	—	Oc1ccc(OCc2ccccc2)cc1
E3 Binder	CHEMBL2337874	ChEMBL	6.17	—	—	Oc1ccc[nH]c1=S
E3 Binder	CHEMBL3110276	ChEMBL	6.02	—	—	Oc1cccn(CCCCCCCn2cc(-c3ccccc3)nn2)c1=S
E3 Binder	CHEMBL3110287	ChEMBL	6.04	—	—	Oc1cccn(CCCCCn2cc(-c3ccccc3)nn2)c1=S
E3 Binder	CHEMBL2337873	ChEMBL	6.07	—	—	Oc1cccn(Cc2ccc(-c3ccccc3)cc2)c1=S
E3 Binder	CHEMBL3657470	ChEMBL	6.27	—	—	Oc1cccn(Cc2ccc(Cn3cc(-c4ccccc4)nn3)cc2)c1=S
E3 Binder	CHEMBL2337875	ChEMBL	6.34	—	—	Oc1cccn(Cc2ccccc2)c1=S
E3 Binder	CHEMBL5288006	ChEMBL	8.8	—	—	[11CH3]n1cc(CCNCc2ccc(/C=C/C(=O)NO)cc2)c2ccccc21
E3 Binder	CHEMBL244830	ChEMBL	6.3	—	—	[C-]#[N+]c1ccc(C(=O)CSC(=S)SCC)cc1
E3 Binder	CHEMBL3657469	ChEMBL	6.43	—	—	[C-]#[N+]c1ccccc1-c1ccc(Cn2cccc(O)c2=S)cc1
E3 Binder	CHEMBL1914708	ChEMBL	6.56	—	—	[N-]=[N+]=NCc1cc(Cn2cc(NC(=O)CCCCCCC(=O)NO)cn2)cc(N=[N+]=[N-])c1
E3 Binder	CHEMBL1914702	ChEMBL	7.33	—	—	[N-]=[N+]=NCc1cc(N=[N+]=[N-])cc(C(=O)Nc2ccc(-c3cc(C(=O)NCCCCCCC(=O)NO)no3)cc2)c1
E3 Binder	CHEMBL270224	ChEMBL	7.01	—	—	[N-]=[N+]=Nc1ccc(C(=O)NC(CCCCNC(=O)CCCCC2SCC3NC(=O)NC32)C(=O)NCCSSCCC(=O)NCCCCCCN(CCc2c[nH]c3ccccc23)Cc2ccc(/C=C/C(=O)NO)cc2)cc1
E3 Binder	CHEMBL625	ChEMBL	6.44	—	—	c1ccc2[nH]c(-c3cscn3)nc2c1